Compile Data Set for Download or QSAR
maximum 50k data
Found 14 Enz. Inhib. hit(s) with all data for entry = 1244
TargetSerine/threonine-protein kinase B-raf [416-766,V600E](Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM313753(US10167282, Compound TBAP-04)
Affinity DataIC50:  8nMAssay Description:Mutant BRAF WM266.4 Cells.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase B-raf [416-766,V600E](Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM313751(US10167282, Compound TBAP-02)
Affinity DataIC50:  12nMAssay Description:Mutant BRAF WM266.4 Cells.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase B-raf [416-766,V600E](Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM313750(US10167282, Compound TBAP-01)
Affinity DataIC50:  18nMAssay Description:Mutant BRAF WM266.4 Cells.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase B-raf [416-766,V600E](Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM313752(US10167282, Compound TBAP-03)
Affinity DataIC50:  19nMAssay Description:Mutant BRAF WM266.4 Cells.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase B-raf [416-766,V600E](Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM313753(US10167282, Compound TBAP-04)
Affinity DataIC50:  47nMAssay Description:V600EBRAF was generated by infection of SF9 insect cells cultured in SF-900 II medium (Invitrogen, Paisley, Scotland) with a baculovirus containing f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase B-raf [416-766,V600E](Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM313750(US10167282, Compound TBAP-01)
Affinity DataIC50:  62nMAssay Description:V600EBRAF was generated by infection of SF9 insect cells cultured in SF-900 II medium (Invitrogen, Paisley, Scotland) with a baculovirus containing f...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase B-raf [416-766,V600E](Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM313751(US10167282, Compound TBAP-02)
Affinity DataIC50:  99nMAssay Description:V600EBRAF was generated by infection of SF9 insect cells cultured in SF-900 II medium (Invitrogen, Paisley, Scotland) with a baculovirus containing f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase B-raf [416-766,V600E](Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM313752(US10167282, Compound TBAP-03)
Affinity DataIC50:  130nMAssay Description:V600EBRAF was generated by infection of SF9 insect cells cultured in SF-900 II medium (Invitrogen, Paisley, Scotland) with a baculovirus containing f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase B-raf [416-766,V600E](Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM313754(US10167282, Compound TBAP-05)
Affinity DataIC50:  390nMAssay Description:V600EBRAF was generated by infection of SF9 insect cells cultured in SF-900 II medium (Invitrogen, Paisley, Scotland) with a baculovirus containing f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase B-raf [416-766,V600E](Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM313754(US10167282, Compound TBAP-05)
Affinity DataIC50:  450nMAssay Description:Mutant BRAF WM266.4 Cells.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM313751(US10167282, Compound TBAP-02)
Affinity DataIC50:  6.50E+4nMAssay Description:Studies were conducted at Cyprotex Discovery in Cheshire, UK according to the contractor's protocol. The studies were performed on an IonWorks¿ H...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM313753(US10167282, Compound TBAP-04)
Affinity DataIC50: >1.00E+5nMAssay Description:Studies were conducted at Cyprotex Discovery in Cheshire, UK according to the contractor's protocol. The studies were performed on an IonWorks¿ H...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM313750(US10167282, Compound TBAP-01)
Affinity DataIC50: >1.00E+5nMAssay Description:Studies were conducted at Cyprotex Discovery in Cheshire, UK according to the contractor's protocol. The studies were performed on an IonWorks¿ H...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM313752(US10167282, Compound TBAP-03)
Affinity DataIC50: >1.00E+5nMAssay Description:Studies were conducted at Cyprotex Discovery in Cheshire, UK according to the contractor's protocol. The studies were performed on an IonWorks¿ H...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent