Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 3013
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Tianjin Institute Of Pharmaceutical Research

US Patent
LigandPNGBDBM254941(US10294259, Compound Table 3.2 | US9505734, I-D1-6)
Affinity DataIC50:  0.670nMAssay Description:IC50 values of inhibition of some compounds described in the present invention and related compounds on SGLT2 and SGLT1 are determined according to t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Tianjin Institute Of Pharmaceutical Research

US Patent
LigandPNGBDBM388440(US10294259, Compound Table 3.1)
Affinity DataIC50:  3.30nMAssay Description:IC50 values of inhibition of some compounds described in the present invention and related compounds on SGLT2 and SGLT1 are determined according to t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Tianjin Institute Of Pharmaceutical Research

US Patent
LigandPNGBDBM388442(US10294259, Compound Table 3.3)
Affinity DataIC50:  7.80nMAssay Description:IC50 values of inhibition of some compounds described in the present invention and related compounds on SGLT2 and SGLT1 are determined according to t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Tianjin Institute Of Pharmaceutical Research

US Patent
LigandPNGBDBM388440(US10294259, Compound Table 3.1)
Affinity DataIC50:  86nMAssay Description:IC50 values of inhibition of some compounds described in the present invention and related compounds on SGLT2 and SGLT1 are determined according to t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Tianjin Institute Of Pharmaceutical Research

US Patent
LigandPNGBDBM388442(US10294259, Compound Table 3.3)
Affinity DataIC50:  187nMAssay Description:IC50 values of inhibition of some compounds described in the present invention and related compounds on SGLT2 and SGLT1 are determined according to t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Tianjin Institute Of Pharmaceutical Research

US Patent
LigandPNGBDBM254941(US10294259, Compound Table 3.2 | US9505734, I-D1-6)
Affinity DataIC50:  251nMAssay Description:IC50 values of inhibition of some compounds described in the present invention and related compounds on SGLT2 and SGLT1 are determined according to t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent