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Found 59 hits Enz. Inhib. hit(s) with Target = 'Diamine oxidase' AND taxid = 9606   
Target
(Institution)
LigandTarget
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Diamine oxidase (DAO)


(Homo sapiens)
BDBM50000999
PNG
(CHEBI:81724 | DIMINAZENE)
Show SMILES NC(=N)c1ccc(N\N=N\c2ccc(cc2)C(N)=N)cc1
Show InChI InChI=1S/C14H15N7/c15-13(16)9-1-5-11(6-2-9)19-21-20-12-7-3-10(4-8-12)14(17)18/h1-8H,(H3,15,16)(H3,17,18)(H,19,20)
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13n/an/an/an/an/an/an/an/a



Xavier University of Louisiana

Curated by ChEMBL


Assay Description
Mixed type inhibition of recombinant human DAO expressed in drosophila S2 cells


Citation and Details
More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM50207159
PNG
(2-aminoguanidine | 2-azanylguanidine | AG | AMINOG...)
Show SMILES NNC(N)=N
Show InChI InChI=1S/CH6N4/c2-1(3)5-4/h4H2,(H4,2,3,5)
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140n/an/an/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Tested for ability of the compound to competitively inhibit hog kidney diamine oxidase (DAO) in a spectrometric assay


Citation and Details
More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM50281515
PNG
((E)-3-(1H-Imidazol-4-yl)-allylamine | CHEMBL119195...)
Show SMILES NCC=Cc1cnc[nH]1
Show InChI InChI=1S/C6H9N3/c7-3-1-2-6-4-8-5-9-6/h1-2,4-5H,3,7H2,(H,8,9)
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170n/an/an/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Tested for ability of the compound to competitively inhibit hog kidney diamine oxidase (DAO) in a spectrometric assay


Citation and Details
More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM50281515
PNG
((E)-3-(1H-Imidazol-4-yl)-allylamine | CHEMBL119195...)
Show SMILES NCC=Cc1cnc[nH]1
Show InChI InChI=1S/C6H9N3/c7-3-1-2-6-4-8-5-9-6/h1-2,4-5H,3,7H2,(H,8,9)
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200n/an/an/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Tested for ability of the compound to competitively inhibit hog kidney diamine oxidase (DAO) in a spectrometric assay


Citation and Details
More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM45440
PNG
(4-[5-(4-amidinophenoxy)pentoxy]benzamidine;2-hydro...)
Show SMILES NC(=N)c1ccc(OCCCCCOc2ccc(cc2)C(N)=N)cc1
Show InChI InChI=1S/C19H24N4O2/c20-18(21)14-4-8-16(9-5-14)24-12-2-1-3-13-25-17-10-6-15(7-11-17)19(22)23/h4-11H,1-3,12-13H2,(H3,20,21)(H3,22,23)
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290n/an/an/an/an/an/an/an/a



Xavier University of Louisiana

Curated by ChEMBL


Assay Description
Mixed type inhibition of recombinant human DAO expressed in drosophila S2 cells


Citation and Details
More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM50281517
PNG
(3-(1H-Imidazol-4-yl)-prop-2-ynylamine | CHEMBL1165...)
Show SMILES NCC#Cc1cnc[nH]1
Show InChI InChI=1S/C6H7N3/c7-3-1-2-6-4-8-5-9-6/h4-5H,3,7H2,(H,8,9)
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1.70E+3n/an/an/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Tested for ability of the compound to competitively inhibit hog kidney diamine oxidase (DAO) in a spectrometric assay


Citation and Details
More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM50020274
PNG
(2,2-Difluoro-hex-5-yne-1,4-diamonium; dichloride |...)
Show SMILES [NH3+]CC(F)(F)CC([NH3+])C#C
Show InChI InChI=1S/C6H10F2N2/c1-2-5(10)3-6(7,8)4-9/h1,5H,3-4,9-10H2/p+2
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2.70E+3n/an/an/an/an/an/an/an/a



Merrell Dow Research Institute

Curated by ChEMBL


Assay Description
In vitro inhibition against hog kidney diamine oxidase


J Med Chem 32: 170-3 (1989)

More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM50121458
PNG
(1-[3-(2-Hydroxy-phenyl)-5-o-tolyl-4,5-dihydro-pyra...)
Show SMILES CC(=O)N1N=C(CC1c1ccccc1C)c1ccccc1O
Show InChI InChI=1S/C18H18N2O2/c1-12-7-3-4-8-14(12)17-11-16(19-20(17)13(2)21)15-9-5-6-10-18(15)22/h3-10,17,22H,11H2,1-2H3
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5.50E+3n/an/an/an/an/an/an/an/a



Università di Roma La Sapienza

Curated by ChEMBL


Assay Description
Inhibitory activity of the compound against Swine kidney diamine oxidase (SKDAO)


Bioorg Med Chem Lett 12: 3629-33 (2002)

More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM50281518
PNG
(2-(1H-Imidazol-4-yl)-allylamine | CHEMBL116538)
Show SMILES NCC(=C)c1cnc[nH]1
Show InChI InChI=1S/C6H9N3/c1-5(2-7)6-3-8-4-9-6/h3-4H,1-2,7H2,(H,8,9)
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7.10E+3n/an/an/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Tested for ability of the compound to competitively inhibit hog kidney diamine oxidase (DAO) in a spectrometric assay


Citation and Details
More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM50121455
PNG
(1-[3-(2-Hydroxy-phenyl)-5-m-tolyl-4,5-dihydro-pyra...)
Show SMILES CC(=O)N1N=C(CC1c1cccc(C)c1)c1ccccc1O
Show InChI InChI=1S/C18H18N2O2/c1-12-6-5-7-14(10-12)17-11-16(19-20(17)13(2)21)15-8-3-4-9-18(15)22/h3-10,17,22H,11H2,1-2H3
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8.00E+3n/an/an/an/an/an/an/an/a



Università di Roma La Sapienza

Curated by ChEMBL


Assay Description
Inhibitory activity of the compound against Swine kidney diamine oxidase (SKDAO)


Bioorg Med Chem Lett 12: 3629-33 (2002)

More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM50121457
PNG
(1-[3-(2,4-Dihydroxy-phenyl)-5-m-tolyl-4,5-dihydro-...)
Show SMILES CC(=O)N1N=C(CC1c1cccc(C)c1)c1ccc(O)cc1O
Show InChI InChI=1S/C18H18N2O3/c1-11-4-3-5-13(8-11)17-10-16(19-20(17)12(2)21)15-7-6-14(22)9-18(15)23/h3-9,17,22-23H,10H2,1-2H3
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2.50E+4n/an/an/an/an/an/an/an/a



Università di Roma La Sapienza

Curated by ChEMBL


Assay Description
Inhibitory activity of the compound against Swine kidney diamine oxidase (SKDAO)


Bioorg Med Chem Lett 12: 3629-33 (2002)

More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM50121456
PNG
(1-[3-(2,4-Dihydroxy-phenyl)-5-o-tolyl-4,5-dihydro-...)
Show SMILES CC(=O)N1N=C(CC1c1ccccc1C)c1ccc(O)cc1O
Show InChI InChI=1S/C18H18N2O3/c1-11-5-3-4-6-14(11)17-10-16(19-20(17)12(2)21)15-8-7-13(22)9-18(15)23/h3-9,17,22-23H,10H2,1-2H3
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1.00E+5n/an/an/an/an/an/an/an/a



Università di Roma La Sapienza

Curated by ChEMBL


Assay Description
Inhibitory activity of the compound against Swine kidney diamine oxidase (SKDAO)


Bioorg Med Chem Lett 12: 3629-33 (2002)

More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM50161146
PNG
(4-(aminomethyl)-5-(dimethyl-lambda~5~-azanyl)-N-me...)
Show SMILES CNc1cncc(N(C)C)c1CN
Show InChI InChI=1S/C9H16N4/c1-11-8-5-12-6-9(13(2)3)7(8)4-10/h5-6,11H,4,10H2,1-3H3
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n/an/a 61n/an/an/an/an/an/a



Universit£ di Genova

Curated by ChEMBL


Assay Description
Inhibition of putrescine binding to against Diamine oxidase of porcine kidney


Citation and Details
More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM220884
PNG
(US9302986, 18)
Show SMILES CN(C)C(=O)c1ccc(OC\C(CN)=C/F)cc1
Show InChI InChI=1S/C13H17FN2O2/c1-16(2)13(17)11-3-5-12(6-4-11)18-9-10(7-14)8-15/h3-7H,8-9,15H2,1-2H3/b10-7-
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n/an/a<100n/an/an/an/an/an/a



BOEHRINGER INGELHEIM INTERNATIONAL GMBH

US Patent


Assay Description
Recombinant human DAO (2.4 μg/mL) was used as source of DAO enzyme activities. The assay was performed as described in the method for human SSAO/V...


US Patent US9302986 (2016)

More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM220869
PNG
(US9302986, 2)
Show SMILES NC\C(COc1ccc(cc1)C(N)=O)=C\F
Show InChI InChI=1S/C11H13FN2O2/c12-5-8(6-13)7-16-10-3-1-9(2-4-10)11(14)15/h1-5H,6-7,13H2,(H2,14,15)/b8-5-
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n/an/a<100n/an/an/an/an/an/a



BOEHRINGER INGELHEIM INTERNATIONAL GMBH

US Patent


Assay Description
Recombinant human DAO (2.4 μg/mL) was used as source of DAO enzyme activities. The assay was performed as described in the method for human SSAO/V...


US Patent US9302986 (2016)

More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM50161153
PNG
(4-(aminomethyl)-N-methyl-5-(methyl-lambda~5~-azany...)
Show SMILES CNc1cncc(NC)c1CN
Show InChI InChI=1S/C8H14N4/c1-10-7-4-12-5-8(11-2)6(7)3-9/h4-5,10-11H,3,9H2,1-2H3
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n/an/a 120n/an/an/an/an/an/a



Universit£ di Genova

Curated by ChEMBL


Assay Description
Inhibition of putrescine binding to against Diamine oxidase of porcine kidney


Citation and Details
More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM50161135
PNG
(4-(aminomethyl)-N-methylpyridin-3-amine dihydrochl...)
Show SMILES CNc1cnccc1CN
Show InChI InChI=1S/C7H11N3/c1-9-7-5-10-3-2-6(7)4-8/h2-3,5,9H,4,8H2,1H3
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n/an/a 160n/an/an/an/an/an/a



Universit£ di Genova

Curated by ChEMBL


Assay Description
Inhibition of putrescine binding to against Diamine oxidase of porcine kidney


Citation and Details
More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM50161138
PNG
(4-(aminomethyl)pyridin-3-amine dihydrochloride | C...)
Show SMILES NCc1ccncc1N
Show InChI InChI=1S/C6H9N3/c7-3-5-1-2-9-4-6(5)8/h1-2,4H,3,7-8H2
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n/an/a 300n/an/an/an/an/an/a



Universit£ di Genova

Curated by ChEMBL


Assay Description
Inhibition of putrescine binding to against Diamine oxidase of porcine kidney


Citation and Details
More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM50161132
PNG
(4-(aminomethyl)-N-ethylpyridin-3-amine dihydrochlo...)
Show SMILES CCNc1cnccc1CN
Show InChI InChI=1S/C8H13N3/c1-2-11-8-6-10-4-3-7(8)5-9/h3-4,6,11H,2,5,9H2,1H3
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n/an/a 500n/an/an/an/an/an/a



Universit£ di Genova

Curated by ChEMBL


Assay Description
Inhibition of putrescine binding to against Diamine oxidase of porcine kidney


Citation and Details
More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM220885
PNG
(US9302986, 9)
Show SMILES NC\C(COc1ccc(cc1)S(N)(=O)=O)=C\F
Show InChI InChI=1S/C10H13FN2O3S/c11-5-8(6-12)7-16-9-1-3-10(4-2-9)17(13,14)15/h1-5H,6-7,12H2,(H2,13,14,15)/b8-5-
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n/an/a<1.00E+3n/an/an/an/an/an/a



BOEHRINGER INGELHEIM INTERNATIONAL GMBH

US Patent


Assay Description
Recombinant human DAO (2.4 μg/mL) was used as source of DAO enzyme activities. The assay was performed as described in the method for human SSAO/V...


US Patent US9302986 (2016)

More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM220873
PNG
(US9302986, 7)
Show SMILES COc1cc(ccc1OCC(CN)=CF)C(=O)N(C)C
Show InChI InChI=1S/C14H19FN2O3/c1-17(2)14(18)11-4-5-12(13(6-11)19-3)20-9-10(7-15)8-16/h4-7H,8-9,16H2,1-3H3/b10-7+
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n/an/a<1.00E+3n/an/an/an/an/an/a



BOEHRINGER INGELHEIM INTERNATIONAL GMBH

US Patent


Assay Description
Recombinant human DAO (2.4 μg/mL) was used as source of DAO enzyme activities. The assay was performed as described in the method for human SSAO/V...


US Patent US9302986 (2016)

More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM220862
PNG
(US9302986, 6)
Show SMILES CN(C)C(=O)c1ccc(OC\C(CN)=C/F)c(Cl)c1
Show InChI InChI=1S/C13H16ClFN2O2/c1-17(2)13(18)10-3-4-12(11(14)5-10)19-8-9(6-15)7-16/h3-6H,7-8,16H2,1-2H3/b9-6-
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n/an/a<1.00E+3n/an/an/an/an/an/a



BOEHRINGER INGELHEIM INTERNATIONAL GMBH

US Patent


Assay Description
Recombinant human DAO (2.4 μg/mL) was used as source of DAO enzyme activities. The assay was performed as described in the method for human SSAO/V...


US Patent US9302986 (2016)

More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM220861
PNG
(US9302986, 4)
Show SMILES CN(C)C(=O)c1ccc(OC\C(CN)=C/F)c(F)c1
Show InChI InChI=1S/C13H16F2N2O2/c1-17(2)13(18)10-3-4-12(11(15)5-10)19-8-9(6-14)7-16/h3-6H,7-8,16H2,1-2H3/b9-6-
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n/an/a<1.00E+3n/an/an/an/an/an/a



BOEHRINGER INGELHEIM INTERNATIONAL GMBH

US Patent


Assay Description
Recombinant human DAO (2.4 μg/mL) was used as source of DAO enzyme activities. The assay was performed as described in the method for human SSAO/V...


US Patent US9302986 (2016)

More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM220883
PNG
(US9302986, 10)
Show SMILES CN(C)S(=O)(=O)c1ccc(OC\C(CN)=C/F)cc1
Show InChI InChI=1S/C12H17FN2O3S/c1-15(2)19(16,17)12-5-3-11(4-6-12)18-9-10(7-13)8-14/h3-7H,8-9,14H2,1-2H3/b10-7-
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n/an/a>1.00E+3n/an/an/an/an/an/a



BOEHRINGER INGELHEIM INTERNATIONAL GMBH

US Patent


Assay Description
Recombinant human DAO (2.4 μg/mL) was used as source of DAO enzyme activities. The assay was performed as described in the method for human SSAO/V...


US Patent US9302986 (2016)

More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM220871
PNG
(US9302986, 13)
Show SMILES CN(C)C(=O)c1ccc(OC\C(CN)=C\F)cc1
Show InChI InChI=1S/C13H17FN2O2/c1-16(2)13(17)11-3-5-12(6-4-11)18-9-10(7-14)8-15/h3-7H,8-9,15H2,1-2H3/b10-7+
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n/an/a>1.00E+3n/an/an/an/an/an/a



BOEHRINGER INGELHEIM INTERNATIONAL GMBH

US Patent


Assay Description
Recombinant human DAO (2.4 μg/mL) was used as source of DAO enzyme activities. The assay was performed as described in the method for human SSAO/V...


US Patent US9302986 (2016)

More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM220863
PNG
(US9302986, 20)
Show SMILES CN(C)C(=O)c1ccc(OC\C(CN)=C/F)c(Br)c1
Show InChI InChI=1S/C13H16BrFN2O2/c1-17(2)13(18)10-3-4-12(11(14)5-10)19-8-9(6-15)7-16/h3-6H,7-8,16H2,1-2H3/b9-6-
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n/an/a<1.00E+3n/an/an/an/an/an/a



BOEHRINGER INGELHEIM INTERNATIONAL GMBH

US Patent


Assay Description
Recombinant human DAO (2.4 μg/mL) was used as source of DAO enzyme activities. The assay was performed as described in the method for human SSAO/V...


US Patent US9302986 (2016)

More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM50161149
PNG
(4-(aminomethyl)-N-isopropyl-5-[isopropyl(methyl)-l...)
Show SMILES CC(C)Nc1cncc(N(C)C(C)C)c1CN
Show InChI InChI=1S/C13H24N4/c1-9(2)16-12-7-15-8-13(11(12)6-14)17(5)10(3)4/h7-10,16H,6,14H2,1-5H3
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n/an/a 1.00E+3n/an/an/an/an/an/a



Universit£ di Genova

Curated by ChEMBL


Assay Description
Inhibition of putrescine binding to against Diamine oxidase of porcine kidney


Citation and Details
More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM220868
PNG
(US9302986, 25)
Show SMILES CNC(=O)c1ccc(OC\C(CN)=C\F)cc1
Show InChI InChI=1S/C12H15FN2O2/c1-15-12(16)10-2-4-11(5-3-10)17-8-9(6-13)7-14/h2-6H,7-8,14H2,1H3,(H,15,16)/b9-6+
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n/an/a<1.00E+3n/an/an/an/an/an/a



BOEHRINGER INGELHEIM INTERNATIONAL GMBH

US Patent


Assay Description
Recombinant human DAO (2.4 μg/mL) was used as source of DAO enzyme activities. The assay was performed as described in the method for human SSAO/V...


US Patent US9302986 (2016)

More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM220872
PNG
(US9302986, 26)
Show SMILES CN(C)C(=O)c1ccc(OC\C(CN)=C/F)cc1C
Show InChI InChI=1S/C14H19FN2O2/c1-10-6-12(19-9-11(7-15)8-16)4-5-13(10)14(18)17(2)3/h4-7H,8-9,16H2,1-3H3/b11-7-
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n/an/a<1.00E+3n/an/an/an/an/an/a



BOEHRINGER INGELHEIM INTERNATIONAL GMBH

US Patent


Assay Description
Recombinant human DAO (2.4 μg/mL) was used as source of DAO enzyme activities. The assay was performed as described in the method for human SSAO/V...


US Patent US9302986 (2016)

More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM220878
PNG
(US9302986, 29)
Show SMILES CNS(=O)(=O)c1ccc(OC\C(CN)=C/F)cc1
Show InChI InChI=1S/C11H15FN2O3S/c1-14-18(15,16)11-4-2-10(3-5-11)17-8-9(6-12)7-13/h2-6,14H,7-8,13H2,1H3/b9-6-
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n/an/a>1.00E+3n/an/an/an/an/an/a



BOEHRINGER INGELHEIM INTERNATIONAL GMBH

US Patent


Assay Description
Recombinant human DAO (2.4 μg/mL) was used as source of DAO enzyme activities. The assay was performed as described in the method for human SSAO/V...


US Patent US9302986 (2016)

More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM220880
PNG
(US9302986, 31)
Show SMILES CCNS(=O)(=O)c1ccc(OC\C(CN)=C/F)cc1
Show InChI InChI=1S/C12H17FN2O3S/c1-2-15-19(16,17)12-5-3-11(4-6-12)18-9-10(7-13)8-14/h3-7,15H,2,8-9,14H2,1H3/b10-7-
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n/an/a<1.00E+3n/an/an/an/an/an/a



BOEHRINGER INGELHEIM INTERNATIONAL GMBH

US Patent


Assay Description
Recombinant human DAO (2.4 μg/mL) was used as source of DAO enzyme activities. The assay was performed as described in the method for human SSAO/V...


