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Patent code US10294214

Compile Data Set for Download or QSAR
Found 80 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387733
PNG
(US10294214, Example 33)
Show SMILES CC(=O)c1nc2ccccc2c1NC(=O)CN1CCN(Cc2ccccc2)CC1
PDB

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US Patent
n/an/an/an/a 2.51E+3n/an/an/an/a



Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387735
PNG
(US10294214, Example 35)
Show SMILES COC(=O)c1nc2ccc(Br)cc2c1NC(=O)CN1CCN(Cc2ccccc2)CC1
PDB

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n/an/an/an/a 1.59E+3n/an/an/an/a



Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387743
PNG
(US10294214, Example 43)
Show SMILES CC(=O)c1nc2ccc(Br)cc2c1NC(=O)CN1CCC(CC1)c1ccccc1
PDB

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n/an/an/an/a 398n/an/an/an/a



Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387747
PNG
(US10294214, Example 47)
Show SMILES COC(=O)c1nc2ccc(Br)cc2c1NC(=O)CN1CCN(CC1)C(c1ccccc1)c1ccccc1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387756
PNG
(US10294214, Example 56)
Show SMILES O=C(CN1CCC(CC1)c1ccccc1)Nc1c(nc2ccccc12)C(=O)C1CCC1
PDB

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n/an/an/an/a 1.26E+3n/an/an/an/a



Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387768
PNG
(US10294214, Example 68)
Show SMILES O=C(CN1CCC2(CCCC2)CC1)Nc1c(nc2ccncc12)C(=O)C1CC1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387769
PNG
(US10294214, Example 69)
Show SMILES O=C(CN1CCC(CC1)c1ccccc1)Nc1c(nc2ccc(cc12)N1CCOCC1)C(=O)C1CC1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387772
PNG
(US10294214, Example 72)
Show SMILES CC(=O)c1nc2ccncc2c1NC(=O)CN1CCC(CC1)C(C)(C)C
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387780
PNG
(US10294214, Example 80)
Show SMILES COC(=O)c1nc2ccc(Cl)cc2c1NC(=O)CN1CCCC(C)(C)C1
PDB

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n/an/an/an/a 1.00E+3n/an/an/an/a



Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387702
PNG
(Synthesis of N-(2-(cyclopropanecarbonyl)-1H-indol-...)
Show SMILES O=C(CN1CCC2(CCCC2)CC1)Nc1c(nc2ccccc12)C(=O)C1CC1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387707
PNG
(US10294214, Example 7)
Show SMILES CC1(C)CCCN(CC(=O)Nc2c(nc3ccc(Br)cc23)C(=O)C2CC2)C1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387711
PNG
(US10294214, Example 11)
Show SMILES COC(=O)c1nc2ccccc2c1NC(=O)CN1CCC(CC1)c1ccccc1
PDB

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n/an/an/an/a 316n/an/an/an/a



Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387714
PNG
(US10294214, Example 14)
Show SMILES Brc1ccc2nc(C(=O)C3CC3)c(NC(=O)CN3CCN(Cc4ccccc4)CC3)c2c1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387721
PNG
(US10294214, Example 21)
Show SMILES COC(=O)c1nc2ccc(Cl)cc2c1NC(=O)CN1CCC(Cc2ccccc2)CC1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387737
PNG
(US10294214, Example 37)
Show SMILES O=C(CN1CCC(CC1)C1CCCCC1)Nc1c(nc2ccccc12)C(=O)C1CC1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387738
PNG
(US10294214, Example 38)
Show SMILES Clc1ccc2nc(C(=O)C3CC3)c(NC(=O)CN3CCC(CC3)C3CCCCC3)c2c1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387750
PNG
(US10294214, Example 50)
Show SMILES CC(C)=C1CCN(CC(=O)Nc2c(nc3ccccc23)C(=O)C2CC2)CC1
PDB

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n/an/an/an/a 794n/an/an/an/a



Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387751
PNG
(US10294214, Example 51)
Show SMILES CC(=O)c1nc2ccc(Br)cc2c1NC(=O)CN1CCCC(C)(C)C1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387752
PNG
(US10294214, Example 52)
Show SMILES CC(=O)c1nc2ccccc2c1NC(=O)CN1CCC(CC1)Oc1ccccc1
PDB

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n/an/an/an/a 1.26E+3n/an/an/an/a



Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387753
PNG
(US10294214, Example 53)
Show SMILES CC1(C)CCCN(CC(=O)Nc2c(nc3ccc(cc23)N2CCOCC2)C(=O)C2CC2)C1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387759
PNG
(US10294214, Example 59)
Show SMILES O=C(CN1CCC(CC1)C1CCCC1)Nc1c(nc2ccncc12)C(=O)C1CC1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387760
PNG
(US10294214, Example 60)
Show SMILES COC(=O)c1nc2ccc(cc2c1NC(=O)CN1CCC(CC1)C1CCCCC1)N1CCOCC1C
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387762
PNG
(US10294214, Example 62)
Show SMILES O=C(CN1CCC(CC1)C1CCCCC1)Nc1c(nc2ccncc12)C(=O)C1CC1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387773
PNG
(US10294214, Example 73)
Show SMILES O=C(CN1CCN(CC1)c1ccccc1)Nc1c(nc2ccncc12)C(=O)C1CC1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387703
PNG
(Synthesis of methyl 3-(2-(4-cyclohexylpiperidin-1-...)
Show SMILES COC(=O)c1nc2ccccc2c1NC(=O)CN1CCC(CC1)C1CCCCC1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387704
PNG
(US10294214, Example 4)
Show SMILES COC(=O)c1nc2ccc(Cl)cc2c1NC(=O)CN1CCC(CC1)c1ccccc1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387717
PNG
(US10294214, Example 17)
Show SMILES COC(=O)c1nc2ccc(Br)cc2c1NC(=O)CN1CCN(CC1)c1ccccc1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387725
PNG
(US10294214, Example 25)
Show SMILES COC(=O)c1nc2ccccc2c1NC(=O)CN1CCC(CC1)Oc1ccccc1
PDB

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n/an/an/an/a 1.00E+3n/an/an/an/a



Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387758
PNG
(US10294214, Example 58)
Show SMILES CS(=O)(=O)c1ccc2nc(C(=O)C3CC3)c(NC(=O)CN3CCC(CC3)C3CCCCC3)c2c1
PDB

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n/an/an/an/a 79.4n/an/an/an/a



Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387706
PNG
(US10294214, Example 6)
Show SMILES COC(=O)c1nc2cc(Br)ccc2c1NC(=O)CN1CCN(CC1)c1ccc(F)cc1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387713
PNG
(US10294214, Example 13)
Show SMILES COC(=O)c1nc2ccc(Br)cc2c1NC(=O)CN1CCN(C(C)C1)c1cccc(OC)c1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387716
PNG
(US10294214, Example 16)
Show SMILES O=C(CN1CCC(CC1)c1ccccc1)Nc1c(nc2ccccc12)C(=O)C1CC1
PDB

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US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387720
PNG
(US10294214, Example 20)
Show SMILES COC(=O)c1nc2ccc(Br)cc2c1NC(=O)C(C)N1CCC(Cc2ccccc2)CC1
PDB

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US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387727
PNG
(US10294214, Example 27)
Show SMILES COC(=O)c1nc2ccc(C)cc2c1NC(=O)CN1CCN(CC1)c1cccc(C)c1C
PDB

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US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387741
PNG
(US10294214, Example 41)
Show SMILES O=C(CN1CCC(CC1)C1CCCC1)Nc1c(nc2ccccc12)C(=O)C1CC1
PDB

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US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387754
PNG
(US10294214, Example 54)
Show SMILES O=C(CN1CCC(CC1)C1CC1)Nc1c(nc2ccccc12)C(=O)C1CC1
PDB

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US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387755
PNG
(US10294214, Example 55)
Show SMILES COC(=O)c1nc2ccccc2c1NC(=O)CN1CCC(CC1)Nc1ccccc1
PDB

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US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387763
PNG
(US10294214, Example 63)
Show SMILES Clc1ccc2nc(C(=O)C3CC3)c(NC(=O)CN3CCC(CC3)C3CCCC3)c2c1
PDB

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US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387775
PNG
(US10294214, Example 75)
Show SMILES COC(=O)c1nc2ccc(C)cc2c1NC(=O)CN1CCC(Cc2ccccc2)CC1
PDB

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US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387705
PNG
(US10294214, Example 5)
Show SMILES COC(=O)c1nc2ccc(Br)cc2c1NC(=O)CN1CCN(CC1)c1cccc(C)c1C
PDB

