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Compile Data Set for Download or QSAR

Found 70 hits Enz. Inhib. hit(s) with Target = 'Voltage-gated potassium channel subunit Kv1.3' AND taxid = 10090   
Target
(Institution)
LigandTarget
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50115772
PNG
(CHEMBL3609094)
Show SMILES CC[C@H](C)[C@@H]1NC(=O)[C@H](CSSC[C@H](NC(=O)[C@@H](NC(=O)CNC(=O)[C@@H]2CSSC[C@@H]3NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](Cc4ccccc4)NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](CSSC[C@H](NC(=O)[C@H](Cc4ccccc4)NC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](Cc4ccc(O)cc4)NC(=O)[C@H](CN)NC(=O)[C@H](CCSC)NC(=O)[C@H](CO)NC(=O)[C@H](Cc4cnc[nH]4)NC(=O)[C@H](CCCCN)NC3=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]([C@@H](C)O)C(=O)N2)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CO)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]2CCCN2C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CC(O)=O)NC1=O)[C@@H](C)O)[C@@H](C)CC)[C@@H](C)O)[C@@H](C)O)C(O)=O)NC(=O)[C@H](CO)NC(=O)[C@@H](N)CCCNC(N)=N
Show InChI InChI=1/C166H268N54O48S7/c1-13-81(5)123-156(261)202-107(65-122(232)233)145(250)218-128(87(11)228)160(265)216-124(82(6)14-2)161(266)220-58-31-43-119(220)155(260)196-95(38-22-25-52-168)135(240)205-110(70-222)147(252)191-99(42-30-57-185-166(179)180)136(241)209-117-77-273-272-75-115-152(257)193-97(40-28-55-183-164(175)176)132(237)189-96(39-23-26-53-169)139(244)217-127(86(10)227)159(264)212-113(131(236)186-68-121(231)214-125(84(8)225)158(263)213-118(162(267)268)78-275-274-76-116(153(258)215-123)211-150(255)109(69-221)204-130(235)93(171)36-27-54-182-163(173)174)73-270-271-74-114(208-137(242)100(48-49-120(172)230)194-141(246)103(61-88-32-17-15-18-33-88)197-129(234)83(7)188-157(262)126(85(9)226)219-154(117)259)151(256)192-94(37-21-24-51-167)133(238)201-106(64-91-67-181-79-187-91)144(249)207-111(71-223)148(253)195-101(50-59-269-12)138(243)203-108(66-170)146(251)199-105(63-90-44-46-92(229)47-45-90)142(247)190-98(41-29-56-184-165(177)178)134(239)198-102(60-80(3)4)140(245)206-112(72-224)149(254)200-104(143(248)210-115)62-89-34-19-16-20-35-89/h15-20,32-35,44-47,67,79-87,93-119,123-128,221-229H,13-14,21-31,36-43,48-66,68-78,167-171H2,1-12H3,(H2,172,230)(H,181,187)(H,186,236)(H,188,262)(H,189,237)(H,190,247)(H,191,252)(H,192,256)(H,193,257)(H,194,246)(H,195,253)(H,196,260)(H,197,234)(H,198,239)(H,199,251)(H,200,254)(H,201,238)(H,202,261)(H,203,243)(H,204,235)(H,205,240)(H,206,245)(H,207,249)(H,208,242)(H,209,241)(H,210,248)(H,211,255)(H,212,264)(H,213,263)(H,214,231)(H,215,258)(H,216,265)(H,217,244)(H,218,250)(H,219,259)(H,232,233)(H,267,268)(H4,173,174,182)(H4,175,176,183)(H4,177,178,184)(H4,179,180,185)/t81-,82-,83-,84+,85+,86+,87+,93-,94-,95-,96-,97-,98-,99-,100-,101-,102-,103-,104-,105-,106-,107-,108-,109-,110-,111-,112-,113-,114-,115-,116-,117-,118-,119-,123-,124-,125-,126-,127-,128-/s2
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n/an/a 23n/an/an/an/an/an/a



Amgen Inc.

Curated by ChEMBL


Assay Description
Displacement of [125I]-ChTX from mouse Kv1.3 after 20 mins by scintillation counting analysis


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50083523
PNG
((1-Benzyl-1H-quinolin-4-ylidene)-pentyl-amine | CH...)
Show SMILES CCCCC\N=c1/ccn(Cc2ccccc2)c2ccccc12
Show InChI InChI=1S/C21H24N2/c1-2-3-9-15-22-20-14-16-23(17-18-10-5-4-6-11-18)21-13-8-7-12-19(20)21/h4-8,10-14,16H,2-3,9,15,17H2,1H3/b22-20+
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n/an/a 230n/an/an/an/an/an/a



University of Kiel

Curated by ChEMBL


Assay Description
Blockade of peak steady-state K+ currents of voltage-gated potassium channel subunit Kv1.3 in mouse fibroblasts L929 at 50 uM


J Med Chem 44: 1249-56 (2001)

More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50098785
PNG
(4-Benzhydryloxymethyl-1-[3-(4-methoxy-phenyl)-prop...)
Show SMILES COc1ccc(CCCN2CCC(COC(c3ccccc3)c3ccccc3)CC2)cc1
Show InChI InChI=1S/C29H35NO2/c1-31-28-16-14-24(15-17-28)9-8-20-30-21-18-25(19-22-30)23-32-29(26-10-4-2-5-11-26)27-12-6-3-7-13-27/h2-7,10-17,25,29H,8-9,18-23H2,1H3
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n/an/a 280n/an/an/an/an/an/a



University of Kiel

Curated by ChEMBL


Assay Description
Blockade of peak steady-state K+ currents of voltage-gated potassium channel subunit Kv1.3 in mouse fibroblasts L929 at 50 uM


J Med Chem 44: 1249-56 (2001)

More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50098782
PNG
(2-Isopropyl-8-methoxy-5-methyl-5H-furo[3,2-c]quino...)
Show SMILES COc1ccc2n(C)c(=O)c3cc(oc3c2c1)C(C)C
Show InChI InChI=1S/C16H17NO3/c1-9(2)14-8-12-15(20-14)11-7-10(19-4)5-6-13(11)17(3)16(12)18/h5-9H,1-4H3
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n/an/a 5.00E+3n/an/an/an/an/an/a



University of Kiel

Curated by ChEMBL


Assay Description
Blockade of peak steady-state K+ currents of voltage-gated potassium channel subunit Kv1.3 in mouse fibroblasts L929 at 50 uM


J Med Chem 44: 1249-56 (2001)

More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50098781
PNG
(9-Methoxy-2,2,6-trimethyl-2,6-dihydro-pyrano[3,2-c...)
Show SMILES COc1ccc2n(C)c(=O)c3C=CC(C)(C)Oc3c2c1
Show InChI InChI=1S/C16H17NO3/c1-16(2)8-7-11-14(20-16)12-9-10(19-4)5-6-13(12)17(3)15(11)18/h5-9H,1-4H3
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n/an/a 1.00E+4n/an/an/an/an/an/a



University of Kiel

Curated by ChEMBL


Assay Description
Blockade of peak steady-state K+ currents of voltage-gated potassium channel subunit Kv1.3 in mouse fibroblasts L929 at 50 uM


J Med Chem 44: 1249-56 (2001)

More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50098784
PNG
(9-Methoxy-2,2,6-trimethyl-2,3,4,6-tetrahydro-pyran...)
Show SMILES COc1ccc2n(C)c(=O)c3CCC(C)(C)Oc3c2c1
Show InChI InChI=1S/C16H19NO3/c1-16(2)8-7-11-14(20-16)12-9-10(19-4)5-6-13(12)17(3)15(11)18/h5-6,9H,7-8H2,1-4H3
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n/an/a 1.80E+4n/an/an/an/an/an/a



University of Kiel

Curated by ChEMBL


Assay Description
Inhibition of voltage-gated potassium channel subunit Kv1.3 expressed in L929 cells


J Med Chem 44: 1249-56 (2001)

More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50098783
PNG
(4,6,7-Trimethoxy-furo[2,3-b]quinoline | CHEMBL2787...)
Show SMILES COc1cc2nc3occc3c(OC)c2cc1OC
Show InChI InChI=1S/C14H13NO4/c1-16-11-6-9-10(7-12(11)17-2)15-14-8(4-5-19-14)13(9)18-3/h4-7H,1-3H3
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n/an/a 4.90E+4n/an/an/an/an/an/a



University of Kiel

Curated by ChEMBL


Assay Description
Blockade of peak steady-state K+ currents of voltage-gated potassium channel subunit Kv1.3 in mouse fibroblasts L929 at 50 uM


J Med Chem 44: 1249-56 (2001)

More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50067879
PNG
(5-Methoxymethyl-3-methyl-furo[3,2-g]chromen-7-one ...)
Show SMILES COCc1cc(=O)oc2cc3occ(C)c3cc12
Show InChI InChI=1S/C14H12O4/c1-8-6-17-12-5-13-11(4-10(8)12)9(7-16-2)3-14(15)18-13/h3-6H,7H2,1-2H3
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n/an/an/a 9.00E+4n/an/an/an/an/a



University of Kiel

Curated by ChEMBL


Assay Description
Blockade of peak Kv1.3 potassium currents


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50067878
PNG
(9-Methoxy-furo[3',2':4,5]benzo[1,2-b][1,4]oxazin-3...)
Show SMILES COc1c2ccoc2cc2oc(=O)cnc12
Show InChI InChI=1S/C11H7NO4/c1-14-11-6-2-3-15-7(6)4-8-10(11)12-5-9(13)16-8/h2-5H,1H3
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n/an/an/a 1.95E+5n/an/an/an/an/a



University of Kiel

Curated by ChEMBL


Assay Description
Blockade of peak Kv1.3 potassium currents


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50067880
PNG
(4-methoxy-7H-furo[3,2-g][1]benzopyran-7-one | 4-me...)
Show SMILES COc1c2ccoc2cc2oc(=O)ccc12
Show InChI InChI=1S/C12H8O4/c1-14-12-7-2-3-11(13)16-10(7)6-9-8(12)4-5-15-9/h2-6H,1H3
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n/an/an/a 1.01E+5n/an/an/an/an/a



University of Kiel

Curated by ChEMBL


Assay Description
Blockade of peak Kv1.3 potassium currents


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50067881
PNG
(4,9-Diethoxy-furo[3,2-g]chromen-7-one | CHEMBL3429...)
Show SMILES CCOc1c2ccoc2c(OCC)c2oc(=O)ccc12
Show InChI InChI=1S/C15H14O5/c1-3-17-12-9-5-6-11(16)20-14(9)15(18-4-2)13-10(12)7-8-19-13/h5-8H,3-4H2,1-2H3
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n/an/an/a 2.80E+4n/an/an/an/an/a



University of Kiel

Curated by ChEMBL


Assay Description
Blockade of peak Kv1.3 potassium currents


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50067882
PNG
(4-Methoxy-9-methoxymethyl-furo[3,2-g]chromen-7-one...)
Show SMILES COCc1c2occc2c(OC)c2ccc(=O)oc12
Show InChI InChI=1S/C14H12O5/c1-16-7-10-13-9(5-6-18-13)12(17-2)8-3-4-11(15)19-14(8)10/h3-6H,7H2,1-2H3
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n/an/an/a 2.80E+4n/an/an/an/an/a



University of Kiel

Curated by ChEMBL


Assay Description
Blockade of peak Kv1.3 potassium currents


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50168302
PNG
(4-Guanidinomethyl-1-phenethyl-1H-indole-7-carboxyl...)
Show SMILES NCCCCNC(=O)c1ccc(CN=C(N)N)c2ccn(CCc3ccccc3)c12
Show InChI InChI=1S/C23H30N6O/c24-12-4-5-13-27-22(30)20-9-8-18(16-28-23(25)26)19-11-15-29(21(19)20)14-10-17-6-2-1-3-7-17/h1-3,6-9,11,15H,4-5,10,12-14,16,24H2,(H,27,30)(H4,25,26,28)
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n/an/an/an/a 7.50E+4n/an/an/an/a



Institute of Medical Research

Curated by ChEMBL


Assay Description
Effective concentration against murine voltage-gated potassium channel subunit Kv1.3 expressed in L929 cells using patch clamp


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182604
PNG
(1-(7-(3-fluorobenzyloxy)-6-hydroxy-4-methoxybenzof...)
Show SMILES COc1c(C(C)=O)c(O)c(OCc2cccc(F)c2)c2occc12
Show InChI InChI=1S/C18H15FO5/c1-10(20)14-15(21)18(17-13(6-7-23-17)16(14)22-2)24-9-11-4-3-5-12(19)8-11/h3-8,21H,9H2,1-2H3
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n/an/an/an/a 750n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182605
PNG
(1-(4-(2-chlorobenzyloxy)-6-hydroxy-7-methoxybenzof...)
Show SMILES COc1c(O)c(C(C)=O)c(OCc2ccccc2Cl)c2ccoc12
Show InChI InChI=1S/C18H15ClO5/c1-10(20)14-15(21)18(22-2)17-12(7-8-23-17)16(14)24-9-11-5-3-4-6-13(11)19/h3-8,21H,9H2,1-2H3
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n/an/an/an/a 1.20E+3n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182606
PNG
(1-(7-(4-isopropylbenzyloxy)-6-hydroxy-4-methoxyben...)
Show SMILES COc1c(C(C)=O)c(O)c(OCc2ccc(cc2)C(C)C)c2occc12
Show InChI InChI=1S/C21H22O5/c1-12(2)15-7-5-14(6-8-15)11-26-21-18(23)17(13(3)22)19(24-4)16-9-10-25-20(16)21/h5-10,12,23H,11H2,1-4H3
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n/an/an/an/a 1.00E+3n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182607
PNG
(1-(7-(3-nitrobenzyloxy)-6-hydroxy-4-methoxybenzofu...)
Show SMILES COc1c(C(C)=O)c(O)c(OCc2cccc(c2)[N+]([O-])=O)c2occc12
Show InChI InChI=1S/C18H15NO7/c1-10(20)14-15(21)18(17-13(6-7-25-17)16(14)24-2)26-9-11-4-3-5-12(8-11)19(22)23/h3-8,21H,9H2,1-2H3
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n/an/an/an/a 600n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182608
PNG
(1-[6-Hydroxy-4-methoxy-7-(3-methyl-benzyloxy)-benz...)
Show SMILES COc1c(C(C)=O)c(O)c(OCc2cccc(C)c2)c2occc12
Show InChI InChI=1S/C19H18O5/c1-11-5-4-6-13(9-11)10-24-19-16(21)15(12(2)20)17(22-3)14-7-8-23-18(14)19/h4-9,21H,10H2,1-3H3
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n/an/an/an/a 1.20E+3n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182597
PNG
(5-acetyl-4,7-benzyloxy-6-hydroxybenzofuran | CHEMB...)
Show SMILES CC(=O)c1c(O)c(OCc2ccccc2)c2occc2c1OCc1ccccc1
Show InChI InChI=1S/C24H20O5/c1-16(25)20-21(26)24(29-15-18-10-6-3-7-11-18)23-19(12-13-27-23)22(20)28-14-17-8-4-2-5-9-17/h2-13,26H,14-15H2,1H3
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n/an/an/an/a 1.20E+3n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182637
PNG
(1,6-bis(5-acetyl-4-ethoxy-7-methoxybenzofuran-6-yl...)
Show SMILES CCOc1c(C(C)=O)c(OCCCCCCOc2c(OC)c3occc3c(OCC)c2C(C)=O)c(OC)c2occc12
Show InChI InChI=1S/C32H38O10/c1-7-37-25-21-13-17-41-27(21)31(35-5)29(23(25)19(3)33)39-15-11-9-10-12-16-40-30-24(20(4)34)26(38-8-2)22-14-18-42-28(22)32(30)36-6/h13-14,17-18H,7-12,15-16H2,1-6H3
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n/an/an/an/a 800n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50145066
PNG
(1-(6-Hydroxy-4,7-dimethoxy-benzofuran-5-yl)-ethano...)
Show SMILES COc1c(O)c(C(C)=O)c(OC)c2ccoc12
Show InChI InChI=1S/C12H12O5/c1-6(13)8-9(14)12(16-3)11-7(4-5-17-11)10(8)15-2/h4-5,14H,1-3H3
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n/an/an/an/a 4.50E+4n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182640
PNG
(1-(7-(2-fluorobenzyloxy)-6-hydroxy-4-methoxybenzof...)
Show SMILES COc1c(C(C)=O)c(O)c(OCc2ccccc2F)c2occc12
Show InChI InChI=1S/C18H15FO5/c1-10(20)14-15(21)18(17-12(7-8-23-17)16(14)22-2)24-9-11-5-3-4-6-13(11)19/h3-8,21H,9H2,1-2H3
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n/an/an/an/a 2.50E+3n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182601
PNG
(1-(4-(3-methoxybenzyloxy)-6-hydroxy-7-methoxybenzo...)
Show SMILES COc1cccc(COc2c(C(C)=O)c(O)c(OC)c3occc23)c1
Show InChI InChI=1S/C19H18O6/c1-11(20)15-16(21)19(23-3)18-14(7-8-24-18)17(15)25-10-12-5-4-6-13(9-12)22-2/h4-9,21H,10H2,1-3H3
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n/an/an/an/a 680n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182602
PNG
(1-(7-(4-tert-butylbenzyloxy)-6-hydroxy-4-methoxybe...)
Show SMILES COc1c(C(C)=O)c(O)c(OCc2ccc(cc2)C(C)(C)C)c2occc12
Show InChI InChI=1S/C22H24O5/c1-13(23)17-18(24)21(20-16(10-11-26-20)19(17)25-5)27-12-14-6-8-15(9-7-14)22(2,3)4/h6-11,24H,12H2,1-5H3
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n/an/an/an/a 5.80E+3n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182603
PNG
(1-(4-(4-bromobenzyloxy)-6-hydroxy-7-methoxybenzofu...)
Show SMILES COc1c(O)c(C(C)=O)c(OCc2ccc(Br)cc2)c2ccoc12
Show InChI InChI=1S/C18H15BrO5/c1-10(20)14-15(21)18(22-2)17-13(7-8-23-17)16(14)24-9-11-3-5-12(19)6-4-11/h3-8,21H,9H2,1-2H3
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n/an/an/an/a 500n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182588
PNG
(1-(7-(4-fluorobenzyloxy)-6-hydroxy-4-methoxybenzof...)
Show SMILES COc1c(C(C)=O)c(O)c(OCc2ccc(F)cc2)c2occc12
Show InChI InChI=1S/C18H15FO5/c1-10(20)14-15(21)18(17-13(7-8-23-17)16(14)22-2)24-9-11-3-5-12(19)6-4-11/h3-8,21H,9H2,1-2H3
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n/an/an/an/a 700n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182591
PNG
(1-(7-(4-(trifluoromethyl)benzyloxy)-6-hydroxy-4-me...)
Show SMILES COc1c(C(C)=O)c(O)c(OCc2ccc(cc2)C(F)(F)F)c2occc12
Show InChI InChI=1S/C19H15F3O5/c1-10(23)14-15(24)18(17-13(7-8-26-17)16(14)25-2)27-9-11-3-5-12(6-4-11)19(20,21)22/h3-8,24H,9H2,1-2H3
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n/an/an/an/a 420n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182589
PNG
(1-[7-(Biphenyl-4-ylmethoxy)-6-hydroxy-4-methoxy-be...)
Show SMILES COc1c(C(C)=O)c(O)c(OCc2ccc(cc2)-c2ccccc2)c2occc12
Show InChI InChI=1S/C24H20O5/c1-15(25)20-21(26)24(23-19(12-13-28-23)22(20)27-2)29-14-16-8-10-18(11-9-16)17-6-4-3-5-7-17/h3-13,26H,14H2,1-2H3
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n/an/an/an/a 1.20E+3n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182590
PNG
(5-acetyl-4-ethoxy-6-hydroxy-7-methoxybenzofuran | ...)
Show SMILES CCOc1c(C(C)=O)c(O)c(OC)c2occc12
Show InChI InChI=1S/C13H14O5/c1-4-17-11-8-5-6-18-12(8)13(16-3)10(15)9(11)7(2)14/h5-6,15H,4H2,1-3H3
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n/an/an/an/a 7.00E+3n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182592
PNG
(1-[7-(Biphenyl-2-ylmethoxy)-6-hydroxy-4-methoxy-be...)
Show SMILES COc1c(C(C)=O)c(O)c(OCc2ccccc2-c2ccccc2)c2occc12
Show InChI InChI=1S/C24H20O5/c1-15(25)20-21(26)24(23-19(12-13-28-23)22(20)27-2)29-14-17-10-6-7-11-18(17)16-8-4-3-5-9-16/h3-13,26H,14H2,1-2H3
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n/an/an/an/a 1.10E+3n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182593
PNG
(1-(7-(3-(trifluoromethoxy)benzyloxy)-6-hydroxy-4-m...)
Show SMILES COc1c(C(C)=O)c(O)c(OCc2cccc(OC(F)(F)F)c2)c2occc12
Show InChI InChI=1S/C19H15F3O6/c1-10(23)14-15(24)18(17-13(6-7-26-17)16(14)25-2)27-9-11-4-3-5-12(8-11)28-19(20,21)22/h3-8,24H,9H2,1-2H3
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n/an/an/an/a 450n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182594
PNG
(1-[4-(1,1'-biphenyl-2-ylmethoxy)-6-hydroxy-7-metho...)
Show SMILES COc1c(O)c(C(C)=O)c(OCc2ccccc2-c2ccccc2)c2ccoc12
Show InChI InChI=1S/C24H20O5/c1-15(25)20-21(26)24(27-2)23-19(12-13-28-23)22(20)29-14-17-10-6-7-11-18(17)16-8-4-3-5-9-16/h3-13,26H,14H2,1-2H3
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n/an/an/an/a 2.00E+3n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182596
PNG
(5-acetyl-4,7-diethoxy-6-hydroxybenzofuran | CHEMBL...)
Show SMILES CCOc1c(O)c(C(C)=O)c(OCC)c2ccoc12
Show InChI InChI=1S/C14H16O5/c1-4-17-12-9-6-7-19-13(9)14(18-5-2)11(16)10(12)8(3)15/h6-7,16H,4-5H2,1-3H3
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n/an/an/an/a 6.00E+3n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182595
PNG
(1-(4-(4-(trifluoromethyl)benzyloxy)-6-hydroxy-7-me...)
Show SMILES COc1c(O)c(C(C)=O)c(OCc2ccc(cc2)C(F)(F)F)c2ccoc12
Show InChI InChI=1S/C19H15F3O5/c1-10(23)14-15(24)18(25-2)17-13(7-8-26-17)16(14)27-9-11-3-5-12(6-4-11)19(20,21)22/h3-8,24H,9H2,1-2H3
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n/an/an/an/a 510n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182598
PNG
(1-[6-Hydroxy-4-methoxy-7-(2-methyl-benzyloxy)-benz...)
Show SMILES COc1c(C(C)=O)c(O)c(OCc2ccccc2C)c2occc12
Show InChI InChI=1S/C19H18O5/c1-11-6-4-5-7-13(11)10-24-19-16(21)15(12(2)20)17(22-3)14-8-9-23-18(14)19/h4-9,21H,10H2,1-3H3
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n/an/an/an/a 1.90E+3n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182599
PNG
(1-(4-(3-(trifluoromethoxy)benzyloxy)-6-hydroxy-7-m...)
Show SMILES COc1c(O)c(C(C)=O)c(OCc2cccc(OC(F)(F)F)c2)c2ccoc12
Show InChI InChI=1S/C19H15F3O6/c1-10(23)14-15(24)18(25-2)17-13(6-7-26-17)16(14)27-9-11-4-3-5-12(8-11)28-19(20,21)22/h3-8,24H,9H2,1-2H3
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n/an/an/an/a 550n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182600
PNG
(1-(4-(4-benzoylbenzyloxy)-6-hydroxy-7-methoxybenzo...)
Show SMILES COc1c(O)c(C(C)=O)c(OCc2ccc(cc2)C(=O)c2ccccc2)c2ccoc12
Show InChI InChI=1S/C25H20O6/c1-15(26)20-22(28)25(29-2)24-19(12-13-30-24)23(20)31-14-16-8-10-18(11-9-16)21(27)17-6-4-3-5-7-17/h3-13,28H,14H2,1-2H3
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n/an/an/an/a 500n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182639
PNG
(1-(4-(2-fluorobenzyloxy)-6-hydroxy-7-methoxybenzof...)
Show SMILES COc1c(O)c(C(C)=O)c(OCc2ccccc2F)c2ccoc12
Show InChI InChI=1S/C18H15FO5/c1-10(20)14-15(21)18(22-2)17-12(7-8-23-17)16(14)24-9-11-5-3-4-6-13(11)19/h3-8,21H,9H2,1-2H3
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n/an/an/an/a 1.70E+3n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182636
PNG
(3-((5-acetyl-6-hydroxy-7-methoxybenzofuran-4-yloxy...)
Show SMILES COc1c(O)c(C(C)=O)c(OCc2cccc(c2)C(O)=O)c2ccoc12
Show InChI InChI=1S/C19H16O7/c1-10(20)14-15(21)18(24-2)17-13(6-7-25-17)16(14)26-9-11-4-3-5-12(8-11)19(22)23/h3-8,21H,9H2,1-2H3,(H,22,23)
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n/an/an/an/a>1.00E+4n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182610
PNG
(1-{6-hydroxy-7-methoxy-4-[(3-methylbenzyl)oxy]-1-b...)
Show SMILES COc1c(O)c(C(C)=O)c(OCc2cccc(C)c2)c2ccoc12
Show InChI InChI=1S/C19H18O5/c1-11-5-4-6-13(9-11)10-24-17-14-7-8-23-18(14)19(22-3)16(21)15(17)12(2)20/h4-9,21H,10H2,1-3H3
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n/an/an/an/a 1.00E+3n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182609
PNG
(1-(4-(3-fluorobenzyloxy)-6-hydroxy-7-methoxybenzof...)
Show SMILES COc1c(O)c(C(C)=O)c(OCc2cccc(F)c2)c2ccoc12
Show InChI InChI=1S/C18H15FO5/c1-10(20)14-15(21)18(22-2)17-13(6-7-23-17)16(14)24-9-11-4-3-5-12(19)8-11/h3-8,21H,9H2,1-2H3
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n/an/an/an/a 1.20E+3n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182614
PNG
(1-(4-(4-(benzyloxy)benzyloxy)-6-hydroxy-7-methoxyb...)
Show SMILES COc1c(O)c(C(C)=O)c(OCc2ccc(OCc3ccccc3)cc2)c2ccoc12
Show InChI InChI=1S/C25H22O6/c1-16(26)21-22(27)25(28-2)24-20(12-13-29-24)23(21)31-15-18-8-10-19(11-9-18)30-14-17-6-4-3-5-7-17/h3-13,27H,14-15H2,1-2H3
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n/an/an/an/a 8.80E+3n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182611
PNG
(1-(4-(4-(trifluoromethoxy)benzyloxy)-6-hydroxy-7-m...)
Show SMILES COc1c(O)c(C(C)=O)c(OCc2ccc(OC(F)(F)F)cc2)c2ccoc12
Show InChI InChI=1S/C19H15F3O6/c1-10(23)14-15(24)18(25-2)17-13(7-8-26-17)16(14)27-9-11-3-5-12(6-4-11)28-19(20,21)22/h3-8,24H,9H2,1-2H3
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n/an/an/an/a 1.80E+3n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182612
PNG
(1-(6-hydroxy-7-methoxy-4-phenoxybenzofuran-5-yl)et...)
Show SMILES COc1c(O)c(C(C)=O)c(Oc2ccccc2)c2ccoc12
Show InChI InChI=1S/C17H14O5/c1-10(18)13-14(19)17(20-2)16-12(8-9-21-16)15(13)22-11-6-4-3-5-7-11/h3-9,19H,1-2H3
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n/an/an/an/a 4.00E+3n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182613
PNG
(5-acetyl-7-benzyloxy-6-hydroxy-4-methoxybenzofuran...)
Show SMILES COc1c(C(C)=O)c(O)c(OCc2ccccc2)c2occc12
Show InChI InChI=1S/C18H16O5/c1-11(19)14-15(20)18(23-10-12-6-4-3-5-7-12)17-13(8-9-22-17)16(14)21-2/h3-9,20H,10H2,1-2H3
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n/an/an/an/a 1.20E+3n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182616
PNG
(3-(4-ethoxy-6-hydroxy-7-methoxybenzofuran-5-yl)-1-...)
Show SMILES CCOc1c(C(=O)\C=C\c2cccc(O)c2)c(O)c(OC)c2occc12
Show InChI InChI=1S/C20H18O6/c1-3-25-18-14-9-10-26-19(14)20(24-2)17(23)16(18)15(22)8-7-12-5-4-6-13(21)11-12/h4-11,21,23H,3H2,1-2H3/b8-7+
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n/an/an/an/a 2.50E+3n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182615
PNG
(1-(4-(3-nitrobenzyloxy)-6-hydroxy-7-methoxybenzofu...)
Show SMILES COc1c(O)c(C(C)=O)c(OCc2cccc(c2)[N+]([O-])=O)c2ccoc12
Show InChI InChI=1S/C18H15NO7/c1-10(20)14-15(21)18(24-2)17-13(6-7-25-17)16(14)26-9-11-4-3-5-12(8-11)19(22)23/h3-8,21H,9H2,1-2H3
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n/an/an/an/a 1.40E+3n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182617
PNG
(1-(4-(4-tert-butylbenzyloxy)-6-hydroxy-7-methoxybe...)
Show SMILES COc1c(O)c(C(C)=O)c(OCc2ccc(cc2)C(C)(C)C)c2ccoc12
Show InChI InChI=1S/C22H24O5/c1-13(23)17-18(24)21(25-5)20-16(10-11-26-20)19(17)27-12-14-6-8-15(9-7-14)22(2,3)4/h6-11,24H,12H2,1-5H3
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n/an/an/an/a 1.50E+3n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182587
PNG
(5-acetyl-4-(4'-chloro)benzyloxy-6-hydroxy-7-methox...)
Show SMILES COc1c(O)c(C(C)=O)c(OCc2ccc(Cl)cc2)c2ccoc12
Show InChI InChI=1S/C18H15ClO5/c1-10(20)14-15(21)18(22-2)17-13(7-8-23-17)16(14)24-9-11-3-5-12(19)6-4-11/h3-8,21H,9H2,1-2H3
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n/an/an/an/a 480n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
Voltage-gated potassium channel subunit Kv1.3


(Mus musculus)
BDBM50182618
PNG
(1-(4-(3-chlorobenzyloxy)-6-hydroxy-7-methoxybenzof...)
Show SMILES COc1c(O)c(C(C)=O)c(OCc2cccc(Cl)c2)c2ccoc12
Show InChI InChI=1S/C18H15ClO5/c1-10(20)14-15(21)18(22-2)17-13(6-7-23-17)16(14)24-9-11-4-3-5-12(19)8-11/h3-8,21H,9H2,1-2H3
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n/an/an/an/a 1.40E+3n/an/an/an/a



Institute of Medical Research Biotechnology Centre

Curated by ChEMBL


Assay Description
Effect on blockade of mouse Kv1.3 channel expressed in L929 cells


Citation and Details
More data for this
Ligand-Target Pair
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