US Patent US9302986 (2016)

More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM220860
PNG
(US9302986, 1)
Show SMILES CC(C)(C)NC(=O)c1ccc(OC\C(CN)=C/F)cc1
Show InChI InChI=1S/C15H21FN2O2/c1-15(2,3)18-14(19)12-4-6-13(7-5-12)20-10-11(8-16)9-17/h4-8H,9-10,17H2,1-3H3,(H,18,19)/b11-8-
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n/an/a<1.00E+3n/an/an/an/an/an/a



BOEHRINGER INGELHEIM INTERNATIONAL GMBH

US Patent


Assay Description
Recombinant human DAO (2.4 μg/mL) was used as source of DAO enzyme activities. The assay was performed as described in the method for human SSAO/V...


US Patent US9302986 (2016)

More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM220882
PNG
(US9302986, 33)
Show SMILES CC(C)NS(=O)(=O)c1ccc(OC\C(CN)=C/F)cc1
Show InChI InChI=1S/C13H19FN2O3S/c1-10(2)16-20(17,18)13-5-3-12(4-6-13)19-9-11(7-14)8-15/h3-7,10,16H,8-9,15H2,1-2H3/b11-7-
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n/an/a<1.00E+3n/an/an/an/an/an/a



BOEHRINGER INGELHEIM INTERNATIONAL GMBH

US Patent


Assay Description
Recombinant human DAO (2.4 μg/mL) was used as source of DAO enzyme activities. The assay was performed as described in the method for human SSAO/V...


US Patent US9302986 (2016)

More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM220870
PNG
(US9302986, 3)
Show SMILES NC\C(COc1ccc(cc1)C(N)=O)=C/F
Show InChI InChI=1S/C11H13FN2O2/c12-5-8(6-13)7-16-10-3-1-9(2-4-10)11(14)15/h1-5H,6-7,13H2,(H2,14,15)/b8-5+
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n/an/a>1.00E+3n/an/an/an/an/an/a



BOEHRINGER INGELHEIM INTERNATIONAL GMBH

US Patent


Assay Description
Recombinant human DAO (2.4 μg/mL) was used as source of DAO enzyme activities. The assay was performed as described in the method for human SSAO/V...


US Patent US9302986 (2016)

More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM50161134
PNG
(4-(aminomethyl)-N-ethyl-5-[ethyl(methyl)-lambda~5~...)
Show SMILES CCNc1cncc(N(C)CC)c1CN
Show InChI InChI=1S/C11H20N4/c1-4-14-10-7-13-8-11(9(10)6-12)15(3)5-2/h7-8,14H,4-6,12H2,1-3H3
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n/an/a 2.50E+3n/an/an/an/an/an/a



Universit£ di Genova

Curated by ChEMBL


Assay Description
Inhibition of putrescine binding to against Diamine oxidase of porcine kidney


Citation and Details
More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM50161147
PNG
(4-(aminomethyl)-N-cyclopropylpyridin-3-amine dihyd...)
Show SMILES NCc1ccncc1NC1CC1
Show InChI InChI=1S/C9H13N3/c10-5-7-3-4-11-6-9(7)12-8-1-2-8/h3-4,6,8,12H,1-2,5,10H2
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Universit£ di Genova

Curated by ChEMBL


Assay Description
Inhibition of putrescine binding to against Diamine oxidase of porcine kidney


Citation and Details
More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM50161151
PNG
(4-(aminomethyl)-5-[methyl(propyl)-lambda~5~-azanyl...)
Show SMILES CCCNc1cncc(N(C)CCC)c1CN
Show InChI InChI=1S/C13H24N4/c1-4-6-16-12-9-15-10-13(11(12)8-14)17(3)7-5-2/h9-10,16H,4-8,14H2,1-3H3
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Universit£ di Genova

Curated by ChEMBL


Assay Description
Inhibition of putrescine binding to against Diamine oxidase of porcine kidney


Citation and Details
More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM50246766
PNG
(CHEMBL489079 | Mofegiline | US9302986, Mofegiline)
Show SMILES NC\C(CCc1ccc(F)cc1)=C\F
Show InChI InChI=1S/C11H13F2N/c12-7-10(8-14)2-1-9-3-5-11(13)6-4-9/h3-7H,1-2,8,14H2/b10-7+
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BOEHRINGER INGELHEIM INTERNATIONAL GMBH

US Patent


Assay Description
Recombinant human DAO (2.4 μg/mL) was used as source of DAO enzyme activities. The assay was performed as described in the method for human SSAO/V...


