Compile Data Set for Download or QSAR
maximum 50k data
Found 118 Enz. Inhib. hit(s) with all data for entry = 8753
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390012(4-amino-1-[(3R)-1-[(E)-4- (dimethylamino)but-2-eno...)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390001(US10323037, Example 18 | US9951077, 18)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390014(4-amino-1-[(3R)-1-[(E)-4- (cyclopropylamino)but-2-...)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390018(4-amino-1-[(3R)-1-[(E)-4- [cyclobutyl(methyl)amino...)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390020(4-amino-1-[(3R)-1-[(E)-4-(azetidin- 1-yl)but-2-eno...)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390021(4-amino-3-(4-phenoxyphenyl)-1- [(3R)-1-[(E)-4-pyrr...)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390022(4-amino-1-[(3R)-1-[(E)-4- morpholinobut-2-enoyl]-3...)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390023(4-amino-1-[(3R)-1-[(E)-4-(4- methylpiperazin-1-yl)...)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390025(4-amino-1-[1-[(E)-4- (dimethylamino)but-2-enoyl]-3...)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390026(4-amino-1-[(3R)-1-[(E)-4- (dimethylamino)but-2- en...)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390032(4-amino-1-[1-[(E)-4- (dimethylamino)but-2-enoyl]-4...)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390034(4-amino-1-[[1-[(E)-4- (dimethylamino)but-2- enoyl]...)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390038(US10323037, Example 51 | US9951077, 51)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390039(US10323037, Example 52 | US9951077, 52)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390040(US10323037, Example 53 | US9951077, 53)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390041(US10323037, Example 54 | US9951077, 54)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390042(US10323037, Example 55 | US9951077, 55)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390043(US10323037, Example 56 | US9951077, 56)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390044(US10323037, Example 57 | US9951077, 57)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM416771((R)-1-(1-acryloylpiperidin-3-yl)-4-amino-3-(4-(2,6...)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390050(US10323037, Example 63 | US9951077, 63)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390054(US10323037, Example 67 | US9951077, 67)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390056(US10323037, Example 69 | US9951077, 69)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390058(US10323037, Example 71 | US9951077, 71)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390062(US10323037, Example 75 | US9951077, 75)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390064(US10323037, Example 77 | US9951077, 77)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390065(US10323037, Example 78 | US9951077, 78)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390066(US10323037, Example 79 | US9951077, 79)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390069(US10323037, Example 82 | US9951077, 82)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390074(US10323037, Example 87 | US9951077, 87)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM416801(N-(3-(4-amino-7-oxo-3-(4-phenoxyphenyl)-6,7-dihydr...)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390087(US10323037, Example 99 | US9951077, 99)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390095(US10323037, Example 107 | US9951077, 107)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390096(US10323037, Example 108 | US9951077, 108)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM416824((R)-4-amino-1-(1-(but-2-ynoyl)pyrrolidin-3-yl)-3-(...)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM416714((R)-1-(1-acryloylpiperidin-3-yl)-4-amino-3-(4-phen...)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM416715(4-amino-3-(4-phenoxyphenyl)-1-(1- prop-2-enoyl-3-p...)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM416726(1-(1-acryloyl-4-fluoropiperidin-3-yl)-4-amino-3-(4...)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM416727((R)-1-(1-acryloyl-5,5-difluoropiperidin-3-yl)-4-am...)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM389999(US10323037, Example 16 | US9951077, 16)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390013(4-amino-1-[(3R)-1-[(E)-4- (diethylamino)but-2-enoy...)
Affinity DataIC50: <10nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390005(4-amino-1-[(3R)-1-(2-chloroacetyl)- 3-piperidyl]-3...)
Affinity DataIC50:  505nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390006(4-amino-1-[(3R)-1- (cyclopropanecarbonyl)-3- piper...)
Affinity DataIC50:  505nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390007(3-[(3R)-3-[4-amino-7-oxo-3-(4- phenoxyphenyl)-6H-p...)
Affinity DataIC50:  505nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390008(4-amino-1-[(3R)-1-[(E)-but-2- enoyl]-3-piperidyl]-...)
Affinity DataIC50:  505nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390016(4-amino-1-[(3R)-1-[(E)-4- (cyclopropyl(methyl)amin...)
Affinity DataIC50:  505nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390017(4-amino-1-[(3R)-1-[(E)-4- [cyclopropyl(ethyl)amino...)
Affinity DataIC50:  505nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390019(4-amino-1-[(3R)-1-[(E)-4- [cyclohexyl(methyl)amino...)
Affinity DataIC50:  505nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390027(4-amino-1-[1-[(E)-4- (dimethylamino)but-2- enoyl]a...)
Affinity DataIC50:  505nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Jiangsu Hengrui Medicine

US Patent
LigandPNGBDBM390028(4-amino-1-[[(2S)-1-[(E)-4- (dimethylamino)but-2- e...)
Affinity DataIC50:  505nMAssay Description:The Btk kinase assay was performed using a ADP-Glo Btk kinase assay kit purchased from Promega (Madison, Wis.). The assay was conducted according to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Displayed 1 to 50 (of 118 total ) | Next | Last >>
Jump to: