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Found 344 hits Enz. Inhib. hit(s) with Target = 'Glutamate [NMDA] receptor subunit epsilon 3/zeta 1' AND taxid = 10116   
Target
(Institution)
LigandTarget
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50111396
PNG
(CHEMBL273636 | [[(S)-1-(4-Bromo-phenyl)-ethylamino...)
Show SMILES C[C@H](NC(c1cccc2[nH]c(=O)c(=O)[nH]c12)P(O)(O)=O)c1ccc(Br)cc1
Show InChI InChI=1S/C17H17BrN3O5P/c1-9(10-5-7-11(18)8-6-10)19-17(27(24,25)26)12-3-2-4-13-14(12)21-16(23)15(22)20-13/h2-9,17,19H,1H3,(H,20,22)(H,21,23)(H2,24,25,26)/t9-,17?/m0/s1
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11.6n/an/an/an/an/an/an/an/a



University Walk

Curated by ChEMBL


Assay Description
Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50419775
PNG
(CHEMBL1950808)
Show SMILES OC(=O)[C@@H]1NCCN([C@@H]1C(O)=O)C(=O)c1ccc2c(ccc3ccccc23)c1
Show InChI InChI=1S/C21H18N2O5/c24-19(23-10-9-22-17(20(25)26)18(23)21(27)28)14-7-8-16-13(11-14)6-5-12-3-1-2-4-15(12)16/h1-8,11,17-18,22H,9-10H2,(H,25,26)(H,27,28)/t17-,18+/m1/s1
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70n/an/an/an/an/an/an/an/a



University of Bristol

Curated by ChEMBL


Assay Description
Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50164540
PNG
((2R,3S)-1-(Phenanthrene-2-carbonyl)-piperazine-2,3...)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc2c(ccc3ccccc23)c1
Show InChI InChI=1S/C21H18N2O5/c24-19(23-10-9-22-17(20(25)26)18(23)21(27)28)14-7-8-16-13(11-14)6-5-12-3-1-2-4-15(12)16/h1-8,11,17-18,22H,9-10H2,(H,25,26)(H,27,28)/t17-,18+/m0/s1
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96n/an/an/an/an/an/an/an/a



University Walk

Curated by ChEMBL


Assay Description
Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50164549
PNG
((2R,3S)-1-(7-Bromo-phenanthrene-2-carbonyl)-pipera...)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc2c(ccc3cc(Br)ccc23)c1
Show InChI InChI=1S/C21H17BrN2O5/c22-14-4-6-16-12(10-14)2-1-11-9-13(3-5-15(11)16)19(25)24-8-7-23-17(20(26)27)18(24)21(28)29/h1-6,9-10,17-18,23H,7-8H2,(H,26,27)(H,28,29)/t17-,18+/m0/s1
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99.4n/an/an/an/an/an/an/an/a



University Walk

Curated by ChEMBL


Assay Description
Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50164540
PNG
((2R,3S)-1-(Phenanthrene-2-carbonyl)-piperazine-2,3...)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc2c(ccc3ccccc23)c1
Show InChI InChI=1S/C21H18N2O5/c24-19(23-10-9-22-17(20(25)26)18(23)21(27)28)14-7-8-16-13(11-14)6-5-12-3-1-2-4-15(12)16/h1-8,11,17-18,22H,9-10H2,(H,25,26)(H,27,28)/t17-,18+/m0/s1
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100n/an/an/an/an/an/an/an/a



University of Bristol

Curated by ChEMBL


Assay Description
Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50164549
PNG
((2R,3S)-1-(7-Bromo-phenanthrene-2-carbonyl)-pipera...)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc2c(ccc3cc(Br)ccc23)c1
Show InChI InChI=1S/C21H17BrN2O5/c22-14-4-6-16-12(10-14)2-1-11-9-13(3-5-15(11)16)19(25)24-8-7-23-17(20(26)27)18(24)21(28)29/h1-6,9-10,17-18,23H,7-8H2,(H,26,27)(H,28,29)/t17-,18+/m0/s1
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100n/an/an/an/an/an/an/an/a



University of Bristol

Curated by ChEMBL


Assay Description
Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50164555
PNG
((2R,3S)-1-(9,10-Dihydro-phenanthrene-2-carbonyl)-p...)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc-2c(CCc3ccccc-23)c1
Show InChI InChI=1S/C21H20N2O5/c24-19(23-10-9-22-17(20(25)26)18(23)21(27)28)14-7-8-16-13(11-14)6-5-12-3-1-2-4-15(12)16/h1-4,7-8,11,17-18,22H,5-6,9-10H2,(H,25,26)(H,27,28)/t17-,18+/m0/s1
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290n/an/an/an/an/an/an/an/a



University Walk

Curated by ChEMBL


Assay Description
Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50164555
PNG
((2R,3S)-1-(9,10-Dihydro-phenanthrene-2-carbonyl)-p...)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc-2c(CCc3ccccc-23)c1
Show InChI InChI=1S/C21H20N2O5/c24-19(23-10-9-22-17(20(25)26)18(23)21(27)28)14-7-8-16-13(11-14)6-5-12-3-1-2-4-15(12)16/h1-4,7-8,11,17-18,22H,5-6,9-10H2,(H,25,26)(H,27,28)/t17-,18+/m0/s1
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290n/an/an/an/an/an/an/an/a



University of Bristol

Curated by ChEMBL


Assay Description
Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50050704
PNG
((R)-4-(3-Phosphono-propyl)-piperazine-2-carboxylic...)
Show SMILES OC(=O)[C@H]1CN(CCCP(O)(O)=O)CCN1
Show InChI InChI=1S/C8H17N2O5P/c11-8(12)7-6-10(4-2-9-7)3-1-5-16(13,14)15/h7,9H,1-6H2,(H,11,12)(H2,13,14,15)/t7-/m1/s1
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630n/an/an/an/an/an/an/an/a



University Walk

Curated by ChEMBL


Assay Description
Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50164548
PNG
((2R,3S)-1-(7-Bromo-9,10-dihydro-phenanthrene-2-car...)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc-2c(CCc3cc(Br)ccc-23)c1
Show InChI InChI=1S/C21H19BrN2O5/c22-14-4-6-16-12(10-14)2-1-11-9-13(3-5-15(11)16)19(25)24-8-7-23-17(20(26)27)18(24)21(28)29/h3-6,9-10,17-18,23H,1-2,7-8H2,(H,26,27)(H,28,29)/t17-,18+/m0/s1
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660n/an/an/an/an/an/an/an/a



University of Bristol

Curated by ChEMBL


Assay Description
Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50164548
PNG
((2R,3S)-1-(7-Bromo-9,10-dihydro-phenanthrene-2-car...)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc-2c(CCc3cc(Br)ccc-23)c1
Show InChI InChI=1S/C21H19BrN2O5/c22-14-4-6-16-12(10-14)2-1-11-9-13(3-5-15(11)16)19(25)24-8-7-23-17(20(26)27)18(24)21(28)29/h3-6,9-10,17-18,23H,1-2,7-8H2,(H,26,27)(H,28,29)/t17-,18+/m0/s1
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660n/an/an/an/an/an/an/an/a



University Walk

Curated by ChEMBL


Assay Description
Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50164556
PNG
((2R,3S)-1-((E)-3-Naphthalen-2-yl-acryloyl)-piperaz...)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)\C=C\c1ccc2ccccc2c1
Show InChI InChI=1S/C19H18N2O5/c22-15(21-10-9-20-16(18(23)24)17(21)19(25)26)8-6-12-5-7-13-3-1-2-4-14(13)11-12/h1-8,11,16-17,20H,9-10H2,(H,23,24)(H,25,26)/b8-6+/t16-,17+/m0/s1
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850n/an/an/an/an/an/an/an/a



University Walk

Curated by ChEMBL


Assay Description
Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50164546
PNG
((2R,3S)-1-(9H-Fluorene-2-carbonyl)-piperazine-2,3-...)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc-2c(Cc3ccccc-23)c1
Show InChI InChI=1S/C20H18N2O5/c23-18(22-8-7-21-16(19(24)25)17(22)20(26)27)12-5-6-15-13(10-12)9-11-3-1-2-4-14(11)15/h1-6,10,16-17,21H,7-9H2,(H,24,25)(H,26,27)/t16-,17+/m0/s1
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1.17E+3n/an/an/an/an/an/an/an/a



University Walk

Curated by ChEMBL


Assay Description
Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50004897
PNG
((APV)2-Amino-5-phosphono-pentanoic acid | (R)-2-Am...)
Show SMILES NC(CCCP(O)(O)=O)C(O)=O
Show InChI InChI=1S/C5H12NO5P/c6-4(5(7)8)2-1-3-12(9,10)11/h4H,1-3,6H2,(H,7,8)(H2,9,10,11)
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1.64E+3n/an/an/an/an/an/an/an/a



University Walk

Curated by ChEMBL


Assay Description
Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50419786
PNG
(CHEMBL1950795)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc2cc(I)ccc2c1
Show InChI InChI=1S/C17H15IN2O5/c18-12-4-3-9-7-11(2-1-10(9)8-12)15(21)20-6-5-19-13(16(22)23)14(20)17(24)25/h1-4,7-8,13-14,19H,5-6H2,(H,22,23)(H,24,25)/t13-,14+/m0/s1
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1.80E+3n/an/an/an/an/an/an/an/a



University of Bristol

Curated by ChEMBL


Assay Description
Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50364074
PNG
(CHEMBL1950805)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc2cc(I)c3ccccc3c2c1
Show InChI InChI=1S/C21H17IN2O5/c22-16-10-11-5-6-12(9-15(11)13-3-1-2-4-14(13)16)19(25)24-8-7-23-17(20(26)27)18(24)21(28)29/h1-6,9-10,17-18,23H,7-8H2,(H,26,27)(H,28,29)/t17-,18+/m0/s1
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1.90E+3n/an/an/an/an/an/an/an/a



University of Bristol

Curated by ChEMBL


Assay Description
Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50419787
PNG
(CHEMBL1950794)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc2cc(Br)ccc2c1
Show InChI InChI=1S/C17H15BrN2O5/c18-12-4-3-9-7-11(2-1-10(9)8-12)15(21)20-6-5-19-13(16(22)23)14(20)17(24)25/h1-4,7-8,13-14,19H,5-6H2,(H,22,23)(H,24,25)/t13-,14+/m0/s1
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2.10E+3n/an/an/an/an/an/an/an/a



University of Bristol

Curated by ChEMBL


Assay Description
Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50164541
PNG
((2R,3S)-1-Phenanthren-2-ylmethyl-piperazine-2,3-di...)
Show SMILES OC(=O)[C@H]1NCCN(Cc2ccc3c(ccc4ccccc34)c2)[C@H]1C(O)=O
Show InChI InChI=1S/C21H20N2O4/c24-20(25)18-19(21(26)27)23(10-9-22-18)12-13-5-8-17-15(11-13)7-6-14-3-1-2-4-16(14)17/h1-8,11,18-19,22H,9-10,12H2,(H,24,25)(H,26,27)/t18-,19+/m0/s1
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2.67E+3n/an/an/an/an/an/an/an/a



University Walk

Curated by ChEMBL


Assay Description
Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50164541
PNG
((2R,3S)-1-Phenanthren-2-ylmethyl-piperazine-2,3-di...)
Show SMILES OC(=O)[C@H]1NCCN(Cc2ccc3c(ccc4ccccc34)c2)[C@H]1C(O)=O
Show InChI InChI=1S/C21H20N2O4/c24-20(25)18-19(21(26)27)23(10-9-22-18)12-13-5-8-17-15(11-13)7-6-14-3-1-2-4-16(14)17/h1-8,11,18-19,22H,9-10,12H2,(H,24,25)(H,26,27)/t18-,19+/m0/s1
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2.70E+3n/an/an/an/an/an/an/an/a



University of Bristol

Curated by ChEMBL


Assay Description
Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50419777
PNG
(CHEMBL1950804)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc2cc(Br)c3ccccc3c2c1
Show InChI InChI=1S/C21H17BrN2O5/c22-16-10-11-5-6-12(9-15(11)13-3-1-2-4-14(13)16)19(25)24-8-7-23-17(20(26)27)18(24)21(28)29/h1-6,9-10,17-18,23H,7-8H2,(H,26,27)(H,28,29)/t17-,18+/m0/s1
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2.80E+3n/an/an/an/an/an/an/an/a



University of Bristol

Curated by ChEMBL


Assay Description
Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50419778
PNG
(CHEMBL1950803)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc2cc(Cl)c3ccccc3c2c1
Show InChI InChI=1S/C21H17ClN2O5/c22-16-10-11-5-6-12(9-15(11)13-3-1-2-4-14(13)16)19(25)24-8-7-23-17(20(26)27)18(24)21(28)29/h1-6,9-10,17-18,23H,7-8H2,(H,26,27)(H,28,29)/t17-,18+/m0/s1
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3.20E+3n/an/an/an/an/an/an/an/a



University of Bristol

Curated by ChEMBL


Assay Description
Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50164540
PNG
((2R,3S)-1-(Phenanthrene-2-carbonyl)-piperazine-2,3...)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc2c(ccc3ccccc23)c1
Show InChI InChI=1S/C21H18N2O5/c24-19(23-10-9-22-17(20(25)26)18(23)21(27)28)14-7-8-16-13(11-14)6-5-12-3-1-2-4-15(12)16/h1-8,11,17-18,22H,9-10H2,(H,25,26)(H,27,28)/t17-,18+/m0/s1
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3.40E+3n/an/an/an/an/an/an/an/a



University of Bristol

Curated by ChEMBL


Assay Description
Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50419776
PNG
(CHEMBL1950806)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc2cc3ccccc3cc2c1
Show InChI InChI=1S/C21H18N2O5/c24-19(23-8-7-22-17(20(25)26)18(23)21(27)28)15-6-5-14-9-12-3-1-2-4-13(12)10-16(14)11-15/h1-6,9-11,17-18,22H,7-8H2,(H,25,26)(H,27,28)/t17-,18+/m0/s1
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3.40E+3n/an/an/an/an/an/an/an/a



University of Bristol

Curated by ChEMBL


Assay Description
Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50419788
PNG
(CHEMBL1950793)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc2cc(F)ccc2c1
Show InChI InChI=1S/C17H15FN2O5/c18-12-4-3-9-7-11(2-1-10(9)8-12)15(21)20-6-5-19-13(16(22)23)14(20)17(24)25/h1-4,7-8,13-14,19H,5-6H2,(H,22,23)(H,24,25)/t13-,14+/m0/s1
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3.60E+3n/an/an/an/an/an/an/an/a



University of Bristol

Curated by ChEMBL


Assay Description
Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50164551
PNG
((2R,3S)-1-(Naphthalene-2-carbonyl)-piperazine-2,3-...)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc2ccccc2c1
Show InChI InChI=1S/C17H16N2O5/c20-15(12-6-5-10-3-1-2-4-11(10)9-12)19-8-7-18-13(16(21)22)14(19)17(23)24/h1-6,9,13-14,18H,7-8H2,(H,21,22)(H,23,24)/t13-,14+/m0/s1
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3.89E+3n/an/an/an/an/an/an/an/a



University Walk

Curated by ChEMBL


Assay Description
Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50164551
PNG
((2R,3S)-1-(Naphthalene-2-carbonyl)-piperazine-2,3-...)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc2ccccc2c1
Show InChI InChI=1S/C17H16N2O5/c20-15(12-6-5-10-3-1-2-4-11(10)9-12)19-8-7-18-13(16(21)22)14(19)17(23)24/h1-6,9,13-14,18H,7-8H2,(H,21,22)(H,23,24)/t13-,14+/m0/s1
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3.90E+3n/an/an/an/an/an/an/an/a



University of Bristol

Curated by ChEMBL


Assay Description
Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50419784
PNG
(CHEMBL1950797)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)CCc1ccc2ccccc2c1
Show InChI InChI=1S/C19H20N2O5/c22-15(21-10-9-20-16(18(23)24)17(21)19(25)26)8-6-12-5-7-13-3-1-2-4-14(13)11-12/h1-5,7,11,16-17,20H,6,8-10H2,(H,23,24)(H,25,26)/t16-,17+/m0/s1
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4.10E+3n/an/an/an/an/an/an/an/a



University of Bristol

Curated by ChEMBL


Assay Description
Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50164553
PNG
((2R,3S)-1-(Phenanthrene-3-carbonyl)-piperazine-2,3...)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc2ccc3ccccc3c2c1
Show InChI InChI=1S/C21H18N2O5/c24-19(23-10-9-22-17(20(25)26)18(23)21(27)28)14-8-7-13-6-5-12-3-1-2-4-15(12)16(13)11-14/h1-8,11,17-18,22H,9-10H2,(H,25,26)(H,27,28)/t17-,18+/m0/s1
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4.22E+3n/an/an/an/an/an/an/an/a



University Walk

Curated by ChEMBL


Assay Description
Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50164545
PNG
((2R,3S)-1-(9-Oxo-9H-fluorene-2-carbonyl)-piperazin...)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc2-c3ccccc3C(=O)c2c1
Show InChI InChI=1S/C20H16N2O6/c23-17-13-4-2-1-3-11(13)12-6-5-10(9-14(12)17)18(24)22-8-7-21-15(19(25)26)16(22)20(27)28/h1-6,9,15-16,21H,7-8H2,(H,25,26)(H,27,28)/t15-,16+/m0/s1
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4.42E+3n/an/an/an/an/an/an/an/a



University Walk

Curated by ChEMBL


Assay Description
Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50164543
PNG
((2R,3R)-1-(Phenanthrene-2-carbonyl)-piperazine-2,3...)
Show SMILES OC(=O)[C@@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc2c(ccc3ccccc23)c1
Show InChI InChI=1S/C21H18N2O5/c24-19(23-10-9-22-17(20(25)26)18(23)21(27)28)14-7-8-16-13(11-14)6-5-12-3-1-2-4-15(12)16/h1-8,11,17-18,22H,9-10H2,(H,25,26)(H,27,28)/t17-,18-/m1/s1
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4.88E+3n/an/an/an/an/an/an/an/a



University Walk

Curated by ChEMBL


Assay Description
Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50164543
PNG
((2R,3R)-1-(Phenanthrene-2-carbonyl)-piperazine-2,3...)
Show SMILES OC(=O)[C@@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc2c(ccc3ccccc23)c1
Show InChI InChI=1S/C21H18N2O5/c24-19(23-10-9-22-17(20(25)26)18(23)21(27)28)14-7-8-16-13(11-14)6-5-12-3-1-2-4-15(12)16/h1-8,11,17-18,22H,9-10H2,(H,25,26)(H,27,28)/t17-,18-/m1/s1
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4.90E+3n/an/an/an/an/an/an/an/a



University of Bristol

Curated by ChEMBL


Assay Description
Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50419785
PNG
(CHEMBL1950796)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc2cc(ccc2c1)-c1ccccc1
Show InChI InChI=1S/C23H20N2O5/c26-21(25-11-10-24-19(22(27)28)20(25)23(29)30)18-9-8-16-12-15(6-7-17(16)13-18)14-4-2-1-3-5-14/h1-9,12-13,19-20,24H,10-11H2,(H,27,28)(H,29,30)/t19-,20+/m0/s1
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5.10E+3n/an/an/an/an/an/an/an/a



University of Bristol

Curated by ChEMBL


Assay Description
Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50164553
PNG
((2R,3S)-1-(Phenanthrene-3-carbonyl)-piperazine-2,3...)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc2ccc3ccccc3c2c1
Show InChI InChI=1S/C21H18N2O5/c24-19(23-10-9-22-17(20(25)26)18(23)21(27)28)14-8-7-13-6-5-12-3-1-2-4-15(12)16(13)11-14/h1-8,11,17-18,22H,9-10H2,(H,25,26)(H,27,28)/t17-,18+/m0/s1
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5.20E+3n/an/an/an/an/an/an/an/a



University of Bristol

Curated by ChEMBL


Assay Description
Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50017226
PNG
((R)-2-Amino-7-phosphono-heptanoic acid | 2-Amino-7...)
Show SMILES N[C@H](CCCCCP(O)(O)=O)C(O)=O
Show InChI InChI=1S/C7H16NO5P/c8-6(7(9)10)4-2-1-3-5-14(11,12)13/h6H,1-5,8H2,(H,9,10)(H2,11,12,13)/t6-/m1/s1
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6.42E+3n/an/an/an/an/an/an/an/a



University Walk

Curated by ChEMBL


Assay Description
Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50164550
PNG
((2R,3S)-1-(4'-Fluoro-biphenyl-4-carbonyl)-piperazi...)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc(cc1)-c1ccc(F)cc1
Show InChI InChI=1S/C19H17FN2O5/c20-14-7-5-12(6-8-14)11-1-3-13(4-2-11)17(23)22-10-9-21-15(18(24)25)16(22)19(26)27/h1-8,15-16,21H,9-10H2,(H,24,25)(H,26,27)/t15-,16+/m0/s1
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7.38E+3n/an/an/an/an/an/an/an/a



University Walk

Curated by ChEMBL


Assay Description
Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50164542
PNG
((2R,3S)-1-(2'-Bromo-biphenyl-4-carbonyl)-piperazin...)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc(cc1)-c1ccccc1Br
Show InChI InChI=1S/C19H17BrN2O5/c20-14-4-2-1-3-13(14)11-5-7-12(8-6-11)17(23)22-10-9-21-15(18(24)25)16(22)19(26)27/h1-8,15-16,21H,9-10H2,(H,24,25)(H,26,27)/t15-,16+/m0/s1
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8.49E+3n/an/an/an/an/an/an/an/a



University Walk

Curated by ChEMBL


Assay Description
Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50164544
PNG
((2R,3S)-1-(Biphenyl-4-sulfonyl)-piperazine-2,3-dic...)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)S(=O)(=O)c1ccc(cc1)-c1ccccc1
Show InChI InChI=1S/C18H18N2O6S/c21-17(22)15-16(18(23)24)20(11-10-19-15)27(25,26)14-8-6-13(7-9-14)12-4-2-1-3-5-12/h1-9,15-16,19H,10-11H2,(H,21,22)(H,23,24)/t15-,16+/m0/s1
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8.67E+3n/an/an/an/an/an/an/an/a



University Walk

Curated by ChEMBL


Assay Description
Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50164544
PNG
((2R,3S)-1-(Biphenyl-4-sulfonyl)-piperazine-2,3-dic...)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)S(=O)(=O)c1ccc(cc1)-c1ccccc1
Show InChI InChI=1S/C18H18N2O6S/c21-17(22)15-16(18(23)24)20(11-10-19-15)27(25,26)14-8-6-13(7-9-14)12-4-2-1-3-5-12/h1-9,15-16,19H,10-11H2,(H,21,22)(H,23,24)/t15-,16+/m0/s1
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8.70E+3n/an/an/an/an/an/an/an/a



University of Bristol

Curated by ChEMBL


Assay Description
Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50164552
PNG
((2R,3S)-1-(Biphenyl-4-carbonyl)-piperazine-2,3-dic...)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc(cc1)-c1ccccc1
Show InChI InChI=1S/C19H18N2O5/c22-17(21-11-10-20-15(18(23)24)16(21)19(25)26)14-8-6-13(7-9-14)12-4-2-1-3-5-12/h1-9,15-16,20H,10-11H2,(H,23,24)(H,25,26)/t15-,16+/m0/s1
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8.98E+3n/an/an/an/an/an/an/an/a



University Walk

Curated by ChEMBL


Assay Description
Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50164552
PNG
((2R,3S)-1-(Biphenyl-4-carbonyl)-piperazine-2,3-dic...)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc(cc1)-c1ccccc1
Show InChI InChI=1S/C19H18N2O5/c22-17(21-11-10-20-15(18(23)24)16(21)19(25)26)14-8-6-13(7-9-14)12-4-2-1-3-5-12/h1-9,15-16,20H,10-11H2,(H,23,24)(H,25,26)/t15-,16+/m0/s1
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9.00E+3n/an/an/an/an/an/an/an/a



University of Bristol

Curated by ChEMBL


Assay Description
Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50419781
PNG
(CHEMBL1950800)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc(cc1)C#Cc1ccccc1
Show InChI InChI=1S/C21H18N2O5/c24-19(23-13-12-22-17(20(25)26)18(23)21(27)28)16-10-8-15(9-11-16)7-6-14-4-2-1-3-5-14/h1-5,8-11,17-18,22H,12-13H2,(H,25,26)(H,27,28)/t17-,18+/m0/s1
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2.14E+4n/an/an/an/an/an/an/an/a



University of Bristol

Curated by ChEMBL


Assay Description
Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50164554
PNG
((2R,3S)-1-[(E)-(3-Phenyl-acryloyl)]-piperazine-2,3...)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)\C=C\c1ccccc1
Show InChI InChI=1S/C15H16N2O5/c18-11(7-6-10-4-2-1-3-5-10)17-9-8-16-12(14(19)20)13(17)15(21)22/h1-7,12-13,16H,8-9H2,(H,19,20)(H,21,22)/b7-6+/t12-,13+/m0/s1
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2.70E+4n/an/an/an/an/an/an/an/a



University Walk

Curated by ChEMBL


Assay Description
Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...


Citation and Details
More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50419780
PNG
(CHEMBL1950801)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc(cc1)\N=N\c1ccccc1
Show InChI InChI=1S/C19H18N4O5/c24-17(23-11-10-20-15(18(25)26)16(23)19(27)28)12-6-8-14(9-7-12)22-21-13-4-2-1-3-5-13/h1-9,15-16,20H,10-11H2,(H,25,26)(H,27,28)/b22-21+/t15-,16+/m0/s1
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2.80E+4n/an/an/an/an/an/an/an/a



University of Bristol

Curated by ChEMBL


Assay Description
Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...


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Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50164547
PNG
((2R,3S)-1-Benzoyl-piperazine-2,3-dicarboxylic acid...)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccccc1
Show InChI InChI=1S/C13H14N2O5/c16-11(8-4-2-1-3-5-8)15-7-6-14-9(12(17)18)10(15)13(19)20/h1-5,9-10,14H,6-7H2,(H,17,18)(H,19,20)/t9-,10+/m0/s1
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>1.00E+5n/an/an/an/an/an/an/an/a



University Walk

Curated by ChEMBL


Assay Description
Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...


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Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50419783
PNG
(CHEMBL1950798)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc2cc(ccc2c1)C(O)=O
Show InChI InChI=1S/C18H16N2O7/c21-15(20-6-5-19-13(17(24)25)14(20)18(26)27)11-3-1-10-8-12(16(22)23)4-2-9(10)7-11/h1-4,7-8,13-14,19H,5-6H2,(H,22,23)(H,24,25)(H,26,27)/t13-,14+/m0/s1
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>1.00E+5n/an/an/an/an/an/an/an/a



University of Bristol

Curated by ChEMBL


Assay Description
Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...


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More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50419782
PNG
(CHEMBL1950799)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc(cc1)-c1ccc(cc1)C(O)=O
Show InChI InChI=1S/C20H18N2O7/c23-17(22-10-9-21-15(19(26)27)16(22)20(28)29)13-5-1-11(2-6-13)12-3-7-14(8-4-12)18(24)25/h1-8,15-16,21H,9-10H2,(H,24,25)(H,26,27)(H,28,29)/t15-,16+/m0/s1
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>1.00E+5n/an/an/an/an/an/an/an/a



University of Bristol

Curated by ChEMBL


Assay Description
Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...


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More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50419779
PNG
(CHEMBL1950802)
Show SMILES OC(=O)[C@H]1NCCN([C@H]1C(O)=O)C(=O)c1ccc(CCc2ccccc2)cc1
Show InChI InChI=1S/C21H22N2O5/c24-19(23-13-12-22-17(20(25)26)18(23)21(27)28)16-10-8-15(9-11-16)7-6-14-4-2-1-3-5-14/h1-5,8-11,17-18,22H,6-7,12-13H2,(H,25,26)(H,27,28)/t17-,18+/m0/s1
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>1.00E+5n/an/an/an/an/an/an/an/a



University of Bristol

Curated by ChEMBL


Assay Description
Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...


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More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50324399
PNG
((E)-4-(6-iodo-2-(3-nitrostyryl)-4-oxoquinazolin-3(...)
Show SMILES OC(=O)c1ccc(cc1)-n1c(\C=C\c2cccc(c2)[N+]([O-])=O)nc2ccc(I)cc2c1=O
Show InChI InChI=1S/C23H14IN3O5/c24-16-7-10-20-19(13-16)22(28)26(17-8-5-15(6-9-17)23(29)30)21(25-20)11-4-14-2-1-3-18(12-14)27(31)32/h1-13H,(H,29,30)/b11-4+
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n/an/a 1.00E+3n/an/an/an/an/an/a



Emory University

Curated by ChEMBL


Assay Description
Antagonist activity at rat recombinant NR1-NR2C receptor expressed in Xenopus oocytes at holding potential of -40mV by two-electrode voltage-clamp el...


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More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50324392
PNG
((E)-4-(6-Chloro-2-(3-nitrostyryl)-4-oxoquinazolin-...)
Show SMILES OC(=O)c1ccc(cc1)-n1c(\C=C\c2cccc(c2)[N+]([O-])=O)nc2ccc(Cl)cc2c1=O
Show InChI InChI=1S/C23H14ClN3O5/c24-16-7-10-20-19(13-16)22(28)26(17-8-5-15(6-9-17)23(29)30)21(25-20)11-4-14-2-1-3-18(12-14)27(31)32/h1-13H,(H,29,30)/b11-4+
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n/an/a 2.00E+3n/an/an/an/an/an/a



Emory University

Curated by ChEMBL


Assay Description
Antagonist activity at rat recombinant NR1-NR2C receptor expressed in Xenopus oocytes at holding potential of -40mV by two-electrode voltage-clamp el...


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More data for this
Ligand-Target Pair
Glutamate [NMDA] receptor subunit epsilon 3/zeta 1


(Rattus norvegicus)
BDBM50324428
PNG
((E)-3-(6-Iodo-2-(3-nitrostyryl)-4-oxoquinazolin-3(...)
Show SMILES OC(=O)c1cccc(c1)-n1c(\C=C\c2cccc(c2)[N+]([O-])=O)nc2ccc(I)cc2c1=O
Show InChI InChI=1S/C23H14IN3O5/c24-16-8-9-20-19(13-16)22(28)26(17-5-2-4-15(12-17)23(29)30)21(25-20)10-7-14-3-1-6-18(11-14)27(31)32/h1-13H,(H,29,30)/b10-7+
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n/an/a 2.00E+3n/an/an/an/an/an/a



Emory University

Curated by ChEMBL


Assay Description
Antagonist activity at rat recombinant NR1-NR2C receptor expressed in Xenopus oocytes at holding potential of -40mV by two-electrode voltage-clamp el...


Citation and Details
More data for this
Ligand-Target Pair
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