Compile Data Set for Download or QSAR
maximum 50k data
Found 48 Enz. Inhib. hit(s) with all data for entry = 3382
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266536(CHEMBL4085664 | US10323016, Example 1)
Affinity DataEC50:  156nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Mus musculus)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398287(US10323016, Example 26)
Affinity DataEC50:  0.5nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266574(CHEMBL4081298 | US10323016, Example 2)
Affinity DataEC50:  299nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Mus musculus)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266574(CHEMBL4081298 | US10323016, Example 2)
Affinity DataEC50:  44nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266537(CHEMBL4075688 | US10323016, Example 3)
Affinity DataEC50:  128nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Mus musculus)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266537(CHEMBL4075688 | US10323016, Example 3)
Affinity DataEC50:  12nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266538(CHEMBL4084668 | US10323016, Example 4)
Affinity DataEC50:  39nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Mus musculus)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266538(CHEMBL4084668 | US10323016, Example 4)
Affinity DataEC50:  1nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266556(CHEMBL4073081 | US10323016, Example 5)
Affinity DataEC50:  880nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Mus musculus)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266556(CHEMBL4073081 | US10323016, Example 5)
Affinity DataEC50:  44nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266560(CHEMBL4104359 | US10323016, Example 6)
Affinity DataEC50:  71nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Mus musculus)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266560(CHEMBL4104359 | US10323016, Example 6)
Affinity DataEC50:  4nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398270(US10323016, Example 7)
Affinity DataEC50:  177nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Mus musculus)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398270(US10323016, Example 7)
Affinity DataEC50:  7nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398271(US10323016, Example 8)
Affinity DataEC50:  260nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Mus musculus)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398271(US10323016, Example 8)
Affinity DataEC50:  17nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398272(US10323016, Example 22 | US10323016, Example 24 | ...)
Affinity DataEC50:  160nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Mus musculus)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398272(US10323016, Example 22 | US10323016, Example 24 | ...)
Affinity DataEC50:  18nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266540(CHEMBL4102610 | US10323016, Example 12)
Affinity DataEC50:  4.30E+3nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Mus musculus)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266540(CHEMBL4102610 | US10323016, Example 12)
Affinity DataEC50:  180nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266573(CHEMBL4104779 | US10323016, Example 13)
Affinity DataEC50:  250nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Mus musculus)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266573(CHEMBL4104779 | US10323016, Example 13)
Affinity DataEC50:  5nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266575(CHEMBL4085777 | US10323016, Example 14)
Affinity DataEC50:  7.70E+3nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Mus musculus)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266575(CHEMBL4085777 | US10323016, Example 14)
Affinity DataEC50:  940nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266572(CHEMBL4060122 | US10323016, Example 15)
Affinity DataEC50:  900nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Mus musculus)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266572(CHEMBL4060122 | US10323016, Example 15)
Affinity DataEC50:  370nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266557(CHEMBL4063932 | US10323016, Example 16)
Affinity DataEC50:  990nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Mus musculus)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266557(CHEMBL4063932 | US10323016, Example 16)
Affinity DataEC50:  90nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266565(CHEMBL4091702 | US10323016, Example 17)
Affinity DataEC50:  1.10E+3nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Mus musculus)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266565(CHEMBL4091702 | US10323016, Example 17)
Affinity DataEC50:  140nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266558(CHEMBL4088938 | US10323016, Example 18)
Affinity DataEC50:  750nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Mus musculus)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266558(CHEMBL4088938 | US10323016, Example 18)
Affinity DataEC50:  510nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266566(CHEMBL4068227 | US10323016, Example 19)
Affinity DataEC50:  47nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Mus musculus)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266566(CHEMBL4068227 | US10323016, Example 19)
Affinity DataEC50:  4.80nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266552(CHEMBL4094487 | US10323016, Example 20)
Affinity DataEC50:  15nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Mus musculus)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266552(CHEMBL4094487 | US10323016, Example 20)
Affinity DataEC50:  1nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266567(CHEMBL4090147 | US10323016, Example 21)
Affinity DataEC50:  35nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Mus musculus)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266567(CHEMBL4090147 | US10323016, Example 21)
Affinity DataEC50:  2nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398283(US10323016, Example 22)
Affinity DataEC50:  580nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Mus musculus)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398283(US10323016, Example 22)
Affinity DataEC50:  29nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398284(US10323016, Example 23)
Affinity DataEC50:  330nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Mus musculus)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398284(US10323016, Example 23)
Affinity DataEC50:  26nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398285(US10323016, Example 24)
Affinity DataEC50:  1.20E+3nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Mus musculus)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398285(US10323016, Example 24)
Affinity DataEC50:  68nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398286(US10323016, Example 25)
Affinity DataEC50:  240nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Mus musculus)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398286(US10323016, Example 25)
Affinity DataEC50:  10nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398287(US10323016, Example 26)
Affinity DataEC50:  40nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Mus musculus)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266536(CHEMBL4085664 | US10323016, Example 1)
Affinity DataEC50:  68nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In DepthDetails US Patent