US Patent US9302986 (2016)

More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM220881
PNG
(US9302986, 32)
Show SMILES CC(C)NS(=O)(=O)c1ccc(OC\C(CN)=C\F)cc1
Show InChI InChI=1S/C13H19FN2O3S/c1-10(2)16-20(17,18)13-5-3-12(4-6-13)19-9-11(7-14)8-15/h3-7,10,16H,8-9,15H2,1-2H3/b11-7+
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n/an/a>1.00E+4n/an/an/an/an/an/a



BOEHRINGER INGELHEIM INTERNATIONAL GMBH

US Patent


Assay Description
Recombinant human DAO (2.4 μg/mL) was used as source of DAO enzyme activities. The assay was performed as described in the method for human SSAO/V...


US Patent US9302986 (2016)

More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM220879
PNG
(US9302986, 30)
Show SMILES CCNS(=O)(=O)c1ccc(OC\C(CN)=C\F)cc1
Show InChI InChI=1S/C12H17FN2O3S/c1-2-15-19(16,17)12-5-3-11(4-6-12)18-9-10(7-13)8-14/h3-7,15H,2,8-9,14H2,1H3/b10-7+
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BOEHRINGER INGELHEIM INTERNATIONAL GMBH

US Patent


Assay Description
Recombinant human DAO (2.4 μg/mL) was used as source of DAO enzyme activities. The assay was performed as described in the method for human SSAO/V...


US Patent US9302986 (2016)

More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM220877
PNG
(US9302986, 28)
Show SMILES CNS(=O)(=O)c1ccc(OC\C(CN)=C\F)cc1
Show InChI InChI=1S/C11H15FN2O3S/c1-14-18(15,16)11-4-2-10(3-5-11)17-8-9(6-12)7-13/h2-6,14H,7-8,13H2,1H3/b9-6+
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n/an/a>1.00E+4n/an/an/an/an/an/a



BOEHRINGER INGELHEIM INTERNATIONAL GMBH

US Patent


Assay Description
Recombinant human DAO (2.4 μg/mL) was used as source of DAO enzyme activities. The assay was performed as described in the method for human SSAO/V...


US Patent US9302986 (2016)

More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM220867
PNG
(US9302986, 24)
Show SMILES CCN(CC)C(=O)c1ccc(OC\C(CN)=C\F)cc1
Show InChI InChI=1S/C15H21FN2O2/c1-3-18(4-2)15(19)13-5-7-14(8-6-13)20-11-12(9-16)10-17/h5-9H,3-4,10-11,17H2,1-2H3/b12-9+
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n/an/a>1.00E+4n/an/an/an/an/an/a



BOEHRINGER INGELHEIM INTERNATIONAL GMBH

US Patent


Assay Description
Recombinant human DAO (2.4 μg/mL) was used as source of DAO enzyme activities. The assay was performed as described in the method for human SSAO/V...


US Patent US9302986 (2016)

More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM220866
PNG
(US9302986, 23)
Show SMILES CC(C)(C)NC(=O)c1ccc(OC\C(CN)=C\F)cc1
Show InChI InChI=1S/C15H21FN2O2/c1-15(2,3)18-14(19)12-4-6-13(7-5-12)20-10-11(8-16)9-17/h4-8H,9-10,17H2,1-3H3,(H,18,19)/b11-8+
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n/an/a>1.00E+4n/an/an/an/an/an/a



BOEHRINGER INGELHEIM INTERNATIONAL GMBH

US Patent


Assay Description
Recombinant human DAO (2.4 μg/mL) was used as source of DAO enzyme activities. The assay was performed as described in the method for human SSAO/V...


US Patent US9302986 (2016)

More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM220875
PNG
(US9302986, 14)
Show SMILES CN(C)S(=O)(=O)c1ccc(OC\C(CN)=C\F)cc1
Show InChI InChI=1S/C12H17FN2O3S/c1-15(2)19(16,17)12-5-3-11(4-6-12)18-9-10(7-13)8-14/h3-7H,8-9,14H2,1-2H3/b10-7+
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n/an/a>1.00E+4n/an/an/an/an/an/a



BOEHRINGER INGELHEIM INTERNATIONAL GMBH

US Patent


Assay Description
Recombinant human DAO (2.4 μg/mL) was used as source of DAO enzyme activities. The assay was performed as described in the method for human SSAO/V...


