Compile Data Set for Download or QSAR
maximum 50k data
Found 104 Enz. Inhib. hit(s) with all data for entry = 3463
TargetAMSH-like protease(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401033(US10005735, Compound 31)
Affinity DataIC50:  170nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCOP9 signalosome complex subunit 5(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM400994(US10005735, Compound 7)
Affinity DataIC50:  200nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401020(US10005735, Compound 19)
Affinity DataIC50: <200nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401033(US10005735, Compound 31)
Affinity DataIC50:  200nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAMSH-like protease(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401021(US10005735, Compound 20)
Affinity DataIC50: <200nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401008(US10005735, Compound 17)
Affinity DataIC50: <200nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401006(US10005735, Compound 15)
Affinity DataIC50:  200nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM400998(US10005735, Compound 11)
Affinity DataIC50:  300nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM224012(Capzimin | US10005735, Compound 12)
Affinity DataIC50:  340nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCOP9 signalosome complex subunit 5(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401023(US10005735, Compound 21)
Affinity DataIC50:  350nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAMSH-like protease(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401034(US10005735, Compound 32)
Affinity DataIC50:  400nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401034(US10005735, Compound 32)
Affinity DataIC50:  400nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM400992(US10005735, Compound 5)
Affinity DataIC50:  450nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM400996(US10005735, Compound 9)
Affinity DataIC50:  500nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAMSH-like protease(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401006(US10005735, Compound 15)
Affinity DataIC50:  500nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCOP9 signalosome complex subunit 5(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401020(US10005735, Compound 19)
Affinity DataIC50:  500nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401029(US10005735, Compound 27)
Affinity DataIC50:  500nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAMSH-like protease(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401029(US10005735, Compound 27)
Affinity DataIC50:  500nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAMSH-like protease(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401020(US10005735, Compound 19)
Affinity DataIC50:  600nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAMSH-like protease(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401030(US10005735, Compound 28)
Affinity DataIC50:  700nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401030(US10005735, Compound 28)
Affinity DataIC50:  700nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401026(US10005735, Compound 24)
Affinity DataIC50:  700nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401009(US10005735, Compound 18)
Affinity DataIC50:  700nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM400995(US10005735, Compound 8)
Affinity DataIC50:  800nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401023(US10005735, Compound 21)
Affinity DataIC50:  800nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAMSH-like protease(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401031(US10005735, Compound 29)
Affinity DataIC50:  800nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAMSH-like protease(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401008(US10005735, Compound 17)
Affinity DataIC50:  850nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAMSH-like protease(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401023(US10005735, Compound 21)
Affinity DataIC50:  880nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAMSH-like protease(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM400994(US10005735, Compound 7)
Affinity DataIC50:  900nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM400994(US10005735, Compound 7)
Affinity DataIC50:  900nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401021(US10005735, Compound 20)
Affinity DataIC50:  900nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM400988(US10005735, Compound 1)
Affinity DataIC50:  1.00E+3nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401028(US10005735, Compound 26)
Affinity DataIC50:  1.00E+3nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAMSH-like protease(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401026(US10005735, Compound 24)
Affinity DataIC50:  1.00E+3nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401031(US10005735, Compound 29)
Affinity DataIC50:  1.10E+3nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401007(US10005735, Compound 16)
Affinity DataIC50:  1.10E+3nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401025(US10005735, Compound 23)
Affinity DataIC50:  1.20E+3nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM400997(US10005735, Compound 10)
Affinity DataIC50:  1.20E+3nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAMSH-like protease(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM400988(US10005735, Compound 1)
Affinity DataIC50:  1.20E+3nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAMSH-like protease(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM400998(US10005735, Compound 11)
Affinity DataIC50:  1.30E+3nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAMSH-like protease(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM400995(US10005735, Compound 8)
Affinity DataIC50:  1.30E+3nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM400989(US10005735, Compound 2)
Affinity DataIC50:  1.60E+3nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAMSH-like protease(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM400997(US10005735, Compound 10)
Affinity DataIC50:  1.70E+3nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAMSH-like protease(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401027(US10005735, Compound 25)
Affinity DataIC50:  2.20E+3nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401027(US10005735, Compound 25)
Affinity DataIC50:  2.20E+3nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAMSH-like protease(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM400990(US10005735, Compound 3)
Affinity DataIC50:  2.20E+3nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAMSH-like protease(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM401025(US10005735, Compound 23)
Affinity DataIC50:  2.27E+3nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM400991(US10005735, Compound 4)
Affinity DataIC50:  2.60E+3nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM400990(US10005735, Compound 3)
Affinity DataIC50:  2.80E+3nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute Of Technology

US Patent
LigandPNGBDBM224013(8-Mercaptoquinoline (8TQ) | US10005735, Example 8T...)
Affinity DataIC50:  2.80E+3nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
In DepthDetails US Patent
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