Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403299![]() (US10329307, Example 46) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 240 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403270![]() (US10329307, Example 17) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 290 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403298![]() (US10329307, Example 45) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 370 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403263![]() (US10329307, Example 10) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 390 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403265![]() (US10329307, Example 12) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 420 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403254![]() (US10329307, Example 1) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 420 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403286![]() (US10329307, Example 33) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 440 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403275![]() (US10329307, Example 22) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 440 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403272![]() (US10329307, Example 19) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 460 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403271![]() (US10329307, Example 18) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 470 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403296![]() (US10329307, Example 43) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 480 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403269![]() (US10329307, Example 16) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 500 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403292![]() (US10329307, Example 39) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 510 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403291![]() (US10329307, Example 38) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 540 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403274![]() (US10329307, Example 21) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 540 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403266![]() (US10329307, Example 13) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 550 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403290![]() (US10329307, Example 37) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 560 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403276![]() (US10329307, Example 23) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 600 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403287![]() (US10329307, Example 34) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 700 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403273![]() (US10329307, Example 20) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 710 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403308![]() (US10329307, Example 55 | US10329307, Example 56 | ...) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 720 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403308![]() (US10329307, Example 55 | US10329307, Example 56 | ...) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 740 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403264![]() (US10329307, Example 11) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 740 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403297![]() (US10329307, Example 44) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 750 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403289![]() (US10329307, Example 36) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 750 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403278![]() (US10329307, Example 25) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 790 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403316![]() (US10329307, Example 63 | US10329307, Example 64 | ...) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 820 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403288![]() (US10329307, Example 35) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 840 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403283![]() (US10329307, Example 30) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 860 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403316![]() (US10329307, Example 63 | US10329307, Example 64 | ...) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 860 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403284![]() (US10329307, Example 31) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 890 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403308![]() (US10329307, Example 55 | US10329307, Example 56 | ...) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 920 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403262![]() (US10329307, Example 9) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 950 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403282![]() (US10329307, Example 29) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 950 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403277![]() (US10329307, Example 24) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 950 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403300![]() (US10329307, Example 47) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403316![]() (US10329307, Example 63 | US10329307, Example 64 | ...) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403305![]() (US10329307, Example 52) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403295![]() (US10329307, Example 42) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403301![]() (US10329307, Example 48) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403256![]() (US10329307, Example 3) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403312![]() (US10329307, Example 59) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403324![]() (US10329307, Example 71) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403268![]() (US10329307, Example 15) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403293![]() (US10329307, Example 40) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403319![]() (US10329307, Example 66) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403311![]() (US10329307, Example 58) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403325![]() (US10329307, Example 72) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403279![]() (US10329307, Example 26) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403307![]() (US10329307, Example 54) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403261![]() (US10329307, Example 8) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403314![]() (US10329307, Example 61) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403306![]() (US10329307, Example 53) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403281![]() (US10329307, Example 28) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403315![]() (US10329307, Example 62) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403321![]() (US10329307, Example 68) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 2.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403294![]() (US10329307, Example 41) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 2.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403280![]() (US10329307, Example 27) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403313![]() (US10329307, Example 60) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 2.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403302![]() (US10329307, Example 49) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 2.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403285![]() (US10329307, Example 32) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 2.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403322![]() (US10329307, Example 69) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403320![]() (US10329307, Example 67) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403323![]() (US10329307, Example 70) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403303![]() (US10329307, Example 50) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 4.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403304![]() (US10329307, Example 51) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403255![]() (US10329307, Example 2) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 9.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403267![]() (US10329307, Example 14) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403259![]() (US10329307, Example 6) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403260![]() (US10329307, Example 7) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403258![]() (US10329307, Example 5) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 2.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403327![]() (US10329307, Example 74) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 2.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403326![]() (US10329307, Example 73) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 4.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PRKC apoptosis WT1 regulator protein (Homo sapiens (Human)) | BDBM403257![]() (US10329307, Example 4) | MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 4.60E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Universite de Montreal US Patent | Assay Description FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th... | US Patent US10329307 (2019) BindingDB Entry DOI: 10.7270/Q26975XD | |||||||||||
More data for this Ligand-Target Pair |