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US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387723
PNG
(US10294214, Example 23)
Show SMILES CC1(C)CCCN(CC(=O)Nc2c(nc3ccccc23)C(=O)C2CC2)C1
PDB

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US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387730
PNG
(US10294214, Example 30)
Show SMILES COC(=O)c1nc2ccccc2c1NC(=O)C(C)N1CCC(Cc2ccccc2)CC1
PDB

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US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387734
PNG
(US10294214, Example 34)
Show SMILES CCOC(=O)c1nc2ncccc2c1NC(=O)CN1CCCC(C)(C)C1
Show InChI InChI=1S/C19H25N4O3/c1-4-26-18(25)16-15(13-7-5-9-20-17(13)22-16)21-14(24)11-23-10-6-8-19(2,3)12-23/h5,7,9H,4,6,8,10-12H2,1-3H3,(H,21,24)
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387742
PNG
(US10294214, Example 42)
Show SMILES CC(=O)c1nc2ccccc2c1NC(=O)CN1CCC(CC1)C1CCCCC1
PDB

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US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387745
PNG
(US10294214, Example 45)
Show SMILES COC(=O)c1nc2ccccc2c1NC(=O)CN1CCC(CC1)N(C)c1ccccc1
PDB

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US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387757
PNG
(US10294214, Example 57)
Show SMILES COC(=O)c1nc2ccccc2c1NC(=O)CN1CCN(Cc2ccccc2)C(C)(C)C1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387761
PNG
(US10294214, Example 61)
Show SMILES COC(=O)c1nc2ccc(cc2c1NC(=O)CN1CCC(CC1)C1CCCCC1)N1CCOCC1
PDB

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US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387770
PNG
(US10294214, Example 70)
Show SMILES CC(N1CCC(CC1)C1CCCC1)C(=O)Nc1c(nc2ccccc12)C(C)=O
PDB

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US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387774
PNG
(US10294214, Example 74)
Show SMILES CC1(C)CCCN(CC(=O)Nc2c(nc3ccncc23)C(=O)C2CC2)C1
PDB

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US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387708
PNG
(US10294214, Example 8)
Show SMILES Brc1ccc2nc(C(=O)C3CC3)c(NC(=O)CN3CCC(CC3)c3ccccc3)c2c1
PDB

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US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387710
PNG
(US10294214, Example 10)
Show SMILES Cc1cccc(N2CCN(CC(=O)Nc3c(nc4ccccc34)C(=O)C3CC3)CC2)c1C
PDB

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US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387715
PNG
(US10294214, Example 15)
Show SMILES COC(=O)c1nc2ccc(Cl)cc2c1NC(=O)CN1CCN(CC1)c1ccccc1
PDB

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US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387718
PNG
(US10294214, Example 18)
Show SMILES CC(=O)c1nc2ccccc2c1NC(=O)CN1CCC(Cc2ccccc2)CC1
PDB

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US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387726
PNG
(US10294214, Example 26)
Show SMILES COC(=O)c1nc2ccc(Br)cc2c1NC(=O)CN1CCCCC1
PDB

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US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387744
PNG
(US10294214, Example 44)
Show SMILES CC(=O)c1nc2ccc(Br)cc2c1NC(=O)CN1CCC(Cc2ccccc2)CC1
PDB

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US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387748
PNG
(US10294214, Example 48)
Show SMILES CC1(C)CCCN(CC(=O)Nc2c(nc3ccc(cc23)S(C)(=O)=O)C(=O)C2CC2)C1
PDB

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US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387767
PNG
(US10294214, Example 67)
Show SMILES O=C(CN1CCC(CC1)c1ccccc1)Nc1c(nc2ccncc12)C(=O)C1CC1
PDB

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US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387778
PNG
(US10294214, Example 78)
Show SMILES COC(=O)c1nc2ccc(Cl)cc2c1NC(=O)C(C)N1CCC(Cc2ccccc2)CC1
PDB

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US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387709
PNG
(US10294214, Example 9)
Show SMILES Cc1cccc(N2CCN(CC(=O)Nc3c(nc4ccc(Br)cc34)C(=O)C3CC3)CC2)c1C
PDB

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US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387719
PNG
(US10294214, Example 19)
Show SMILES CC(=O)c1nc2ccccc2c1NC(=O)CN1CCC(CC1)c1ccccc1
PDB