US Patent US9302986 (2016)

More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM220874
PNG
(US9302986, 11)
Show SMILES NC\C(COc1ccc(cc1)S(N)(=O)=O)=C/F
Show InChI InChI=1S/C10H13FN2O3S/c11-5-8(6-12)7-16-9-1-3-10(4-2-9)17(13,14)15/h1-5H,6-7,12H2,(H2,13,14,15)/b8-5+
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n/an/a>1.00E+4n/an/an/an/an/an/a



BOEHRINGER INGELHEIM INTERNATIONAL GMBH

US Patent


Assay Description
Recombinant human DAO (2.4 μg/mL) was used as source of DAO enzyme activities. The assay was performed as described in the method for human SSAO/V...


US Patent US9302986 (2016)

More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM50161148
PNG
(4-(aminomethyl)-N-cyclohexylpyridin-3-amine dihydr...)
Show SMILES NCc1ccncc1NC1CCCCC1
Show InChI InChI=1S/C12H19N3/c13-8-10-6-7-14-9-12(10)15-11-4-2-1-3-5-11/h6-7,9,11,15H,1-5,8,13H2
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n/an/a 1.60E+4n/an/an/an/an/an/a



Universit£ di Genova

Curated by ChEMBL


Assay Description
Inhibition of putrescine binding to against Diamine oxidase of porcine kidney


Citation and Details
More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM50161152
PNG
(4-(aminomethyl)-N-isopropylpyridin-3-amine dihydro...)
Show SMILES CC(C)Nc1cnccc1CN
Show InChI InChI=1S/C9H15N3/c1-7(2)12-9-6-11-4-3-8(9)5-10/h3-4,6-7,12H,5,10H2,1-2H3
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n/an/a 1.60E+4n/an/an/an/an/an/a



Universit£ di Genova

Curated by ChEMBL


Assay Description
Inhibition of putrescine binding to Diamine oxidase of porcine kidney


Citation and Details
More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM50161133
PNG
(4-(aminomethyl)-N-cycloheptylpyridin-3-amine dihyd...)
Show SMILES NCc1ccncc1NC1CCCCCC1
Show InChI InChI=1S/C13H21N3/c14-9-11-7-8-15-10-13(11)16-12-5-3-1-2-4-6-12/h7-8,10,12,16H,1-6,9,14H2
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n/an/a 1.80E+4n/an/an/an/an/an/a



Universit£ di Genova

Curated by ChEMBL


Assay Description
Inhibition of putrescine binding to against Diamine oxidase of porcine kidney


Citation and Details
More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM50161139
PNG
(4-(aminomethyl)-N-cyclopentylpyridin-3-amine dihyd...)
Show SMILES NCc1ccncc1NC1CCCC1
Show InChI InChI=1S/C11H17N3/c12-7-9-5-6-13-8-11(9)14-10-3-1-2-4-10/h5-6,8,10,14H,1-4,7,12H2
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n/an/a 1.90E+4n/an/an/an/an/an/a



Universit£ di Genova

Curated by ChEMBL


Assay Description
Inhibition of putrescine binding to against Diamine oxidase of porcine kidney


Citation and Details
More data for this
Ligand-Target Pair
Diamine oxidase (DAO)


(Homo sapiens)
BDBM50161140
PNG
(4-(aminomethyl)-N-(cyclohexylmethyl)pyridin-3-amin...)
Show SMILES NCc1ccncc1NCC1CCCCC1
Show InChI InChI=1S/C13H21N3/c14-8-12-6-7-15-10-13(12)16-9-11-4-2-1-3-5-11/h6-7,10-11,16H,1-5,8-9,14H2
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n/an/a 5.00E+4n/an/an/an/an/an/a



Universit£ di Genova

Curated by ChEMBL


Assay Description
Inhibition of putrescine binding to against Diamine oxidase of porcine kidney


Citation and Details
More data for this
Ligand-Target Pair
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