Compile Data Set for Download or QSAR
maximum 50k data
Found 20 Enz. Inhib. hit(s) with all data for entry = 8954
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM431915(((S)-6-{(R)-7-Fluoro-4-[4-(3-hydroxy-3-methyl-buto...)
Affinity DataEC50:  15nMAssay Description:IP1 accumulation measurements using the IPOne assay system—1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM431934(US10550127, Example 20 | {(S)-6-[(R)-4-(2,6-Dimeth...)
Affinity DataEC50:  9nMAssay Description:IP1 accumulation measurements using the IPOne assay system—1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM431917(((S)-6-{(R)-4-[4-(3-Hydroxy-3-methyl-butoxy)-2,6-d...)
Affinity DataEC50:  21nMAssay Description:IP1 accumulation measurements using the IPOne assay system—1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM431918(((R)-6-{(R)-4-[4-(3-Hydroxy-3-methyl-butoxy)-2,6-d...)
Affinity DataEC50:  751nMAssay Description:IP1 accumulation measurements using the IPOne assay system—1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM431919(((S)-6-{(R)-4-[2,6-Dimethyl-4-(2-methyl-2H-tetrazo...)
Affinity DataEC50:  6nMAssay Description:IP1 accumulation measurements using the IPOne assay system—1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM431920(((R)-6-{(R)-4-[2,6-Dimethyl-4-(2-methyl-2H-tetrazo...)
Affinity DataEC50:  382nMAssay Description:IP1 accumulation measurements using the IPOne assay system—1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM431921(((S)-6-{(R)-4-[2,6-Dimethyl-4-(2-methyl-2H-tetrazo...)
Affinity DataEC50:  7nMAssay Description:IP1 accumulation measurements using the IPOne assay system—1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM431922(((R)-6-{(R)-4-[2,6-Dimethyl-4-(2-methyl-2H-tetrazo...)
Affinity DataEC50:  378nMAssay Description:IP1 accumulation measurements using the IPOne assay system—1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM431923(US10550127, Example 9 | [(S)-6-((R)-4-{2,6-Dimethy...)
Affinity DataEC50:  57nMAssay Description:IP1 accumulation measurements using the IPOne assay system—1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM431924(((S)-6-{(R)-4-[2,6-Dimethyl-4-(tetrahydro-pyran-4-...)
Affinity DataEC50:  56nMAssay Description:IP1 accumulation measurements using the IPOne assay system—1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM431925(((S)-6-{(R)-4-[2,6-Dimethyl-4-(3-methyl-oxetan-3-y...)
Affinity DataEC50:  37nMAssay Description:IP1 accumulation measurements using the IPOne assay system—1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM431926(US10550127, Example 12 | [(S)-6-((R)-4-{2,6-Dimeth...)
Affinity DataEC50:  73nMAssay Description:IP1 accumulation measurements using the IPOne assay system—1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM431927(((S)-6-{(R)-7-Fluoro-4-[4-(2-hydroxo-2-methyl-prop...)
Affinity DataEC50:  35nMAssay Description:IP1 accumulation measurements using the IPOne assay system—1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM431928(((S)-6-{(R)-4-[2,6-Dimethyl-4-(tetrahydro-furan-3-...)
Affinity DataEC50:  27nMAssay Description:IP1 accumulation measurements using the IPOne assay system—1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM431929(US10550127, Example 15 | [(S)-6-((R)-7-Fluoro-4-{4...)
Affinity DataEC50:  9nMAssay Description:IP1 accumulation measurements using the IPOne assay system—1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM431930(((S)-6-{(R)-4-[2,6-Dimethyl-4-(1-methyl-2-oxo-1,2-...)
Affinity DataEC50:  27nMAssay Description:IP1 accumulation measurements using the IPOne assay system—1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM431931(((S)-6-{(R)-4-[2,6-Dimethyl-4-(1-methyl-2-oxo-1,2-...)
Affinity DataEC50:  12nMAssay Description:IP1 accumulation measurements using the IPOne assay system—1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM431932(((S)-6-{(R)-4-[2,6-Dimethyl-4-(1-methyl-6-oxo-1,6-...)
Affinity DataEC50:  14nMAssay Description:IP1 accumulation measurements using the IPOne assay system—1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM431933(((S)-6-{(R)-4-[2,6-Dimethyl-4-(1-methyl-6-oxo-1,6-...)
Affinity DataEC50:  27nMAssay Description:IP1 accumulation measurements using the IPOne assay system—1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM431916(((R)-6-{(R)-7-Fluoro-4-[4-(3-hydroxy-3-methyl-buto...)
Affinity DataEC50:  764nMAssay Description:IP1 accumulation measurements using the IPOne assay system—1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent