Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 9045
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Centaurus Biopharma

US Patent
LigandPNGBDBM433323(US10561657, Ruxolitinib | US10617692, Ruxolitinib ...)
Affinity DataIC50: <10nMAssay Description:A testing platform for kinase activity of JAK2 was established based on Homogeneous Time-Resolved Fluorescence (HTRF) assay, and the activities of th...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Centaurus Biopharma

US Patent
LigandPNGBDBM437665(US10617692, Compound II)
Affinity DataIC50: <10nMAssay Description:A testing platform for kinase activity of JAK2 was established based on Homogeneous Time-Resolved Fluorescence (HTRF) assay, and the activities of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Centaurus Biopharma

US Patent
LigandPNGBDBM437666(US10617692, Compound III)
Affinity DataIC50: <10nMAssay Description:A testing platform for kinase activity of JAK2 was established based on Homogeneous Time-Resolved Fluorescence (HTRF) assay, and the activities of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Centaurus Biopharma

US Patent
LigandPNGBDBM437667(US10617692, Compound IV)
Affinity DataIC50: <30nMAssay Description:A testing platform for kinase activity of JAK2 was established based on Homogeneous Time-Resolved Fluorescence (HTRF) assay, and the activities of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent