Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with all data for entry = 733
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

US Patent
LigandPNGBDBM288689(TC001262 | US10092529, Compound 38)
Affinity DataKi:  13.7nM ΔG°:  -44.9kJ/moleT: 2°CAssay Description:Materials: Recombinant full-length RIPK1 protein with N-terminal GST-tag (Cat#R07-34G) was purchased from SignalChem. The ADP-Glo kinase assay kit (C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

US Patent
LigandPNGBDBM288691(TC001207 | US10092529, Compound 24)
Affinity DataKi:  19.8nM ΔG°:  -44.0kJ/moleT: 2°CAssay Description:Materials: Recombinant full-length RIPK1 protein with N-terminal GST-tag (Cat#R07-34G) was purchased from SignalChem. The ADP-Glo kinase assay kit (C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

US Patent
LigandPNGBDBM288686(TC001124 | US10092529, Compound 10)
Affinity DataKi:  22.5nM ΔG°:  -43.7kJ/moleT: 2°CAssay Description:Materials: Recombinant full-length RIPK1 protein with N-terminal GST-tag (Cat#R07-34G) was purchased from SignalChem. The ADP-Glo kinase assay kit (C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

US Patent
LigandPNGBDBM288687(TC001129 | US10092529, Compound 2)
Affinity DataKi:  34.8nM ΔG°:  -42.6kJ/moleT: 2°CAssay Description:Materials: Recombinant full-length RIPK1 protein with N-terminal GST-tag (Cat#R07-34G) was purchased from SignalChem. The ADP-Glo kinase assay kit (C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

US Patent
LigandPNGBDBM288688(TC001273 | US10092529, Compound 25)
Affinity DataKi:  152nM ΔG°:  -38.9kJ/moleT: 2°CAssay Description:Materials: Recombinant full-length RIPK1 protein with N-terminal GST-tag (Cat#R07-34G) was purchased from SignalChem. The ADP-Glo kinase assay kit (C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

US Patent
LigandPNGBDBM288690(TC001287 | US10092529, Compound 15)
Affinity DataKi:  460nM ΔG°:  -36.2kJ/moleT: 2°CAssay Description:Materials: Recombinant full-length RIPK1 protein with N-terminal GST-tag (Cat#R07-34G) was purchased from SignalChem. The ADP-Glo kinase assay kit (C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

US Patent
LigandPNGBDBM288692(TC001265 | US10092529, Compound 31)
Affinity DataKi:  1.07E+3nM ΔG°:  -34.1kJ/moleT: 2°CAssay Description:Materials: Recombinant full-length RIPK1 protein with N-terminal GST-tag (Cat#R07-34G) was purchased from SignalChem. The ADP-Glo kinase assay kit (C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent