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Found 29 hits Enz. Inhib. hit(s) with Target = 'Arachidonate 12-lipoxygenase' AND taxid = 10090   
Target
(Institution)
LigandTarget
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Arachidonate 12-lipoxygenase


(Mus musculus)
BDBM50447175
PNG
(CHEMBL3113165)
Show SMILES COc1cccc(CNc2ccc(cc2)S(=O)(=O)Nc2nc3ccccc3s2)c1O
Show InChI InChI=1S/C21H19N3O4S2/c1-28-18-7-4-5-14(20(18)25)13-22-15-9-11-16(12-10-15)30(26,27)24-21-23-17-6-2-3-8-19(17)29-21/h2-12,22,25H,13H2,1H3,(H,23,24)
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n/an/a 1.00E+3n/an/an/an/an/an/a



National Institutes of Health

Curated by ChEMBL


Assay Description
Inhibition of 12-LOX in mouse BTC3 cells assessed as inhibition of arachidonic acid/calcium ionophore-induced 12-HETE production after 4 hrs by ELISA


Citation and Details
More data for this
Ligand-Target Pair
Arachidonate 12-lipoxygenase


(Mus musculus)
BDBM50052450
PNG
(1,8-Dihydroxy-10-(2-methoxy-phenylsulfanyl)-10H-an...)
Show SMILES COc1ccccc1SC1c2cccc(O)c2C(=O)c2c(O)cccc12
Show InChI InChI=1S/C21H16O4S/c1-25-16-10-2-3-11-17(16)26-21-12-6-4-8-14(22)18(12)20(24)19-13(21)7-5-9-15(19)23/h2-11,21-23H,1H3
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n/an/a 3.00E+3n/an/an/an/an/an/a



Universität Regensburg

Curated by ChEMBL


Assay Description
Tested for inhibition of 12-LO (12-lipoxygenase) as an inhibitor of 12(S)-HETE biosynthesis in mouse epidermal homogenates


Citation and Details
More data for this
Ligand-Target Pair
Arachidonate 12-lipoxygenase


(Mus musculus)
BDBM50052464
PNG
(1,8-Dihydroxy-10-(4-hydroxy-phenylsulfanyl)-10H-an...)
Show SMILES Oc1ccc(SC2c3cccc(O)c3C(=O)c3c(O)cccc23)cc1
Show InChI InChI=1S/C20H14O4S/c21-11-7-9-12(10-8-11)25-20-13-3-1-5-15(22)17(13)19(24)18-14(20)4-2-6-16(18)23/h1-10,20-23H
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n/an/a 3.00E+3n/an/an/an/an/an/a



Universität Regensburg

Curated by ChEMBL


Assay Description
Tested for inhibition of 12-LO (12-lipoxygenase) as an inhibitor of 12(S)-HETE biosynthesis in mouse epidermal homogenates


Citation and Details
More data for this
Ligand-Target Pair
Arachidonate 12-lipoxygenase


(Mus musculus)
BDBM50052462
PNG
(10-(2-Amino-phenylsulfanyl)-1,8-dihydroxy-10H-anth...)
Show SMILES Nc1ccccc1SC1c2cccc(O)c2C(=O)c2c(O)cccc12
Show InChI InChI=1S/C20H15NO3S/c21-13-7-1-2-10-16(13)25-20-11-5-3-8-14(22)17(11)19(24)18-12(20)6-4-9-15(18)23/h1-10,20,22-23H,21H2
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n/an/a 6.00E+3n/an/an/an/an/an/a



Universität Regensburg

Curated by ChEMBL


Assay Description
Tested for inhibition of 12-LO (12-lipoxygenase) as an inhibitor of 12(S)-HETE biosynthesis in mouse epidermal homogenates


Citation and Details
More data for this
Ligand-Target Pair
Arachidonate 12-lipoxygenase


(Mus musculus)
BDBM50350396
PNG
(CHEMBL1573436)
Show SMILES CC(=O)NC(c1cccs1)c1cc(Br)c2cccnc2c1O
Show InChI InChI=1S/C16H13BrN2O2S/c1-9(20)19-14(13-5-3-7-22-13)11-8-12(17)10-4-2-6-18-15(10)16(11)21/h2-8,14,21H,1H3,(H,19,20)
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n/an/a 1.40E+4n/an/an/an/an/an/a



National Human Genome Research Institute

Curated by ChEMBL


Assay Description
Inhibition of mouse N-terminally His6-tagged 12-lipoxygenase expressed in SF9 insect cells assessed as 12-HPETE formation using arachidonic acid by U...


Citation and Details
More data for this
Ligand-Target Pair
Arachidonate 12-lipoxygenase


(Mus musculus)
BDBM50052454
PNG
(2-(4,5-Dihydroxy-10-oxo-9,10-dihydro-anthracen-9-y...)
Show SMILES CC(SC1c2cccc(O)c2C(=O)c2c(O)cccc12)C(O)=O
Show InChI InChI=1S/C17H14O5S/c1-8(17(21)22)23-16-9-4-2-6-11(18)13(9)15(20)14-10(16)5-3-7-12(14)19/h2-8,16,18-19H,1H3,(H,21,22)
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n/an/a 1.50E+4n/an/an/an/an/an/a



Universität Regensburg

Curated by ChEMBL


Assay Description
Tested for inhibition of 12-LO (12-lipoxygenase) as an inhibitor of 12(S)-HETE biosynthesis in mouse epidermal homogenates


Citation and Details
More data for this
Ligand-Target Pair
Arachidonate 12-lipoxygenase


(Mus musculus)
BDBM50052458
PNG
(3-(4,5-Dihydroxy-10-oxo-9,10-dihydro-anthracen-9-y...)
Show SMILES COC(=O)CCSC1c2cccc(O)c2C(=O)c2c(O)cccc12
Show InChI InChI=1S/C18H16O5S/c1-23-14(21)8-9-24-18-10-4-2-6-12(19)15(10)17(22)16-11(18)5-3-7-13(16)20/h2-7,18-20H,8-9H2,1H3
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n/an/a 2.70E+4n/an/an/an/an/an/a



Universität Regensburg

Curated by ChEMBL


Assay Description
Tested for inhibition of 12-LO (12-lipoxygenase) as an inhibitor of 12(S)-HETE biosynthesis in mouse epidermal homogenates


Citation and Details
More data for this
Ligand-Target Pair
Arachidonate 12-lipoxygenase


(Mus musculus)
BDBM50052459
PNG
(10-(4-Amino-phenylsulfanyl)-1,8-dihydroxy-10H-anth...)
Show SMILES Nc1ccc(SC2c3cccc(O)c3C(=O)c3c(O)cccc23)cc1
Show InChI InChI=1S/C20H15NO3S/c21-11-7-9-12(10-8-11)25-20-13-3-1-5-15(22)17(13)19(24)18-14(20)4-2-6-16(18)23/h1-10,20,22-23H,21H2
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n/an/a>3.00E+4n/an/an/an/an/an/a



Universität Regensburg

Curated by ChEMBL


Assay Description
Tested for inhibition of 12-LO (12-lipoxygenase) as an inhibitor of 12(S)-HETE biosynthesis in mouse epidermal homogenates


Citation and Details
More data for this
Ligand-Target Pair
Arachidonate 12-lipoxygenase


(Mus musculus)
BDBM50052461
PNG
(1,8-Dihydroxy-10-(3-mercapto-propylsulfanyl)-10H-a...)
Show SMILES Oc1cccc2C(SCCCS)c3cccc(O)c3C(=O)c12
Show InChI InChI=1S/C17H16O3S2/c18-12-6-1-4-10-14(12)16(20)15-11(5-2-7-13(15)19)17(10)22-9-3-8-21/h1-2,4-7,17-19,21H,3,8-9H2
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n/an/a 3.00E+4n/an/an/an/an/an/a



Universität Regensburg

Curated by ChEMBL


Assay Description
Tested for inhibition of 12-LO (12-lipoxygenase) as an inhibitor of 12(S)-HETE biosynthesis in mouse epidermal homogenates


Citation and Details
More data for this
Ligand-Target Pair
Arachidonate 12-lipoxygenase


(Mus musculus)
BDBM50052473
PNG
(1,8-Dihydroxy-10-(3-methoxy-phenylsulfanyl)-10H-an...)
Show SMILES COc1cccc(SC2c3cccc(O)c3C(=O)c3c(O)cccc23)c1
Show InChI InChI=1S/C21H16O4S/c1-25-12-5-2-6-13(11-12)26-21-14-7-3-9-16(22)18(14)20(24)19-15(21)8-4-10-17(19)23/h2-11,21-23H,1H3
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n/an/a 3.00E+4n/an/an/an/an/an/a



Universität Regensburg

Curated by ChEMBL


Assay Description
Tested for inhibition of 12-LO (12-lipoxygenase) as an inhibitor of 12(S)-HETE biosynthesis in mouse epidermal homogenates


Citation and Details
More data for this
Ligand-Target Pair
Arachidonate 12-lipoxygenase


(Mus musculus)
BDBM50052474
PNG
((4,5-Dihydroxy-10-oxo-9,10-dihydro-anthracen-9-yls...)
Show SMILES OC(=O)CSC1c2cccc(O)c2C(=O)c2c(O)cccc12
Show InChI InChI=1S/C16H12O5S/c17-10-5-1-3-8-13(10)15(21)14-9(4-2-6-11(14)18)16(8)22-7-12(19)20/h1-6,16-18H,7H2,(H,19,20)
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n/an/a 3.00E+4n/an/an/an/an/an/a



Universität Regensburg

Curated by ChEMBL


Assay Description
Tested for inhibition of 12-LO (12-lipoxygenase) as an inhibitor of 12(S)-HETE biosynthesis in mouse epidermal homogenates


Citation and Details
More data for this
Ligand-Target Pair
Arachidonate 12-lipoxygenase


(Mus musculus)
BDBM50052457
PNG
(1,8-Dihydroxy-10-(2-hydroxy-ethylsulfanyl)-10H-ant...)
Show SMILES OCCSC1c2cccc(O)c2C(=O)c2c(O)cccc12
Show InChI InChI=1S/C16H14O4S/c17-7-8-21-16-9-3-1-5-11(18)13(9)15(20)14-10(16)4-2-6-12(14)19/h1-6,16-19H,7-8H2
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n/an/a>3.00E+4n/an/an/an/an/an/a



Universität Regensburg

Curated by ChEMBL


Assay Description
Tested for inhibition of 12-LO (12-lipoxygenase) as an inhibitor of 12(S)-HETE biosynthesis in mouse epidermal homogenates


Citation and Details
More data for this
Ligand-Target Pair
Arachidonate 12-lipoxygenase


(Mus musculus)
BDBM50052456
PNG
(1,8-Dihydroxy-10-(2-hydroxy-phenylsulfanyl)-10H-an...)
Show SMILES Oc1ccccc1SC1c2cccc(O)c2C(=O)c2c(O)cccc12
Show InChI InChI=1S/C20H14O4S/c21-13-7-1-2-10-16(13)25-20-11-5-3-8-14(22)17(11)19(24)18-12(20)6-4-9-15(18)23/h1-10,20-23H
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n/an/a 3.00E+4n/an/an/an/an/an/a



Universität Regensburg

Curated by ChEMBL


Assay Description
Tested for inhibition of 12-LO (12-lipoxygenase) as an inhibitor of 12(S)-HETE biosynthesis in mouse epidermal homogenates


Citation and Details
More data for this
Ligand-Target Pair
Arachidonate 12-lipoxygenase


(Mus musculus)
BDBM50052469
PNG
((4,5-Dihydroxy-10-oxo-9,10-dihydro-anthracen-9-yls...)
Show SMILES COC(=O)CSC1c2cccc(O)c2C(=O)c2c(O)cccc12
Show InChI InChI=1S/C17H14O5S/c1-22-13(20)8-23-17-9-4-2-6-11(18)14(9)16(21)15-10(17)5-3-7-12(15)19/h2-7,17-19H,8H2,1H3
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n/an/a>3.00E+4n/an/an/an/an/an/a



Universität Regensburg

Curated by ChEMBL


Assay Description
Tested for inhibition of 12-LO (12-lipoxygenase) as an inhibitor of 12(S)-HETE biosynthesis in mouse epidermal homogenates


Citation and Details
More data for this
Ligand-Target Pair
Arachidonate 12-lipoxygenase


(Mus musculus)
BDBM50052466
PNG
(3-(4,5-Dihydroxy-10-oxo-9,10-dihydro-anthracen-9-y...)
Show SMILES OC(=O)CCSC1c2cccc(O)c2C(=O)c2c(O)cccc12
Show InChI InChI=1S/C17H14O5S/c18-11-5-1-3-9-14(11)16(22)15-10(4-2-6-12(15)19)17(9)23-8-7-13(20)21/h1-6,17-19H,7-8H2,(H,20,21)
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n/an/a 3.00E+4n/an/an/an/an/an/a



Universität Regensburg

Curated by ChEMBL


Assay Description
Tested for inhibition of 12-LO (12-lipoxygenase) as an inhibitor of 12(S)-HETE biosynthesis in mouse epidermal homogenates


Citation and Details
More data for this
Ligand-Target Pair
Arachidonate 12-lipoxygenase


(Mus musculus)
BDBM50052470
PNG
(1,8-Dihydroxy-10-(4-methoxy-phenylsulfanyl)-10H-an...)
Show SMILES COc1ccc(SC2c3cccc(O)c3C(=O)c3c(O)cccc23)cc1
Show InChI InChI=1S/C21H16O4S/c1-25-12-8-10-13(11-9-12)26-21-14-4-2-6-16(22)18(14)20(24)19-15(21)5-3-7-17(19)23/h2-11,21-23H,1H3
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n/an/a 3.00E+4n/an/an/an/an/an/a



Universität Regensburg

Curated by ChEMBL


Assay Description
Tested for inhibition of 12-LO (12-lipoxygenase) as an inhibitor of 12(S)-HETE biosynthesis in mouse epidermal homogenates


Citation and Details
More data for this
Ligand-Target Pair
Arachidonate 12-lipoxygenase


(Mus musculus)
BDBM50052471
PNG
(10-(2,3-Dihydroxy-propylsulfanyl)-1,8-dihydroxy-10...)
Show SMILES OCC(O)CSC1c2cccc(O)c2C(=O)c2c(O)cccc12
Show InChI InChI=1S/C17H16O5S/c18-7-9(19)8-23-17-10-3-1-5-12(20)14(10)16(22)15-11(17)4-2-6-13(15)21/h1-6,9,17-21H,7-8H2
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n/an/a>3.00E+4n/an/an/an/an/an/a



Universität Regensburg

Curated by ChEMBL


Assay Description
Tested for inhibition of 12-LO (12-lipoxygenase) as an inhibitor of 12(S)-HETE biosynthesis in mouse epidermal homogenates


Citation and Details
More data for this
Ligand-Target Pair
Arachidonate 12-lipoxygenase


(Mus musculus)
BDBM50052475
PNG
((4,5-Dihydroxy-10-oxo-9,10-dihydro-anthracen-9-yls...)
Show SMILES CCCCOC(=O)CSC1c2cccc(O)c2C(=O)c2c(O)cccc12
Show InChI InChI=1S/C20H20O5S/c1-2-3-10-25-16(23)11-26-20-12-6-4-8-14(21)17(12)19(24)18-13(20)7-5-9-15(18)22/h4-9,20-22H,2-3,10-11H2,1H3
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n/an/a 3.00E+4n/an/an/an/an/an/a



Universität Regensburg

Curated by ChEMBL


Assay Description
Tested for inhibition of 12-LO (12-lipoxygenase) as an inhibitor of 12(S)-HETE biosynthesis in mouse epidermal homogenates


Citation and Details
More data for this
Ligand-Target Pair
Arachidonate 12-lipoxygenase


(Mus musculus)
BDBM50052449
PNG
(10-Benzylsulfanyl-1,8-dihydroxy-10H-anthracen-9-on...)
Show SMILES Oc1cccc2C(SCc3ccccc3)c3cccc(O)c3C(=O)c12
Show InChI InChI=1S/C21H16O3S/c22-16-10-4-8-14-18(16)20(24)19-15(9-5-11-17(19)23)21(14)25-12-13-6-2-1-3-7-13/h1-11,21-23H,12H2
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n/an/a 3.00E+4n/an/an/an/an/an/a



Universität Regensburg

Curated by ChEMBL


Assay Description
Tested for inhibition of 12-LO (12-lipoxygenase) as an inhibitor of 12(S)-HETE biosynthesis in mouse epidermal homogenates


Citation and Details
More data for this
Ligand-Target Pair
Arachidonate 12-lipoxygenase


(Mus musculus)
BDBM50052453
PNG
((4,5-Dihydroxy-10-oxo-9,10-dihydro-anthracen-9-yls...)
Show SMILES CCOC(=O)CSC1c2cccc(O)c2C(=O)c2c(O)cccc12
Show InChI InChI=1S/C18H16O5S/c1-2-23-14(21)9-24-18-10-5-3-7-12(19)15(10)17(22)16-11(18)6-4-8-13(16)20/h3-8,18-20H,2,9H2,1H3
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n/an/a>3.00E+4n/an/an/an/an/an/a



Universität Regensburg

Curated by ChEMBL


Assay Description
Tested for inhibition of 12-LO (12-lipoxygenase) as an inhibitor of 12(S)-HETE biosynthesis in mouse epidermal homogenates


Citation and Details
More data for this
Ligand-Target Pair
Arachidonate 12-lipoxygenase


(Mus musculus)
BDBM50052455
PNG
(1,8-Dihydroxy-10-phenethylsulfanyl-10H-anthracen-9...)
Show SMILES Oc1cccc2C(SCCc3ccccc3)c3cccc(O)c3C(=O)c12
Show InChI InChI=1S/C22H18O3S/c23-17-10-4-8-15-19(17)21(25)20-16(9-5-11-18(20)24)22(15)26-13-12-14-6-2-1-3-7-14/h1-11,22-24H,12-13H2
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n/an/a>3.00E+4n/an/an/an/an/an/a



Universität Regensburg

Curated by ChEMBL


Assay Description
Tested for inhibition of 12-LO (12-lipoxygenase) as an inhibitor of 12(S)-HETE biosynthesis in mouse epidermal homogenates


Citation and Details
More data for this
Ligand-Target Pair
Arachidonate 12-lipoxygenase


(Mus musculus)
BDBM50052452
PNG
(1,8-Dihydroxy-10-(3-phenyl-propylsulfanyl)-10H-ant...)
Show SMILES Oc1cccc2C(SCCCc3ccccc3)c3cccc(O)c3C(=O)c12
Show InChI InChI=1S/C23H20O3S/c24-18-12-4-10-16-20(18)22(26)21-17(11-5-13-19(21)25)23(16)27-14-6-9-15-7-2-1-3-8-15/h1-5,7-8,10-13,23-25H,6,9,14H2
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n/an/a>3.00E+4n/an/an/an/an/an/a



Universität Regensburg

Curated by ChEMBL


Assay Description
Tested for inhibition of 12-LO (12-lipoxygenase) as an inhibitor of 12(S)-HETE biosynthesis in mouse epidermal homogenates


Citation and Details
More data for this
Ligand-Target Pair
Arachidonate 12-lipoxygenase


(Mus musculus)
BDBM50052460
PNG
(1,8-Dihydroxy-10-phenylsulfanyl-10H-anthracen-9-on...)
Show SMILES Oc1cccc2C(Sc3ccccc3)c3cccc(O)c3C(=O)c12
Show InChI InChI=1S/C20H14O3S/c21-15-10-4-8-13-17(15)19(23)18-14(9-5-11-16(18)22)20(13)24-12-6-2-1-3-7-12/h1-11,20-22H
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n/an/a 3.00E+4n/an/an/an/an/an/a



Universität Regensburg

Curated by ChEMBL


Assay Description
Tested for inhibition of 12-LO (12-lipoxygenase) as an inhibitor of 12(S)-HETE biosynthesis in mouse epidermal homogenates


Citation and Details
More data for this
Ligand-Target Pair
Arachidonate 12-lipoxygenase


(Mus musculus)
BDBM50052463
PNG
(1,8-Dihydroxy-10-propylsulfanyl-10H-anthracen-9-on...)
Show SMILES CCCSC1c2cccc(O)c2C(=O)c2c(O)cccc12
Show InChI InChI=1S/C17H16O3S/c1-2-9-21-17-10-5-3-7-12(18)14(10)16(20)15-11(17)6-4-8-13(15)19/h3-8,17-19H,2,9H2,1H3
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n/an/a>3.00E+4n/an/an/an/an/an/a



Universität Regensburg

Curated by ChEMBL


Assay Description
Tested for inhibition of 12-LO (12-lipoxygenase) as an inhibitor of 12(S)-HETE biosynthesis in mouse epidermal homogenates


Citation and Details
More data for this
Ligand-Target Pair
Arachidonate 12-lipoxygenase


