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Found 462 Enz. Inhib. hit(s) with all data for entry = 2569
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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US Patent
LigandPNGBDBM50192240(CHEMBL3941818 | US10239870, Example 278)
Affinity DataKi:  0.0630nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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LigandPNGBDBM372015(US10239870, Example 275)
Affinity DataKi:  0.117nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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LigandPNGBDBM50192317(CHEMBL3899125 | US10239870, Example 281)
Affinity DataKi:  0.158nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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LigandPNGBDBM372014(US10239870, Example 274)
Affinity DataKi:  0.162nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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LigandPNGBDBM50192319(CHEMBL3920167 | US10239870, Example 279)
Affinity DataKi:  0.182nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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LigandPNGBDBM371876(US10239870, Example 89 | US10239870, Example 94)
Affinity DataKi:  0.186nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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LigandPNGBDBM372012(US10239870, Example 272)
Affinity DataKi:  0.234nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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LigandPNGBDBM50192318(CHEMBL3979523 | US10239870, Example 284)
Affinity DataKi:  0.245nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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LigandPNGBDBM50192449(CHEMBL3950540 | US10239870, Example 283)
Affinity DataKi:  0.263nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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LigandPNGBDBM50192333(CHEMBL3958201 | US10239870, Example 97)
Affinity DataKi:  0.275nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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LigandPNGBDBM371953(US10239870, Example 190)
Affinity DataKi:  0.282nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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LigandPNGBDBM50192445(CHEMBL3959240 | US10239870, Example 285)
Affinity DataKi:  0.316nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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LigandPNGBDBM371952(US10239870, Example 189)
Affinity DataKi:  0.339nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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LigandPNGBDBM50192023(CHEMBL3950254 | US10239870, Example 184)
Affinity DataKi:  0.339nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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US Patent
LigandPNGBDBM371980(US10239870, Example 228)
Affinity DataKi:  0.355nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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US Patent
LigandPNGBDBM372016(US10239870, Example 276)
Affinity DataKi:  0.363nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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LigandPNGBDBM371948(US10239870, Example 185)
Affinity DataKi:  0.417nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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LigandPNGBDBM371858(US10239870, Example 59 | US10239870, Example 60)
Affinity DataKi:  0.417nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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LigandPNGBDBM372000(US10239870, Example 258)
Affinity DataKi:  0.417nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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LigandPNGBDBM50192248(CHEMBL3927895 | US10239870, Example 30)
Affinity DataKi:  0.417nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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LigandPNGBDBM50192030(CHEMBL3970323 | US10239870, Example 289)
Affinity DataKi:  0.468nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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US Patent
LigandPNGBDBM372023(US10239870, Example 286)
Affinity DataKi:  0.525nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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LigandPNGBDBM372005(US10239870, Example 263)
Affinity DataKi:  0.550nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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LigandPNGBDBM50192447(CHEMBL3975989 | US10239870, Example 53)
Affinity DataKi:  0.550nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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LigandPNGBDBM371999(US10239870, Example 257)
Affinity DataKi:  0.575nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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LigandPNGBDBM50192326(CHEMBL3955608 | US10239870, Example 220)
Affinity DataKi:  0.575nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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US Patent
LigandPNGBDBM371998(US10239870, Example 256)
Affinity DataKi:  0.603nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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US Patent
LigandPNGBDBM50192454(CHEMBL3911264 | US10239870, Example 12)
Affinity DataKi:  0.631nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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LigandPNGBDBM50192230(CHEMBL3908174 | US10239870, Example 253)
Affinity DataKi:  0.631nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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US Patent
LigandPNGBDBM371954(US10239870, Example 191)
Affinity DataKi:  0.724nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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US Patent
LigandPNGBDBM371943(US10239870, Example 179 | US10239870, Example 182)
Affinity DataKi:  0.724nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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US Patent
LigandPNGBDBM372004(US10239870, Example 262)
Affinity DataKi:  0.759nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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US Patent
LigandPNGBDBM371877(US10239870, Example 92)
Affinity DataKi:  0.776nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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US Patent
LigandPNGBDBM372013(US10239870, Example 273)
Affinity DataKi:  0.776nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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US Patent
LigandPNGBDBM371914(US10239870, Example 140 | US10239870, Example 141)
Affinity DataKi:  0.794nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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LigandPNGBDBM50192029(CHEMBL3917887 | US10239870, Example 39)
Affinity DataKi:  0.813nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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LigandPNGBDBM371975(US10239870, Example 221)
Affinity DataKi:  0.832nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM371876(US10239870, Example 89 | US10239870, Example 94)
Affinity DataKi:  0.832nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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US Patent
LigandPNGBDBM371894(US10239870, Example 118)
Affinity DataKi:  0.851nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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US Patent
LigandPNGBDBM371978(US10239870, Example 224 | US10239870, Example 227)
Affinity DataKi:  0.851nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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LigandPNGBDBM50192315(CHEMBL3981856 | US10239870, Example 287)
Affinity DataKi:  0.851nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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US Patent
LigandPNGBDBM371878(US10239870, Example 93)
Affinity DataKi:  0.871nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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LigandPNGBDBM50192239(CHEMBL3922143 | US10239870, Example 48)
Affinity DataKi:  0.912nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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LigandPNGBDBM371870(US10239870, Example 79)
Affinity DataKi:  0.955nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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LigandPNGBDBM371928(US10239870, Example 162 | US10239870, Example 163)
Affinity DataKi:  0.955nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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LigandPNGBDBM50192099(CHEMBL3914556 | US10239870, Example 244)
Affinity DataKi:  0.977nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
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LigandPNGBDBM371858(US10239870, Example 59 | US10239870, Example 60)
Affinity DataKi:  0.977nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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LigandPNGBDBM371965(US10239870, Example 207 | US10239870, Example 212)
Affinity DataKi:  1.02nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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LigandPNGBDBM50192316(CHEMBL3985877 | US10239870, Example 57)
Affinity DataKi:  1.05nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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LigandPNGBDBM371969(US10239870, Example 213)
Affinity DataKi:  1.05nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
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