Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Acetylcholine receptor protein epsilon chain (Rattus norvegicus) | BDBM50524696![]() (CHEMBL4571835) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Zhejiang Academy of Medical Sciences Curated by ChEMBL | Assay Description Inhibition of rat brain cortex AChE using acetylthiocholine iodide as substrate incubated for 15 mins by spectrophotometry | Eur J Med Chem 177: 247-258 (2019) Article DOI: 10.1016/j.ejmech.2019.05.051 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine receptor protein epsilon chain (Rattus norvegicus) | BDBM50524701![]() (CHEMBL4594074) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Zhejiang Academy of Medical Sciences Curated by ChEMBL | Assay Description Inhibition of rat brain cortex AChE using acetylthiocholine iodide as substrate incubated for 15 mins by spectrophotometry | Eur J Med Chem 177: 247-258 (2019) Article DOI: 10.1016/j.ejmech.2019.05.051 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine receptor protein epsilon chain (Rattus norvegicus) | BDBM50524708![]() (CHEMBL4459614) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8.80 | n/a | n/a | n/a | n/a | n/a | n/a |
Zhejiang Academy of Medical Sciences Curated by ChEMBL | Assay Description Inhibition of rat brain cortex AChE using acetylthiocholine iodide as substrate incubated for 15 mins by spectrophotometry | Eur J Med Chem 177: 247-258 (2019) Article DOI: 10.1016/j.ejmech.2019.05.051 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine receptor protein epsilon chain (Rattus norvegicus) | BDBM11682![]() (2,3-dihydroxybutanedioic acid; 3-[(1S)-1-(dimethyl...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | Purchase DrugBank KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9 | n/a | n/a | n/a | n/a | n/a | n/a |
Zhejiang Academy of Medical Sciences Curated by ChEMBL | Assay Description Inhibition of rat brain cortex AChE using acetylthiocholine iodide as substrate incubated for 15 mins by spectrophotometry | Eur J Med Chem 177: 247-258 (2019) Article DOI: 10.1016/j.ejmech.2019.05.051 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine receptor protein epsilon chain (Rattus norvegicus) | BDBM50524697![]() (CHEMBL4470950) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
Zhejiang Academy of Medical Sciences Curated by ChEMBL | Assay Description Inhibition of rat brain cortex AChE using acetylthiocholine iodide as substrate incubated for 15 mins by spectrophotometry | Eur J Med Chem 177: 247-258 (2019) Article DOI: 10.1016/j.ejmech.2019.05.051 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine receptor protein epsilon chain (Rattus norvegicus) | BDBM50524707![]() (CHEMBL4468053) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | n/a |
Zhejiang Academy of Medical Sciences Curated by ChEMBL | Assay Description Inhibition of rat brain cortex AChE using acetylthiocholine iodide as substrate incubated for 15 mins by spectrophotometry | Eur J Med Chem 177: 247-258 (2019) Article DOI: 10.1016/j.ejmech.2019.05.051 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine receptor protein epsilon chain (Rattus norvegicus) | BDBM50524705![]() (CHEMBL4452617) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
Zhejiang Academy of Medical Sciences Curated by ChEMBL | Assay Description Inhibition of rat brain cortex AChE using acetylthiocholine iodide as substrate incubated for 15 mins by spectrophotometry | Eur J Med Chem 177: 247-258 (2019) Article DOI: 10.1016/j.ejmech.2019.05.051 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine receptor protein epsilon chain (Rattus norvegicus) | BDBM50524698![]() (CHEMBL4452986) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 21 | n/a | n/a | n/a | n/a | n/a | n/a |
Zhejiang Academy of Medical Sciences Curated by ChEMBL | Assay Description Inhibition of rat brain cortex AChE using acetylthiocholine iodide as substrate incubated for 15 mins by spectrophotometry | Eur J Med Chem 177: 247-258 (2019) Article DOI: 10.1016/j.ejmech.2019.05.051 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine receptor protein epsilon chain (Rattus norvegicus) | BDBM50524706![]() (CHEMBL4566337) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 29 | n/a | n/a | n/a | n/a | n/a | n/a |
Zhejiang Academy of Medical Sciences Curated by ChEMBL | Assay Description Inhibition of rat brain cortex AChE using acetylthiocholine iodide as substrate incubated for 15 mins by spectrophotometry | Eur J Med Chem 177: 247-258 (2019) Article DOI: 10.1016/j.ejmech.2019.05.051 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine receptor protein epsilon chain (Rattus norvegicus) | BDBM50524703![]() (CHEMBL4443818) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 29 | n/a | n/a | n/a | n/a | n/a | n/a |
Zhejiang Academy of Medical Sciences Curated by ChEMBL | Assay Description Inhibition of rat brain cortex AChE using acetylthiocholine iodide as substrate incubated for 15 mins by spectrophotometry | Eur J Med Chem 177: 247-258 (2019) Article DOI: 10.1016/j.ejmech.2019.05.051 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine receptor protein epsilon chain (Rattus norvegicus) | BDBM50524709![]() (CHEMBL4471688) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 41 | n/a | n/a | n/a | n/a | n/a | n/a |
Zhejiang Academy of Medical Sciences Curated by ChEMBL | Assay Description Inhibition of rat brain cortex AChE using acetylthiocholine iodide as substrate incubated for 15 mins by spectrophotometry | Eur J Med Chem 177: 247-258 (2019) Article DOI: 10.1016/j.ejmech.2019.05.051 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine receptor protein epsilon chain (Rattus norvegicus) | BDBM50524702![]() (CHEMBL4517494) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 41 | n/a | n/a | n/a | n/a | n/a | n/a |
Zhejiang Academy of Medical Sciences Curated by ChEMBL | Assay Description Inhibition of rat brain cortex AChE using acetylthiocholine iodide as substrate incubated for 15 mins by spectrophotometry | Eur J Med Chem 177: 247-258 (2019) Article DOI: 10.1016/j.ejmech.2019.05.051 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine receptor protein epsilon chain (Rattus norvegicus) | BDBM50524700![]() (CHEMBL4535921) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 49 | n/a | n/a | n/a | n/a | n/a | n/a |
Zhejiang Academy of Medical Sciences Curated by ChEMBL | Assay Description Inhibition of rat brain cortex AChE using acetylthiocholine iodide as substrate incubated for 15 mins by spectrophotometry | Eur J Med Chem 177: 247-258 (2019) Article DOI: 10.1016/j.ejmech.2019.05.051 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine receptor protein epsilon chain (Rattus norvegicus) | BDBM50524704![]() (CHEMBL4446271) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 55 | n/a | n/a | n/a | n/a | n/a | n/a |
Zhejiang Academy of Medical Sciences Curated by ChEMBL | Assay Description Inhibition of rat brain cortex AChE using acetylthiocholine iodide as substrate incubated for 15 mins by spectrophotometry | Eur J Med Chem 177: 247-258 (2019) Article DOI: 10.1016/j.ejmech.2019.05.051 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine receptor protein epsilon chain (Rattus norvegicus) | BDBM50524699![]() (CHEMBL4557064) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 70 | n/a | n/a | n/a | n/a | n/a | n/a |
Zhejiang Academy of Medical Sciences Curated by ChEMBL | Assay Description Inhibition of rat brain cortex AChE using acetylthiocholine iodide as substrate incubated for 15 mins by spectrophotometry | Eur J Med Chem 177: 247-258 (2019) Article DOI: 10.1016/j.ejmech.2019.05.051 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine receptor protein epsilon chain (Rattus norvegicus) | BDBM50448370![]() (CHEMBL3120178) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.94E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Milano Curated by ChEMBL | Assay Description Inhibition of acetylcholinesterase in rat brain homogenate after 15 mins by Ellman assay | Eur J Med Chem 75: 222-32 (2014) Article DOI: 10.1016/j.ejmech.2014.01.032 BindingDB Entry DOI: 10.7270/Q2K075RG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine receptor protein epsilon chain (Rattus norvegicus) | BDBM50448375![]() (CHEMBL3121479) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Milano Curated by ChEMBL | Assay Description Inhibition of acetylcholinesterase in rat brain homogenate after 15 mins by Ellman assay | Eur J Med Chem 75: 222-32 (2014) Article DOI: 10.1016/j.ejmech.2014.01.032 BindingDB Entry DOI: 10.7270/Q2K075RG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine receptor protein epsilon chain (Rattus norvegicus) | BDBM50448374![]() (CHEMBL3121478) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.02E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Milano Curated by ChEMBL | Assay Description Inhibition of acetylcholinesterase in rat brain homogenate after 15 mins by Ellman assay | Eur J Med Chem 75: 222-32 (2014) Article DOI: 10.1016/j.ejmech.2014.01.032 BindingDB Entry DOI: 10.7270/Q2K075RG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine receptor protein epsilon chain (Rattus norvegicus) | BDBM50448369![]() (CHEMBL3121476) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.95E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Milano Curated by ChEMBL | Assay Description Inhibition of acetylcholinesterase in rat brain homogenate after 15 mins by Ellman assay | Eur J Med Chem 75: 222-32 (2014) Article DOI: 10.1016/j.ejmech.2014.01.032 BindingDB Entry DOI: 10.7270/Q2K075RG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine receptor protein epsilon chain (Rattus norvegicus) | BDBM50448371![]() (CHEMBL3121480) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.29E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Milano Curated by ChEMBL | Assay Description Inhibition of acetylcholinesterase in rat brain homogenate after 15 mins by Ellman assay | Eur J Med Chem 75: 222-32 (2014) Article DOI: 10.1016/j.ejmech.2014.01.032 BindingDB Entry DOI: 10.7270/Q2K075RG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine receptor protein epsilon chain (Rattus norvegicus) | BDBM50448372![]() (CHEMBL3121475) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.16E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Milano Curated by ChEMBL | Assay Description Inhibition of acetylcholinesterase in rat brain homogenate after 15 mins by Ellman assay | Eur J Med Chem 75: 222-32 (2014) Article DOI: 10.1016/j.ejmech.2014.01.032 BindingDB Entry DOI: 10.7270/Q2K075RG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine receptor protein epsilon chain (Rattus norvegicus) | BDBM50448376![]() (NAPHMETHONIUM | Naphmethonium) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.17E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Milano Curated by ChEMBL | Assay Description Inhibition of acetylcholinesterase in rat brain homogenate after 15 mins by Ellman assay | Eur J Med Chem 75: 222-32 (2014) Article DOI: 10.1016/j.ejmech.2014.01.032 BindingDB Entry DOI: 10.7270/Q2K075RG | |||||||||||
More data for this Ligand-Target Pair |