Compile Data Set for Download or QSAR
maximum 50k data
Found 140 Enz. Inhib. hit(s) with all data for entry = 3480
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401715(US10005792, Compound 135 | US10005792, Compound 77)
Affinity DataIC50:  15nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401715(US10005792, Compound 135 | US10005792, Compound 77)
Affinity DataIC50:  29nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401764(US10005792, Compound 123)
Affinity DataIC50:  40nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401765(US10005792, Compound 124)
Affinity DataIC50:  48nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401672(US10005792, Compound 35)
Affinity DataIC50:  50nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401741(US10005792, Compound 103 | US10005792, Compound 13...)
Affinity DataIC50:  50nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401677(US10005792, Compound 40)
Affinity DataIC50:  57nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401713(US10005792, Compound 75)
Affinity DataIC50:  64nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401755(US10005792, Compound 114)
Affinity DataIC50:  66nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401673(US10005792, Compound 37)
Affinity DataIC50:  95nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401693(US10005792, Compound 56)
Affinity DataIC50:  98nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401741(US10005792, Compound 103 | US10005792, Compound 13...)
Affinity DataIC50:  120nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401676(US10005792, Compound 39)
Affinity DataIC50:  120nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401762(US10005792, Compound 121)
Affinity DataIC50:  130nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401774(US10005792, Compound 133)
Affinity DataIC50:  131nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401768(US10005792, Compound 127)
Affinity DataIC50:  137nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401679(US10005792, Compound 42)
Affinity DataIC50:  137nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401672(US10005792, Compound 35)
Affinity DataIC50:  155nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401678(US10005792, Compound 41)
Affinity DataIC50:  157nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401708(US10005792, Compound 70)
Affinity DataIC50:  157nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401673(US10005792, Compound 37)
Affinity DataIC50:  163nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401690(US10005792, Compound 53)
Affinity DataIC50:  164nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401751(US10005792, Compound 110)
Affinity DataIC50:  166nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401763(US10005792, Compound 122)
Affinity DataIC50:  166nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401658(US10005792, Compound 22)
Affinity DataIC50:  171nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401698(US10005792, Compound 61)
Affinity DataIC50:  180nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401743(US10005792, Compound 105)
Affinity DataIC50:  196nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401714(US10005792, Compound 76)
Affinity DataIC50:  209nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401675(US10005792, Compound 38)
Affinity DataIC50:  210nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401652(US10005792, Compound 15)
Affinity DataIC50:  218nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401767(US10005792, Compound 126)
Affinity DataIC50:  226nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401727(US10005792, Compound 88)
Affinity DataIC50:  229nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401709(US10005792, Compound 71)
Affinity DataIC50:  237nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401655(US10005792, Compound 18)
Affinity DataIC50:  238nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401775(US10005792, Compound 134)
Affinity DataIC50:  238nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401718(US10005792, Compound 80)
Affinity DataIC50:  253nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401645(US10005792, Compound 8)
Affinity DataIC50:  263nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401757(US10005792, Compound 116)
Affinity DataIC50:  276nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401737(US10005792, Compound 98)
Affinity DataIC50:  281nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401653(US10005792, Compound 16)
Affinity DataIC50:  301nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401756(US10005792, Compound 115)
Affinity DataIC50:  305nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401618(US10005792, Compound 3)
Affinity DataIC50:  309nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401675(US10005792, Compound 38)
Affinity DataIC50:  310nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401617(US10005792, Compound 2)
Affinity DataIC50:  310nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401710(US10005792, Compound 72)
Affinity DataIC50:  341nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401681(US10005792, Compound 44)
Affinity DataIC50:  373nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401660(US10005792, Compound 24)
Affinity DataIC50:  425nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401664(US10005792, Compound 27)
Affinity DataIC50:  434nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401651(US10005792, Compound 14)
Affinity DataIC50:  445nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Ctxt

US Patent
LigandPNGBDBM401692(US10005792, Compound 55)
Affinity DataIC50:  450nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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