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US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387729
PNG
(US10294214, Example 29)
Show SMILES COC(=O)c1nc2ccccc2c1NC(=O)CN1CCCC2(CCC2)C1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387731
PNG
(US10294214, Example 31)
Show SMILES COC(=O)c1nc2ccc(C)cc2c1NC(=O)CN1CCN(C(C)C1)c1cccc(OC)c1
PDB

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US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387740
PNG
(US10294214, Example 40)
Show SMILES CC(=O)c1nc2ccccc2c1NC(=O)CN1CCC(CC1)C1CCCC1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387764
PNG
(US10294214, Example 64)
Show SMILES CC(=O)c1nc2ccncc2c1NC(=O)CN1CCC(CC1)C1CCCC1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387765
PNG
(US10294214, Example 65)
Show SMILES O=C(CN1CCC2(CCCCC2)CC1)Nc1c(nc2ccccc12)C(=O)C1CC1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387766
PNG
(US10294214, Example 66)
Show SMILES O=C(CN1CCC(CC1)C1CCCCC1)Nc1c(nc2ccc(cc12)N1CCOCC1)C(=O)C1CC1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387776
PNG
(US10294214, Example 76)
Show SMILES CC1COCCN1c1ccc2nc(C(=O)C3CC3)c(NC(=O)CN3CCCC(C)(C)C3)c2c1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387777
PNG
(US10294214, Example 77)
Show SMILES CC(=O)c1nc2ccccc2c1NC(=O)CN1CCC(CC1)OC1CCCCC1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387701
PNG
(Synthesis of 2-(4-(tert-butyl)piperidin-1-yl)-N-(2...)
Show SMILES CC(C)(C)C1CCN(CC(=O)Nc2c(nc3ccccc23)C(=O)C2CC2)CC1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387712
PNG
(US10294214, Example 12)
Show SMILES COC(=O)c1nc2ccccc2c1NC(=O)CN1CCN(CC1)c1cccc(c1)C(F)(F)F
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387722
PNG
(US10294214, Example 22)
Show SMILES COC(=O)c1nc2ccc(Br)cc2c1NC(=O)CN1CCC(Cc2ccccc2)CC1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387724
PNG
(US10294214, Example 24)
Show SMILES COC(=O)c1nc2ccccc2c1NC(=O)CN1CCC(Cc2ccccc2)CC1
PDB

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n/an/an/an/a 1.00E+3n/an/an/an/a



Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387728
PNG
(US10294214, Example 28)
Show SMILES CCOC(=O)c1nc2ccncc2c1NC(=O)CN1CCCC(C)(C)C1
PDB

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n/an/an/an/a 1.59E+3n/an/an/an/a



Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387732
PNG
(US10294214, Example 32)
Show SMILES COC(=O)c1nc2ccccc2c1NC(=O)CN1CCC(CC1)Oc1ccccn1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387736
PNG
(US10294214, Example 36)
Show SMILES COC(=O)c1nc2ccc(Br)cc2c1NC(=O)CN1CCSCC1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387739
PNG
(US10294214, Example 39)
Show SMILES COC(=O)c1nc2ccc(Br)cc2c1NC(=O)CN1CCC(CC1)c1ccccc1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387746
PNG
(US10294214, Example 46)
Show SMILES COC(=O)c1nc2ccc(Br)cc2c1NC(=O)CN1CCN(CC1)C1c2ccccc2-c2ccccc12
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387749
PNG
(US10294214, Example 49)
Show SMILES COC(=O)c1nc2ccccc2c1NC(=O)CN1CCC(CC1)N1CCc2ccccc12
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387771
PNG
(US10294214, Example 71)
Show SMILES CC(N1CCC(CC1)C1CCCC1)C(=O)Nc1c(nc2ccccc12)C(=O)C1CC1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM387779
PNG
(US10294214, Example 79)
Show SMILES COC(=O)c1nc2ccc(Br)cc2c1NC(=O)CN1CCCC(C)(C)C1
PDB

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Vanderbilt University

US Patent


Assay Description
Analysis of pharmacological properties of compounds was performed using the LANCE cAMP kit (Perkin Elmer). HEK293 cells stably expressing the hMC4R w...

US Patent US10294214 (2019)


BindingDB Entry DOI: 10.7270/Q20V8G3D
More data for this
Ligand-Target Pair
* indicates data uncertainty>20%