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Found 6 Enz. Inhib. hit(s) with all data for entry = 8636
LigandPNGBDBM409778(2-oxo-4-[3- (pyridin-3-yl) pyrrolidin-1- yl]-1,2- ...)
Affinity DataKi:  3.40nMAssay Description:The fluorescence polarization assay for cyclic nucleotide phosphodiesterases was performed using an IMAP® FP kit supplied by Molecular Devices, Sunny...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM409949(4-(2-fluoro- 4-methyl- phenyl)-2- oxo-1H- quinolin...)
Affinity DataKi:  7.20nMAssay Description:The fluorescence polarization assay for cyclic nucleotide phosphodiesterases was performed using an IMAP® FP kit supplied by Molecular Devices, Sunny...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM409781(2-oxo-4- (p-tolyl)-1H- quinoline-3- carbonitrile |...)
Affinity DataKi:  8.90nMAssay Description:The fluorescence polarization assay for cyclic nucleotide phosphodiesterases was performed using an IMAP® FP kit supplied by Molecular Devices, Sunny...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM409783(4-(2-naphthyl)- 2-oxo-1H- quinoline-3- carbonitril...)
Affinity DataKi:  14.8nMAssay Description:The fluorescence polarization assay for cyclic nucleotide phosphodiesterases was performed using an IMAP® FP kit supplied by Molecular Devices, Sunny...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM409774(US10370336, Example 1-14 | US10370336, Example 1-7)
Affinity DataKi:  66nMAssay Description:The fluorescence polarization assay for cyclic nucleotide phosphodiesterases was performed using an IMAP® FP kit supplied by Molecular Devices, Sunny...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM409774(US10370336, Example 1-14 | US10370336, Example 1-7)
Affinity DataKi:  444nMAssay Description:The fluorescence polarization assay for cyclic nucleotide phosphodiesterases was performed using an IMAP® FP kit supplied by Molecular Devices, Sunny...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent