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Found 10 Enz. Inhib. hit(s) with all data for entry = 1136
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM310926(((5-Bromo-2-(Carboxy)Benzo[b]Thiophen-6-yl)Difluor...)
Affinity DataIC50:  170nMAssay Description:The assay was carried out at room temperature in 96 well plates. The reaction mixture in 170 μl contained 50 mM Bis-Tris (pH=6.3), 2 mM EDTA, 5 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM310919(6-Bromo-5-(Difluoro(Phosphonato)Methyl)Benzo[b]Thi...)
Affinity DataIC50:  260nMAssay Description:The assay was carried out at room temperature in 96 well plates. The reaction mixture in 170 μl contained 50 mM Bis-Tris (pH=6.3), 2 mM EDTA, 5 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM310920(((6-Bromo-2-Carbamoylbenzo[b]Thiophen-5-yl)Difluor...)
Affinity DataIC50:  280nMAssay Description:The assay was carried out at room temperature in 96 well plates. The reaction mixture in 170 μl contained 50 mM Bis-Tris (pH=6.3), 2 mM EDTA, 5 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM310923(((6-Bromo-2-(Cyanomethyl)Benzo[b]Thiophen-5-yl)Dif...)
Affinity DataIC50:  370nMAssay Description:The assay was carried out at room temperature in 96 well plates. The reaction mixture in 170 μl contained 50 mM Bis-Tris (pH=6.3), 2 mM EDTA, 5 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM310918(((6-Bromo-2-(Ethoxycarbonyl)Benzo[b]Thiophen-5-yl)...)
Affinity DataIC50:  450nMAssay Description:The assay was carried out at room temperature in 96 well plates. The reaction mixture in 170 μl contained 50 mM Bis-Tris (pH=6.3), 2 mM EDTA, 5 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50239833((3-bromo-7-cyanonaphthalen-2-yl)difluoromethylphos...)
Affinity DataIC50:  490nMAssay Description:The assay was carried out at room temperature in 96 well plates. The reaction mixture in 170 μl contained 50 mM Bis-Tris (pH=6.3), 2 mM EDTA, 5 ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM310924(((5-Bromo-2-(Ethoxycarbonyl)Benzo[b]Thiophen-6-yl)...)
Affinity DataIC50:  740nMAssay Description:The assay was carried out at room temperature in 96 well plates. The reaction mixture in 170 μl contained 50 mM Bis-Tris (pH=6.3), 2 mM EDTA, 5 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM310921(((6-Bromo-2-Cyanobenzo[b]Thiophen-5-yl)Difluoromet...)
Affinity DataIC50:  1.20E+3nMAssay Description:The assay was carried out at room temperature in 96 well plates. The reaction mixture in 170 μl contained 50 mM Bis-Tris (pH=6.3), 2 mM EDTA, 5 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM310922(((6-Bromo-2-(Hydroxymethyl)Benzo[b]Thiophen-5-yl)D...)
Affinity DataIC50:  1.50E+3nMAssay Description:The assay was carried out at room temperature in 96 well plates. The reaction mixture in 170 μl contained 50 mM Bis-Tris (pH=6.3), 2 mM EDTA, 5 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM310925(((5-Bromo-2-(Methoxycarbonyl)Benzo[b]Thiophen-6-yl...)
Affinity DataIC50:  2.90E+3nMAssay Description:The assay was carried out at room temperature in 96 well plates. The reaction mixture in 170 μl contained 50 mM Bis-Tris (pH=6.3), 2 mM EDTA, 5 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent