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Found 130 hits Enz. Inhib. hit(s) with Target = 'SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635' AND taxid = 9606   
Target
(Institution)
LigandTarget
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM50400044
PNG
(CHEMBL2177726 | US9169259, I-54)
Show SMILES COc1ccc(Nc2cc(nn3ccnc23)-c2cccc(c2)C(=O)Nc2ccc(cc2)C(O)=O)nc1OC
Show InChI InChI=1S/C27H22N6O5/c1-37-22-10-11-23(31-26(22)38-2)30-21-15-20(32-33-13-12-28-24(21)33)17-4-3-5-18(14-17)25(34)29-19-8-6-16(7-9-19)27(35)36/h3-15H,1-2H3,(H,29,34)(H,30,31)(H,35,36)
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n/an/a 1n/an/an/an/an/an/a



HOFFMANN-LA ROCHE INC.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 um filter plates (Millipore Cat. No.: MADVNOB10)Streptavidin coated beads: Streptavidin Sepharose, suspension ...


US Patent US9169259 (2015)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM188174
PNG
(US9169259, I-57)
Show SMILES COc1ccc(Nc2cc(nn3ccnc23)-c2cccc(c2)C(=O)Nc2ccc(C(O)=O)c(OC)c2)nc1OC
Show InChI InChI=1S/C28H24N6O6/c1-38-22-9-10-24(32-27(22)40-3)31-21-15-20(33-34-12-11-29-25(21)34)16-5-4-6-17(13-16)26(35)30-18-7-8-19(28(36)37)23(14-18)39-2/h4-15H,1-3H3,(H,30,35)(H,31,32)(H,36,37)
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n/an/a 1.55n/an/an/an/an/an/a



HOFFMANN-LA ROCHE INC.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 um filter plates (Millipore Cat. No.: MADVNOB10)Streptavidin coated beads: Streptavidin Sepharose, suspension ...


US Patent US9169259 (2015)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM188128
PNG
(US9169259, I-10)
Show SMILES CC1CCCN1c1cccc(Nc2cc(nn3ccnc23)-c2cccc(c2)C(=O)Nc2ccc(cc2)C(O)=O)n1
Show InChI InChI=1/C30H27N7O3/c1-19-5-4-15-36(19)27-9-3-8-26(34-27)33-25-18-24(35-37-16-14-31-28(25)37)21-6-2-7-22(17-21)29(38)32-23-12-10-20(11-13-23)30(39)40/h2-3,6-14,16-19H,4-5,15H2,1H3,(H,32,38)(H,33,34)(H,39,40)
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n/an/a 1.65n/an/an/an/an/an/a



HOFFMANN-LA ROCHE INC.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 um filter plates (Millipore Cat. No.: MADVNOB10)Streptavidin coated beads: Streptavidin Sepharose, suspension ...


US Patent US9169259 (2015)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM227529
PNG
(US9334278, I-18)
Show SMILES Cc1cc(Nc2cnc3[nH]cc(C(=O)NC(C)(C)C)c3n2)sn1
Show InChI InChI=1S/C15H18N6OS/c1-8-5-11(23-21-8)18-10-7-17-13-12(19-10)9(6-16-13)14(22)20-15(2,3)4/h5-7H,1-4H3,(H,16,17)(H,18,19)(H,20,22)
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n/an/a 2n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 μm filter plates (Millipore Cat. No.: MADVNOB 10) Streptavidin coated beads: Streptavidin Sepharose™,...


US Patent US9334278 (2016)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM188188
PNG
(US9169259, I-72)
Show SMILES COc1ccc(Nc2cc(nn3ccnc23)N2CCCC(C2)NC(=O)c2ccc(cc2)C(O)=O)nc1OC
Show InChI InChI=1/C26H27N7O5/c1-37-20-9-10-21(30-25(20)38-2)29-19-14-22(31-33-13-11-27-23(19)33)32-12-3-4-18(15-32)28-24(34)16-5-7-17(8-6-16)26(35)36/h5-11,13-14,18H,3-4,12,15H2,1-2H3,(H,28,34)(H,29,30)(H,35,36)
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n/an/a 2.20n/an/an/an/an/an/a



HOFFMANN-LA ROCHE INC.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 um filter plates (Millipore Cat. No.: MADVNOB10)Streptavidin coated beads: Streptavidin Sepharose, suspension ...


US Patent US9169259 (2015)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM227523
PNG
(US9334278, I-12)
Show SMILES Cc1ccc(Nc2cnc3[nH]cc(C(=O)NC(C)(C)C)c3n2)cc1
Show InChI InChI=1S/C18H21N5O/c1-11-5-7-12(8-6-11)21-14-10-20-16-15(22-14)13(9-19-16)17(24)23-18(2,3)4/h5-10H,1-4H3,(H,19,20)(H,21,22)(H,23,24)
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n/an/a 3.20n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 μm filter plates (Millipore Cat. No.: MADVNOB 10) Streptavidin coated beads: Streptavidin Sepharose™,...


US Patent US9334278 (2016)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM227549
PNG
(US9334278, I-37)
Show SMILES Cc1nc2[nH]cc(C(=O)NC(C)(C)C)c2nc1Nc1ccccc1
Show InChI InChI=1S/C18H21N5O/c1-11-15(21-12-8-6-5-7-9-12)22-14-13(10-19-16(14)20-11)17(24)23-18(2,3)4/h5-10H,1-4H3,(H,19,20)(H,21,22)(H,23,24)
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n/an/a 4.80n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 μm filter plates (Millipore Cat. No.: MADVNOB 10) Streptavidin coated beads: Streptavidin Sepharose™,...


US Patent US9334278 (2016)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM227537
PNG
(US9334278, I-26)
Show SMILES CC(C)(CO)NC(=O)c1c[nH]c2ncc(Nc3cccnc3)nc12
Show InChI InChI=1S/C16H18N6O2/c1-16(2,9-23)22-15(24)11-7-18-14-13(11)21-12(8-19-14)20-10-4-3-5-17-6-10/h3-8,23H,9H2,1-2H3,(H,18,19)(H,20,21)(H,22,24)
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n/an/a 5.60n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 μm filter plates (Millipore Cat. No.: MADVNOB 10) Streptavidin coated beads: Streptavidin Sepharose™,...


US Patent US9334278 (2016)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM227535
PNG
(US9334278, I-24)
Show SMILES CC(O)c1cccc(Nc2cnc3[nH]cc(C(=O)NC(C)(C)C)c3n2)c1
Show InChI InChI=1/C19H23N5O2/c1-11(25)12-6-5-7-13(8-12)22-15-10-21-17-16(23-15)14(9-20-17)18(26)24-19(2,3)4/h5-11,25H,1-4H3,(H,20,21)(H,22,23)(H,24,26)
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n/an/a 5.90n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 μm filter plates (Millipore Cat. No.: MADVNOB 10) Streptavidin coated beads: Streptavidin Sepharose™,...


US Patent US9334278 (2016)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM188172
PNG
(US9169259, I-55)
Show SMILES COc1ccc(Nc2cc(nn3ccnc23)-c2cccc(c2)C(=O)Nc2ccc3[nH]ncc3c2)nc1OC
Show InChI InChI=1S/C27H22N8O3/c1-37-23-8-9-24(32-27(23)38-2)31-22-14-21(34-35-11-10-28-25(22)35)16-4-3-5-17(12-16)26(36)30-19-6-7-20-18(13-19)15-29-33-20/h3-15H,1-2H3,(H,29,33)(H,30,36)(H,31,32)
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n/an/a 7.33n/an/an/an/an/an/a



HOFFMANN-LA ROCHE INC.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 um filter plates (Millipore Cat. No.: MADVNOB10)Streptavidin coated beads: Streptavidin Sepharose, suspension ...


US Patent US9169259 (2015)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM227512
PNG
(US9334278, I-1)
Show SMILES Cc1ccc(Nc2cnc3[nH]cc(C(=O)NC(C)(C)C)c3n2)nc1
Show InChI InChI=1S/C17H20N6O/c1-10-5-6-12(18-7-10)21-13-9-20-15-14(22-13)11(8-19-15)16(24)23-17(2,3)4/h5-9H,1-4H3,(H,19,20)(H,23,24)(H,18,21,22)
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n/an/a 8.5n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 μm filter plates (Millipore Cat. No.: MADVNOB 10) Streptavidin coated beads: Streptavidin Sepharose™,...


US Patent US9334278 (2016)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM227522
PNG
(US9334278, I-11)
Show SMILES Cc1ccc(Nc2cnc3[nH]cc(C(=O)NC(C)(C)C)c3n2)c(F)c1
Show InChI InChI=1S/C18H20FN5O/c1-10-5-6-13(12(19)7-10)22-14-9-21-16-15(23-14)11(8-20-16)17(25)24-18(2,3)4/h5-9H,1-4H3,(H,20,21)(H,22,23)(H,24,25)
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n/an/a 10.9n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 μm filter plates (Millipore Cat. No.: MADVNOB 10) Streptavidin coated beads: Streptavidin Sepharose™,...


US Patent US9334278 (2016)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM227524
PNG
(US9334278, I-13)
Show SMILES CC(C)(C)NC(=O)c1c[nH]c2ncc(Nc3cccc(c3)S(C)(=O)=O)nc12
Show InChI InChI=1S/C18H21N5O3S/c1-18(2,3)23-17(24)13-9-19-16-15(13)22-14(10-20-16)21-11-6-5-7-12(8-11)27(4,25)26/h5-10H,1-4H3,(H,19,20)(H,21,22)(H,23,24)
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n/an/a 12.8n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 μm filter plates (Millipore Cat. No.: MADVNOB 10) Streptavidin coated beads: Streptavidin Sepharose™,...


US Patent US9334278 (2016)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM227516
PNG
(US9334278, I-5)
Show SMILES Cn1cc(Nc2cnc3[nH]cc(C(=O)NC(C)(C)C)c3n2)cn1
Show InChI InChI=1S/C15H19N7O/c1-15(2,3)21-14(23)10-6-16-13-12(10)20-11(7-17-13)19-9-5-18-22(4)8-9/h5-8H,1-4H3,(H,16,17)(H,19,20)(H,21,23)
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n/an/a 13.7n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 μm filter plates (Millipore Cat. No.: MADVNOB 10) Streptavidin coated beads: Streptavidin Sepharose™,...


US Patent US9334278 (2016)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM188190
PNG
(US9169259, I-74)
Show SMILES COc1ccc(Nc2cc(nn3ccnc23)N2CCCC(C2)C(=O)Nc2ccc(cc2)C(O)=O)nc1OC
Show InChI InChI=1/C26H27N7O5/c1-37-20-9-10-21(30-25(20)38-2)29-19-14-22(31-33-13-11-27-23(19)33)32-12-3-4-17(15-32)24(34)28-18-7-5-16(6-8-18)26(35)36/h5-11,13-14,17H,3-4,12,15H2,1-2H3,(H,28,34)(H,29,30)(H,35,36)
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n/an/a 14.9n/an/an/an/an/an/a



HOFFMANN-LA ROCHE INC.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 um filter plates (Millipore Cat. No.: MADVNOB10)Streptavidin coated beads: Streptavidin Sepharose, suspension ...


US Patent US9169259 (2015)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM227520
PNG
(US9334278, I-9)
Show SMILES Cc1cc(Nc2cnc3[nH]cc(C(=O)NC(C)(C)C)c3n2)[nH]n1
Show InChI InChI=1S/C15H19N7O/c1-8-5-10(22-21-8)18-11-7-17-13-12(19-11)9(6-16-13)14(23)20-15(2,3)4/h5-7H,1-4H3,(H,16,17)(H,20,23)(H2,18,19,21,22)
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n/an/a 15.5n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 μm filter plates (Millipore Cat. No.: MADVNOB 10) Streptavidin coated beads: Streptavidin Sepharose™,...


US Patent US9334278 (2016)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM50400035
PNG
(CHEMBL2177735 | US9169259, I-84)
Show SMILES CC1CCCN1c1cccc(Nc2cc(nn3ccnc23)-c2cccc(CN)c2)n1
Show InChI InChI=1S/C23H25N7/c1-16-5-4-11-29(16)22-9-3-8-21(27-22)26-20-14-19(28-30-12-10-25-23(20)30)18-7-2-6-17(13-18)15-24/h2-3,6-10,12-14,16H,4-5,11,15,24H2,1H3,(H,26,27)
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n/an/a 15.6n/an/an/an/an/an/a



HOFFMANN-LA ROCHE INC.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 um filter plates (Millipore Cat. No.: MADVNOB10)Streptavidin coated beads: Streptavidin Sepharose, suspension ...


US Patent US9169259 (2015)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM188169
PNG
(US9169259, I-51)
Show SMILES C[C@H]1CCCN1c1cccc(Nc2cc(nn3ccnc23)-c2cccc(c2)C(N)=O)n1
Show InChI InChI=1/C23H23N7O/c1-15-5-4-11-29(15)21-9-3-8-20(27-21)26-19-14-18(28-30-12-10-25-23(19)30)16-6-2-7-17(13-16)22(24)31/h2-3,6-10,12-15H,4-5,11H2,1H3,(H2,24,31)(H,26,27)/t15-/s2
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n/an/a 16.1n/an/an/an/an/an/a



HOFFMANN-LA ROCHE INC.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 um filter plates (Millipore Cat. No.: MADVNOB10)Streptavidin coated beads: Streptavidin Sepharose, suspension ...


US Patent US9169259 (2015)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM227521
PNG
(US9334278, I-10)
Show SMILES CC(C)(C)NC(=O)c1c[nH]c2ncc(Nc3cccnc3)nc12
Show InChI InChI=1S/C16H18N6O/c1-16(2,3)22-15(23)11-8-18-14-13(11)21-12(9-19-14)20-10-5-4-6-17-7-10/h4-9H,1-3H3,(H,18,19)(H,20,21)(H,22,23)
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n/an/a 16.3n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 μm filter plates (Millipore Cat. No.: MADVNOB 10) Streptavidin coated beads: Streptavidin Sepharose™,...


US Patent US9334278 (2016)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM227517
PNG
(US9334278, I-6)
Show SMILES Cc1ccc(Nc2cnc3[nH]cc(C(=O)NC(C)(C)C)c3n2)cn1
Show InChI InChI=1S/C17H20N6O/c1-10-5-6-11(7-18-10)21-13-9-20-15-14(22-13)12(8-19-15)16(24)23-17(2,3)4/h5-9H,1-4H3,(H,19,20)(H,21,22)(H,23,24)
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n/an/a 17.1n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 μm filter plates (Millipore Cat. No.: MADVNOB 10) Streptavidin coated beads: Streptavidin Sepharose™,...


US Patent US9334278 (2016)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM227542
PNG
(US9334278, I-31)
Show SMILES Cc1nsc(Nc2cnc3[nH]cc(C(=O)NC(C)(C)C)c3n2)n1
Show InChI InChI=1S/C14H17N7OS/c1-7-17-13(23-21-7)19-9-6-16-11-10(18-9)8(5-15-11)12(22)20-14(2,3)4/h5-6H,1-4H3,(H,15,16)(H,20,22)(H,17,18,19,21)
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n/an/a 17.8n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 μm filter plates (Millipore Cat. No.: MADVNOB 10) Streptavidin coated beads: Streptavidin Sepharose™,...


US Patent US9334278 (2016)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM227538
PNG
(US9334278, I-27)
Show SMILES CC(N)c1cccc(Nc2cnc3[nH]cc(C(=O)NC(C)(C)C)c3n2)c1
Show InChI InChI=1/C19H24N6O/c1-11(20)12-6-5-7-13(8-12)23-15-10-22-17-16(24-15)14(9-21-17)18(26)25-19(2,3)4/h5-11H,20H2,1-4H3,(H,21,22)(H,23,24)(H,25,26)
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n/an/a 18.8n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 μm filter plates (Millipore Cat. No.: MADVNOB 10) Streptavidin coated beads: Streptavidin Sepharose™,...


US Patent US9334278 (2016)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM188168
PNG
(US9169259, I-50)
Show SMILES C[C@H]1CCCN1c1cccc(Nc2cc(nn3ccnc23)-c2ccc(cc2)C(N)=O)n1
Show InChI InChI=1/C23H23N7O/c1-15-4-3-12-29(15)21-6-2-5-20(27-21)26-19-14-18(28-30-13-11-25-23(19)30)16-7-9-17(10-8-16)22(24)31/h2,5-11,13-15H,3-4,12H2,1H3,(H2,24,31)(H,26,27)/t15-/s2
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n/an/a 18.9n/an/an/an/an/an/a



HOFFMANN-LA ROCHE INC.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 um filter plates (Millipore Cat. No.: MADVNOB10)Streptavidin coated beads: Streptavidin Sepharose, suspension ...


US Patent US9169259 (2015)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM227514
PNG
(US9334278, I-3)
Show SMILES Cn1ccc(Nc2cnc3[nH]cc(C(=O)NC(C)(C)C)c3n2)n1
Show InChI InChI=1S/C15H19N7O/c1-15(2,3)20-14(23)9-7-16-13-12(9)19-11(8-17-13)18-10-5-6-22(4)21-10/h5-8H,1-4H3,(H,16,17)(H,20,23)(H,18,19,21)
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n/an/a 21.1n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 μm filter plates (Millipore Cat. No.: MADVNOB 10) Streptavidin coated beads: Streptavidin Sepharose™,...


US Patent US9334278 (2016)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM188208
PNG
(US9169259, I-93)
Show SMILES CC1CCCN1c1cccc(Nc2cc(nn3ccnc23)-c2cccc(CNC3CCNCC3)c2)n1
Show InChI InChI=1/C28H34N8/c1-20-5-4-15-35(20)27-9-3-8-26(33-27)32-25-18-24(34-36-16-14-30-28(25)36)22-7-2-6-21(17-22)19-31-23-10-12-29-13-11-23/h2-3,6-9,14,16-18,20,23,29,31H,4-5,10-13,15,19H2,1H3,(H,32,33)
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n/an/a 24.4n/an/an/an/an/an/a



HOFFMANN-LA ROCHE INC.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 um filter plates (Millipore Cat. No.: MADVNOB10)Streptavidin coated beads: Streptavidin Sepharose, suspension ...


US Patent US9169259 (2015)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM50400036
PNG
(CHEMBL2177734 | US9169259, I-68)
Show SMILES CC1CCCN1c1cccc(Nc2cc(nn3ccnc23)-c2cccc(CO)c2)n1
Show InChI InChI=1S/C23H24N6O/c1-16-5-4-11-28(16)22-9-3-8-21(26-22)25-20-14-19(27-29-12-10-24-23(20)29)18-7-2-6-17(13-18)15-30/h2-3,6-10,12-14,16,30H,4-5,11,15H2,1H3,(H,25,26)
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n/an/a 24.7n/an/an/an/an/an/a



HOFFMANN-LA ROCHE INC.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 um filter plates (Millipore Cat. No.: MADVNOB10)Streptavidin coated beads: Streptavidin Sepharose, suspension ...


US Patent US9169259 (2015)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM227533
PNG
(US9334278, I-22)
Show SMILES Cc1cc(Nc2cnc3[nH]cc(C(=O)NC(C)(C)C)c3n2)on1
Show InChI InChI=1S/C15H18N6O2/c1-8-5-11(23-21-8)18-10-7-17-13-12(19-10)9(6-16-13)14(22)20-15(2,3)4/h5-7H,1-4H3,(H,16,17)(H,18,19)(H,20,22)
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n/an/a 25.1n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 μm filter plates (Millipore Cat. No.: MADVNOB 10) Streptavidin coated beads: Streptavidin Sepharose™,...


US Patent US9334278 (2016)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM227513
PNG
(US9334278, I-2)
Show SMILES Cc1ccc(Nc2cnc3[nH]cc(C(=O)NC(C)(C)CO)c3n2)nc1
Show InChI InChI=1S/C17H20N6O2/c1-10-4-5-12(18-6-10)21-13-8-20-15-14(22-13)11(7-19-15)16(25)23-17(2,3)9-24/h4-8,24H,9H2,1-3H3,(H,19,20)(H,23,25)(H,18,21,22)
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n/an/a 27.4n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 μm filter plates (Millipore Cat. No.: MADVNOB 10) Streptavidin coated beads: Streptavidin Sepharose™,...


US Patent US9334278 (2016)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM227531
PNG
(US9334278, I-20)
Show SMILES CC(C)(C)NC(=O)c1c[nH]c2ncc(Nc3ccc(cc3)S(C)(=O)=O)nc12
Show InChI InChI=1S/C18H21N5O3S/c1-18(2,3)23-17(24)13-9-19-16-15(13)22-14(10-20-16)21-11-5-7-12(8-6-11)27(4,25)26/h5-10H,1-4H3,(H,19,20)(H,21,22)(H,23,24)
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n/an/a 30n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 μm filter plates (Millipore Cat. No.: MADVNOB 10) Streptavidin coated beads: Streptavidin Sepharose™,...


US Patent US9334278 (2016)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM188135
PNG
(US9169259, I-17)
Show SMILES CC1CCCN1c1cccc(Nc2cc(nn3ccnc23)-c2ccc(cc2)C(N)=O)n1
Show InChI InChI=1/C23H23N7O/c1-15-4-3-12-29(15)21-6-2-5-20(27-21)26-19-14-18(28-30-13-11-25-23(19)30)16-7-9-17(10-8-16)22(24)31/h2,5-11,13-15H,3-4,12H2,1H3,(H2,24,31)(H,26,27)
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n/an/a 33.1n/an/an/an/an/an/a



HOFFMANN-LA ROCHE INC.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 um filter plates (Millipore Cat. No.: MADVNOB10)Streptavidin coated beads: Streptavidin Sepharose, suspension ...


US Patent US9169259 (2015)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM227525
PNG
(US9334278, I-14)
Show SMILES CCn1cc(Nc2cnc3[nH]cc(C(=O)NC(C)(C)C)c3n2)cn1
Show InChI InChI=1S/C16H21N7O/c1-5-23-9-10(6-19-23)20-12-8-18-14-13(21-12)11(7-17-14)15(24)22-16(2,3)4/h6-9H,5H2,1-4H3,(H,17,18)(H,20,21)(H,22,24)
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n/an/a 35.9n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 μm filter plates (Millipore Cat. No.: MADVNOB 10) Streptavidin coated beads: Streptavidin Sepharose™,...


US Patent US9334278 (2016)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM188170
PNG
(US9169259, I-52)
Show SMILES C[C@H]1CCCN1c1cccc(Nc2cc(nn3ccnc23)-c2ccc3ncsc3c2)n1
Show InChI InChI=1/C23H21N7S/c1-15-4-3-10-29(15)22-6-2-5-21(27-22)26-19-13-18(28-30-11-9-24-23(19)30)16-7-8-17-20(12-16)31-14-25-17/h2,5-9,11-15H,3-4,10H2,1H3,(H,26,27)/t15-/s2
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n/an/a 36.1n/an/an/an/an/an/a



HOFFMANN-LA ROCHE INC.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 um filter plates (Millipore Cat. No.: MADVNOB10)Streptavidin coated beads: Streptavidin Sepharose, suspension ...


US Patent US9169259 (2015)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM188192
PNG
(US9169259, I-76)
Show SMILES COc1ccc(Nc2cc(nn3ccnc23)N2CCC(C2)NC(=O)c2ccc(cc2)C(O)=O)nc1OC
Show InChI InChI=1/C25H25N7O5/c1-36-19-7-8-20(29-24(19)37-2)28-18-13-21(30-32-12-10-26-22(18)32)31-11-9-17(14-31)27-23(33)15-3-5-16(6-4-15)25(34)35/h3-8,10,12-13,17H,9,11,14H2,1-2H3,(H,27,33)(H,28,29)(H,34,35)
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n/an/a 42.1n/an/an/an/an/an/a



HOFFMANN-LA ROCHE INC.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 um filter plates (Millipore Cat. No.: MADVNOB10)Streptavidin coated beads: Streptavidin Sepharose, suspension ...


US Patent US9169259 (2015)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM188158
PNG
(US9169259, I-40)
Show SMILES CC1CCCN1c1cccc(Nc2cc(nn3ccnc23)-c2cccc(c2)C(=O)NCCO)n1
Show InChI InChI=1/C25H27N7O2/c1-17-5-4-12-31(17)23-9-3-8-22(29-23)28-21-16-20(30-32-13-10-26-24(21)32)18-6-2-7-19(15-18)25(34)27-11-14-33/h2-3,6-10,13,15-17,33H,4-5,11-12,14H2,1H3,(H,27,34)(H,28,29)
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n/an/a 42.5n/an/an/an/an/an/a



HOFFMANN-LA ROCHE INC.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 um filter plates (Millipore Cat. No.: MADVNOB10)Streptavidin coated beads: Streptavidin Sepharose, suspension ...


US Patent US9169259 (2015)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM227515
PNG
(US9334278, I-4)
Show SMILES CC(C)NC(=O)c1c[nH]c2ncc(Nc3ccc(C)cn3)nc12
Show InChI InChI=1S/C16H18N6O/c1-9(2)20-16(23)11-7-18-15-14(11)22-13(8-19-15)21-12-5-4-10(3)6-17-12/h4-9H,1-3H3,(H,18,19)(H,20,23)(H,17,21,22)
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n/an/a 42.8n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 μm filter plates (Millipore Cat. No.: MADVNOB 10) Streptavidin coated beads: Streptavidin Sepharose™,...


US Patent US9334278 (2016)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM227543
PNG
(US9334278, I-32)
Show SMILES Cn1cc2N(CCCc2n1)c1cnc2[nH]cc(C(=O)NC(C)(C)C)c2n1
Show InChI InChI=1S/C18H23N7O/c1-18(2,3)22-17(26)11-8-19-16-15(11)21-14(9-20-16)25-7-5-6-12-13(25)10-24(4)23-12/h8-10H,5-7H2,1-4H3,(H,19,20)(H,22,26)
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n/an/a 43.7n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 μm filter plates (Millipore Cat. No.: MADVNOB 10) Streptavidin coated beads: Streptavidin Sepharose™,...


US Patent US9334278 (2016)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM188199
PNG
(US9169259, I-83)
Show SMILES CC1CCCN1c1cccc(Nc2cc(nn3ccnc23)-c2ccc(OCCN3CCCC3)cc2)n1
Show InChI InChI=1/C28H33N7O/c1-21-6-5-16-34(21)27-8-4-7-26(31-27)30-25-20-24(32-35-17-13-29-28(25)35)22-9-11-23(12-10-22)36-19-18-33-14-2-3-15-33/h4,7-13,17,20-21H,2-3,5-6,14-16,18-19H2,1H3,(H,30,31)
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n/an/a 47.5n/an/an/an/an/an/a



HOFFMANN-LA ROCHE INC.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 um filter plates (Millipore Cat. No.: MADVNOB10)Streptavidin coated beads: Streptavidin Sepharose, suspension ...


US Patent US9169259 (2015)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM188162
PNG
(US9169259, I-44)
Show SMILES COc1ccc(Nc2cc(nn3ccnc23)-c2ccccc2)nc1OC
Show InChI InChI=1S/C19H17N5O2/c1-25-16-8-9-17(22-19(16)26-2)21-15-12-14(13-6-4-3-5-7-13)23-24-11-10-20-18(15)24/h3-12H,1-2H3,(H,21,22)
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n/an/a 47.6n/an/an/an/an/an/a



HOFFMANN-LA ROCHE INC.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 um filter plates (Millipore Cat. No.: MADVNOB10)Streptavidin coated beads: Streptavidin Sepharose, suspension ...


US Patent US9169259 (2015)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM188130
PNG
(US9169259, I-12)
Show SMILES CC1CCCN1c1cccc(Nc2cc(nn3ccnc23)-c2cccc(c2)C(N)=O)n1
Show InChI InChI=1/C23H23N7O/c1-15-5-4-11-29(15)21-9-3-8-20(27-21)26-19-14-18(28-30-12-10-25-23(19)30)16-6-2-7-17(13-16)22(24)31/h2-3,6-10,12-15H,4-5,11H2,1H3,(H2,24,31)(H,26,27)
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n/an/a 48.6n/an/an/an/an/an/a



HOFFMANN-LA ROCHE INC.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 um filter plates (Millipore Cat. No.: MADVNOB10)Streptavidin coated beads: Streptavidin Sepharose, suspension ...


US Patent US9169259 (2015)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM227528
PNG
(US9334278, I-17)
Show SMILES Cn1cc(Nc2cnc3[nH]cc(C(=O)NC(C)(C)CO)c3n2)cn1
Show InChI InChI=1S/C15H19N7O2/c1-15(2,8-23)21-14(24)10-5-16-13-12(10)20-11(6-17-13)19-9-4-18-22(3)7-9/h4-7,23H,8H2,1-3H3,(H,16,17)(H,19,20)(H,21,24)
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n/an/a 49.9n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 μm filter plates (Millipore Cat. No.: MADVNOB 10) Streptavidin coated beads: Streptavidin Sepharose™,...


US Patent US9334278 (2016)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM188203
PNG
(US9169259, I-88)
Show SMILES CC1CCCN1c1cccc(Nc2cc(nn3ccnc23)-c2cccc(OCCN3CCOCC3)c2)n1
Show InChI InChI=1/C28H33N7O2/c1-21-5-4-11-34(21)27-9-3-8-26(31-27)30-25-20-24(32-35-12-10-29-28(25)35)22-6-2-7-23(19-22)37-18-15-33-13-16-36-17-14-33/h2-3,6-10,12,19-21H,4-5,11,13-18H2,1H3,(H,30,31)
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n/an/a 51.0n/an/an/an/an/an/a



HOFFMANN-LA ROCHE INC.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 um filter plates (Millipore Cat. No.: MADVNOB10)Streptavidin coated beads: Streptavidin Sepharose, suspension ...


US Patent US9169259 (2015)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM227519
PNG
(US9334278, I-8)
Show SMILES Cc1cnc(Nc2cnc3[nH]cc(C(=O)NC(C)(C)C)c3n2)cn1
Show InChI InChI=1S/C16H19N7O/c1-9-5-18-11(7-17-9)21-12-8-20-14-13(22-12)10(6-19-14)15(24)23-16(2,3)4/h5-8H,1-4H3,(H,19,20)(H,23,24)(H,18,21,22)
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n/an/a 51.3n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 μm filter plates (Millipore Cat. No.: MADVNOB 10) Streptavidin coated beads: Streptavidin Sepharose™,...


US Patent US9334278 (2016)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM188181
PNG
(US9169259, I-64)
Show SMILES CC1CCCN1c1cccc(Nc2cc(nn3ccnc23)-c2ccc3CCN(Cc3c2)C(C)=O)n1
Show InChI InChI=1/C27H29N7O/c1-18-5-4-12-33(18)26-7-3-6-25(30-26)29-24-16-23(31-34-14-11-28-27(24)34)21-9-8-20-10-13-32(19(2)35)17-22(20)15-21/h3,6-9,11,14-16,18H,4-5,10,12-13,17H2,1-2H3,(H,29,30)
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n/an/a 56.6n/an/an/an/an/an/a



HOFFMANN-LA ROCHE INC.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 um filter plates (Millipore Cat. No.: MADVNOB10)Streptavidin coated beads: Streptavidin Sepharose, suspension ...


US Patent US9169259 (2015)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM188198
PNG
(US9169259, I-82)
Show SMILES COc1cncc(c1)-c1cc(Nc2cccc(n2)N2CCCC2C)c2nccn2n1
Show InChI InChI=1/C22H23N7O/c1-15-5-4-9-28(15)21-7-3-6-20(26-21)25-19-12-18(27-29-10-8-24-22(19)29)16-11-17(30-2)14-23-13-16/h3,6-8,10-15H,4-5,9H2,1-2H3,(H,25,26)
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n/an/a 59.9n/an/an/an/an/an/a



HOFFMANN-LA ROCHE INC.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 um filter plates (Millipore Cat. No.: MADVNOB10)Streptavidin coated beads: Streptavidin Sepharose, suspension ...


US Patent US9169259 (2015)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM188207
PNG
(US9169259, I-92)
Show SMILES CCN(CC)CCOc1ccc(cc1)-c1cc(Nc2cccc(n2)N2CCCC2C)c2nccn2n1
Show InChI InChI=1/C28H35N7O/c1-4-33(5-2)18-19-36-23-13-11-22(12-14-23)24-20-25(28-29-15-17-35(28)32-24)30-26-9-6-10-27(31-26)34-16-7-8-21(34)3/h6,9-15,17,20-21H,4-5,7-8,16,18-19H2,1-3H3,(H,30,31)
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n/an/a 60.6n/an/an/an/an/an/a



HOFFMANN-LA ROCHE INC.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 um filter plates (Millipore Cat. No.: MADVNOB10)Streptavidin coated beads: Streptavidin Sepharose, suspension ...


US Patent US9169259 (2015)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM188186
PNG
(US9169259, I-70)
Show SMILES CC1CCCN1c1cccc(Nc2cc(nn3ccnc23)-c2cccc(CN3CCCC3)c2)n1
Show InChI InChI=1/C27H31N7/c1-20-7-6-15-33(20)26-11-5-10-25(30-26)29-24-18-23(31-34-16-12-28-27(24)34)22-9-4-8-21(17-22)19-32-13-2-3-14-32/h4-5,8-12,16-18,20H,2-3,6-7,13-15,19H2,1H3,(H,29,30)
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n/an/a 60.8n/an/an/an/an/an/a



HOFFMANN-LA ROCHE INC.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 um filter plates (Millipore Cat. No.: MADVNOB10)Streptavidin coated beads: Streptavidin Sepharose, suspension ...


US Patent US9169259 (2015)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM188193
PNG
(US9169259, I-77)
Show SMILES CC1CCCN1c1cccc(Nc2cc(nn3ccnc23)-c2ccc(O)cc2)n1
Show InChI InChI=1/C22H22N6O/c1-15-4-3-12-27(15)21-6-2-5-20(25-21)24-19-14-18(16-7-9-17(29)10-8-16)26-28-13-11-23-22(19)28/h2,5-11,13-15,29H,3-4,12H2,1H3,(H,24,25)
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n/an/a 63.9n/an/an/an/an/an/a



HOFFMANN-LA ROCHE INC.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 um filter plates (Millipore Cat. No.: MADVNOB10)Streptavidin coated beads: Streptavidin Sepharose, suspension ...


US Patent US9169259 (2015)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM188194
PNG
(US9169259, I-78)
Show SMILES CC1CCCN1c1cccc(Nc2cc(nn3ccnc23)-c2cccnc2)n1
Show InChI InChI=1/C21H21N7/c1-15-5-4-11-27(15)20-8-2-7-19(25-20)24-18-13-17(16-6-3-9-22-14-16)26-28-12-10-23-21(18)28/h2-3,6-10,12-15H,4-5,11H2,1H3,(H,24,25)
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n/an/a 65.2n/an/an/an/an/an/a



HOFFMANN-LA ROCHE INC.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 um filter plates (Millipore Cat. No.: MADVNOB10)Streptavidin coated beads: Streptavidin Sepharose, suspension ...


US Patent US9169259 (2015)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM227536
PNG
(US9334278, I-25)
Show SMILES COc1ncc(Nc2cnc3[nH]cc(C(=O)NC(C)(C)C)c3n2)cn1
Show InChI InChI=1S/C16H19N7O2/c1-16(2,3)23-14(24)10-7-17-13-12(10)22-11(8-18-13)21-9-5-19-15(25-4)20-6-9/h5-8H,1-4H3,(H,17,18)(H,21,22)(H,23,24)
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n/an/a 71.2n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 μm filter plates (Millipore Cat. No.: MADVNOB 10) Streptavidin coated beads: Streptavidin Sepharose™,...


US Patent US9334278 (2016)

More data for this
Ligand-Target Pair
SYK RPA purified, truncated construct of Spleen Tyrosine Kinase aa 360-635


(Homo sapiens (human))
BDBM188163
PNG
(US9169259, I-45)
Show SMILES CC1CCCN1c1cccc(Nc2cc(nn3ccnc23)-c2ccccc2Cl)n1
Show InChI InChI=1/C22H21ClN6/c1-15-6-5-12-28(15)21-10-4-9-20(26-21)25-19-14-18(16-7-2-3-8-17(16)23)27-29-13-11-24-22(19)29/h2-4,7-11,13-15H,5-6,12H2,1H3,(H,25,26)
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n/an/a 71.2n/an/an/an/an/an/a



HOFFMANN-LA ROCHE INC.

US Patent


Assay Description
Assay plates: 96-well MultiScreen 0.65 um filter plates (Millipore Cat. No.: MADVNOB10)Streptavidin coated beads: Streptavidin Sepharose, suspension ...


US Patent US9169259 (2015)

More data for this
Ligand-Target Pair
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