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Patent code US10464907

Compile Data Set for Download or QSAR
Found 29 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Heat shock protein HSP 90-alpha


(Bovine)
BDBM50464556
PNG
(CHEMBL4289811 | US10464907, Compound 21f)
Show SMILES CCCNC(=O)c1ccc(CN(C)C(=O)c2cc(C(C)C)c(O)cc2O)cc1
Show InChI InChI=1S/C22H28N2O4/c1-5-10-23-21(27)16-8-6-15(7-9-16)13-24(4)22(28)18-11-17(14(2)3)19(25)12-20(18)26/h6-9,11-12,14,25-26H,5,10,13H2,1-4H3,(H,23,27)
PDB

UniProtKB/SwissProt

GoogleScholar
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US Patent
n/an/a 5.30n/an/an/an/an/an/a



INDUSTRY ACADEMIC COOPERATION FOUNDATION KEIMYUNG UNIVERSITY

US Patent


Assay Description
Fluorescence polarization assay was performed to confirm the binding ability to the compound synthesized with HSP90 according the concentration. 1 M ...


US Patent US10464907 (2019)

More data for this
Ligand-Target Pair
Heat shock protein HSP 90-alpha


(Bovine)
BDBM50464557
PNG
(CHEMBL4279132 | US10464907, Compound 21e)
Show SMILES CCNC(=O)c1ccc(CN(C)C(=O)c2cc(C(C)C)c(O)cc2O)cc1
Show InChI InChI=1S/C21H26N2O4/c1-5-22-20(26)15-8-6-14(7-9-15)12-23(4)21(27)17-10-16(13(2)3)18(24)11-19(17)25/h6-11,13,24-25H,5,12H2,1-4H3,(H,22,26)
PDB

UniProtKB/SwissProt

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US Patent
n/an/a 6.5n/an/an/an/an/an/a



INDUSTRY ACADEMIC COOPERATION FOUNDATION KEIMYUNG UNIVERSITY

US Patent


Assay Description
Fluorescence polarization assay was performed to confirm the binding ability to the compound synthesized with HSP90 according the concentration. 1 M ...


US Patent US10464907 (2019)

More data for this
Ligand-Target Pair
Heat shock protein HSP 90-alpha


(Bovine)
BDBM50464562
PNG
(CHEMBL4293186 | US10464907, Compound 21d)
Show SMILES CNC(=O)c1ccc(CN(C)C(=O)c2cc(C(C)C)c(O)cc2O)cc1
Show InChI InChI=1S/C20H24N2O4/c1-12(2)15-9-16(18(24)10-17(15)23)20(26)22(4)11-13-5-7-14(8-6-13)19(25)21-3/h5-10,12,23-24H,11H2,1-4H3,(H,21,25)
PDB

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US Patent
n/an/a 11.4n/an/an/an/an/an/a



INDUSTRY ACADEMIC COOPERATION FOUNDATION KEIMYUNG UNIVERSITY

US Patent


Assay Description
Fluorescence polarization assay was performed to confirm the binding ability to the compound synthesized with HSP90 according the concentration. 1 M ...


US Patent US10464907 (2019)

More data for this
Ligand-Target Pair
Heat shock protein HSP 90-alpha


(Bovine)
BDBM419585
PNG
(US10464907, Compound 21g)
Show SMILES CC(C)c1cc(C(=O)N(C)Cc2ccccc2)c(O)cc1O
Show InChI InChI=1S/C18H21NO3/c1-12(2)14-9-15(17(21)10-16(14)20)18(22)19(3)11-13-7-5-4-6-8-13/h4-10,12,20-21H,11H2,1-3H3
PDB

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US Patent
n/an/a 33n/an/an/an/an/an/a



INDUSTRY ACADEMIC COOPERATION FOUNDATION KEIMYUNG UNIVERSITY

US Patent


Assay Description
Fluorescence polarization assay was performed to confirm the binding ability to the compound synthesized with HSP90 according the concentration. 1 M ...


US Patent US10464907 (2019)

More data for this
Ligand-Target Pair
Heat shock protein HSP 90-alpha


(Bovine)
BDBM419586
PNG
(US10464907, Compound 17)
Show SMILES CC(C)c1cc(C(=O)N2CCN(C)CC2c2ccccc2)c(O)cc1O
Show InChI InChI=1/C21H26N2O3/c1-14(2)16-11-17(20(25)12-19(16)24)21(26)23-10-9-22(3)13-18(23)15-7-5-4-6-8-15/h4-8,11-12,14,18,24-25H,9-10,13H2,1-3H3
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US Patent
n/an/a 49.5n/an/an/an/an/an/a



INDUSTRY ACADEMIC COOPERATION FOUNDATION KEIMYUNG UNIVERSITY

US Patent


Assay Description
Fluorescence polarization assay was performed to confirm the binding ability to the compound synthesized with HSP90 according the concentration. 1 M ...


US Patent US10464907 (2019)

More data for this
Ligand-Target Pair
Heat shock protein HSP 90-alpha


(Bovine)
BDBM419566
PNG
(US10464907, Compound 11j)
Show SMILES CN1CCN(C(C1)c1ccccc1)C(=O)c1cc(Cl)c(O)cc1O
Show InChI InChI=1/C18H19ClN2O3/c1-20-7-8-21(15(11-20)12-5-3-2-4-6-12)18(24)13-9-14(19)17(23)10-16(13)22/h2-6,9-10,15,22-23H,7-8,11H2,1H3
PDB

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US Patent
n/an/a 70n/an/an/an/an/an/a



INDUSTRY ACADEMIC COOPERATION FOUNDATION KEIMYUNG UNIVERSITY

US Patent


Assay Description
Fluorescence polarization assay was performed to confirm the binding ability to the compound synthesized with HSP90 according the concentration. 1 M ...


US Patent US10464907 (2019)

More data for this
Ligand-Target Pair
Heat shock protein HSP 90-alpha


(Bovine)
BDBM50464555
PNG
(CHEMBL4292004 | US10464907, Compound 14c)
Show SMILES COc1ccc(CN(C)C(=O)c2cc(Cl)c(O)cc2O)cc1
Show InChI InChI=1S/C16H16ClNO4/c1-18(9-10-3-5-11(22-2)6-4-10)16(21)12-7-13(17)15(20)8-14(12)19/h3-8,19-20H,9H2,1-2H3
PDB

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US Patent
n/an/a 135n/an/an/an/an/an/a



INDUSTRY ACADEMIC COOPERATION FOUNDATION KEIMYUNG UNIVERSITY

US Patent


Assay Description
Fluorescence polarization assay was performed to confirm the binding ability to the compound synthesized with HSP90 according the concentration. 1 M ...


US Patent US10464907 (2019)

More data for this
Ligand-Target Pair
Heat shock protein HSP 90-alpha


(Bovine)
BDBM419561
PNG
(US10464907, Compound 11e)
Show SMILES CN1CCN(CC1)C(=O)c1cc(Cl)c(O)cc1O
Show InChI InChI=1S/C12H15ClN2O3/c1-14-2-4-15(5-3-14)12(18)8-6-9(13)11(17)7-10(8)16/h6-7,16-17H,2-5H2,1H3
PDB

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US Patent
n/an/a 253n/an/an/an/an/an/a



INDUSTRY ACADEMIC COOPERATION FOUNDATION KEIMYUNG UNIVERSITY

US Patent


Assay Description
Fluorescence polarization assay was performed to confirm the binding ability to the compound synthesized with HSP90 according the concentration. 1 M ...


US Patent US10464907 (2019)

More data for this
Ligand-Target Pair
Heat shock protein HSP 90-alpha


(Bovine)
BDBM419317
PNG
(US10464907, Compound 11a)
Show SMILES Oc1cc(O)c(cc1Cl)C(=O)N1CCCC1
Show InChI InChI=1S/C11H12ClNO3/c12-8-5-7(9(14)6-10(8)15)11(16)13-3-1-2-4-13/h5-6,14-15H,1-4H2
PDB

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US Patent
n/an/a 348n/an/an/an/an/an/a



INDUSTRY ACADEMIC COOPERATION FOUNDATION KEIMYUNG UNIVERSITY

US Patent


Assay Description
Fluorescence polarization assay was performed to confirm the binding ability to the compound synthesized with HSP90 according the concentration. 1 M ...


US Patent US10464907 (2019)

More data for this
Ligand-Target Pair
Heat shock protein HSP 90-alpha


(Bovine)
BDBM50464564
PNG
(CHEMBL4280551 | US10464907, Compound 14d)
Show SMILES COc1ccc(CN(C)C(=O)c2cc(Cl)c(O)cc2O)cc1OC
Show InChI InChI=1S/C17H18ClNO5/c1-19(9-10-4-5-15(23-2)16(6-10)24-3)17(22)11-7-12(18)14(21)8-13(11)20/h4-8,20-21H,9H2,1-3H3
PDB

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US Patent
n/an/a 362n/an/an/an/an/an/a



INDUSTRY ACADEMIC COOPERATION FOUNDATION KEIMYUNG UNIVERSITY

US Patent


Assay Description
Fluorescence polarization assay was performed to confirm the binding ability to the compound synthesized with HSP90 according the concentration. 1 M ...


US Patent US10464907 (2019)

More data for this
Ligand-Target Pair
Heat shock protein HSP 90-alpha


(Bovine)
BDBM419559
PNG
(US10464907, Compound 11c)
Show SMILES Oc1cc(O)c(cc1Cl)C(=O)N1CCOCC1
Show InChI InChI=1S/C11H12ClNO4/c12-8-5-7(9(14)6-10(8)15)11(16)13-1-3-17-4-2-13/h5-6,14-15H,1-4H2
PDB

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US Patent
n/an/a 383n/an/an/an/an/an/a



INDUSTRY ACADEMIC COOPERATION FOUNDATION KEIMYUNG UNIVERSITY

US Patent


Assay Description
Fluorescence polarization assay was performed to confirm the binding ability to the compound synthesized with HSP90 according the concentration. 1 M ...


US Patent US10464907 (2019)

More data for this
Ligand-Target Pair
Heat shock protein HSP 90-alpha


(Bovine)
BDBM50464560
PNG
(CHEMBL4281389 | US10464907, Compound 14b)
Show SMILES CN(Cc1ccccc1)C(=O)c1cc(Cl)c(O)cc1O
Show InChI InChI=1S/C15H14ClNO3/c1-17(9-10-5-3-2-4-6-10)15(20)11-7-12(16)14(19)8-13(11)18/h2-8,18-19H,9H2,1H3
PDB

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US Patent
n/an/a 413n/an/an/an/an/an/a



INDUSTRY ACADEMIC COOPERATION FOUNDATION KEIMYUNG UNIVERSITY

US Patent


Assay Description
Fluorescence polarization assay was performed to confirm the binding ability to the compound synthesized with HSP90 according the concentration. 1 M ...


US Patent US10464907 (2019)

More data for this
Ligand-Target Pair
Heat shock protein HSP 90-alpha


(Bovine)
BDBM50464552
PNG
(CHEMBL4291855 | US10464907, Compound 14g)
Show SMILES COc1cc(CN(C)C(=O)c2cc(Cl)c(O)cc2O)c(Cl)c(OC)c1OC
Show InChI InChI=1S/C18H19Cl2NO6/c1-21(18(24)10-6-11(19)13(23)7-12(10)22)8-9-5-14(25-2)16(26-3)17(27-4)15(9)20/h5-7,22-23H,8H2,1-4H3
PDB

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US Patent
n/an/a 429n/an/an/an/an/an/a



INDUSTRY ACADEMIC COOPERATION FOUNDATION KEIMYUNG UNIVERSITY

US Patent


Assay Description
Fluorescence polarization assay was performed to confirm the binding ability to the compound synthesized with HSP90 according the concentration. 1 M ...


US Patent US10464907 (2019)

More data for this
Ligand-Target Pair
Heat shock protein HSP 90-alpha


(Bovine)
BDBM50464558
PNG
(CHEMBL4282602 | US10464907, Compound 21c)
Show SMILES CCCNC(=O)c1ccc(CN(C)C(=O)c2cc(Cl)c(O)cc2O)cc1
Show InChI InChI=1S/C19H21ClN2O4/c1-3-8-21-18(25)13-6-4-12(5-7-13)11-22(2)19(26)14-9-15(20)17(24)10-16(14)23/h4-7,9-10,23-24H,3,8,11H2,1-2H3,(H,21,25)
PDB

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US Patent
n/an/a 454n/an/an/an/an/an/a



INDUSTRY ACADEMIC COOPERATION FOUNDATION KEIMYUNG UNIVERSITY

US Patent


Assay Description
Fluorescence polarization assay was performed to confirm the binding ability to the compound synthesized with HSP90 according the concentration. 1 M ...


US Patent US10464907 (2019)

More data for this
Ligand-Target Pair
Heat shock protein HSP 90-alpha


(Bovine)
BDBM50464550
PNG
(CHEMBL4294168 | US10464907, Compound 21a)
Show SMILES CNC(=O)c1ccc(CN(C)C(=O)c2cc(Cl)c(O)cc2O)cc1
Show InChI InChI=1S/C17H17ClN2O4/c1-19-16(23)11-5-3-10(4-6-11)9-20(2)17(24)12-7-13(18)15(22)8-14(12)21/h3-8,21-22H,9H2,1-2H3,(H,19,23)
PDB

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US Patent
n/an/a 496n/an/an/an/an/an/a



INDUSTRY ACADEMIC COOPERATION FOUNDATION KEIMYUNG UNIVERSITY

US Patent


Assay Description
Fluorescence polarization assay was performed to confirm the binding ability to the compound synthesized with HSP90 according the concentration. 1 M ...


US Patent US10464907 (2019)

More data for this
Ligand-Target Pair
Heat shock protein HSP 90-alpha


(Bovine)
BDBM50464563
PNG
(CHEMBL4292279 | US10464907, Compound 14h)
Show SMILES COc1cc(CN(C)C(=O)c2cc(Cl)c(O)cc2O)c(Br)c(OC)c1OC
Show InChI InChI=1S/C18H19BrClNO6/c1-21(18(24)10-6-11(20)13(23)7-12(10)22)8-9-5-14(25-2)16(26-3)17(27-4)15(9)19/h5-7,22-23H,8H2,1-4H3
PDB

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US Patent
n/an/a 528n/an/an/an/an/an/a



INDUSTRY ACADEMIC COOPERATION FOUNDATION KEIMYUNG UNIVERSITY

US Patent


Assay Description
Fluorescence polarization assay was performed to confirm the binding ability to the compound synthesized with HSP90 according the concentration. 1 M ...


US Patent US10464907 (2019)

More data for this
Ligand-Target Pair
Heat shock protein HSP 90-alpha


(Bovine)
BDBM419557
PNG
(US10464907, Compound 11b)
Show SMILES Oc1cc(O)c(cc1Cl)C(=O)N1CCCCC1
Show InChI InChI=1S/C12H14ClNO3/c13-9-6-8(10(15)7-11(9)16)12(17)14-4-2-1-3-5-14/h6-7,15-16H,1-5H2
PDB

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US Patent
n/an/a 541n/an/an/an/an/an/a



INDUSTRY ACADEMIC COOPERATION FOUNDATION KEIMYUNG UNIVERSITY

US Patent


Assay Description
Fluorescence polarization assay was performed to confirm the binding ability to the compound synthesized with HSP90 according the concentration. 1 M ...


US Patent US10464907 (2019)

More data for this
Ligand-Target Pair
Heat shock protein HSP 90-alpha


(Bovine)
BDBM50464565
PNG
(CHEMBL4285068 | US10464907, Compound 16b)
Show SMILES CN(Cc1ccc(C)cc1)C(=O)c1cc(Cl)c(O)cc1O
Show InChI InChI=1S/C16H16ClNO3/c1-10-3-5-11(6-4-10)9-18(2)16(21)12-7-13(17)15(20)8-14(12)19/h3-8,19-20H,9H2,1-2H3
PDB

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US Patent
n/an/a 558n/an/an/an/an/an/a



INDUSTRY ACADEMIC COOPERATION FOUNDATION KEIMYUNG UNIVERSITY

US Patent


Assay Description
Fluorescence polarization assay was performed to confirm the binding ability to the compound synthesized with HSP90 according the concentration. 1 M ...


US Patent US10464907 (2019)

More data for this
Ligand-Target Pair
Heat shock protein HSP 90-alpha


(Bovine)
BDBM50464554
PNG
(CHEMBL4288435 | US10464907, Compound 14e)
Show SMILES CN(Cc1ccc2OCOc2c1)C(=O)c1cc(Cl)c(O)cc1O
Show InChI InChI=1S/C16H14ClNO5/c1-18(7-9-2-3-14-15(4-9)23-8-22-14)16(21)10-5-11(17)13(20)6-12(10)19/h2-6,19-20H,7-8H2,1H3
PDB

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US Patent
n/an/a 585n/an/an/an/an/an/a



INDUSTRY ACADEMIC COOPERATION FOUNDATION KEIMYUNG UNIVERSITY

US Patent


Assay Description
Fluorescence polarization assay was performed to confirm the binding ability to the compound synthesized with HSP90 according the concentration. 1 M ...


US Patent US10464907 (2019)

More data for this
Ligand-Target Pair
Heat shock protein HSP 90-alpha


(Bovine)
BDBM50464561
PNG
(CHEMBL4283580 | US10464907, Compound 21b)
Show SMILES CCNC(=O)c1ccc(CN(C)C(=O)c2cc(Cl)c(O)cc2O)cc1
Show InChI InChI=1S/C18H19ClN2O4/c1-3-20-17(24)12-6-4-11(5-7-12)10-21(2)18(25)13-8-14(19)16(23)9-15(13)22/h4-9,22-23H,3,10H2,1-2H3,(H,20,24)
PDB

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US Patent
n/an/a 612n/an/an/an/an/an/a



INDUSTRY ACADEMIC COOPERATION FOUNDATION KEIMYUNG UNIVERSITY

US Patent


Assay Description
Fluorescence polarization assay was performed to confirm the binding ability to the compound synthesized with HSP90 according the concentration. 1 M ...


US Patent US10464907 (2019)

More data for this
Ligand-Target Pair
Heat shock protein HSP 90-alpha


(Bovine)
BDBM419565
PNG
(US10464907, Compound 11i)
Show SMILES Oc1cc(O)c(cc1Cl)C(=O)N1CCC(=O)CC1
Show InChI InChI=1S/C12H12ClNO4/c13-9-5-8(10(16)6-11(9)17)12(18)14-3-1-7(15)2-4-14/h5-6,16-17H,1-4H2
PDB

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n/an/a 670n/an/an/an/an/an/a



INDUSTRY ACADEMIC COOPERATION FOUNDATION KEIMYUNG UNIVERSITY

US Patent


Assay Description
Fluorescence polarization assay was performed to confirm the binding ability to the compound synthesized with HSP90 according the concentration. 1 M ...


US Patent US10464907 (2019)

More data for this
Ligand-Target Pair
Heat shock protein HSP 90-alpha


(Bovine)
BDBM50464551
PNG
(CHEMBL4281643 | US10464907, Compound 16a)
Show SMILES CN(Cc1ccccc1C)C(=O)c1cc(Cl)c(O)cc1O
Show InChI InChI=1S/C16H16ClNO3/c1-10-5-3-4-6-11(10)9-18(2)16(21)12-7-13(17)15(20)8-14(12)19/h3-8,19-20H,9H2,1-2H3
PDB

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n/an/a 830n/an/an/an/an/an/a



INDUSTRY ACADEMIC COOPERATION FOUNDATION KEIMYUNG UNIVERSITY

US Patent


Assay Description
Fluorescence polarization assay was performed to confirm the binding ability to the compound synthesized with HSP90 according the concentration. 1 M ...


US Patent US10464907 (2019)

More data for this
Ligand-Target Pair
Heat shock protein HSP 90-alpha


(Bovine)
BDBM50464559
PNG
(CHEMBL4277126 | US10464907, Compound 14i)
Show SMILES CN(Cc1cccc(C)c1)C(=O)c1cc(Cl)c(O)cc1O
Show InChI InChI=1S/C16H16ClNO3/c1-10-4-3-5-11(6-10)9-18(2)16(21)12-7-13(17)15(20)8-14(12)19/h3-8,19-20H,9H2,1-2H3
PDB

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US Patent
n/an/a 995n/an/an/an/an/an/a



INDUSTRY ACADEMIC COOPERATION FOUNDATION KEIMYUNG UNIVERSITY

US Patent


Assay Description
Fluorescence polarization assay was performed to confirm the binding ability to the compound synthesized with HSP90 according the concentration. 1 M ...


US Patent US10464907 (2019)

More data for this
Ligand-Target Pair
Heat shock protein HSP 90-alpha


(Bovine)
BDBM419563
PNG
(US10464907, Compound 11g)
Show SMILES Oc1cc(O)c(cc1Cl)C(=O)N1CCNC(=O)C1
Show InChI InChI=1S/C11H11ClN2O4/c12-7-3-6(8(15)4-9(7)16)11(18)14-2-1-13-10(17)5-14/h3-4,15-16H,1-2,5H2,(H,13,17)
PDB

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US Patent
n/an/a 1.37E+3n/an/an/an/an/an/a



INDUSTRY ACADEMIC COOPERATION FOUNDATION KEIMYUNG UNIVERSITY

US Patent


Assay Description
Fluorescence polarization assay was performed to confirm the binding ability to the compound synthesized with HSP90 according the concentration. 1 M ...


US Patent US10464907 (2019)

More data for this
Ligand-Target Pair
Heat shock protein HSP 90-alpha


(Bovine)
BDBM419573
PNG
(US10464907, Compound 14f)
Show SMILES COc1cc(CN(C)C(=O)c2cc(Cl)c(O)c(O)c2O)c(Cl)c(OC)c1OC
Show InChI InChI=1S/C18H19Cl2NO7/c1-21(18(25)9-6-10(19)14(23)15(24)13(9)22)7-8-5-11(26-2)16(27-3)17(28-4)12(8)20/h5-6,22-24H,7H2,1-4H3
PDB

UniProtKB/SwissProt

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US Patent
n/an/a 1.46E+3n/an/an/an/an/an/a



INDUSTRY ACADEMIC COOPERATION FOUNDATION KEIMYUNG UNIVERSITY

US Patent


Assay Description
Fluorescence polarization assay was performed to confirm the binding ability to the compound synthesized with HSP90 according the concentration. 1 M ...


US Patent US10464907 (2019)

More data for this
Ligand-Target Pair
Heat shock protein HSP 90-alpha


(Bovine)
BDBM419562
PNG
(US10464907, Compound 11f)
Show SMILES CC(=O)N1CCN(CC1)C(=O)c1cc(Cl)c(O)cc1O
Show InChI InChI=1S/C13H15ClN2O4/c1-8(17)15-2-4-16(5-3-15)13(20)9-6-10(14)12(19)7-11(9)18/h6-7,18-19H,2-5H2,1H3
PDB

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UniChem
US Patent
n/an/a 3.21E+3n/an/an/an/an/an/a



INDUSTRY ACADEMIC COOPERATION FOUNDATION KEIMYUNG UNIVERSITY

US Patent


Assay Description
Fluorescence polarization assay was performed to confirm the binding ability to the compound synthesized with HSP90 according the concentration. 1 M ...


US Patent US10464907 (2019)

More data for this
Ligand-Target Pair
Heat shock protein HSP 90-alpha


(Bovine)
BDBM419564
PNG
(US10464907, Compound 11h)
Show SMILES Oc1cc(O)c(cc1Cl)C(=O)N1CCC(=O)C1
Show InChI InChI=1S/C11H10ClNO4/c12-8-3-7(9(15)4-10(8)16)11(17)13-2-1-6(14)5-13/h3-4,15-16H,1-2,5H2
PDB

UniProtKB/SwissProt

GoogleScholar
UniChem
US Patent
n/an/a 3.92E+3n/an/an/an/an/an/a



INDUSTRY ACADEMIC COOPERATION FOUNDATION KEIMYUNG UNIVERSITY

US Patent


Assay Description
Fluorescence polarization assay was performed to confirm the binding ability to the compound synthesized with HSP90 according the concentration. 1 M ...


US Patent US10464907 (2019)

More data for this
Ligand-Target Pair
Heat shock protein HSP 90-alpha


(Bovine)
BDBM419560
PNG
(US10464907, Compound 11d)
Show SMILES Oc1cc(O)c(cc1Cl)C(=O)N1CCNCC1
Show InChI InChI=1S/C11H13ClN2O3/c12-8-5-7(9(15)6-10(8)16)11(17)14-3-1-13-2-4-14/h5-6,13,15-16H,1-4H2
PDB

UniProtKB/SwissProt

GoogleScholar
UniChem
US Patent
n/an/a 5.59E+3n/an/an/an/an/an/a



INDUSTRY ACADEMIC COOPERATION FOUNDATION KEIMYUNG UNIVERSITY

US Patent


Assay Description
Fluorescence polarization assay was performed to confirm the binding ability to the compound synthesized with HSP90 according the concentration. 1 M ...


US Patent US10464907 (2019)

More data for this
Ligand-Target Pair
Heat shock protein HSP 90-alpha


(Bovine)
BDBM50464549
PNG
(CHEMBL4278768 | US10464907, Compound 14a)
Show SMILES Oc1cc(O)c(cc1Cl)C(=O)NCc1ccccc1
Show InChI InChI=1S/C14H12ClNO3/c15-11-6-10(12(17)7-13(11)18)14(19)16-8-9-4-2-1-3-5-9/h1-7,17-18H,8H2,(H,16,19)
PDB

UniProtKB/SwissProt

GoogleScholar
UniChem
US Patent
n/an/a 6.68E+3n/an/an/an/an/an/a



INDUSTRY ACADEMIC COOPERATION FOUNDATION KEIMYUNG UNIVERSITY

US Patent


Assay Description
Fluorescence polarization assay was performed to confirm the binding ability to the compound synthesized with HSP90 according the concentration. 1 M ...


US Patent US10464907 (2019)

More data for this
Ligand-Target Pair
* indicates data uncertainty>20%