Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
lxrbeta () | BDBM19992![]() (2-[3-[3-[[2-chloro-3-(trifluoromethyl)phenyl]methy...) | GoogleScholar | Purchase CHEMBL KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | US Patent | n/a | n/a | n/a | n/a | 40 | n/a | n/a | n/a | n/a |
Rgenix, Inc. US Patent | Assay Description TBD | US Patent US10669296 (2020) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
lxralpha () | BDBM426493![]() (US10543183, Compound SB742881 | US10669296, Compou...) | GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 74 | n/a | n/a | n/a | n/a |
Rgenix, Inc. US Patent | Assay Description TBD | US Patent US10669296 (2020) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
lxrbeta () | BDBM426493![]() (US10543183, Compound SB742881 | US10669296, Compou...) | GoogleScholar | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 25 | n/a | n/a | n/a | n/a |
Rgenix, Inc. US Patent | Assay Description TBD | US Patent US10669296 (2020) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
lxralpha () | BDBM19992![]() (2-[3-[3-[[2-chloro-3-(trifluoromethyl)phenyl]methy...) | GoogleScholar | Purchase CHEMBL KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | US Patent | n/a | n/a | n/a | n/a | 200 | n/a | n/a | n/a | n/a |
Rgenix, Inc. US Patent | Assay Description TBD | US Patent US10669296 (2020) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
lxralpha () | BDBM26066![]() (2-[(2-chloro-4-fluorophenyl)methyl]-3-(4-fluorophe...) | GoogleScholar | Purchase PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 179 | n/a | n/a | n/a | n/a |
Rgenix, Inc. US Patent | Assay Description TBD | US Patent US10669296 (2020) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
lxralpha () | BDBM19993![]() (CHEMBL62136 | N-[4-(1,1,1,3,3,3-hexafluoro-2-hydro...) | GoogleScholar | Purchase CHEMBL DrugBank KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | US Patent | n/a | n/a | n/a | n/a | 20 | n/a | n/a | n/a | n/a |
Rgenix, Inc. US Patent | Assay Description TBD | US Patent US10669296 (2020) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
lxrbeta () | BDBM26066![]() (2-[(2-chloro-4-fluorophenyl)methyl]-3-(4-fluorophe...) | GoogleScholar | Purchase PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 24 | n/a | n/a | n/a | n/a |
Rgenix, Inc. US Patent | Assay Description TBD | US Patent US10669296 (2020) | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
lxrbeta () | BDBM19993![]() (CHEMBL62136 | N-[4-(1,1,1,3,3,3-hexafluoro-2-hydro...) | GoogleScholar | Purchase CHEMBL DrugBank KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | US Patent | n/a | n/a | n/a | n/a | 50 | n/a | n/a | n/a | n/a |
Rgenix, Inc. US Patent | Assay Description TBD | US Patent US10669296 (2020) | |||||||||||
More data for this Ligand-Target Pair |