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| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Equilibrative nucleoside transporter 1 (Mus musculus (Mouse)) | BDBM409054 (3,3-Dimethyl-6-(2-methylpyrimidin-5-yl)-1-(5-(meth...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 27 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well... | US Patent US10377746 (2019) BindingDB Entry DOI: 10.7270/Q2H997JV | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Equilibrative nucleoside transporter 1 (Mus musculus (Mouse)) | BDBM409053 (6-(5-Fluoro-6-methylpyridin-3-yl)-3,3-dimethyl-1-(...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 27 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well... | US Patent US10377746 (2019) BindingDB Entry DOI: 10.7270/Q2H997JV | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Equilibrative nucleoside transporter 1 (Mus musculus (Mouse)) | BDBM409033 (3,3-Dimethyl-6-(2-methylpyrimidin-5-yl)-1-(5-(meth...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 32.1 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well... | US Patent US10377746 (2019) BindingDB Entry DOI: 10.7270/Q2H997JV | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Equilibrative nucleoside transporter 1 (Mus musculus (Mouse)) | BDBM409050 (1-(6-Cyclopropyl-5-(methylsulfonyl)pyridin-3-yl)-3...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 38.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well... | US Patent US10377746 (2019) BindingDB Entry DOI: 10.7270/Q2H997JV | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Equilibrative nucleoside transporter 1 (Mus musculus (Mouse)) | BDBM409044 (1-(5-(Cyclopropylsulfonyl)pyridin-3-yl)-3,3-dimeth...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well... | US Patent US10377746 (2019) BindingDB Entry DOI: 10.7270/Q2H997JV | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Equilibrative nucleoside transporter 1 (Mus musculus (Mouse)) | BDBM409034 (3,3-Dimethyl-6-(2-methylpyrimidin-5-yl)-1-(6-(meth...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 40.1 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well... | US Patent US10377746 (2019) BindingDB Entry DOI: 10.7270/Q2H997JV | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Equilibrative nucleoside transporter 1 (Mus musculus (Mouse)) | BDBM409037 (5-(3,3-Dimethyl-6-(2-methylpyrimidin-5-yl)-2-oxoin...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 44.9 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well... | US Patent US10377746 (2019) BindingDB Entry DOI: 10.7270/Q2H997JV | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Equilibrative nucleoside transporter 1 (Mus musculus (Mouse)) | BDBM409049 (5-(3,3-Dimethyl-6-(2-methylpyrimidin-5-yl)-2-oxoin...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 71.7 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well... | US Patent US10377746 (2019) BindingDB Entry DOI: 10.7270/Q2H997JV | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Equilibrative nucleoside transporter 1 (Mus musculus (Mouse)) | BDBM409048 (5-(3,3-dimethyl-6-(2-methylpyrimidin-5-yl)-2-oxoin...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 79.3 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well... | US Patent US10377746 (2019) BindingDB Entry DOI: 10.7270/Q2H997JV | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Equilibrative nucleoside transporter 1 (Mus musculus (Mouse)) | BDBM409035 (3,3-Dimethyl-6-(2-methylpyrimidin-5-yl)-1-(3-(meth...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 106 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well... | US Patent US10377746 (2019) BindingDB Entry DOI: 10.7270/Q2H997JV | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Equilibrative nucleoside transporter 1 (Mus musculus (Mouse)) | BDBM409046 (5-(3,3-Dimethyl-6-(2-methylpyrimidin-5-yl)-2-oxoin...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 128 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well... | US Patent US10377746 (2019) BindingDB Entry DOI: 10.7270/Q2H997JV | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Equilibrative nucleoside transporter 1 (Mus musculus (Mouse)) | BDBM409043 (1-(5-(Isopropylsulfonyl)pyridin-3-yl)-3,3-dimethyl...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 135 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well... | US Patent US10377746 (2019) BindingDB Entry DOI: 10.7270/Q2H997JV | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Equilibrative nucleoside transporter 1 (Mus musculus (Mouse)) | BDBM409055 (3,3-Dimethyl-6-(2-methylpyrimidin-5-yl)-1-(5-(meth...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 157 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well... | US Patent US10377746 (2019) BindingDB Entry DOI: 10.7270/Q2H997JV | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Equilibrative nucleoside transporter 1 (Mus musculus (Mouse)) | BDBM409047 (1-(5-(Azetidin-1-ylsulfonyl)pyridin-3-yl)-3,3-dime...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 169 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well... | US Patent US10377746 (2019) BindingDB Entry DOI: 10.7270/Q2H997JV | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Equilibrative nucleoside transporter 1 (Mus musculus (Mouse)) | BDBM409031 (1-(Benzo[b]thiophen-6-yl)-3,3-dimethyl-6-(2-methyl...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 189 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well... | US Patent US10377746 (2019) BindingDB Entry DOI: 10.7270/Q2H997JV | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Equilibrative nucleoside transporter 1 (Mus musculus (Mouse)) | BDBM409051 (3,3-Dimethyl-6-(2-methyl-1-oxidopyrimidin-1-ium-5-...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 218 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well... | US Patent US10377746 (2019) BindingDB Entry DOI: 10.7270/Q2H997JV | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Equilibrative nucleoside transporter 1 (Mus musculus (Mouse)) | BDBM409045 (3,3-Dimethyl-6-(2-methylpyrimidin-5-yl)-1-(5-(meth...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 218 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well... | US Patent US10377746 (2019) BindingDB Entry DOI: 10.7270/Q2H997JV | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Equilibrative nucleoside transporter 1 (Mus musculus (Mouse)) | BDBM409056 (6'-(2-Methylpyrimidin-5-yl)-1'-(5-(methylsulfonyl)...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 230 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well... | US Patent US10377746 (2019) BindingDB Entry DOI: 10.7270/Q2H997JV | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Equilibrative nucleoside transporter 1 (Mus musculus (Mouse)) | BDBM409052 (3,3-Dimethyl-6-(5-methylpyridin-3-yl)-1-(5-(methyl...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 313 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well... | US Patent US10377746 (2019) BindingDB Entry DOI: 10.7270/Q2H997JV | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Equilibrative nucleoside transporter 1 (Mus musculus (Mouse)) | BDBM409032 (1-(Benzo[b]thiophen-4-yl)-3,3-dimethyl-6-(2-methyl...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | 844 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well... | US Patent US10377746 (2019) BindingDB Entry DOI: 10.7270/Q2H997JV | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
