Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435105![]() (US10584120, Compound 39) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435104![]() (US10584120, Compound 38) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435111![]() (US10584120, Compound 45) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435108![]() (US10584120, Compound 42) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435128![]() (US10584120, Compound 62) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435114![]() (US10584120, Compound 47) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435123![]() (US10584120, Compound 56) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 7 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435126![]() (US10584120, Compound 60) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 7 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435109![]() (US10584120, Compound 43) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 8 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435112![]() (US10584120, Compound 46) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 8 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435106![]() (US10584120, Compound 40) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 9 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435110![]() (US10584120, Compound 44) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435115![]() (US10584120, Compound 48) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435116![]() (US10584120, Compound 49) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435129![]() (US10584120, Compound 63) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 11 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435107![]() (US10584120, Compound 41) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 12 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435130![]() (US10584120, Compound 64) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435117![]() (US10584120, Compound 50) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435127![]() (US10584120, Compound 61) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 16 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435078![]() (US10584120, Compound 9) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 16 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435103![]() (US10584120, Compound 37) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 18 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435125![]() (US10584120, Compound 59) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 19 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435131![]() (US10584120, Compound 65) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435075![]() (US10584120, Compound 7) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 21 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435121![]() (US10584120, Compound 54) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 23 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435118![]() (US10584120, Compound 51) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 24 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435102![]() (US10584120, Compound 36) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 32 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435090![]() (US10584120, Compound 21) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 36 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435097![]() (US10584120, Compound 28) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 39 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435076![]() (US10584120, Compound 8) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 49 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435072![]() (US10584120, Compound 1) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 53 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435089![]() (US10584120, Compound 20) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 57 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435088![]() (US10584120, Compound 19) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 58 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435096![]() (US10584120, Compound 27) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 66 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435100![]() (US10584120, Compound 34) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 69 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435094![]() (US10584120, Compound 25) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 71 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435098![]() (US10584120, Compound 29) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 72 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435084![]() (US10584120, Compound 15) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 76 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435124![]() (US10584120, Compound 57) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 87 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435080![]() (US10584120, Compound 11) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435073![]() (US10584120, Compound 2) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435093![]() (US10584120, Compound 24) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 101 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435083![]() (US10584120, Compound 14) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 106 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435085![]() (US10584120, Compound 16) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 112 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435095![]() (US10584120, Compound 26) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 114 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435092![]() (US10584120, Compound 23) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 124 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435082![]() (US10584120, Compound 13) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 124 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435081![]() (US10584120, Compound 12) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 132 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435087![]() (US10584120, Compound 18) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 134 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435086![]() (US10584120, Compound 17) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 151 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435091![]() (US10584120, Compound 22) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 156 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435074![]() (US10584120, Compound 3) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 348 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435119![]() (US10584120, Compound 52) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 397 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435099![]() (US10584120, Compound 33) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 736 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435079![]() (US10584120, Compound 10) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 964 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435122![]() (US10584120, Compound 55) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 1.59E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435101![]() (US10584120, Compound 35) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 2.05E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutaminyl-peptide cyclotransferase (Homo sapiens (Human)) | BDBM435120![]() (US10584120, Compound 53) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | UniChem | US Patent | 3.42E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Health Research Institutes; Academia Sinica US Patent | Assay Description An inhibition activity assay of QC inhibitors was conducted. See Huang et al., J. Biol. Chem. 2011, 286, 12439-12449. A reaction mixture containing 3... | US Patent US10584120 (2020) BindingDB Entry DOI: 10.7270/Q2ZK5K20 | |||||||||||
More data for this Ligand-Target Pair |