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Found 44 Enz. Inhib. hit(s) with all data for entry = 1609
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332706(US10196378, Compound C09 | US10196378, Compound C1...)
Affinity DataKi:  0.640nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332705(US10196378, Compound C08)
Affinity DataKi:  0.960nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332699(US10196378, Compound C02)
Affinity DataKi: <1nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1 [Y253F](Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332702(US10196378, Compound C05)
Affinity DataKi: <1nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332700(US10196378, Compound C03)
Affinity DataKi: <1nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1 [Y253F](Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332699(US10196378, Compound C02)
Affinity DataKi: <1nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332700(US10196378, Compound C03)
Affinity DataKi: <1nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332702(US10196378, Compound C05)
Affinity DataKi: <1nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1 [T315I](Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332699(US10196378, Compound C02)
Affinity DataKi: <1nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332702(US10196378, Compound C05)
Affinity DataKi: <1nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332698(US10196378, Compound C01)
Affinity DataKi: <1nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1 [Y253F](Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332700(US10196378, Compound C03)
Affinity DataKi: <1nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1 [T315I](Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332700(US10196378, Compound C03)
Affinity DataKi: <1nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1 [T315I](Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332702(US10196378, Compound C05)
Affinity DataKi: <1nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332698(US10196378, Compound C01)
Affinity DataKi: <1nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1 [T315I](Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332698(US10196378, Compound C01)
Affinity DataKi: <1nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1 [Y253F](Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332698(US10196378, Compound C01)
Affinity DataKi: <1nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332699(US10196378, Compound C02)
Affinity DataKi: <1nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332701(US10196378, Compound C04)
Affinity DataKi:  1.70nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332701(US10196378, Compound C04)
Affinity DataKi:  1.70nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332703(US10196378, Compound C06)
Affinity DataKi:  2nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332703(US10196378, Compound C06)
Affinity DataKi:  2nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1 [T315I](Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332701(US10196378, Compound C04)
Affinity DataKi:  2.10nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1 [Y253F](Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332706(US10196378, Compound C09 | US10196378, Compound C1...)
Affinity DataKi:  2.5nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332706(US10196378, Compound C09 | US10196378, Compound C1...)
Affinity DataKi:  3.30nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1 [Y253F](Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332705(US10196378, Compound C08)
Affinity DataKi:  3.40nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1 [T315I](Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332703(US10196378, Compound C06)
Affinity DataKi:  4nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1 [Y253F](Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332703(US10196378, Compound C06)
Affinity DataKi:  6.20nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1 [Y253F](Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332706(US10196378, Compound C09 | US10196378, Compound C1...)
Affinity DataKi:  7.60nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332699(US10196378, Compound C02)
Affinity DataKi:  28nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332698(US10196378, Compound C01)
Affinity DataKi:  36nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1 [Y253F](Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332701(US10196378, Compound C04)
Affinity DataKi:  50nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1 [T315I](Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332704(US10196378, Compound C07)
Affinity DataKi:  119nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332700(US10196378, Compound C03)
Affinity DataKi:  120nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332706(US10196378, Compound C09 | US10196378, Compound C1...)
Affinity DataKi:  143nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332704(US10196378, Compound C07)
Affinity DataKi:  155nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332704(US10196378, Compound C07)
Affinity DataKi:  155nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332702(US10196378, Compound C05)
Affinity DataKi:  216nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332706(US10196378, Compound C09 | US10196378, Compound C1...)
Affinity DataKi:  345nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332705(US10196378, Compound C08)
Affinity DataKi:  518nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332701(US10196378, Compound C04)
Affinity DataKi:  4.50E+3nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1 [Y253F](Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332704(US10196378, Compound C07)
Affinity DataKi: >9.00E+3nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332703(US10196378, Compound C06)
Affinity DataKi:  1.20E+4nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM332704(US10196378, Compound C07)
Affinity DataKi: >2.70E+4nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent