Compile Data Set for Download or QSAR
maximum 50k data
Found 17 Enz. Inhib. hit(s) with all data for entry = 9225
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Merch Sharp & Dohne Corp. Rahway

US Patent
LigandPNGBDBM450607((2S,3R)-3-(2-(1-(2,5-bis(Trifluoromethyl)benzyl)pi...)
Affinity DataEC50:  611nMAssay Description:The assay was performed in 384-well format. HEK cells stably expressing human GPR40 were plated at 7500 cells per well in growth medium (DMEM/10% fet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Merch Sharp & Dohne Corp. Rahway

US Patent
LigandPNGBDBM450622(Sodium (2S,3R)-3-cyclopropyl-3-((R or S)-3-(2̸...)
Affinity DataEC50:  12nMAssay Description:The assay was performed in 384-well format. HEK cells stably expressing human GPR40 were plated at 7500 cells per well in growth medium (DMEM/10% fet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Merch Sharp & Dohne Corp. Rahway

US Patent
LigandPNGBDBM450609(Sodium (2S,3R)-methyl 3- ((S or R)-3-(1-(2,5- bis(...)
Affinity DataEC50:  642nMAssay Description:The assay was performed in 384-well format. HEK cells stably expressing human GPR40 were plated at 7500 cells per well in growth medium (DMEM/10% fet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Merch Sharp & Dohne Corp. Rahway

US Patent
LigandPNGBDBM450610(Sodium (2S,3S)-3-((R or S)-3-(1-(2,5-bis(trifluoro...)
Affinity DataEC50:  4.70E+3nMAssay Description:The assay was performed in 384-well format. HEK cells stably expressing human GPR40 were plated at 7500 cells per well in growth medium (DMEM/10% fet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Merch Sharp & Dohne Corp. Rahway

US Patent
LigandPNGBDBM450610(Sodium (2S,3S)-3-((R or S)-3-(1-(2,5-bis(trifluoro...)
Affinity DataEC50:  2.10E+3nMAssay Description:The assay was performed in 384-well format. HEK cells stably expressing human GPR40 were plated at 7500 cells per well in growth medium (DMEM/10% fet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Merch Sharp & Dohne Corp. Rahway

US Patent
LigandPNGBDBM450612(Sodium (2S,3R)-3-((R or S)-2-(1-(2,5-bis(trifluoro...)
Affinity DataEC50:  35nMAssay Description:The assay was performed in 384-well format. HEK cells stably expressing human GPR40 were plated at 7500 cells per well in growth medium (DMEM/10% fet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Merch Sharp & Dohne Corp. Rahway

US Patent
LigandPNGBDBM450612(Sodium (2S,3R)-3-((R or S)-2-(1-(2,5-bis(trifluoro...)
Affinity DataEC50:  99nMAssay Description:The assay was performed in 384-well format. HEK cells stably expressing human GPR40 were plated at 7500 cells per well in growth medium (DMEM/10% fet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Merch Sharp & Dohne Corp. Rahway

US Patent
LigandPNGBDBM450614((2S,3R)-3-((R or S)-2-(1-(2,5-bis(trifluoromethyl)...)
Affinity DataEC50:  439nMAssay Description:The assay was performed in 384-well format. HEK cells stably expressing human GPR40 were plated at 7500 cells per well in growth medium (DMEM/10% fet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Merch Sharp & Dohne Corp. Rahway

US Patent
LigandPNGBDBM450615((2S,3R)-3-((S or R)-2-(1- (2,5-bis(trifluoromethyl...)
Affinity DataEC50:  289nMAssay Description:The assay was performed in 384-well format. HEK cells stably expressing human GPR40 were plated at 7500 cells per well in growth medium (DMEM/10% fet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Merch Sharp & Dohne Corp. Rahway

US Patent
LigandPNGBDBM450616(Sodium (2S,3R)-3-cyclopropyl-3-((R or S)-2-(2̸...)
Affinity DataEC50:  0.790nMAssay Description:The assay was performed in 384-well format. HEK cells stably expressing human GPR40 were plated at 7500 cells per well in growth medium (DMEM/10% fet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Merch Sharp & Dohne Corp. Rahway

US Patent
LigandPNGBDBM450616(Sodium (2S,3R)-3-cyclopropyl-3-((R or S)-2-(2̸...)
Affinity DataEC50:  0.200nMAssay Description:The assay was performed in 384-well format. HEK cells stably expressing human GPR40 were plated at 7500 cells per well in growth medium (DMEM/10% fet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Merch Sharp & Dohne Corp. Rahway

US Patent
LigandPNGBDBM450618((2S,3R)-3-cyclopropyl-3-((R or S)-2-(2′-fluo...)
Affinity DataEC50:  1nMAssay Description:The assay was performed in 384-well format. HEK cells stably expressing human GPR40 were plated at 7500 cells per well in growth medium (DMEM/10% fet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Merch Sharp & Dohne Corp. Rahway

US Patent
LigandPNGBDBM450618((2S,3R)-3-cyclopropyl-3-((R or S)-2-(2′-fluo...)
Affinity DataEC50:  12nMAssay Description:The assay was performed in 384-well format. HEK cells stably expressing human GPR40 were plated at 7500 cells per well in growth medium (DMEM/10% fet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Merch Sharp & Dohne Corp. Rahway

US Patent
LigandPNGBDBM450620(Sodium (2S,3R)-3-cyclopropyl-3-((R or S)-3-(2̸...)
Affinity DataEC50:  10nMAssay Description:The assay was performed in 384-well format. HEK cells stably expressing human GPR40 were plated at 7500 cells per well in growth medium (DMEM/10% fet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Merch Sharp & Dohne Corp. Rahway

US Patent
LigandPNGBDBM450620(Sodium (2S,3R)-3-cyclopropyl-3-((R or S)-3-(2̸...)
Affinity DataEC50:  0.800nMAssay Description:The assay was performed in 384-well format. HEK cells stably expressing human GPR40 were plated at 7500 cells per well in growth medium (DMEM/10% fet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Merch Sharp & Dohne Corp. Rahway

US Patent
LigandPNGBDBM450622(Sodium (2S,3R)-3-cyclopropyl-3-((R or S)-3-(2̸...)
Affinity DataEC50:  0.800nMAssay Description:The assay was performed in 384-well format. HEK cells stably expressing human GPR40 were plated at 7500 cells per well in growth medium (DMEM/10% fet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Merch Sharp & Dohne Corp. Rahway

US Patent
LigandPNGBDBM450608(Sodium (2S,3S)-3-((R or S)-3-(1-(2,5-Bis(trifluoro...)
Affinity DataEC50:  388nMAssay Description:The assay was performed in 384-well format. HEK cells stably expressing human GPR40 were plated at 7500 cells per well in growth medium (DMEM/10% fet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent