Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Rho-associated protein kinase 1 (Homo sapiens (human)) | BDBM50173310![]() (CHEMBL3808660 | US10023564, Example 1) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem Patents | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rho-associated protein kinase 1 (Homo sapiens (human)) | BDBM50173307![]() (CHEMBL3809796 | US10023564, Example 8) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem Patents | n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rho-associated protein kinase 1 (Homo sapiens (human)) | BDBM50173315![]() (CHEMBL3809100 | US10023564, Example 4) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 21 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rho-associated protein kinase 1 (Homo sapiens (human)) | BDBM50173305![]() (CHEMBL3810107 | US10023564, Example 3) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 23 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rho-associated protein kinase 1 (Homo sapiens (human)) | BDBM50173311![]() (CHEMBL3810073 | US10023564, Example 6) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rho-associated protein kinase 1 (Homo sapiens (human)) | BDBM50173325![]() (CHEMBL3809965 | US10023564, Example 5) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 57 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM50173325![]() (CHEMBL3809965 | US10023564, Example 5) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 60 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rho-associated protein kinase 1 (Homo sapiens (human)) | BDBM50173323![]() (CHEMBL3808621 | US10023564, Example 2) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | n/a | n/a | 61 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rho-associated protein kinase 1 (Homo sapiens (human)) | BDBM50173314![]() (CHEMBL3808840 | US10023564, Example 16) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 69 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM50173309![]() (CHEMBL3809913 | US10023564, Example 10) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 70 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM50173307![]() (CHEMBL3809796 | US10023564, Example 8) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem Patents | n/a | n/a | 70 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rho-associated protein kinase 1 (Homo sapiens (human)) | BDBM50173320![]() (GSK-180736A | GSK180736A | US10023564, Compound GS...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | n/a | n/a | 78 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rho-associated protein kinase 1 (Homo sapiens (human)) | BDBM50173312![]() (CHEMBL3810312 | US10023564, Example 18) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | n/a | n/a | 97 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM50173323![]() (CHEMBL3808621 | US10023564, Example 2) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | n/a | n/a | 120 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM50173308![]() (CHEMBL3810271 | US10023564, Example 9) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM50173319![]() (CHEMBL3809020 | US10023564, Example 11) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem Patents Similars | PDB | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a | n/a |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM283998![]() (E24 | US10023564, Example 24) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 140 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rho-associated protein kinase 1 (Homo sapiens (human)) | BDBM50173329![]() (CHEMBL3809697 | US10023564, Example 15) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 150 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM50173310![]() (CHEMBL3808660 | US10023564, Example 1) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem Patents | PDB | n/a | n/a | 150 | n/a | n/a | n/a | n/a | n/a | n/a |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM283996![]() (E22 | US10023564, Example 22) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 180 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rho-associated protein kinase 1 (Homo sapiens (human)) | BDBM50173317![]() (CHEMBL3810349 | US10023564, Example 12) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 190 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM50173315![]() (CHEMBL3809100 | US10023564, Example 4) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rho-associated protein kinase 1 (Homo sapiens (human)) | BDBM50173324![]() (CHEMBL3809124 | US10023564, Example 30) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM50173328![]() (CHEMBL3808918 | US10023564, Example 14) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem Similars | PDB | n/a | n/a | 230 | n/a | n/a | n/a | n/a | n/a | n/a |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM283998![]() (E24 | US10023564, Example 24) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 240 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM50173305![]() (CHEMBL3810107 | US10023564, Example 3) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 280 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rho-associated protein kinase 1 (Homo sapiens (human)) | BDBM50173328![]() (CHEMBL3808918 | US10023564, Example 14) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem Similars | n/a | n/a | 290 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM284001![]() (E27 | US10023564, Example 27) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 320 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM50173310![]() (CHEMBL3808660 | US10023564, Example 1) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem Patents | PDB | n/a | n/a | 380 | n/a | n/a | n/a | n/a | n/a | n/a |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Rho-associated protein kinase 1 (Homo sapiens (human)) | BDBM50173326![]() (CHEMBL3809604 | US10023564, Example 29) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 400 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM283996![]() (E22 | US10023564, Example 22) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 410 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM50173312![]() (CHEMBL3810312 | US10023564, Example 18) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | n/a | n/a | 420 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rho-associated protein kinase 1 (Homo sapiens (human)) | BDBM50173327![]() (CHEMBL3808499 | US10023564, Example 28) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 450 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM50173324![]() (CHEMBL3809124 | US10023564, Example 30) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 450 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM50173311![]() (CHEMBL3810073 | US10023564, Example 6) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 460 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM284006![]() (E32 | US10023564, Example 32) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 500 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM284007![]() (E33 | US10023564, Example 33) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 680 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM50173314![]() (CHEMBL3808840 | US10023564, Example 16) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 690 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM283994![]() (E20 | US10023564, Example 20) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 740 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM50173320![]() (GSK-180736A | GSK180736A | US10023564, Compound GS...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | n/a | n/a | 770 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM50173315![]() (CHEMBL3809100 | US10023564, Example 4) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM283997![]() (E23 | US10023564, Example 23) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 820 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM284009![]() (E35 | US10023564, Example 35) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 960 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM50173318![]() (CHEMBL3809788 | US10023564, Example 17) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM284000![]() (E26 | US10023564, Example 26) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM284008![]() (E34 | US10023564, Example 34) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM284005![]() (E31 | US10023564, Example 31) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM284006![]() (E32 | US10023564, Example 32) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rho-associated protein kinase 1 (Homo sapiens (human)) | BDBM50173330![]() (CHEMBL3808657 | US10023564, Example 13) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 1.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM50173329![]() (CHEMBL3809697 | US10023564, Example 15) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 1.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM50173325![]() (CHEMBL3809965 | US10023564, Example 5) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM284001![]() (E27 | US10023564, Example 27) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 2.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM50173307![]() (CHEMBL3809796 | US10023564, Example 8) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem Patents | PDB | n/a | n/a | 2.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM284010![]() (E36 | US10023564, Example 36) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 2.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM50173330![]() (CHEMBL3808657 | US10023564, Example 13) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 2.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM283996![]() (E22 | US10023564, Example 22) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 3.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM50173312![]() (CHEMBL3810312 | US10023564, Example 18) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | n/a | n/a | 3.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM50173310![]() (CHEMBL3808660 | US10023564, Example 1) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem Patents | n/a | n/a | 3.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM284011![]() (E37 | US10023564, Example 37) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM50173317![]() (CHEMBL3810349 | US10023564, Example 12) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 4.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM284009![]() (E35 | US10023564, Example 35) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 4.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM50173314![]() (CHEMBL3808840 | US10023564, Example 16) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 4.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM50173323![]() (CHEMBL3808621 | US10023564, Example 2) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | n/a | n/a | 5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM50173306![]() (CHEMBL3808565 | US10023564, Example 7) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 5.15E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM283999![]() (E25 | US10023564, Example 25) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 5.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM50173307![]() (CHEMBL3809796 | US10023564, Example 8) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem Patents | n/a | n/a | 5.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rho-associated protein kinase 1 (Homo sapiens (human)) | BDBM50173309![]() (CHEMBL3809913 | US10023564, Example 10) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 5.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM50173305![]() (CHEMBL3810107 | US10023564, Example 3) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 6.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rho-associated protein kinase 1 (Homo sapiens (human)) | BDBM50173308![]() (CHEMBL3810271 | US10023564, Example 9) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | n/a | n/a | 6.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM284012![]() (E38 | US10023564, Example 38) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 7.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM50173311![]() (CHEMBL3810073 | US10023564, Example 6) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 8.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM284010![]() (E36 | US10023564, Example 36) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 8.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rho-associated protein kinase 1 (Homo sapiens (human)) | BDBM50173318![]() (CHEMBL3809788 | US10023564, Example 17) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rho-associated protein kinase 1 (Homo sapiens (human)) | BDBM50173319![]() (CHEMBL3809020 | US10023564, Example 11) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem Patents Similars | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM284005![]() (E31 | US10023564, Example 31) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 1.08E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM284007![]() (E33 | US10023564, Example 33) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 1.18E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM50173315![]() (CHEMBL3809100 | US10023564, Example 4) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 1.19E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM284001![]() (E27 | US10023564, Example 27) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 1.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM283995![]() (E21 | US10023564, Example 21) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 1.46E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM50173325![]() (CHEMBL3809965 | US10023564, Example 5) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 1.63E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM283998![]() (E24 | US10023564, Example 24) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 1.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM284006![]() (E32 | US10023564, Example 32) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 2.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM283997![]() (E23 | US10023564, Example 23) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 2.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM50173327![]() (CHEMBL3808499 | US10023564, Example 28) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 2.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM284008![]() (E34 | US10023564, Example 34) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 4.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM284000![]() (E26 | US10023564, Example 26) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 4.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM283993![]() (E19 | US10023564, Example 19) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 5.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM50173328![]() (CHEMBL3808918 | US10023564, Example 14) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem Similars | n/a | n/a | 5.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM50173309![]() (CHEMBL3809913 | US10023564, Example 10) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 6.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM284011![]() (E37 | US10023564, Example 37) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 6.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM283997![]() (E23 | US10023564, Example 23) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 6.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM50173329![]() (CHEMBL3809697 | US10023564, Example 15) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 6.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM50173314![]() (CHEMBL3808840 | US10023564, Example 16) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | 7.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM284011![]() (E37 | US10023564, Example 37) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 7.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM283999![]() (E25 | US10023564, Example 25) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 8.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM283994![]() (E20 | US10023564, Example 20) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | 9.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM284009![]() (E35 | US10023564, Example 35) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM284012![]() (E38 | US10023564, Example 38) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM50173311![]() (CHEMBL3810073 | US10023564, Example 6) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM50173309![]() (CHEMBL3809913 | US10023564, Example 10) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM50173330![]() (CHEMBL3808657 | US10023564, Example 13) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM284005![]() (E31 | US10023564, Example 31) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rho-associated protein kinase 1 (Homo sapiens (human)) | BDBM50173306![]() (CHEMBL3808565 | US10023564, Example 7) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM50173312![]() (CHEMBL3810312 | US10023564, Example 18) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM50173326![]() (CHEMBL3809604 | US10023564, Example 29) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM50173317![]() (CHEMBL3810349 | US10023564, Example 12) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM50173329![]() (CHEMBL3809697 | US10023564, Example 15) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM283993![]() (E19 | US10023564, Example 19) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM283999![]() (E25 | US10023564, Example 25) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM284007![]() (E33 | US10023564, Example 33) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM284010![]() (E36 | US10023564, Example 36) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM50173308![]() (CHEMBL3810271 | US10023564, Example 9) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM50173319![]() (CHEMBL3809020 | US10023564, Example 11) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem Patents Similars | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM50173328![]() (CHEMBL3808918 | US10023564, Example 14) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem Similars | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM283994![]() (E20 | US10023564, Example 20) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM283995![]() (E21 | US10023564, Example 21) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM50173327![]() (CHEMBL3808499 | US10023564, Example 28) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM50173324![]() (CHEMBL3809124 | US10023564, Example 30) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM284012![]() (E38 | US10023564, Example 38) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM50173320![]() (GSK-180736A | GSK180736A | US10023564, Compound GS...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM50173320![]() (GSK-180736A | GSK180736A | US10023564, Compound GS...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | n/a | n/a | 1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM50173306![]() (CHEMBL3808565 | US10023564, Example 7) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM50173306![]() (CHEMBL3808565 | US10023564, Example 7) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM50173319![]() (CHEMBL3809020 | US10023564, Example 11) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem Patents Similars | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM50173317![]() (CHEMBL3810349 | US10023564, Example 12) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM50173326![]() (CHEMBL3809604 | US10023564, Example 29) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM284008![]() (E34 | US10023564, Example 34) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM50173330![]() (CHEMBL3808657 | US10023564, Example 13) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM50173318![]() (CHEMBL3809788 | US10023564, Example 17) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM283993![]() (E19 | US10023564, Example 19) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM50173327![]() (CHEMBL3808499 | US10023564, Example 28) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human)) | BDBM50173326![]() (CHEMBL3809604 | US10023564, Example 29) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM50173324![]() (CHEMBL3809124 | US10023564, Example 30) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM50173323![]() (CHEMBL3808621 | US10023564, Example 2) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM50173305![]() (CHEMBL3810107 | US10023564, Example 3) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM50173308![]() (CHEMBL3810271 | US10023564, Example 9) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM50173318![]() (CHEMBL3809788 | US10023564, Example 17) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein-coupled receptor kinase 5 (Homo sapiens) | BDBM283995![]() (E21 | US10023564, Example 21) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Rhodopsin kinase (Homo sapiens) | BDBM284000![]() (E26 | US10023564, Example 26) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | UniChem | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description GRK1, 2 and 5 kinetic assays were conducted in a buffer containing 20 mM HEPES pH 7.0, 5 μM ATP, 2 mM MgCl2, and 0.025% DDM with 50 nM GRK and e... | US Patent US10023564 (2018) | |||||||||||
More data for this Ligand-Target Pair |