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Compile Data Set for Download or QSAR

Found 121 hits Enz. Inhib. hit(s) with Target = 'Secreted frizzled-related protein 1' AND taxid = 9606   
Target
(Institution)
LigandTarget
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50308711
PNG
(4-{[4-({[5-(Phenylsulfonyl)-2-(trifluoromethyl)phe...)
Show SMILES OC(=O)c1ccc(cc1)S(=O)(=O)N1CCC(CC1)NS(=O)(=O)c1cc(ccc1C(F)(F)F)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C25H23F3N2O8S3/c26-25(27,28)22-11-10-21(39(33,34)19-4-2-1-3-5-19)16-23(22)40(35,36)29-18-12-14-30(15-13-18)41(37,38)20-8-6-17(7-9-20)24(31)32/h1-11,16,18,29H,12-15H2,(H,31,32)
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Wyeth Research

Curated by ChEMBL


Assay Description
Displacement of fluorescence probe compound from human SFRP1 after 30 mins by fluorescence polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50265555
PNG
((2S)-N-Phenyl-2-{[4-({[5-(phenylsulfonyl)-2-(trifl...)
Show SMILES FC(F)(F)c1ccc(cc1S(=O)(=O)NC1CCN(CC1)C(=O)[C@@H]1CCCN1C(=O)Nc1ccccc1)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C30H31F3N4O6S2/c31-30(32,33)25-14-13-24(44(40,41)23-10-5-2-6-11-23)20-27(25)45(42,43)35-22-15-18-36(19-16-22)28(38)26-12-7-17-37(26)29(39)34-21-8-3-1-4-9-21/h1-6,8-11,13-14,20,22,26,35H,7,12,15-19H2,(H,34,39)/t26-/m0/s1
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Wyeth Research

Curated by ChEMBL


Assay Description
Binding affinity to human purified SARP2 by fluorescent polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50265554
PNG
((2S)-N-(tert-Butyl)-2-{[4-({[5-(phenylsulfonyl)-2-...)
Show SMILES CC(C)(C)NC(=O)N1CCC[C@H]1C(=O)N1CCC(CC1)NS(=O)(=O)c1cc(ccc1C(F)(F)F)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C28H35F3N4O6S2/c1-27(2,3)32-26(37)35-15-7-10-23(35)25(36)34-16-13-19(14-17-34)33-43(40,41)24-18-21(11-12-22(24)28(29,30)31)42(38,39)20-8-5-4-6-9-20/h4-6,8-9,11-12,18-19,23,33H,7,10,13-17H2,1-3H3,(H,32,37)/t23-/m0/s1
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Wyeth Research

Curated by ChEMBL


Assay Description
Binding affinity to human purified SARP2 by fluorescent polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50265547
PNG
(CHEMBL455476 | N-{1-[1-(3,3-Dimethylbutanoyl)-L-pr...)
Show SMILES CC(C)(C)CC(=O)N1CCC[C@H]1C(=O)N1CCC(CC1)NS(=O)(=O)c1cc(ccc1C(F)(F)F)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C29H36F3N3O6S2/c1-28(2,3)19-26(36)35-15-7-10-24(35)27(37)34-16-13-20(14-17-34)33-43(40,41)25-18-22(11-12-23(25)29(30,31)32)42(38,39)21-8-5-4-6-9-21/h4-6,8-9,11-12,18,20,24,33H,7,10,13-17,19H2,1-3H3/t24-/m0/s1
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Wyeth Research

Curated by ChEMBL


Assay Description
Binding affinity to human purified SARP2 by fluorescent polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50308710
PNG
(3-{[4-({[5-(Phenylsulfonyl)-2-(trifluoromethyl)phe...)
Show SMILES OC(=O)c1cccc(c1)S(=O)(=O)N1CCC(CC1)NS(=O)(=O)c1cc(ccc1C(F)(F)F)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C25H23F3N2O8S3/c26-25(27,28)22-10-9-20(39(33,34)19-6-2-1-3-7-19)16-23(22)40(35,36)29-18-11-13-30(14-12-18)41(37,38)21-8-4-5-17(15-21)24(31)32/h1-10,15-16,18,29H,11-14H2,(H,31,32)
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Wyeth Research

Curated by ChEMBL


Assay Description
Displacement of fluorescence probe compound from human SFRP1 after 30 mins by fluorescence polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50265580
PNG
((2S)-N,N-Dimethyl-2-{[4-({[5-(phenylsulfonyl)-2-(t...)
Show SMILES CN(C)C(=O)N1CCC[C@H]1C(=O)N1CCC(CC1)NS(=O)(=O)c1cc(ccc1C(F)(F)F)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C26H31F3N4O6S2/c1-31(2)25(35)33-14-6-9-22(33)24(34)32-15-12-18(13-16-32)30-41(38,39)23-17-20(10-11-21(23)26(27,28)29)40(36,37)19-7-4-3-5-8-19/h3-5,7-8,10-11,17-18,22,30H,6,9,12-16H2,1-2H3/t22-/m0/s1
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Wyeth Research

Curated by ChEMBL


Assay Description
Binding affinity to human purified SARP2 by fluorescent polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50265553
PNG
((2S)-N-Ethyl-2-{[4-({[5-(phenylsulfonyl)-2-(triflu...)
Show SMILES CCNC(=O)N1CCC[C@H]1C(=O)N1CCC(CC1)NS(=O)(=O)c1cc(ccc1C(F)(F)F)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C26H31F3N4O6S2/c1-2-30-25(35)33-14-6-9-22(33)24(34)32-15-12-18(13-16-32)31-41(38,39)23-17-20(10-11-21(23)26(27,28)29)40(36,37)19-7-4-3-5-8-19/h3-5,7-8,10-11,17-18,22,31H,2,6,9,12-16H2,1H3,(H,30,35)/t22-/m0/s1
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Wyeth Research

Curated by ChEMBL


Assay Description
Binding affinity to human purified SARP2 by fluorescent polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50265499
PNG
(CHEMBL495534 | N-[1-(1H-Imidazol-1-ylacetyl)piperi...)
Show SMILES FC(F)(F)c1ccc(cc1S(=O)(=O)NC1CCN(CC1)C(=O)Cn1ccnc1)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C23H23F3N4O5S2/c24-23(25,26)20-7-6-19(36(32,33)18-4-2-1-3-5-18)14-21(20)37(34,35)28-17-8-11-30(12-9-17)22(31)15-29-13-10-27-16-29/h1-7,10,13-14,16-17,28H,8-9,11-12,15H2
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Wyeth Research

Curated by ChEMBL


Assay Description
Binding affinity to human purified SARP2 by fluorescent polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50265583
PNG
(CHEMBL451431 | N-{1-[1-(3,3-Dimethylbutyl)-L-proly...)
Show SMILES CC(C)(C)CCN1CCC[C@H]1C(=O)N1CCC(CC1)NS(=O)(=O)c1cc(ccc1C(F)(F)F)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C29H38F3N3O5S2/c1-28(2,3)15-19-34-16-7-10-25(34)27(36)35-17-13-21(14-18-35)33-42(39,40)26-20-23(11-12-24(26)29(30,31)32)41(37,38)22-8-5-4-6-9-22/h4-6,8-9,11-12,20-21,25,33H,7,10,13-19H2,1-3H3/t25-/m0/s1
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Wyeth Research

Curated by ChEMBL


Assay Description
Binding affinity to human purified SARP2 by fluorescent polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50308712
PNG
(5-(Phenylsulfonyl)-N-(1-{[3-(2H-tetrazol-5-yl)phen...)
Show SMILES FC(F)(F)c1ccc(cc1S(=O)(=O)NC1CCN(CC1)S(=O)(=O)c1cccc(c1)-c1nnn[nH]1)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C25H23F3N6O6S3/c26-25(27,28)22-10-9-20(41(35,36)19-6-2-1-3-7-19)16-23(22)42(37,38)31-18-11-13-34(14-12-18)43(39,40)21-8-4-5-17(15-21)24-29-32-33-30-24/h1-10,15-16,18,31H,11-14H2,(H,29,30,32,33)
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Wyeth Research

Curated by ChEMBL


Assay Description
Displacement of fluorescence probe compound from human SFRP1 after 30 mins by fluorescence polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50265584
PNG
(CHEMBL503281 | N-{1-[1-(Cyclohexylmethyl)-L-prolyl...)
Show SMILES FC(F)(F)c1ccc(cc1S(=O)(=O)NC1CCN(CC1)C(=O)[C@@H]1CCCN1CC1CCCCC1)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C30H38F3N3O5S2/c31-30(32,33)26-14-13-25(42(38,39)24-10-5-2-6-11-24)20-28(26)43(40,41)34-23-15-18-35(19-16-23)29(37)27-12-7-17-36(27)21-22-8-3-1-4-9-22/h2,5-6,10-11,13-14,20,22-23,27,34H,1,3-4,7-9,12,15-19,21H2/t27-/m0/s1
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Wyeth Research

Curated by ChEMBL


Assay Description
Binding affinity to human purified SARP2 by fluorescent polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50308701
PNG
(5-(Phenylsulfonyl)-N-{1-[(3S)-pyrrolidin-3-ylcarbo...)
Show SMILES FC(F)(F)c1ccc(cc1S(=O)(=O)NC1CCN(CC1)C(=O)[C@H]1CCNC1)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C23H26F3N3O5S2/c24-23(25,26)20-7-6-19(35(31,32)18-4-2-1-3-5-18)14-21(20)36(33,34)28-17-9-12-29(13-10-17)22(30)16-8-11-27-15-16/h1-7,14,16-17,27-28H,8-13,15H2/t16-/m0/s1
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Wyeth Research

Curated by ChEMBL


Assay Description
Displacement of fluorescence probe compound from human SFRP1 after 30 mins by fluorescence polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50265545
PNG
(CHEMBL500903 | N-[1-(1-Isobutyryl-L-prolyl)piperid...)
Show SMILES CC(C)C(=O)N1CCC[C@H]1C(=O)N1CCC(CC1)NS(=O)(=O)c1cc(ccc1C(F)(F)F)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C27H32F3N3O6S2/c1-18(2)25(34)33-14-6-9-23(33)26(35)32-15-12-19(13-16-32)31-41(38,39)24-17-21(10-11-22(24)27(28,29)30)40(36,37)20-7-4-3-5-8-20/h3-5,7-8,10-11,17-19,23,31H,6,9,12-16H2,1-2H3/t23-/m0/s1
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Wyeth Research

Curated by ChEMBL


Assay Description
Binding affinity to human purified SARP2 by fluorescent polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50265546
PNG
(CHEMBL447079 | N-{1-[1-(2,2-Dimethylpropanoyl)-L-p...)
Show SMILES CC(C)(C)C(=O)N1CCC[C@H]1C(=O)N1CCC(CC1)NS(=O)(=O)c1cc(ccc1C(F)(F)F)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C28H34F3N3O6S2/c1-27(2,3)26(36)34-15-7-10-23(34)25(35)33-16-13-19(14-17-33)32-42(39,40)24-18-21(11-12-22(24)28(29,30)31)41(37,38)20-8-5-4-6-9-20/h4-6,8-9,11-12,18-19,23,32H,7,10,13-17H2,1-3H3/t23-/m0/s1
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Wyeth Research

Curated by ChEMBL


Assay Description
Binding affinity to human purified SARP2 by fluorescent polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50265581
PNG
(CHEMBL505036 | N-{1-[1-(Morpholin-4-ylcarbonyl)-L-...)
Show SMILES FC(F)(F)c1ccc(cc1S(=O)(=O)NC1CCN(CC1)C(=O)[C@@H]1CCCN1C(=O)N1CCOCC1)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C28H33F3N4O7S2/c29-28(30,31)23-9-8-22(43(38,39)21-5-2-1-3-6-21)19-25(23)44(40,41)32-20-10-13-33(14-11-20)26(36)24-7-4-12-35(24)27(37)34-15-17-42-18-16-34/h1-3,5-6,8-9,19-20,24,32H,4,7,10-18H2/t24-/m0/s1
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Wyeth Research

Curated by ChEMBL


Assay Description
Binding affinity to human purified SARP2 by fluorescent polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50308692
PNG
(CHEMBL606033 | N-(1-{[6-(Dimethylamino)pyridin-3-y...)
Show SMILES CN(C)c1ccc(cn1)C(=O)N1CCC(CC1)NS(=O)(=O)c1cc(ccc1C(F)(F)F)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C26H27F3N4O5S2/c1-32(2)24-11-8-18(17-30-24)25(34)33-14-12-19(13-15-33)31-40(37,38)23-16-21(9-10-22(23)26(27,28)29)39(35,36)20-6-4-3-5-7-20/h3-11,16-17,19,31H,12-15H2,1-2H3
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Wyeth Research

Curated by ChEMBL


Assay Description
Displacement of fluorescence probe compound from human SFRP1 after 30 mins by fluorescence polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50308698
PNG
(CHEMBL600050 | tert-Butyl(3R)-3-{[4-({[5-(phenylsu...)
Show SMILES CC(C)(C)OC(=O)N1CC[C@H](C1)C(=O)N1CCC(CC1)NS(=O)(=O)c1cc(ccc1C(F)(F)F)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C28H34F3N3O7S2/c1-27(2,3)41-26(36)34-14-11-19(18-34)25(35)33-15-12-20(13-16-33)32-43(39,40)24-17-22(9-10-23(24)28(29,30)31)42(37,38)21-7-5-4-6-8-21/h4-10,17,19-20,32H,11-16,18H2,1-3H3/t19-/m1/s1
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Wyeth Research

Curated by ChEMBL


Assay Description
Displacement of fluorescence probe compound from human SFRP1 after 30 mins by fluorescence polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50308691
PNG
(5-(Phenylsulfonyl)-2-(trifluoromethyl)-N-(1-{[6-(t...)
Show SMILES FC(F)(F)c1ccc(cn1)C(=O)N1CCC(CC1)NS(=O)(=O)c1cc(ccc1C(F)(F)F)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C25H21F6N3O5S2/c26-24(27,28)20-8-7-19(40(36,37)18-4-2-1-3-5-18)14-21(20)41(38,39)33-17-10-12-34(13-11-17)23(35)16-6-9-22(32-15-16)25(29,30)31/h1-9,14-15,17,33H,10-13H2
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Wyeth Research

Curated by ChEMBL


Assay Description
Displacement of fluorescence probe compound from human SFRP1 after 30 mins by fluorescence polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50265549
PNG
(CHEMBL507695 | N-{1-[1-(Cyclohexylcarbonyl)-L-prol...)
Show SMILES FC(F)(F)c1ccc(cc1S(=O)(=O)NC1CCN(CC1)C(=O)[C@@H]1CCCN1C(=O)C1CCCCC1)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C30H36F3N3O6S2/c31-30(32,33)25-14-13-24(43(39,40)23-10-5-2-6-11-23)20-27(25)44(41,42)34-22-15-18-35(19-16-22)29(38)26-12-7-17-36(26)28(37)21-8-3-1-4-9-21/h2,5-6,10-11,13-14,20-22,26,34H,1,3-4,7-9,12,15-19H2/t26-/m0/s1
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n/an/a 50n/an/an/an/an/an/a



Wyeth Research

Curated by ChEMBL


Assay Description
Binding affinity to human purified SARP2 by fluorescent polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50308703
PNG
(2-[4-({[5-(Phenylsulfonyl)-2-(trifluoromethyl)phen...)
Show SMILES NC(=O)CN1CCC(CC1)NS(=O)(=O)c1cc(ccc1C(F)(F)F)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C20H22F3N3O5S2/c21-20(22,23)17-7-6-16(32(28,29)15-4-2-1-3-5-15)12-18(17)33(30,31)25-14-8-10-26(11-9-14)13-19(24)27/h1-7,12,14,25H,8-11,13H2,(H2,24,27)
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n/an/a 60n/an/an/an/an/an/a



Wyeth Research

Curated by ChEMBL


Assay Description
Displacement of fluorescence probe compound from human SFRP1 after 30 mins by fluorescence polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50265500
PNG
((S)-tert-butyl 2-(4-(5-(phenylsulfonyl)-2-(trifluo...)
Show SMILES CC(C)(C)OC(=O)N1CCC[C@H]1C(=O)N1CCC(CC1)NS(=O)(=O)c1cc(ccc1C(F)(F)F)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C28H34F3N3O7S2/c1-27(2,3)41-26(36)34-15-7-10-23(34)25(35)33-16-13-19(14-17-33)32-43(39,40)24-18-21(11-12-22(24)28(29,30)31)42(37,38)20-8-5-4-6-9-20/h4-6,8-9,11-12,18-19,23,32H,7,10,13-17H2,1-3H3/t23-/m0/s1
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n/an/a 60n/an/an/an/an/an/a



Wyeth Research

Curated by ChEMBL


Assay Description
Binding affinity to human purified SARP2 by fluorescent polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50308688
PNG
(5-(Phenylsulfonyl)-N-[1-(pyridin-3-ylcarbonyl)pipe...)
Show SMILES FC(F)(F)c1ccc(cc1S(=O)(=O)NC1CCN(CC1)C(=O)c1ccccn1)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C24H22F3N3O5S2/c25-24(26,27)20-10-9-19(36(32,33)18-6-2-1-3-7-18)16-22(20)37(34,35)29-17-11-14-30(15-12-17)23(31)21-8-4-5-13-28-21/h1-10,13,16-17,29H,11-12,14-15H2
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n/an/a 60n/an/an/an/an/an/a



Wyeth Research

Curated by ChEMBL


Assay Description
Displacement of fluorescence probe compound from human SFRP1 after 30 mins by fluorescence polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50265500
PNG
((S)-tert-butyl 2-(4-(5-(phenylsulfonyl)-2-(trifluo...)
Show SMILES CC(C)(C)OC(=O)N1CCC[C@H]1C(=O)N1CCC(CC1)NS(=O)(=O)c1cc(ccc1C(F)(F)F)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C28H34F3N3O7S2/c1-27(2,3)41-26(36)34-15-7-10-23(34)25(35)33-16-13-19(14-17-33)32-43(39,40)24-18-21(11-12-22(24)28(29,30)31)42(37,38)20-8-5-4-6-9-20/h4-6,8-9,11-12,18-19,23,32H,7,10,13-17H2,1-3H3/t23-/m0/s1
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Wyeth Research

Curated by ChEMBL


Assay Description
Displacement of fluorescence probe compound from human SFRP1 after 30 mins by fluorescence polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50308702
PNG
(5-(Phenylsulfonyl)-N-{1-[(3R)-pyrrolidin-3-ylcarbo...)
Show SMILES FC(F)(F)c1ccc(cc1S(=O)(=O)NC1CCN(CC1)C(=O)[C@@H]1CCNC1)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C23H26F3N3O5S2/c24-23(25,26)20-7-6-19(35(31,32)18-4-2-1-3-5-18)14-21(20)36(33,34)28-17-9-12-29(13-10-17)22(30)16-8-11-27-15-16/h1-7,14,16-17,27-28H,8-13,15H2/t16-/m1/s1
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Wyeth Research

Curated by ChEMBL


Assay Description
Displacement of fluorescence probe compound from human SFRP1 after 30 mins by fluorescence polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50308681
PNG
(CHEMBL589088 | N-(1-Benzoylpiperidin-4-yl)-5-(phen...)
Show SMILES FC(F)(F)c1ccc(cc1S(=O)(=O)NC1CCN(CC1)C(=O)c1ccccc1)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C25H23F3N2O5S2/c26-25(27,28)22-12-11-21(36(32,33)20-9-5-2-6-10-20)17-23(22)37(34,35)29-19-13-15-30(16-14-19)24(31)18-7-3-1-4-8-18/h1-12,17,19,29H,13-16H2
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n/an/a 70n/an/an/an/an/an/a



Wyeth Research

Curated by ChEMBL


Assay Description
Displacement of fluorescence probe compound from human SFRP1 after 30 mins by fluorescence polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50265552
PNG
(CHEMBL454478 | N-[1-(1-Isonicotinoyl-L-prolyl)pipe...)
Show SMILES FC(F)(F)c1ccc(cc1S(=O)(=O)NC1CCN(CC1)C(=O)[C@@H]1CCCN1C(=O)c1ccncc1)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C29H29F3N4O6S2/c30-29(31,32)24-9-8-23(43(39,40)22-5-2-1-3-6-22)19-26(24)44(41,42)34-21-12-17-35(18-13-21)28(38)25-7-4-16-36(25)27(37)20-10-14-33-15-11-20/h1-3,5-6,8-11,14-15,19,21,25,34H,4,7,12-13,16-18H2/t25-/m0/s1
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n/an/a 70n/an/an/an/an/an/a



Wyeth Research

Curated by ChEMBL


Assay Description
Binding affinity to human purified SARP2 by fluorescent polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50265550
PNG
(CHEMBL510748 | N-[1-(1-Benzoyl-L-prolyl)piperidin-...)
Show SMILES FC(F)(F)c1ccc(cc1S(=O)(=O)NC1CCN(CC1)C(=O)[C@@H]1CCCN1C(=O)c1ccccc1)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C30H30F3N3O6S2/c31-30(32,33)25-14-13-24(43(39,40)23-10-5-2-6-11-23)20-27(25)44(41,42)34-22-15-18-35(19-16-22)29(38)26-12-7-17-36(26)28(37)21-8-3-1-4-9-21/h1-6,8-11,13-14,20,22,26,34H,7,12,15-19H2/t26-/m0/s1
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n/an/a 70n/an/an/an/an/an/a



Wyeth Research

Curated by ChEMBL


Assay Description
Binding affinity to human purified SARP2 by fluorescent polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50308697
PNG
(CHEMBL600049 | tert-Butyl(3S)-3-{[4-({[5-(phenylsu...)
Show SMILES CC(C)(C)OC(=O)N1CC[C@@H](C1)C(=O)N1CCC(CC1)NS(=O)(=O)c1cc(ccc1C(F)(F)F)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C28H34F3N3O7S2/c1-27(2,3)41-26(36)34-14-11-19(18-34)25(35)33-15-12-20(13-16-33)32-43(39,40)24-17-22(9-10-23(24)28(29,30)31)42(37,38)21-7-5-4-6-8-21/h4-10,17,19-20,32H,11-16,18H2,1-3H3/t19-/m0/s1
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Wyeth Research

Curated by ChEMBL


Assay Description
Displacement of fluorescence probe compound from human SFRP1 after 30 mins by fluorescence polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50308689
PNG
(CHEMBL589067 | N-(1-Isonicotinoylpiperidin-4-yl)-5...)
Show SMILES FC(F)(F)c1ccc(cc1S(=O)(=O)NC1CCN(CC1)C(=O)c1cccnc1)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C24H22F3N3O5S2/c25-24(26,27)21-9-8-20(36(32,33)19-6-2-1-3-7-19)15-22(21)37(34,35)29-18-10-13-30(14-11-18)23(31)17-5-4-12-28-16-17/h1-9,12,15-16,18,29H,10-11,13-14H2
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n/an/a 80n/an/an/an/an/an/a



Wyeth Research

Curated by ChEMBL


Assay Description
Displacement of fluorescence probe compound from human SFRP1 after 30 mins by fluorescence polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50308713
PNG
(CHEMBL592455 | N-{1-[(3-Cyanophenyl)sulfonyl]piper...)
Show SMILES FC(F)(F)c1ccc(cc1S(=O)(=O)NC1CCN(CC1)S(=O)(=O)c1cccc(c1)C#N)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C25H22F3N3O6S3/c26-25(27,28)23-10-9-21(38(32,33)20-6-2-1-3-7-20)16-24(23)39(34,35)30-19-11-13-31(14-12-19)40(36,37)22-8-4-5-18(15-22)17-29/h1-10,15-16,19,30H,11-14H2
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n/an/a 90n/an/an/an/an/an/a



Wyeth Research

Curated by ChEMBL


Assay Description
Displacement of fluorescence probe compound from human SFRP1 after 30 mins by fluorescence polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50265548
PNG
(CHEMBL501332 | N-[1-(N,N-Dimethylglycyl-L-prolyl)p...)
Show SMILES CN(C)CC(=O)N1CCC[C@H]1C(=O)N1CCC(CC1)NS(=O)(=O)c1cc(ccc1C(F)(F)F)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C27H33F3N4O6S2/c1-32(2)18-25(35)34-14-6-9-23(34)26(36)33-15-12-19(13-16-33)31-42(39,40)24-17-21(10-11-22(24)27(28,29)30)41(37,38)20-7-4-3-5-8-20/h3-5,7-8,10-11,17,19,23,31H,6,9,12-16,18H2,1-2H3/t23-/m0/s1
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n/an/a 90n/an/an/an/an/an/a



Wyeth Research

Curated by ChEMBL


Assay Description
Binding affinity to human purified SARP2 by fluorescent polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50265505
PNG
(CHEMBL525899 | N-[1-(5-oxo-L-Prolyl)piperidin-4-yl...)
Show SMILES FC(F)(F)c1ccc(cc1S(=O)(=O)NC1CCN(CC1)C(=O)[C@@H]1CCC(=O)N1)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C23H24F3N3O6S2/c24-23(25,26)18-7-6-17(36(32,33)16-4-2-1-3-5-16)14-20(18)37(34,35)28-15-10-12-29(13-11-15)22(31)19-8-9-21(30)27-19/h1-7,14-15,19,28H,8-13H2,(H,27,30)/t19-/m0/s1
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n/an/a 90n/an/an/an/an/an/a



Wyeth Research

Curated by ChEMBL


Assay Description
Binding affinity to human purified SARP2 by fluorescent polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50265480
PNG
(CHEMBL523726 | N-[1-(Morpholin-4-ylacetyl)piperidi...)
Show SMILES FC(F)(F)c1ccc(cc1S(=O)(=O)NC1CCN(CC1)C(=O)CN1CCOCC1)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C24H28F3N3O6S2/c25-24(26,27)21-7-6-20(37(32,33)19-4-2-1-3-5-19)16-22(21)38(34,35)28-18-8-10-30(11-9-18)23(31)17-29-12-14-36-15-13-29/h1-7,16,18,28H,8-15,17H2
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n/an/a 100n/an/an/an/an/an/a



Wyeth Research

Curated by ChEMBL


Assay Description
Binding affinity to human purified SARP2 by fluorescent polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50308714
PNG
(3-[4-({[5-(Phenylsulfonyl)-2-(trifluoromethyl)phen...)
Show SMILES OC(=O)c1cccc(c1)N1CCC(CC1)NS(=O)(=O)c1cc(ccc1C(F)(F)F)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C25H23F3N2O6S2/c26-25(27,28)22-10-9-21(37(33,34)20-7-2-1-3-8-20)16-23(22)38(35,36)29-18-11-13-30(14-12-18)19-6-4-5-17(15-19)24(31)32/h1-10,15-16,18,29H,11-14H2,(H,31,32)
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n/an/a 100n/an/an/an/an/an/a



Wyeth Research

Curated by ChEMBL


Assay Description
Displacement of fluorescence probe compound from human SFRP1 after 30 mins by fluorescence polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50308700
PNG
(5-(Phenylsulfonyl)-N-[1-(piperidin-4-ylacetyl)pipe...)
Show SMILES FC(F)(F)c1ccc(cc1S(=O)(=O)NC1CCN(CC1)C(=O)CC1CCNCC1)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C25H30F3N3O5S2/c26-25(27,28)22-7-6-21(37(33,34)20-4-2-1-3-5-20)17-23(22)38(35,36)30-19-10-14-31(15-11-19)24(32)16-18-8-12-29-13-9-18/h1-7,17-19,29-30H,8-16H2
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Wyeth Research

Curated by ChEMBL


Assay Description
Displacement of fluorescence probe compound from human SFRP1 after 30 mins by fluorescence polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50308690
PNG
(CHEMBL605196 | N-{1-[(6-Chloropyridin-3-yl)carbony...)
Show SMILES FC(F)(F)c1ccc(cc1S(=O)(=O)NC1CCN(CC1)C(=O)c1ccc(Cl)nc1)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C24H21ClF3N3O5S2/c25-22-9-6-16(15-29-22)23(32)31-12-10-17(11-13-31)30-38(35,36)21-14-19(7-8-20(21)24(26,27)28)37(33,34)18-4-2-1-3-5-18/h1-9,14-15,17,30H,10-13H2
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n/an/a 110n/an/an/an/an/an/a



Wyeth Research

Curated by ChEMBL


Assay Description
Displacement of fluorescence probe compound from human SFRP1 after 30 mins by fluorescence polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50265551
PNG
(CHEMBL462363 | N-(1-{1-[4-(Dimethylamino)benzoyl]-...)
Show SMILES CN(C)c1ccc(cc1)C(=O)N1CCC[C@H]1C(=O)N1CCC(CC1)NS(=O)(=O)c1cc(ccc1C(F)(F)F)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C32H35F3N4O6S2/c1-37(2)24-12-10-22(11-13-24)30(40)39-18-6-9-28(39)31(41)38-19-16-23(17-20-38)36-47(44,45)29-21-26(14-15-27(29)32(33,34)35)46(42,43)25-7-4-3-5-8-25/h3-5,7-8,10-15,21,23,28,36H,6,9,16-20H2,1-2H3/t28-/m0/s1
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Wyeth Research

Curated by ChEMBL


Assay Description
Binding affinity to human purified SARP2 by fluorescent polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50265503
PNG
((S)-5-(phenylsulfonyl)-N-(1-(pyrrolidine-2-carbony...)
Show SMILES FC(F)(F)c1ccc(cc1S(=O)(=O)NC1CCN(CC1)C(=O)[C@@H]1CCCN1)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C23H26F3N3O5S2/c24-23(25,26)19-9-8-18(35(31,32)17-5-2-1-3-6-17)15-21(19)36(33,34)28-16-10-13-29(14-11-16)22(30)20-7-4-12-27-20/h1-3,5-6,8-9,15-16,20,27-28H,4,7,10-14H2/t20-/m0/s1
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n/an/a 110n/an/an/an/an/an/a



Wyeth Research

Curated by ChEMBL


Assay Description
Binding affinity to human purified SARP2 by fluorescent polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50265503
PNG
((S)-5-(phenylsulfonyl)-N-(1-(pyrrolidine-2-carbony...)
Show SMILES FC(F)(F)c1ccc(cc1S(=O)(=O)NC1CCN(CC1)C(=O)[C@@H]1CCCN1)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C23H26F3N3O5S2/c24-23(25,26)19-9-8-18(35(31,32)17-5-2-1-3-6-17)15-21(19)36(33,34)28-16-10-13-29(14-11-16)22(30)20-7-4-12-27-20/h1-3,5-6,8-9,15-16,20,27-28H,4,7,10-14H2/t20-/m0/s1
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n/an/a 110n/an/an/an/an/an/a



Wyeth Research

Curated by ChEMBL


Assay Description
Displacement of fluorescence probe compound from human SFRP1 after 30 mins by fluorescence polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50265479
PNG
(5-(Phenylsulfonyl)-N-[1-(pyrrolidin-1-ylacetyl)pip...)
Show SMILES FC(F)(F)c1ccc(cc1S(=O)(=O)NC1CCN(CC1)C(=O)CN1CCCC1)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C24H28F3N3O5S2/c25-24(26,27)21-9-8-20(36(32,33)19-6-2-1-3-7-19)16-22(21)37(34,35)28-18-10-14-30(15-11-18)23(31)17-29-12-4-5-13-29/h1-3,6-9,16,18,28H,4-5,10-15,17H2
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n/an/a 110n/an/an/an/an/an/a



Wyeth Research

Curated by ChEMBL


Assay Description
Binding affinity to human purified SARP2 by fluorescent polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50265501
PNG
((R)-tert-butyl 2-(4-(5-(phenylsulfonyl)-2-(trifluo...)
Show SMILES CC(C)(C)OC(=O)N1CCC[C@@H]1C(=O)N1CCC(CC1)NS(=O)(=O)c1cc(ccc1C(F)(F)F)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C28H34F3N3O7S2/c1-27(2,3)41-26(36)34-15-7-10-23(34)25(35)33-16-13-19(14-17-33)32-43(39,40)24-18-21(11-12-22(24)28(29,30)31)42(37,38)20-8-5-4-6-9-20/h4-6,8-9,11-12,18-19,23,32H,7,10,13-17H2,1-3H3/t23-/m1/s1
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n/an/a 120n/an/an/an/an/an/a



Wyeth Research

Curated by ChEMBL


Assay Description
Binding affinity to human purified SARP2 by fluorescent polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50265501
PNG
((R)-tert-butyl 2-(4-(5-(phenylsulfonyl)-2-(trifluo...)
Show SMILES CC(C)(C)OC(=O)N1CCC[C@@H]1C(=O)N1CCC(CC1)NS(=O)(=O)c1cc(ccc1C(F)(F)F)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C28H34F3N3O7S2/c1-27(2,3)41-26(36)34-15-7-10-23(34)25(35)33-16-13-19(14-17-33)32-43(39,40)24-18-21(11-12-22(24)28(29,30)31)42(37,38)20-8-5-4-6-9-20/h4-6,8-9,11-12,18-19,23,32H,7,10,13-17H2,1-3H3/t23-/m1/s1
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n/an/a 120n/an/an/an/an/an/a



Wyeth Research

Curated by ChEMBL


Assay Description
Displacement of fluorescence probe compound from human SFRP1 after 30 mins by fluorescence polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50308715
PNG
(4-[4-({[5-(Phenylsulfonyl)-2-(trifluoromethyl)phen...)
Show SMILES OC(=O)c1ccc(cc1)N1CCC(CC1)NS(=O)(=O)c1cc(ccc1C(F)(F)F)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C25H23F3N2O6S2/c26-25(27,28)22-11-10-21(37(33,34)20-4-2-1-3-5-20)16-23(22)38(35,36)29-18-12-14-30(15-13-18)19-8-6-17(7-9-19)24(31)32/h1-11,16,18,29H,12-15H2,(H,31,32)
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n/an/a 120n/an/an/an/an/an/a



Wyeth Research

Curated by ChEMBL


Assay Description
Displacement of fluorescence probe compound from human SFRP1 after 30 mins by fluorescence polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50308699
PNG
(5-(Phenylsulfonyl)-N-[1-(piperidin-4-ylcarbonyl)pi...)
Show SMILES FC(F)(F)c1ccc(cc1S(=O)(=O)NC1CCN(CC1)C(=O)C1CCNCC1)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C24H28F3N3O5S2/c25-24(26,27)21-7-6-20(36(32,33)19-4-2-1-3-5-19)16-22(21)37(34,35)29-18-10-14-30(15-11-18)23(31)17-8-12-28-13-9-17/h1-7,16-18,28-29H,8-15H2
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n/an/a 120n/an/an/an/an/an/a



Wyeth Research

Curated by ChEMBL


Assay Description
Displacement of fluorescence probe compound from human SFRP1 after 30 mins by fluorescence polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50265582
PNG
(CHEMBL496581 | N-[1-(1-Methyl-L-prolyl)piperidin-4...)
Show SMILES CN1CCC[C@H]1C(=O)N1CCC(CC1)NS(=O)(=O)c1cc(ccc1C(F)(F)F)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C24H28F3N3O5S2/c1-29-13-5-8-21(29)23(31)30-14-11-17(12-15-30)28-37(34,35)22-16-19(9-10-20(22)24(25,26)27)36(32,33)18-6-3-2-4-7-18/h2-4,6-7,9-10,16-17,21,28H,5,8,11-15H2,1H3/t21-/m0/s1
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n/an/a 120n/an/an/an/an/an/a



Wyeth Research

Curated by ChEMBL


Assay Description
Binding affinity to human purified SARP2 by fluorescent polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50308694
PNG
(CHEMBL590478 | N-{1-[(6-Morpholin-4-ylpyridin-3-yl...)
Show SMILES FC(F)(F)c1ccc(cc1S(=O)(=O)NC1CCN(CC1)C(=O)c1ccc(nc1)N1CCOCC1)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C28H29F3N4O6S2/c29-28(30,31)24-8-7-23(42(37,38)22-4-2-1-3-5-22)18-25(24)43(39,40)33-21-10-12-35(13-11-21)27(36)20-6-9-26(32-19-20)34-14-16-41-17-15-34/h1-9,18-19,21,33H,10-17H2
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n/an/a 130n/an/an/an/an/an/a



Wyeth Research

Curated by ChEMBL


Assay Description
Displacement of fluorescence probe compound from human SFRP1 after 30 mins by fluorescence polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50308716
PNG
(5-(Phenylsulfonyl)-N-[1-(phenylsulfonyl)piperidin-...)
Show SMILES FC(F)(F)c1ccc(cc1S(=O)(=O)NC1CCN(CC1)S(=O)(=O)c1ccccc1)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C24H23F3N2O6S3/c25-24(26,27)22-12-11-21(36(30,31)19-7-3-1-4-8-19)17-23(22)37(32,33)28-18-13-15-29(16-14-18)38(34,35)20-9-5-2-6-10-20/h1-12,17-18,28H,13-16H2
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n/an/a 130n/an/an/an/an/an/a



Wyeth Research

Curated by ChEMBL


Assay Description
Displacement of fluorescence probe compound from human SFRP1 after 30 mins by fluorescence polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50265502
PNG
(CHEMBL504979 | tert-Butyl(5S)-2-oxo-5-{[4-({[5-(Ph...)
Show SMILES CC(C)(C)OC(=O)N1[C@@H](CCC1=O)C(=O)N1CCC(CC1)NS(=O)(=O)c1cc(ccc1C(F)(F)F)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C28H32F3N3O8S2/c1-27(2,3)42-26(37)34-22(11-12-24(34)35)25(36)33-15-13-18(14-16-33)32-44(40,41)23-17-20(9-10-21(23)28(29,30)31)43(38,39)19-7-5-4-6-8-19/h4-10,17-18,22,32H,11-16H2,1-3H3/t22-/m0/s1
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n/an/a 130n/an/an/an/an/an/a



Wyeth Research

Curated by ChEMBL


Assay Description
Binding affinity to human purified SARP2 by fluorescent polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50265481
PNG
(5-(Phenylsulfonyl)-N-[1-(piperazin-1-ylacetyl)pipe...)
Show SMILES FC(F)(F)c1ccc(cc1S(=O)(=O)NC1CCN(CC1)C(=O)CN1CCNCC1)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C24H29F3N4O5S2/c25-24(26,27)21-7-6-20(37(33,34)19-4-2-1-3-5-19)16-22(21)38(35,36)29-18-8-12-31(13-9-18)23(32)17-30-14-10-28-11-15-30/h1-7,16,18,28-29H,8-15,17H2
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n/an/a 140n/an/an/an/an/an/a



Wyeth Research

Curated by ChEMBL


Assay Description
Binding affinity to human purified SARP2 by fluorescent polarization assay


Citation and Details
More data for this
Ligand-Target Pair
Secreted frizzled-related protein 1


(Homo sapiens)
BDBM50265544
PNG
(CHEMBL525970 | N-[1-(1-Acetyl-L-prolyl)piperidin-4...)
Show SMILES CC(=O)N1CCC[C@H]1C(=O)N1CCC(CC1)NS(=O)(=O)c1cc(ccc1C(F)(F)F)S(=O)(=O)c1ccccc1
Show InChI InChI=1S/C25H28F3N3O6S2/c1-17(32)31-13-5-8-22(31)24(33)30-14-11-18(12-15-30)29-39(36,37)23-16-20(9-10-21(23)25(26,27)28)38(34,35)19-6-3-2-4-7-19/h2-4,6-7,9-10,16,18,22,29H,5,8,11-15H2,1H3/t22-/m0/s1
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n/an/a 160n/an/an/an/an/an/a



Wyeth Research

Curated by ChEMBL


Assay Description
Binding affinity to human purified SARP2 by fluorescent polarization assay


Citation and Details
More data for this
Ligand-Target Pair
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