Compile Data Set for Download or QSAR
maximum 50k data
Found 22 Enz. Inhib. hit(s) with all data for entry = 1390
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Shanghai Huilun Life Science & Technology

US Patent
LigandPNGBDBM320266(4-(3-(4-(1H-imidazo[4,5-b]pyridin-5-yl)piperazine-...)
Affinity DataIC50:  1nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Shanghai Huilun Life Science & Technology

US Patent
LigandPNGBDBM320275(4-(3-(4-(1H-imidazo[4,5-b]pyridin-5-yl)piperazine-...)
Affinity DataIC50:  1nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Shanghai Huilun Life Science & Technology

US Patent
LigandPNGBDBM320267(4-(4-fluoro-3-(4-(2-oxo-2,3-dihydro-1H-imidazo[4,5...)
Affinity DataIC50:  1nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Shanghai Huilun Life Science & Technology

US Patent
LigandPNGBDBM320277(4-(3-(4-(1H-imidazo[4,5-b]pyridin-5-yl)piperazine-...)
Affinity DataIC50:  2nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Shanghai Huilun Life Science & Technology

US Patent
LigandPNGBDBM320263(4-(3-(4-(1H[1,2,3]triazolo[4,5-b]pyridin-5-yl)pipe...)
Affinity DataIC50:  2nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Shanghai Huilun Life Science & Technology

US Patent
LigandPNGBDBM320282(4-(3-(4-(3H-imidazo[4,5-b]pyridin-6-yl)piperazine-...)
Affinity DataIC50:  2nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Shanghai Huilun Life Science & Technology

US Patent
LigandPNGBDBM320271(4-(3-(4-(2-carbonyl-2,3-dihydro-1H-imidazo[4,5-b]p...)
Affinity DataIC50:  2nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Shanghai Huilun Life Science & Technology

US Patent
LigandPNGBDBM320268(4-(3-(4-(3H-imidazo[4,5-c]pyridin-6-yl)piperazine-...)
Affinity DataIC50:  3nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Shanghai Huilun Life Science & Technology

US Patent
LigandPNGBDBM320276(4-(3-(4-(1H-imidazo[4,5-b]pyridin-5-yl)piperazine-...)
Affinity DataIC50:  4nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Shanghai Huilun Life Science & Technology

US Patent
LigandPNGBDBM320272(4-(3-(4-(1H-[1,2,3]triazolo[4,5-b]pyridin-5-yl)pip...)
Affinity DataIC50:  5nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Shanghai Huilun Life Science & Technology

US Patent
LigandPNGBDBM320279(4-(3-(4-(2-oxo-2,3-dihydro-1H-imidazo[4,5-]pyridin...)
Affinity DataIC50:  6nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Shanghai Huilun Life Science & Technology

US Patent
LigandPNGBDBM320265(4-(4-fluoro-3-(4-(2-trifluoromethyl)-1H-imidazo[4,...)
Affinity DataIC50:  6nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Shanghai Huilun Life Science & Technology

US Patent
LigandPNGBDBM320278(4-(3-(4-(1H-[1,2,3]triazolo[4,5-b]pyridin-5-yl)pip...)
Affinity DataIC50:  7nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Shanghai Huilun Life Science & Technology

US Patent
LigandPNGBDBM27566(4-({3-[(4-cyclopropanecarbonylpiperazin-1-yl)carbo...)
Affinity DataIC50:  8nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Shanghai Huilun Life Science & Technology

US Patent
LigandPNGBDBM320269(4-(3-(4-(3H-imidazo[4,5-b]pyridin-6-yl)piperazine-...)
Affinity DataIC50:  8nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Shanghai Huilun Life Science & Technology

US Patent
LigandPNGBDBM320281(4-(3-(4-(3H-imidazo[4,5-c]pyridin-6-yl)piperazine-...)
Affinity DataIC50:  8nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Shanghai Huilun Life Science & Technology

US Patent
LigandPNGBDBM320264(4-(4-fluoro-3-(4-(2-methyl-1H-imidazo[4,5-b]pyridi...)
Affinity DataIC50:  9nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Shanghai Huilun Life Science & Technology

US Patent
LigandPNGBDBM320274(4-(3-(4-(2-trifluoromethyl)-1H-imidazo[4,5-b]pyrid...)
Affinity DataIC50:  10nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Shanghai Huilun Life Science & Technology

US Patent
LigandPNGBDBM320270(4-(3-(4-(7H-purin-2-yl)piperazine-1-carbonyl)-4-fl...)
Affinity DataIC50:  11nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Shanghai Huilun Life Science & Technology

US Patent
LigandPNGBDBM320280(4-(3-(4-(3H-imidazo[4,5-c]pyridin-6-yl)piperazine-...)
Affinity DataIC50:  13nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Shanghai Huilun Life Science & Technology

US Patent
LigandPNGBDBM320283(4-(3-(4-(3H-imidazo[4,5-b]pyridin-6-yl)piperazine-...)
Affinity DataIC50:  15nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Shanghai Huilun Life Science & Technology

US Patent
LigandPNGBDBM320273(4-(3-(4-(2-methyl-1H-imidazo[4,5-b]pyridin-5-yl)pi...)
Affinity DataIC50:  17nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent