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Found 5 Enz. Inhib. hit(s) with all data for entry = 748
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Eli Lilly

US Patent
LigandPNGBDBM289087(N-[(1S)-2-[4-[2-[4-Amino- 6-methyl-2- (trifluorome...)
Affinity DataIC50:  55.7nMpH: 7.5Assay Description:Prepare test compounds in DMSO to make up a 0.2 mM stock solution. Serially dilute the stock solution in DMSO to obtain a ten-point dilution curve wi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Eli Lilly

US Patent
LigandPNGBDBM289086(N-[(1 S)-2-[4-[2-[4-Amino-6-methyl-2-(trifluoromet...)
Affinity DataIC50:  69.5nMpH: 7.5Assay Description:Prepare test compounds in DMSO to make up a 0.2 mM stock solution. Serially dilute the stock solution in DMSO to obtain a ten-point dilution curve wi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Eli Lilly

US Patent
LigandPNGBDBM289089(N-[(1S)-2-[4-[2-[4-Amino- 6-methyl-2- (trifluorome...)
Affinity DataIC50:  276nMpH: 7.5Assay Description:Prepare test compounds in DMSO to make up a 0.2 mM stock solution. Serially dilute the stock solution in DMSO to obtain a ten-point dilution curve wi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Eli Lilly

US Patent
LigandPNGBDBM289088(N-[(1S)-2-[4-[2-[4-Amino- 6-methyl-2- (trifluorome...)
Affinity DataIC50:  420nMpH: 7.5Assay Description:Prepare test compounds in DMSO to make up a 0.2 mM stock solution. Serially dilute the stock solution in DMSO to obtain a ten-point dilution curve wi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Eli Lilly

US Patent
LigandPNGBDBM289090(Methyl-[(1S)-2-[4-[2-[4-amino-6-methyl-2-(trifluor...)
Affinity DataIC50:  615nMpH: 7.5Assay Description:Prepare test compounds in DMSO to make up a 0.2 mM stock solution. Serially dilute the stock solution in DMSO to obtain a ten-point dilution curve wi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent