Compile Data Set for Download or QSAR
maximum 50k data
Found 26 Enz. Inhib. hit(s) with all data for entry = 3493
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402040(Preparation of N-(3-(5-chloro-2-(4-fluoro-3-(N-met...)
Affinity DataIC50:  11nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402042(Preparation of N-(3-(5-chloro-2-(4-fluoro-3-(N-met...)
Affinity DataIC50:  11nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402041(Preparation of N-(3-(5-chloro-2-(4-fluoro-3-(N-met...)
Affinity DataIC50:  21nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402042(Preparation of N-(3-(5-chloro-2-(4-fluoro-3-(N-met...)
Affinity DataIC50:  42nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402040(Preparation of N-(3-(5-chloro-2-(4-fluoro-3-(N-met...)
Affinity DataIC50:  105nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402040(Preparation of N-(3-(5-chloro-2-(4-fluoro-3-(N-met...)
Affinity DataIC50:  107nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402040(Preparation of N-(3-(5-chloro-2-(4-fluoro-3-(N-met...)
Affinity DataIC50:  162nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402042(Preparation of N-(3-(5-chloro-2-(4-fluoro-3-(N-met...)
Affinity DataIC50:  173nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402041(Preparation of N-(3-(5-chloro-2-(4-fluoro-3-(N-met...)
Affinity DataIC50:  279nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Blk(Homo sapiens (Human))
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402040(Preparation of N-(3-(5-chloro-2-(4-fluoro-3-(N-met...)
Affinity DataIC50:  286nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402040(Preparation of N-(3-(5-chloro-2-(4-fluoro-3-(N-met...)
Affinity DataIC50:  319nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402042(Preparation of N-(3-(5-chloro-2-(4-fluoro-3-(N-met...)
Affinity DataIC50:  664nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402040(Preparation of N-(3-(5-chloro-2-(4-fluoro-3-(N-met...)
Affinity DataIC50:  698nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase Blk(Homo sapiens (Human))
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402042(Preparation of N-(3-(5-chloro-2-(4-fluoro-3-(N-met...)
Affinity DataIC50:  855nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402042(Preparation of N-(3-(5-chloro-2-(4-fluoro-3-(N-met...)
Affinity DataIC50:  1.23E+3nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402040(Preparation of N-(3-(5-chloro-2-(4-fluoro-3-(N-met...)
Affinity DataIC50:  1.40E+3nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase Blk(Homo sapiens (Human))
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402041(Preparation of N-(3-(5-chloro-2-(4-fluoro-3-(N-met...)
Affinity DataIC50:  1.66E+3nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402042(Preparation of N-(3-(5-chloro-2-(4-fluoro-3-(N-met...)
Affinity DataIC50:  1.92E+3nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402041(Preparation of N-(3-(5-chloro-2-(4-fluoro-3-(N-met...)
Affinity DataIC50: >1.00E+4nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402041(Preparation of N-(3-(5-chloro-2-(4-fluoro-3-(N-met...)
Affinity DataIC50: >1.00E+4nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402041(Preparation of N-(3-(5-chloro-2-(4-fluoro-3-(N-met...)
Affinity DataIC50: >1.00E+4nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402042(Preparation of N-(3-(5-chloro-2-(4-fluoro-3-(N-met...)
Affinity DataIC50: >1.00E+4nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402041(Preparation of N-(3-(5-chloro-2-(4-fluoro-3-(N-met...)
Affinity DataIC50: >1.00E+4nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402040(Preparation of N-(3-(5-chloro-2-(4-fluoro-3-(N-met...)
Affinity DataIC50: >1.00E+4nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402041(Preparation of N-(3-(5-chloro-2-(4-fluoro-3-(N-met...)
Affinity DataIC50: >1.00E+4nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402041(Preparation of N-(3-(5-chloro-2-(4-fluoro-3-(N-met...)
Affinity DataIC50: >1.00E+4nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent