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Found 625 hits Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily A member 1 (TRPA1)' AND taxid = 9606   
Target
(Institution)
LigandTarget
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM50318511
PNG
(CHEMBL1085100 | dibenzo[b,f][1,4]oxazepine)
Show SMILES O1c2ccccc2C=Nc2ccccc12
Show InChI InChI=1S/C13H9NO/c1-3-7-12-10(5-1)9-14-11-6-2-4-8-13(11)15-12/h1-9H
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PubMed
n/an/a 0.700n/an/an/an/an/an/a



Johnson& Johnson Pharmaceutical Research& Development

Curated by ChEMBL


Assay Description
Agonist activity at human TRPA1 expressed in T-REx-HEK293 cells assessed as concentration required to incapacitate 50% of the population exposed to t...


Citation and Details
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191653
PNG
(US9186360, 57)
Show SMILES Cn1c2occ(CC(=O)Nc3nc(cs3)-c3cc(Cl)c(OCC(F)(F)F)c(Cl)c3)c2c(=O)n(C)c1=O
Show InChI InChI=1S/C21H15Cl2F3N4O5S/c1-29-17(32)15-10(6-34-18(15)30(2)20(29)33)5-14(31)28-19-27-13(7-36-19)9-3-11(22)16(12(23)4-9)35-8-21(24,25)26/h3-4,6-7H,5,8H2,1-2H3,(H,27,28,31)
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US Patent
n/an/a 1.45n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM60874
PNG
(US9186360, 62)
Show SMILES Cc1oc2n(C)c(=O)n(C)c(=O)c2c1CC(=O)Nc1nc(cs1)-c1cc(F)c(OCC(F)(F)F)c(F)c1
Show InChI InChI=1S/C22H17F5N4O5S/c1-9-11(16-18(33)30(2)21(34)31(3)19(16)36-9)6-15(32)29-20-28-14(7-37-20)10-4-12(23)17(13(24)5-10)35-8-22(25,26)27/h4-5,7H,6,8H2,1-3H3,(H,28,29,32)
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US Patent
n/an/a 1.68n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191709
PNG
(US9186360, 55)
Show SMILES Cn1c2occ(CC(=O)Nc3nc(cs3)-c3cc(F)cc(c3)C(F)(F)F)c2c(=O)n(C)c1=O
Show InChI InChI=1S/C20H14F4N4O4S/c1-27-16(30)15-10(7-32-17(15)28(2)19(27)31)5-14(29)26-18-25-13(8-33-18)9-3-11(20(22,23)24)6-12(21)4-9/h3-4,6-8H,5H2,1-2H3,(H,25,26,29)
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n/an/a 2.15n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191712
PNG
(US9186360, 59)
Show SMILES Cn1c2occ(CC(=O)Nc3nc(cs3)-c3cccc(c3F)C(F)(F)F)c2c(=O)n(C)c1=O
Show InChI InChI=1S/C20H14F4N4O4S/c1-27-16(30)14-9(7-32-17(14)28(2)19(27)31)6-13(29)26-18-25-12(8-33-18)10-4-3-5-11(15(10)21)20(22,23)24/h3-5,7-8H,6H2,1-2H3,(H,25,26,29)
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US Patent
n/an/a 2.21n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191652
PNG
(US9186360, 51 | US9186360, 52)
Show SMILES Cn1c2scc(CC(=O)Nc3nc(cs3)-c3ccc(F)c(c3F)C(F)(F)F)c2c(=O)n(C)c1=O
Show InChI InChI=1S/C20H13F5N4O3S2/c1-28-16(31)13-8(6-33-17(13)29(2)19(28)32)5-12(30)27-18-26-11(7-34-18)9-3-4-10(21)14(15(9)22)20(23,24)25/h3-4,6-7H,5H2,1-2H3,(H,26,27,30)
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US Patent
n/an/a 2.49n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191713
PNG
(US9186360, 61)
Show SMILES Cc1oc2n(C)c(=O)n(C)c(=O)c2c1CC(=O)Nc1nc(cs1)-c1cc(F)cc(c1)C(F)(F)F
Show InChI InChI=1S/C21H16F4N4O4S/c1-9-13(16-17(31)28(2)20(32)29(3)18(16)33-9)7-15(30)27-19-26-14(8-34-19)10-4-11(21(23,24)25)6-12(22)5-10/h4-6,8H,7H2,1-3H3,(H,26,27,30)
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n/an/a 2.93n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191722
PNG
(US9186360, 71)
Show SMILES Cc1oc2n(C)c(=O)n(C)c(=O)c2c1CC(=O)Nc1nc(cs1)-c1ccc(Cl)c(c1)C(F)(F)F
Show InChI InChI=1S/C21H16ClF3N4O4S/c1-9-11(16-17(31)28(2)20(32)29(3)18(16)33-9)7-15(30)27-19-26-14(8-34-19)10-4-5-13(22)12(6-10)21(23,24)25/h4-6,8H,7H2,1-3H3,(H,26,27,30)
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n/an/a 3.18n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191656
PNG
(US9186360, 75)
Show SMILES CC(C)COc1c(Cl)cc(cc1Cl)-c1csc(NC(=O)Cc2c(C)oc3n(C)c(=O)n(C)c(=O)c23)n1
Show InChI InChI=1S/C24H24Cl2N4O5S/c1-11(2)9-34-20-15(25)6-13(7-16(20)26)17-10-36-23(27-17)28-18(31)8-14-12(3)35-22-19(14)21(32)29(4)24(33)30(22)5/h6-7,10-11H,8-9H2,1-5H3,(H,27,28,31)
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n/an/a 3.34n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191710
PNG
(US9186360, 56)
Show SMILES Cn1c2occ(CC(=O)Nc3nc(cs3)-c3cc(F)c(CCC(F)(F)F)c(F)c3)c2c(=O)n(C)c1=O
Show InChI InChI=1S/C22H17F5N4O4S/c1-30-18(33)17-11(8-35-19(17)31(2)21(30)34)7-16(32)29-20-28-15(9-36-20)10-5-13(23)12(14(24)6-10)3-4-22(25,26)27/h5-6,8-9H,3-4,7H2,1-2H3,(H,28,29,32)
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US Patent
n/an/a 3.38n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191654
PNG
(US9186360, 60)
Show SMILES Cn1c2occ(CC(=O)Nc3nc(cs3)-c3cc(F)c(OCC(F)(F)F)c(Cl)c3)c2c(=O)n(C)c1=O
Show InChI InChI=1S/C21H15ClF4N4O5S/c1-29-17(32)15-10(6-34-18(15)30(2)20(29)33)5-14(31)28-19-27-13(7-36-19)9-3-11(22)16(12(23)4-9)35-8-21(24,25)26/h3-4,6-7H,5,8H2,1-2H3,(H,27,28,31)
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US Patent
n/an/a 3.54n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM50327657
PNG
(2-chlorobenzylidenemalononitrile | CHEMBL1256101)
Show SMILES Clc1ccccc1C=C(C#N)C#N
Show InChI InChI=1S/C10H5ClN2/c11-10-4-2-1-3-9(10)5-8(6-12)7-13/h1-5H
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n/an/a 3.60n/an/an/an/an/an/a



Johnson& Johnson Pharmaceutical Research& Development

Curated by ChEMBL


Assay Description
Agonist activity at human TRPA1 expressed in T-REx-HEK293 cells assessed as concentration required to incapacitate 50% of the population exposed to t...


Citation and Details
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191655
PNG
(US9186360, 62 | US9186360, 66)
Show SMILES Cc1oc2n(C)c(=O)n(C)c(=O)c2c1CC(=O)Nc1nc(cs1)-c1cc(F)c(OCC(C)(C)C)c(F)c1
Show InChI InChI=1S/C25H26F2N4O5S/c1-12-14(19-21(33)30(5)24(34)31(6)22(19)36-12)9-18(32)29-23-28-17(10-37-23)13-7-15(26)20(16(27)8-13)35-11-25(2,3)4/h7-8,10H,9,11H2,1-6H3,(H,28,29,32)
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US Patent
n/an/a 3.63n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191705
PNG
(US9186360, 49)
Show SMILES CCc1sc2n(C)c(=O)n(C)c(=O)c2c1CC(=O)Nc1nc(cs1)-c1cc(F)c(OCC(F)(F)F)c(F)c1
Show InChI InChI=1S/C23H19F5N4O4S2/c1-4-15-11(17-19(34)31(2)22(35)32(3)20(17)38-15)7-16(33)30-21-29-14(8-37-21)10-5-12(24)18(13(25)6-10)36-9-23(26,27)28/h5-6,8H,4,7,9H2,1-3H3,(H,29,30,33)
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US Patent
n/an/a 3.98n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191725
PNG
(US9186360, 76)
Show SMILES Cc1oc2n(C)c(=O)n(C)c(=O)c2c1CC(=O)Nc1nc(cs1)-c1ccc(c(F)c1F)C(F)(F)F
Show InChI InChI=1S/C21H15F5N4O4S/c1-8-10(14-17(32)29(2)20(33)30(3)18(14)34-8)6-13(31)28-19-27-12(7-35-19)9-4-5-11(21(24,25)26)16(23)15(9)22/h4-5,7H,6H2,1-3H3,(H,27,28,31)
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n/an/a 4.02n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191723
PNG
(US9186360, 72)
Show SMILES Cc1oc2n(C)c(=O)n(C)c(=O)c2c1CC(=O)Nc1nc(cs1)-c1cc(F)c(c(F)c1)C(F)(F)F
Show InChI InChI=1S/C21H15F5N4O4S/c1-8-10(15-17(32)29(2)20(33)30(3)18(15)34-8)6-14(31)28-19-27-13(7-35-19)9-4-11(22)16(12(23)5-9)21(24,25)26/h4-5,7H,6H2,1-3H3,(H,27,28,31)
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n/an/a 4.16n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191731
PNG
(US9186360, 83)
Show SMILES Cn1c2snc(CC(=O)Nc3nc(cs3)-c3cc(F)cc(c3)C(F)(F)F)c2c(=O)n(C)c1=O
Show InChI InChI=1S/C19H13F4N5O3S2/c1-27-15(30)14-11(26-33-16(14)28(2)18(27)31)6-13(29)25-17-24-12(7-32-17)8-3-9(19(21,22)23)5-10(20)4-8/h3-5,7H,6H2,1-2H3,(H,24,25,29)
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n/an/a 4.40n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191715
PNG
(US9186360, 64)
Show SMILES Cc1oc2n(C)c(=O)n(C)c(=O)c2c1CC(=O)Nc1nc(cs1)-c1ccc(F)c(c1F)C(F)(F)F
Show InChI InChI=1S/C21H15F5N4O4S/c1-8-10(14-17(32)29(2)20(33)30(3)18(14)34-8)6-13(31)28-19-27-12(7-35-19)9-4-5-11(22)15(16(9)23)21(24,25)26/h4-5,7H,6H2,1-3H3,(H,27,28,31)
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US Patent
n/an/a 4.52n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191652
PNG
(US9186360, 51 | US9186360, 52)
Show SMILES Cn1c2scc(CC(=O)Nc3nc(cs3)-c3ccc(F)c(c3F)C(F)(F)F)c2c(=O)n(C)c1=O
Show InChI InChI=1S/C20H13F5N4O3S2/c1-28-16(31)13-8(6-33-17(13)29(2)19(28)32)5-12(30)27-18-26-11(7-34-18)9-3-4-10(21)14(15(9)22)20(23,24)25/h3-4,6-7H,5H2,1-2H3,(H,26,27,30)
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US Patent
n/an/a 4.84n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191719
PNG
(US9186360, 68)
Show SMILES Cc1oc2n(C)c(=O)n(C)c(=O)c2c1CC(=O)Nc1nc(cs1)-c1ccc(F)c(OC(F)(F)F)c1
Show InChI InChI=1S/C21H16F4N4O5S/c1-9-11(16-17(31)28(2)20(32)29(3)18(16)33-9)7-15(30)27-19-26-13(8-35-19)10-4-5-12(22)14(6-10)34-21(23,24)25/h4-6,8H,7H2,1-3H3,(H,26,27,30)
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n/an/a 4.84n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191740
PNG
(US9186360, 99)
Show SMILES Cn1c2oc(Cl)c(CC(=O)Nc3nc(cs3)-c3ccc(c(F)c3)C(F)(F)F)c2c(=O)n(C)c1=O
Show InChI InChI=1S/C20H13ClF4N4O4S/c1-28-16(31)14-9(15(21)33-17(14)29(2)19(28)32)6-13(30)27-18-26-12(7-34-18)8-3-4-10(11(22)5-8)20(23,24)25/h3-5,7H,6H2,1-2H3,(H,26,27,30)
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n/an/a 5.06n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191741
PNG
(US9186360, 100)
Show SMILES Cn1c2oc(Cl)c(CC(=O)Nc3nc(cs3)-c3cc(F)cc(c3)C(F)(F)F)c2c(=O)n(C)c1=O
Show InChI InChI=1S/C20H13ClF4N4O4S/c1-28-16(31)14-11(15(21)33-17(14)29(2)19(28)32)6-13(30)27-18-26-12(7-34-18)8-3-9(20(23,24)25)5-10(22)4-8/h3-5,7H,6H2,1-2H3,(H,26,27,30)
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n/an/a 5.15n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191724
PNG
(US9186360, 74)
Show SMILES Cc1oc2n(C)c(=O)n(C)c(=O)c2c1CC(=O)Nc1nc(cs1)-c1ccc(OCC(F)(F)F)c(Cl)c1
Show InChI InChI=1S/C22H18ClF3N4O5S/c1-10-12(17-18(32)29(2)21(33)30(3)19(17)35-10)7-16(31)28-20-27-14(8-36-20)11-4-5-15(13(23)6-11)34-9-22(24,25)26/h4-6,8H,7,9H2,1-3H3,(H,27,28,31)
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n/an/a 5.29n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191728
PNG
(US9186360, 79)
Show SMILES Cn1c2snc(CC(=O)Nc3nc(cs3)-c3cccc(c3F)C(F)(F)F)c2c(=O)n(C)c1=O
Show InChI InChI=1S/C19H13F4N5O3S2/c1-27-15(30)13-10(26-33-16(13)28(2)18(27)31)6-12(29)25-17-24-11(7-32-17)8-4-3-5-9(14(8)20)19(21,22)23/h3-5,7H,6H2,1-2H3,(H,24,25,29)
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n/an/a 5.29n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191666
PNG
(US9186360, 84)
Show SMILES Cn1c2snc(CC(=O)Nc3nc(cs3)-c3ccc(c(F)c3F)C(F)(F)F)c2c(=O)n(C)c1=O
Show InChI InChI=1S/C19H12F5N5O3S2/c1-28-15(31)12-9(27-34-16(12)29(2)18(28)32)5-11(30)26-17-25-10(6-33-17)7-3-4-8(19(22,23)24)14(21)13(7)20/h3-4,6H,5H2,1-2H3,(H,25,26,30)
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n/an/a 5.35n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191648
PNG
(US9186360, 33)
Show SMILES Cn1c2cccc(CC(=O)Nc3nc(cs3)-c3cc(F)c(c(F)c3)C(F)(F)F)c2c(=O)n(C)c1=O
Show InChI InChI=1S/C22H15F5N4O3S/c1-30-15-5-3-4-10(17(15)19(33)31(2)21(30)34)8-16(32)29-20-28-14(9-35-20)11-6-12(23)18(13(24)7-11)22(25,26)27/h3-7,9H,8H2,1-2H3,(H,28,29,32)
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n/an/a 5.37n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191726
PNG
(US9186360, 77)
Show SMILES Cn1c2snc(CC(=O)Nc3nc(cs3)-c3ccc(F)c(c3F)C(F)(F)F)c2c(=O)n(C)c1=O
Show InChI InChI=1S/C19H12F5N5O3S2/c1-28-15(31)12-9(27-34-16(12)29(2)18(28)32)5-11(30)26-17-25-10(6-33-17)7-3-4-8(20)13(14(7)21)19(22,23)24/h3-4,6H,5H2,1-2H3,(H,25,26,30)
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n/an/a 5.60n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM50046740
PNG
(CHEMBL1939972 | US9186360, 90)
Show SMILES COCCCOc1cccc(c1)C1NC(=S)NC2=C1C(=O)c1ccccc21
Show InChI InChI=1/C21H20N2O3S/c1-25-10-5-11-26-14-7-4-6-13(12-14)18-17-19(23-21(27)22-18)15-8-2-3-9-16(15)20(17)24/h2-4,6-9,12,18H,5,10-11H2,1H3,(H2,22,23,27)
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n/an/a 5.61n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191647
PNG
(US9186360, 32)
Show SMILES Cn1c2cccc(CC(=O)Nc3nc(cs3)-c3cc(F)c(OCC(F)(F)F)c(F)c3)c2c(=O)n(C)c1=O
Show InChI InChI=1S/C23H17F5N4O4S/c1-31-16-5-3-4-11(18(16)20(34)32(2)22(31)35)8-17(33)30-21-29-15(9-37-21)12-6-13(24)19(14(25)7-12)36-10-23(26,27)28/h3-7,9H,8,10H2,1-2H3,(H,29,30,33)
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n/an/a 5.96n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191657
PNG
(US9186360, 80)
Show SMILES Cn1c2snc(CC(=O)Nc3nc(cs3)-c3ccc(OC(F)(F)F)c(Cl)c3)c2c(=O)n(C)c1=O
Show InChI InChI=1S/C19H13ClF3N5O4S2/c1-27-15(30)14-10(26-34-16(14)28(2)18(27)31)6-13(29)25-17-24-11(7-33-17)8-3-4-12(9(20)5-8)32-19(21,22)23/h3-5,7H,6H2,1-2H3,(H,24,25,29)
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n/an/a 6.28n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191689
PNG
(US9186360, 28)
Show SMILES Cn1c2cccc(CC(=O)Nc3nc(cs3)-c3ccc(c(F)c3F)C(F)(F)F)c2c(=O)n(C)c1=O
Show InChI InChI=1S/C22H15F5N4O3S/c1-30-14-5-3-4-10(16(14)19(33)31(2)21(30)34)8-15(32)29-20-28-13(9-35-20)11-6-7-12(22(25,26)27)18(24)17(11)23/h3-7,9H,8H2,1-2H3,(H,28,29,32)
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n/an/a 6.49n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191716
PNG
(US9186360, 65)
Show SMILES Cc1oc2n(C)c(=O)n(C)c(=O)c2c1CC(=O)Nc1nc(cs1)-c1ccc(cc1F)C(F)(F)F
Show InChI InChI=1S/C21H16F4N4O4S/c1-9-12(16-17(31)28(2)20(32)29(3)18(16)33-9)7-15(30)27-19-26-14(8-34-19)11-5-4-10(6-13(11)22)21(23,24)25/h4-6,8H,7H2,1-3H3,(H,26,27,30)
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n/an/a 6.65n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191729
PNG
(US9186360, 81)
Show SMILES Cn1c2snc(CC(=O)Nc3nc(cs3)-c3ccc(c(F)c3)C(F)(F)F)c2c(=O)n(C)c1=O
Show InChI InChI=1S/C19H13F4N5O3S2/c1-27-15(30)14-11(26-33-16(14)28(2)18(27)31)6-13(29)25-17-24-12(7-32-17)8-3-4-9(10(20)5-8)19(21,22)23/h3-5,7H,6H2,1-2H3,(H,24,25,29)
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n/an/a 6.74n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191658
PNG
(US9186360, 86)
Show SMILES Cn1c2nccc(CC(=O)Nc3nc(cs3)-c3cc(F)c(OCC(F)(F)F)c(F)c3)c2c(=O)n(C)c1=O
Show InChI InChI=1S/C22H16F5N5O4S/c1-31-18-16(19(34)32(2)21(31)35)10(3-4-28-18)7-15(33)30-20-29-14(8-37-20)11-5-12(23)17(13(24)6-11)36-9-22(25,26)27/h3-6,8H,7,9H2,1-2H3,(H,29,30,33)
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n/an/a 6.91n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM50318455
PNG
(AMG-9090 | CHEMBL1086371 | N-(2,2,2-trichloro-1-(4...)
Show SMILES Clc1ccc(SC(NC(=O)c2ccccc2)C(Cl)(Cl)Cl)cc1
Show InChI InChI=1S/C15H11Cl4NOS/c16-11-6-8-12(9-7-11)22-14(15(17,18)19)20-13(21)10-4-2-1-3-5-10/h1-9,14H,(H,20,21)
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n/an/a 7n/an/an/an/an/an/a



Ferrara University

Curated by ChEMBL


Assay Description
Antagonist activity at human TRPA1 channel assessed as inhibition of noxious cold-induced receptor activation


Citation and Details
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191720
PNG
(US9186360, 69)
Show SMILES Cc1oc2n(C)c(=O)n(C)c(=O)c2c1CC(=O)Nc1nc(cs1)-c1ccc(F)c(c1)C(F)(F)F
Show InChI InChI=1S/C21H16F4N4O4S/c1-9-11(16-17(31)28(2)20(32)29(3)18(16)33-9)7-15(30)27-19-26-14(8-34-19)10-4-5-13(22)12(6-10)21(23,24)25/h4-6,8H,7H2,1-3H3,(H,26,27,30)
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n/an/a 7.10n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191663
PNG
(US9186360, 104)
Show SMILES Cn1c2oc(Cl)c(CC(=O)Nc3nc(cs3)-c3ccc(c(F)c3F)C(F)(F)F)c2c(=O)n(C)c1=O
Show InChI InChI=1S/C20H12ClF5N4O4S/c1-29-16(32)12-8(15(21)34-17(12)30(2)19(29)33)5-11(31)28-18-27-10(6-35-18)7-3-4-9(20(24,25)26)14(23)13(7)22/h3-4,6H,5H2,1-2H3,(H,27,28,31)
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n/an/a 7.58n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191742
PNG
(US9186360, 102)
Show SMILES Cn1c2oc(Cl)c(CC(=O)Nc3nc(cs3)-c3ccc(OC(F)(F)F)c(F)c3)c2c(=O)n(C)c1=O
Show InChI InChI=1S/C20H13ClF4N4O5S/c1-28-16(31)14-9(15(21)33-17(14)29(2)19(28)32)6-13(30)27-18-26-11(7-35-18)8-3-4-12(10(22)5-8)34-20(23,24)25/h3-5,7H,6H2,1-2H3,(H,26,27,30)
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n/an/a 7.67n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191730
PNG
(US9186360, 82)
Show SMILES Cn1c2snc(CC(=O)Nc3nc(cs3)-c3ccc(OC(F)(F)F)c(F)c3)c2c(=O)n(C)c1=O
Show InChI InChI=1S/C19H13F4N5O4S2/c1-27-15(30)14-10(26-34-16(14)28(2)18(27)31)6-13(29)25-17-24-11(7-33-17)8-3-4-12(9(20)5-8)32-19(21,22)23/h3-5,7H,6H2,1-2H3,(H,24,25,29)
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n/an/a 8.04n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191700
PNG
(US9186360, 44)
Show SMILES Cn1c2c[nH]n(CC(=O)Nc3nc(cs3)-c3cc(Cl)c(OCC(C)(C)C)c(Cl)c3)c2c(=O)n(C)c1=O
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US Patent
n/an/a 8.36n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191665
PNG
(US9186360, 73)
Show SMILES Cc1oc2n(C)c(=O)n(C)c(=O)c2c1CC(=O)Nc1nc(cs1)-c1ccc(OC(F)(F)F)c(Cl)c1
Show InChI InChI=1S/C21H16ClF3N4O5S/c1-9-11(16-17(31)28(2)20(32)29(3)18(16)33-9)7-15(30)27-19-26-13(8-35-19)10-4-5-14(12(22)6-10)34-21(23,24)25/h4-6,8H,7H2,1-3H3,(H,26,27,30)
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US Patent
n/an/a 8.54n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191732
PNG
(US9186360, 85)
Show SMILES Cn1c2nccc(CC(=O)Nc3nc(cs3)-c3ccc(c(F)c3)C(F)(F)F)c2c(=O)n(C)c1=O
Show InChI InChI=1S/C21H15F4N5O3S/c1-29-17-16(18(32)30(2)20(29)33)11(5-6-26-17)8-15(31)28-19-27-14(9-34-19)10-3-4-12(13(22)7-10)21(23,24)25/h3-7,9H,8H2,1-2H3,(H,27,28,31)
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US Patent
n/an/a 8.92n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191714
PNG
(US9186360, 63)
Show SMILES Cc1oc2n(C)c(=O)n(C)c(=O)c2c1CC(=O)Nc1nc(cs1)-c1ccc(Cl)c(OC(F)(F)F)c1
Show InChI InChI=1S/C21H16ClF3N4O5S/c1-9-11(16-17(31)28(2)20(32)29(3)18(16)33-9)7-15(30)27-19-26-13(8-35-19)10-4-5-12(22)14(6-10)34-21(23,24)25/h4-6,8H,7H2,1-3H3,(H,26,27,30)
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US Patent
n/an/a 9.04n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM50390485
PNG
(CHEMBL2071601)
Show SMILES CC(C)C(NC(=O)c1cc(Cl)ccc1C(F)(F)F)C(=O)c1ccc(cc1)[N+]([O-])=O
Show InChI InChI=1S/C19H16ClF3N2O4/c1-10(2)16(17(26)11-3-6-13(7-4-11)25(28)29)24-18(27)14-9-12(20)5-8-15(14)19(21,22)23/h3-10,16H,1-2H3,(H,24,27)
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PubMed
n/an/a 10n/an/an/an/an/an/a



AstraZeneca

Curated by ChEMBL


Assay Description
Antagonist activity at human TRPA1 expressed in HEK293 cells assessed as inhibition of Zn2+-induced intracellular calcium flux by FLIPR assay


Citation and Details
More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191662
PNG
(US9186360, 101)
Show SMILES Cn1c2oc(Cl)c(CC(=O)Nc3nc(cs3)-c3ccc(F)c(c3F)C(F)(F)F)c2c(=O)n(C)c1=O
Show InChI InChI=1S/C20H12ClF5N4O4S/c1-29-16(32)12-8(15(21)34-17(12)30(2)19(29)33)5-11(31)28-18-27-10(6-35-18)7-3-4-9(22)13(14(7)23)20(24,25)26/h3-4,6H,5H2,1-2H3,(H,27,28,31)
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US Patent
n/an/a 10.1n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191727
PNG
(US9186360, 78)
Show SMILES Cn1c2snc(CC(=O)Nc3nc(cs3)-c3ccc(cc3F)C(F)(F)F)c2c(=O)n(C)c1=O
Show InChI InChI=1S/C19H13F4N5O3S2/c1-27-15(30)14-11(26-33-16(14)28(2)18(27)31)6-13(29)25-17-24-12(7-32-17)9-4-3-8(5-10(9)20)19(21,22)23/h3-5,7H,6H2,1-2H3,(H,24,25,29)
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US Patent
n/an/a 10.6n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191697
PNG
(US9186360, 41)
Show SMILES Cn1nc2n(C)c(=O)n(C)c(=O)c2c1CC(=O)Nc1nc(cs1)-c1ccc(OC(F)(F)F)c(F)c1
Show InChI InChI=1S/C20H16F4N6O4S/c1-28-16-15(17(32)29(2)19(28)33)12(30(3)27-16)7-14(31)26-18-25-11(8-35-18)9-4-5-13(10(21)6-9)34-20(22,23)24/h4-6,8H,7H2,1-3H3,(H,25,26,31)
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US Patent
n/an/a 11.0n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191698
PNG
(US9186360, 42)
Show SMILES Cn1c2c[nH]n(CC(=O)Nc3nc(cs3)-c3cc(F)c(OCC(C)(C)C)c(Cl)c3)c2c(=O)n(C)c1=O
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US Patent
n/an/a 11.4n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191690
PNG
(US9186360, 29)
Show SMILES Cn1c2cccc(CC(=O)Nc3nc(cs3)-c3ccc(OC(F)(F)F)c(F)c3)c2c(=O)n(C)c1=O
Show InChI InChI=1S/C22H16F4N4O4S/c1-29-15-5-3-4-12(18(15)19(32)30(2)21(29)33)9-17(31)28-20-27-14(10-35-20)11-6-7-16(13(23)8-11)34-22(24,25)26/h3-8,10H,9H2,1-2H3,(H,27,28,31)
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n/an/a 11.4n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
Transient receptor potential cation channel subfamily A member 1 (TRPA1)


(Homo sapiens (Human))
BDBM191734
PNG
(US9186360, 88)
Show SMILES Cn1c2nccc(CC(=O)Nc3nc(cs3)-c3ccc(OC(F)(F)F)c(F)c3)c2c(=O)n(C)c1=O
Show InChI InChI=1S/C21H15F4N5O4S/c1-29-17-16(18(32)30(2)20(29)33)11(5-6-26-17)8-15(31)28-19-27-13(9-35-19)10-3-4-14(12(22)7-10)34-21(23,24)25/h3-7,9H,8H2,1-2H3,(H,27,28,31)
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n/an/a 11.4n/an/an/an/an/an/a



GLENMARK PHARMACEUTICALS S.A.

US Patent


Assay Description
The inhibition of TRPA1 receptor activation was measured as inhibition of allylisothiocyanate (AITC) induced cellular uptake of radioactive calcium. ...


US Patent US9186360 (2015)

More data for this
Ligand-Target Pair
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