(Mus musculus)
BDBM50052465
PNG
(1,8-Dihydroxy-10-(4-methoxy-benzylsulfanyl)-10H-an...)
Show SMILES COc1ccc(CSC2c3cccc(O)c3C(=O)c3c(O)cccc23)cc1
Show InChI InChI=1S/C22H18O4S/c1-26-14-10-8-13(9-11-14)12-27-22-15-4-2-6-17(23)19(15)21(25)20-16(22)5-3-7-18(20)24/h2-11,22-24H,12H2,1H3
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n/an/a 3.00E+4n/an/an/an/an/an/a



Universität Regensburg

Curated by ChEMBL


Assay Description
Tested for inhibition of 12-LO (12-lipoxygenase) as an inhibitor of 12(S)-HETE biosynthesis in mouse epidermal homogenates


Citation and Details
More data for this
Ligand-Target Pair
Arachidonate 12-lipoxygenase


(Mus musculus)
BDBM50052467
PNG
(3-(4,5-Dihydroxy-10-oxo-9,10-dihydro-anthracen-9-y...)
Show SMILES CCCCOC(=O)CCSC1c2cccc(O)c2C(=O)c2c(O)cccc12
Show InChI InChI=1S/C21H22O5S/c1-2-3-11-26-17(24)10-12-27-21-13-6-4-8-15(22)18(13)20(25)19-14(21)7-5-9-16(19)23/h4-9,21-23H,2-3,10-12H2,1H3
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n/an/a 3.00E+4n/an/an/an/an/an/a



Universität Regensburg

Curated by ChEMBL


Assay Description
Tested for inhibition of 12-LO (12-lipoxygenase) as an inhibitor of 12(S)-HETE biosynthesis in mouse epidermal homogenates


Citation and Details
More data for this
Ligand-Target Pair
Arachidonate 12-lipoxygenase


(Mus musculus)
BDBM50052451
PNG
(10-Ethylsulfanyl-1,8-dihydroxy-10H-anthracen-9-one...)
Show SMILES CCSC1c2cccc(O)c2C(=O)c2c(O)cccc12
Show InChI InChI=1S/C16H14O3S/c1-2-20-16-9-5-3-7-11(17)13(9)15(19)14-10(16)6-4-8-12(14)18/h3-8,16-18H,2H2,1H3
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n/an/a>3.00E+4n/an/an/an/an/an/a



Universität Regensburg

Curated by ChEMBL


Assay Description
Tested for inhibition of 12-LO (12-lipoxygenase) as an inhibitor of 12(S)-HETE biosynthesis in mouse epidermal homogenates


Citation and Details
More data for this
Ligand-Target Pair
Arachidonate 12-lipoxygenase


(Mus musculus)
BDBM50052472
PNG
(3-(4,5-Dihydroxy-10-oxo-9,10-dihydro-anthracen-9-y...)
Show SMILES CCOC(=O)CCSC1c2cccc(O)c2C(=O)c2c(O)cccc12
Show InChI InChI=1S/C19H18O5S/c1-2-24-15(22)9-10-25-19-11-5-3-7-13(20)16(11)18(23)17-12(19)6-4-8-14(17)21/h3-8,19-21H,2,9-10H2,1H3
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n/an/a 3.00E+4n/an/an/an/an/an/a



Universität Regensburg

Curated by ChEMBL


Assay Description
Tested for inhibition of 12-LO (12-lipoxygenase) as an inhibitor of 12(S)-HETE biosynthesis in mouse epidermal homogenates


Citation and Details
More data for this
Ligand-Target Pair
Arachidonate 12-lipoxygenase


(Mus musculus)
BDBM50052468
PNG
(2-Amino-3-(4,5-dihydroxy-10-oxo-9,10-dihydro-anthr...)
Show SMILES NC(CSC1c2cccc(O)c2C(=O)c2c(O)cccc12)C(O)=O
Show InChI InChI=1S/C17H15NO5S/c18-10(17(22)23)7-24-16-8-3-1-5-11(19)13(8)15(21)14-9(16)4-2-6-12(14)20/h1-6,10,16,19-20H,7,18H2,(H,22,23)
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n/an/a 3.00E+4n/an/an/an/an/an/a



Universität Regensburg

Curated by ChEMBL


Assay Description
Tested for inhibition of 12-LO (12-lipoxygenase) as an inhibitor of 12(S)-HETE biosynthesis in mouse epidermal homogenates


Citation and Details
More data for this
Ligand-Target Pair