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Found 27 hits Enz. Inhib. hit(s) with Target = 'Dihydrofolate reductase (DHFR)' AND taxid = 226900   
Target
(Institution)
LigandTarget
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Dihydrofolate Reductase (DHFR)


(Bacillus cereus (ATCC 14579))
BDBM18050
PNG
(2-[(4-{[(2,4-diaminopteridin-6-yl)methyl](methyl)a...)
Show SMILES CN(Cc1cnc2nc(N)nc(N)c2n1)c1ccc(cc1)C(=O)N[C@@H](CCC(O)=O)C(O)=O
Show InChI InChI=1S/C20H22N8O5/c1-28(9-11-8-23-17-15(24-11)16(21)26-20(22)27-17)12-4-2-10(3-5-12)18(31)25-13(19(32)33)6-7-14(29)30/h2-5,8,13H,6-7,9H2,1H3,(H,25,31)(H,29,30)(H,32,33)(H4,21,22,23,26,27)/t13-/m0/s1
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PubMed
n/an/a 24n/an/an/an/a7.025



University of Connecticut at Storrs



Assay Description
Enzyme activity assays were performed by monitoring the rate of enzyme-dependent NADPH consumption at an absorbance of 340 nm over a period of severa...


Citation and Details
More data for this
Ligand-Target Pair
3D
3D Structure (crystal)
Dihydrofolate Reductase (DHFR)


(Bacillus cereus (ATCC 14579))
BDBM18231
PNG
(2,4-diamino-5-deazapteridine, 2 | 7-[3-({2,4-diami...)
Show SMILES COc1ccc(cc1Cc1cnc2nc(N)nc(N)c2c1C)C#CCCCCC(O)=O
Show InChI InChI=1S/C23H25N5O3/c1-14-17(13-26-22-20(14)21(24)27-23(25)28-22)12-16-11-15(9-10-18(16)31-2)7-5-3-4-6-8-19(29)30/h9-11,13H,3-4,6,8,12H2,1-2H3,(H,29,30)(H4,24,25,26,27,28)
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PubMed
n/an/a 270n/an/an/an/a7.025



University of Connecticut at Storrs



Assay Description
Enzyme activity assays were performed by monitoring the rate of enzyme-dependent NADPH consumption at an absorbance of 340 nm over a period of severa...


Citation and Details
More data for this
Ligand-Target Pair
Dihydrofolate Reductase (DHFR)


(Bacillus cereus (ATCC 14579))
BDBM18239
PNG
(2,4-diamino-5-deazapteridine, 8 | Piritrexim analo...)
Show SMILES CCOC(=O)CCCCOc1ccc(OC)c(Cc2cnc3nc(N)nc(N)c3c2C)c1
Show InChI InChI=1S/C23H29N5O4/c1-4-31-19(29)7-5-6-10-32-17-8-9-18(30-3)15(12-17)11-16-13-26-22-20(14(16)2)21(24)27-23(25)28-22/h8-9,12-13H,4-7,10-11H2,1-3H3,(H4,24,25,26,27,28)
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PubMed
n/an/a 350n/an/an/an/a7.025



University of Connecticut at Storrs



Assay Description
Enzyme activity assays were performed by monitoring the rate of enzyme-dependent NADPH consumption at an absorbance of 340 nm over a period of severa...


Citation and Details
More data for this
Ligand-Target Pair
Dihydrofolate Reductase (DHFR)


(Bacillus cereus (ATCC 14579))
BDBM18227
PNG
(2,4-diamino-5-deazapteridine, 6 | 6-[3-({2,4-diami...)
Show SMILES COc1ccc(OCCCCCC(O)=O)cc1Cc1cnc2nc(N)nc(N)c2c1C
Show InChI InChI=1S/C22H27N5O4/c1-13-15(12-25-21-19(13)20(23)26-22(24)27-21)10-14-11-16(7-8-17(14)30-2)31-9-5-3-4-6-18(28)29/h7-8,11-12H,3-6,9-10H2,1-2H3,(H,28,29)(H4,23,24,25,26,27)
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n/an/a 510n/an/an/an/a7.025



University of Connecticut at Storrs



Assay Description
Enzyme activity assays were performed by monitoring the rate of enzyme-dependent NADPH consumption at an absorbance of 340 nm over a period of severa...


Citation and Details
More data for this
Ligand-Target Pair
Dihydrofolate Reductase (DHFR)


(Bacillus cereus (ATCC 14579))
BDBM18225
PNG
(2,4-diamino-5-deazapteridine, 4 | 4-[3-({2,4-diami...)
Show SMILES COc1ccc(OCCCC(O)=O)cc1Cc1cnc2nc(N)nc(N)c2c1C
Show InChI InChI=1S/C20H23N5O4/c1-11-13(10-23-19-17(11)18(21)24-20(22)25-19)8-12-9-14(5-6-15(12)28-2)29-7-3-4-16(26)27/h5-6,9-10H,3-4,7-8H2,1-2H3,(H,26,27)(H4,21,22,23,24,25)
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PubMed
n/an/a 600n/an/an/an/a7.025



University of Connecticut at Storrs



Assay Description
Enzyme activity assays were performed by monitoring the rate of enzyme-dependent NADPH consumption at an absorbance of 340 nm over a period of severa...


Citation and Details
More data for this
Ligand-Target Pair
Dihydrofolate Reductase (DHFR)


(Bacillus cereus (ATCC 14579))
BDBM18238
PNG
(2,4-diamino-5-deazapteridine, 7 | Piritrexim analo...)
Show SMILES CCOC(=O)CCCOc1ccc(OC)c(Cc2cnc3nc(N)nc(N)c3c2C)c1
Show InChI InChI=1S/C22H27N5O4/c1-4-30-18(28)6-5-9-31-16-7-8-17(29-3)14(11-16)10-15-12-25-21-19(13(15)2)20(23)26-22(24)27-21/h7-8,11-12H,4-6,9-10H2,1-3H3,(H4,23,24,25,26,27)
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n/an/a 880n/an/an/an/a7.025



University of Connecticut at Storrs



Assay Description
Enzyme activity assays were performed by monitoring the rate of enzyme-dependent NADPH consumption at an absorbance of 340 nm over a period of severa...


Citation and Details
More data for this
Ligand-Target Pair
Dihydrofolate Reductase (DHFR)


(Bacillus cereus (ATCC 14579))
BDBM18499
PNG
(6-{[(2-bromo-3,4,5-trimethoxyphenyl)amino]methyl}q...)
Show SMILES COc1cc(NCc2ccc3nc(N)nc(N)c3c2)c(Br)c(OC)c1OC
Show InChI InChI=1S/C18H20BrN5O3/c1-25-13-7-12(14(19)16(27-3)15(13)26-2)22-8-9-4-5-11-10(6-9)17(20)24-18(21)23-11/h4-7,22H,8H2,1-3H3,(H4,20,21,23,24)
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PubMed
n/an/a 1.10E+3n/an/an/an/a7.025



University of Connecticut at Storrs



Assay Description
Enzyme activity assays were performed by monitoring the rate of enzyme-dependent NADPH consumption at an absorbance of 340 nm over a period of severa...


Citation and Details
More data for this
Ligand-Target Pair
Dihydrofolate Reductase (DHFR)


(Bacillus cereus (ATCC 14579))
BDBM18226
PNG
(2,4-diamino-5-deazapteridine, 5 | 5-[3-({2,4-diami...)
Show SMILES COc1ccc(OCCCCC(O)=O)cc1Cc1cnc2nc(N)nc(N)c2c1C
Show InChI InChI=1S/C21H25N5O4/c1-12-14(11-24-20-18(12)19(22)25-21(23)26-20)9-13-10-15(6-7-16(13)29-2)30-8-4-3-5-17(27)28/h6-7,10-11H,3-5,8-9H2,1-2H3,(H,27,28)(H4,22,23,24,25,26)
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PubMed
n/an/a 1.67E+3n/an/an/an/a7.025



University of Connecticut at Storrs



Assay Description
Enzyme activity assays were performed by monitoring the rate of enzyme-dependent NADPH consumption at an absorbance of 340 nm over a period of severa...


Citation and Details
More data for this
Ligand-Target Pair
Dihydrofolate Reductase (DHFR)


(Bacillus cereus (ATCC 14579))
BDBM18240
PNG
(2,4-diamino-5-deazapteridine, 9 | Piritrexim analo...)
Show SMILES CCOC(=O)CCCCCOc1ccc(OC)c(Cc2cnc3nc(N)nc(N)c3c2C)c1
Show InChI InChI=1S/C24H31N5O4/c1-4-32-20(30)8-6-5-7-11-33-18-9-10-19(31-3)16(13-18)12-17-14-27-23-21(15(17)2)22(25)28-24(26)29-23/h9-10,13-14H,4-8,11-12H2,1-3H3,(H4,25,26,27,28,29)
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n/an/a 1.85E+3n/an/an/an/a7.025



University of Connecticut at Storrs



Assay Description
Enzyme activity assays were performed by monitoring the rate of enzyme-dependent NADPH consumption at an absorbance of 340 nm over a period of severa...


Citation and Details
More data for this
Ligand-Target Pair
Dihydrofolate Reductase (DHFR)


(Bacillus cereus (ATCC 14579))
BDBM18230
PNG
(2,4-diamino-5-deazapteridine, 10 | 6-[3-({2,4-diam...)
Show SMILES COc1ccc(cc1Cc1cnc2nc(N)nc(N)c2c1C)C#CCCCC(O)=O
Show InChI InChI=1S/C22H23N5O3/c1-13-16(12-25-21-19(13)20(23)26-22(24)27-21)11-15-10-14(8-9-17(15)30-2)6-4-3-5-7-18(28)29/h8-10,12H,3,5,7,11H2,1-2H3,(H,28,29)(H4,23,24,25,26,27)
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n/an/a 1.90E+3n/an/an/an/a7.025



University of Connecticut at Storrs



Assay Description
Enzyme activity assays were performed by monitoring the rate of enzyme-dependent NADPH consumption at an absorbance of 340 nm over a period of severa...


Citation and Details
More data for this
Ligand-Target Pair
Dihydrofolate Reductase (DHFR)


(Bacillus cereus (ATCC 14579))
BDBM18502
PNG
(6-{[(6-chloronaphthalen-2-yl)(methyl)amino]methyl}...)
Show SMILES CN(Cc1cnc2nc(N)nc(N)c2n1)c1ccc2cc(Cl)ccc2c1
Show InChI InChI=1S/C18H16ClN7/c1-26(14-5-3-10-6-12(19)4-2-11(10)7-14)9-13-8-22-17-15(23-13)16(20)24-18(21)25-17/h2-8H,9H2,1H3,(H4,20,21,22,24,25)
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PubMed
n/an/a 2.26E+3n/an/an/an/a7.025



University of Connecticut at Storrs



Assay Description
Enzyme activity assays were performed by monitoring the rate of enzyme-dependent NADPH consumption at an absorbance of 340 nm over a period of severa...


Citation and Details
More data for this
Ligand-Target Pair
Dihydrofolate Reductase (DHFR)


(Bacillus cereus (ATCC 14579))
BDBM18500
PNG
(6-{[(6,7-dichloronaphthalen-2-yl)amino]methyl}pter...)
Show SMILES Nc1nc(N)c2nc(CNc3ccc4cc(Cl)c(Cl)cc4c3)cnc2n1
Show InChI InChI=1S/C17H13Cl2N7/c18-12-4-8-1-2-10(3-9(8)5-13(12)19)22-6-11-7-23-16-14(24-11)15(20)25-17(21)26-16/h1-5,7,22H,6H2,(H4,20,21,23,25,26)
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PubMed
n/an/a 4.82E+3n/an/an/an/a7.025



University of Connecticut at Storrs



Assay Description
Enzyme activity assays were performed by monitoring the rate of enzyme-dependent NADPH consumption at an absorbance of 340 nm over a period of severa...


Citation and Details
More data for this
Ligand-Target Pair
Dihydrofolate Reductase (DHFR)


(Bacillus cereus (ATCC 14579))
BDBM18501
PNG
(6-{[(6-chloronaphthalen-2-yl)amino]methyl}pteridin...)
Show SMILES Nc1nc(N)c2nc(CNc3ccc4cc(Cl)ccc4c3)cnc2n1
Show InChI InChI=1S/C17H14ClN7/c18-11-3-1-10-6-12(4-2-9(10)5-11)21-7-13-8-22-16-14(23-13)15(19)24-17(20)25-16/h1-6,8,21H,7H2,(H4,19,20,22,24,25)
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PubMed
n/an/a 6.32E+3n/an/an/an/a7.025



University of Connecticut at Storrs



Assay Description
Enzyme activity assays were performed by monitoring the rate of enzyme-dependent NADPH consumption at an absorbance of 340 nm over a period of severa...


Citation and Details
More data for this
Ligand-Target Pair
Dihydrofolate Reductase (DHFR)


(Bacillus cereus (ATCC 14579))
BDBM18503
PNG
(6-{[(5,7-dichloronaphthalen-2-yl)amino]methyl}pter...)
Show SMILES Nc1nc(N)c2nc(CNc3ccc4c(Cl)cc(Cl)cc4c3)cnc2n1
Show InChI InChI=1S/C17H13Cl2N7/c18-9-3-8-4-10(1-2-12(8)13(19)5-9)22-6-11-7-23-16-14(24-11)15(20)25-17(21)26-16/h1-5,7,22H,6H2,(H4,20,21,23,25,26)
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n/an/a 7.58E+3n/an/an/an/a7.025



University of Connecticut at Storrs



Assay Description
Enzyme activity assays were performed by monitoring the rate of enzyme-dependent NADPH consumption at an absorbance of 340 nm over a period of severa...


Citation and Details
More data for this
Ligand-Target Pair
Dihydrofolate Reductase (DHFR)


(Bacillus cereus (ATCC 14579))
BDBM18506
PNG
(6-{2-azatricyclo[9.4.0.0^{3,8}]pentadeca-1(11),3(8...)
Show SMILES Nc1nc(N)c2nc(CN3c4ccccc4C=Cc4ccccc34)cnc2n1
Show InChI InChI=1S/C21H17N7/c22-19-18-20(27-21(23)26-19)24-11-15(25-18)12-28-16-7-3-1-5-13(16)9-10-14-6-2-4-8-17(14)28/h1-11H,12H2,(H4,22,23,24,26,27)
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n/an/a 1.67E+4n/an/an/an/a7.025



University of Connecticut at Storrs



Assay Description
Enzyme activity assays were performed by monitoring the rate of enzyme-dependent NADPH consumption at an absorbance of 340 nm over a period of severa...


Citation and Details
More data for this
Ligand-Target Pair
Dihydrofolate Reductase (DHFR)


(Bacillus cereus (ATCC 14579))
BDBM18504
PNG
(6-{[(5,7-dichloronaphthalen-2-yl)(methyl)amino]met...)
Show SMILES CN(Cc1cnc2nc(N)nc(N)c2n1)c1ccc2c(Cl)cc(Cl)cc2c1
Show InChI InChI=1S/C18H15Cl2N7/c1-27(12-2-3-13-9(5-12)4-10(19)6-14(13)20)8-11-7-23-17-15(24-11)16(21)25-18(22)26-17/h2-7H,8H2,1H3,(H4,21,22,23,25,26)
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n/an/a 1.76E+4n/an/an/an/a7.025



University of Connecticut at Storrs



Assay Description
Enzyme activity assays were performed by monitoring the rate of enzyme-dependent NADPH consumption at an absorbance of 340 nm over a period of severa...


Citation and Details
More data for this
Ligand-Target Pair
Dihydrofolate Reductase (DHFR)


(Bacillus cereus (ATCC 14579))
BDBM18508
PNG
(5-[(5-iodo-2-methoxyphenyl)methyl]pyrimidine-2,4-d...)
Show SMILES COc1ccc(I)cc1Cc1cnc(N)nc1N
Show InChI InChI=1S/C12H13IN4O/c1-18-10-3-2-9(13)5-7(10)4-8-6-16-12(15)17-11(8)14/h2-3,5-6H,4H2,1H3,(H4,14,15,16,17)
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n/an/a 3.73E+4n/an/an/an/a7.025



University of Connecticut at Storrs



Assay Description
Enzyme activity assays were performed by monitoring the rate of enzyme-dependent NADPH consumption at an absorbance of 340 nm over a period of severa...


Citation and Details
More data for this
Ligand-Target Pair
Dihydrofolate Reductase (DHFR)


(Bacillus cereus (ATCC 14579))
BDBM18069
PNG
(5-[(3,4,5-trimethoxyphenyl)methyl]pyrimidine-2,4-d...)
Show SMILES COc1cc(Cc2cnc(N)nc2N)cc(OC)c1OC
Show InChI InChI=1S/C14H18N4O3/c1-19-10-5-8(6-11(20-2)12(10)21-3)4-9-7-17-14(16)18-13(9)15/h5-7H,4H2,1-3H3,(H4,15,16,17,18)
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PubMed
n/an/a 4.30E+4n/an/an/an/a7.025



University of Connecticut at Storrs



Assay Description
Enzyme activity assays were performed by monitoring the rate of enzyme-dependent NADPH consumption at an absorbance of 340 nm over a period of severa...


Citation and Details
More data for this
Ligand-Target Pair
3D
3D Structure (crystal)
Dihydrofolate Reductase (DHFR)


(Bacillus cereus (ATCC 14579))
BDBM18509
PNG
(7-{3-[(2,4-diaminopyrimidin-5-yl)methyl]-4-methoxy...)
Show SMILES COc1ccc(cc1Cc1cnc(N)nc1N)C#CCCCCC(O)=O
Show InChI InChI=1S/C19H22N4O3/c1-26-16-9-8-13(6-4-2-3-5-7-17(24)25)10-14(16)11-15-12-22-19(21)23-18(15)20/h8-10,12H,2-3,5,7,11H2,1H3,(H,24,25)(H4,20,21,22,23)
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PubMed
n/an/a 6.93E+4n/an/an/an/a7.025



University of Connecticut at Storrs



Assay Description
Enzyme activity assays were performed by monitoring the rate of enzyme-dependent NADPH consumption at an absorbance of 340 nm over a period of severa...


Citation and Details
More data for this
Ligand-Target Pair
Dihydrofolate Reductase (DHFR)


(Bacillus cereus (ATCC 14579))
BDBM18510
PNG
(5-{3-[(2,4-diaminopyrimidin-5-yl)methyl]-4-methoxy...)
Show SMILES COc1ccc(OCCCCC(O)=O)cc1Cc1cnc(N)nc1N
Show InChI InChI=1S/C17H22N4O4/c1-24-14-6-5-13(25-7-3-2-4-15(22)23)9-11(14)8-12-10-20-17(19)21-16(12)18/h5-6,9-10H,2-4,7-8H2,1H3,(H,22,23)(H4,18,19,20,21)
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PubMed
n/an/a 7.37E+4n/an/an/an/a7.025



University of Connecticut at Storrs



Assay Description
Enzyme activity assays were performed by monitoring the rate of enzyme-dependent NADPH consumption at an absorbance of 340 nm over a period of severa...


Citation and Details
More data for this
Ligand-Target Pair
Dihydrofolate Reductase (DHFR)


(Bacillus cereus (ATCC 14579))
BDBM18511
PNG
(6-{3-[(2,4-diaminopyrimidin-5-yl)methyl]-4-methoxy...)
Show SMILES COc1ccc(CCCCCC(O)=O)cc1Cc1cnc(N)nc1N
Show InChI InChI=1S/C18H24N4O3/c1-25-15-8-7-12(5-3-2-4-6-16(23)24)9-13(15)10-14-11-21-18(20)22-17(14)19/h7-9,11H,2-6,10H2,1H3,(H,23,24)(H4,19,20,21,22)
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n/an/a 1.50E+5n/an/an/an/a7.025



University of Connecticut at Storrs



Assay Description
Enzyme activity assays were performed by monitoring the rate of enzyme-dependent NADPH consumption at an absorbance of 340 nm over a period of severa...


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More data for this
Ligand-Target Pair
Dihydrofolate Reductase (DHFR)


(Bacillus cereus (ATCC 14579))
BDBM18507
PNG
(5-[2-(3,4,5-trimethoxyphenyl)ethyl]-7H-pyrrolo[2,3...)
Show SMILES COc1cc(CCc2c[nH]c3nc(N)nc(N)c23)cc(OC)c1OC
Show InChI InChI=1S/C17H21N5O3/c1-23-11-6-9(7-12(24-2)14(11)25-3)4-5-10-8-20-16-13(10)15(18)21-17(19)22-16/h6-8H,4-5H2,1-3H3,(H5,18,19,20,21,22)
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n/an/a 2.52E+5n/an/an/an/a7.025



University of Connecticut at Storrs



Assay Description
Enzyme activity assays were performed by monitoring the rate of enzyme-dependent NADPH consumption at an absorbance of 340 nm over a period of severa...


Citation and Details
More data for this
Ligand-Target Pair
Dihydrofolate Reductase (DHFR)


(Bacillus cereus (ATCC 14579))
BDBM18514
PNG
(4,6-diazatetracyclo[8.8.0.0^{2,7}.0^{11,16}]octade...)
Show SMILES Nc1nc(N)c2c(ccc3c4ccccc4ccc23)n1
Show InChI InChI=1S/C16H12N4/c17-15-14-12-6-5-9-3-1-2-4-10(9)11(12)7-8-13(14)19-16(18)20-15/h1-8H,(H4,17,18,19,20)
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n/an/a>1.00E+6n/an/an/an/a7.025



University of Connecticut at Storrs



Assay Description
Enzyme activity assays were performed by monitoring the rate of enzyme-dependent NADPH consumption at an absorbance of 340 nm over a period of severa...


Citation and Details
More data for this
Ligand-Target Pair
Dihydrofolate Reductase (DHFR)


(Bacillus cereus (ATCC 14579))
BDBM18513
PNG
(1,3-diazatetraphene-2,4-diamine | Diaminonaphthoqu...)
Show SMILES Nc1nc(N)c2cc3c(ccc4ccccc34)cc2n1
Show InChI InChI=1S/C16H12N4/c17-15-13-8-12-10(7-14(13)19-16(18)20-15)6-5-9-3-1-2-4-11(9)12/h1-8H,(H4,17,18,19,20)
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n/an/a>1.00E+6n/an/an/an/a7.025



University of Connecticut at Storrs



Assay Description
Enzyme activity assays were performed by monitoring the rate of enzyme-dependent NADPH consumption at an absorbance of 340 nm over a period of severa...


Citation and Details
More data for this
Ligand-Target Pair
Dihydrofolate Reductase (DHFR)


(Bacillus cereus (ATCC 14579))
BDBM18512
PNG
(5-(4-chlorophenyl)-6-ethylpyrimidine-2,4-diamine |...)
Show SMILES CCc1nc(N)nc(N)c1-c1ccc(Cl)cc1
Show InChI InChI=1S/C12H13ClN4/c1-2-9-10(11(14)17-12(15)16-9)7-3-5-8(13)6-4-7/h3-6H,2H2,1H3,(H4,14,15,16,17)
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n/an/a>1.00E+6n/an/an/an/a7.025



University of Connecticut at Storrs



Assay Description
Enzyme activity assays were performed by monitoring the rate of enzyme-dependent NADPH consumption at an absorbance of 340 nm over a period of severa...


Citation and Details
More data for this
Ligand-Target Pair
Dihydrofolate Reductase (DHFR)


(Bacillus cereus (ATCC 14579))
BDBM18505
PNG
(6-{[(5,7-dichloronaphthalen-2-yl)(methyl)amino]met...)
Show SMILES CN(Cc1nc2c(N)nc(N)nc2nc1C)c1ccc2c(Cl)cc(Cl)cc2c1
Show InChI InChI=1S/C19H17Cl2N7/c1-9-15(25-16-17(22)26-19(23)27-18(16)24-9)8-28(2)12-3-4-13-10(6-12)5-11(20)7-14(13)21/h3-7H,8H2,1-2H3,(H4,22,23,24,26,27)
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n/an/a>1.00E+6n/an/an/an/a7.025



University of Connecticut at Storrs



Assay Description
Enzyme activity assays were performed by monitoring the rate of enzyme-dependent NADPH consumption at an absorbance of 340 nm over a period of severa...


Citation and Details
More data for this
Ligand-Target Pair
Dihydrofolate Reductase (DHFR)


(Bacillus cereus (ATCC 14579))
BDBM18515
PNG
(1,3-diazatetraphene-2,4-diamine | Diaminonaphthoqu...)
Show SMILES Nc1nc(N)c2c(ccc3cc4ccccc4cc23)n1
Show InChI InChI=1S/C16H12N4/c17-15-14-12-8-10-4-2-1-3-9(10)7-11(12)5-6-13(14)19-16(18)20-15/h1-8H,(H4,17,18,19,20)
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n/an/a>1.00E+6n/an/an/an/a7.025



University of Connecticut at Storrs



Assay Description
Enzyme activity assays were performed by monitoring the rate of enzyme-dependent NADPH consumption at an absorbance of 340 nm over a period of severa...


Citation and Details
More data for this
Ligand-Target Pair