Compile Data Set for Download or QSAR
maximum 50k data
Found 185 Enz. Inhib. hit(s) with all data for entry = 9831
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492438(5-(1-tert-butyl-1H- pyrazol-4-yl)-6-(1- methylethy...)
Affinity DataIC50:  5.08nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492457(6-(1-methylethyl)-5-[1- (1-methylethyl)-1H-pyrazol...)
Affinity DataIC50:  5.08nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492546(5-(1-cyclobutyl-1H- pyrazol-4-yl)-6-(1- methylethy...)
Affinity DataIC50:  5.08nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492545(6-(1-methylethyl)-5-[5- (morpholin-4- ylmethyl)thi...)
Affinity DataIC50:  5.08nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492544(5-[1-(2-hydroxy-1,1- dimethylethyl)-1H- pyrazol-4-...)
Affinity DataIC50:  5.08nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492458(6-(1-methylethyl)-5-(1- propyl-1H-pyrazol-4- yl)[1...)
Affinity DataIC50:  5.08nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492571(5-(1-tert-butyl-1H-pyrrol- 3-yl)-6-(1- methylethyl...)
Affinity DataIC50:  5.08nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492449(6-(1-methylethyl)-5-[1- (2-methylpropyl)-1H- pyraz...)
Affinity DataIC50:  5.08nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492450(5-{1-[(1- fluorocyclopentyl)methyl]- 1H-pyrazol-4-...)
Affinity DataIC50:  5.08nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492451(5-[1- (cyclopropylmethyl)-1H- pyrazol-4-yl]-6-(1- ...)
Affinity DataIC50:  5.08nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492439(5-[1-(3-methylbutyl)-1H- pyrazol-4-yl]-6-(1- methy...)
Affinity DataIC50:  5.22nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492529(5-[1-(2-methoxy-1,1- dimethylethyl)-1H- pyrazol-4-...)
Affinity DataIC50:  5.29nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492453(5-[1-(2-methoxyethyl)- 1H-pyrazol-4-yl]-6-(1- meth...)
Affinity DataIC50:  5.73nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492455(5-(1-cyclopropyl-1H- pyrazol-4-yl)-6-(1- methyleth...)
Affinity DataIC50:  5.74nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492477(6-(1-methylethyl)-5-[1- (pyridin-3-ylmethyl)-1H- p...)
Affinity DataIC50:  5.77nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492476(6-(1-methylethyl)-5-[1- (pyridin-2-ylmethyl)-1H- p...)
Affinity DataIC50:  5.83nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492456(5-(1-ethyl-1H-pyrazol-4- yl)-6-(1- methylethyl)[1,...)
Affinity DataIC50:  6.27nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492445(6-(1-methylethyl)-5-(1- phenyl-1H-pyrazol-4- yl)[1...)
Affinity DataIC50:  6.28nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492454(5-[1-(4-fluorophenyl)- 1H-pyrazol-4-yl]-6-(1- meth...)
Affinity DataIC50:  6.47nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492547(6-(1-methylethyl)-5-[1- (thiophen-2-ylmethyl)- 1H-...)
Affinity DataIC50:  6.70nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492560(6-(1-methylethyl)-5-(2- oxo-2,3-dihydro-1H- indol-...)
Affinity DataIC50:  6.93nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492484(6-(1-methylethyl)-5-{1- [2-(methylsulfonyl)ethyl]-...)
Affinity DataIC50:  6.93nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492489(6-(1-methylethyl)-5-[1- (2-morpholin-4-ylethyl)- 1...)
Affinity DataIC50:  6.96nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492527(6-(1-methylethyl)-5-[4- (1-methyl-1H-imidazol-2- y...)
Affinity DataIC50:  7.26nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492446(5-(1-benzyl-1H-pyrazol- 4-yl)-6-(1- methylethyl)[1...)
Affinity DataIC50:  7.30nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492562(6-(1-methylethyl)-5-[1- (tetrahydro-2H-pyran-2- yl...)
Affinity DataIC50:  7.36nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492452(6-(1-methylethyl)-5-[1- (pyridin-4-ylmethyl)-1H- p...)
Affinity DataIC50:  7.5nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492447(6-(1-methylethyl)-5-(4- morpholin-4- ylphenyl)[1,2...)
Affinity DataIC50:  7.52nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492538(6-[6-(1-methylethyl)-7- oxo-4,7- dihydro[1,2,4]tri...)
Affinity DataIC50:  7.57nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492525(6-(1-methylethyl)-5-(4-pyridin-4- ylphenyl)[1,2,4]...)
Affinity DataIC50:  8.57nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492532(6-(1-methylethyl)-5-[4- (1H-1,2,3-triazol-1- yl)ph...)
Affinity DataIC50:  8.59nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492561(N-{4-[6-(1-methylethyl)- 7-oxo-4,7- dihydro[1,2,4]...)
Affinity DataIC50:  8.76nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492519(6-(1-methylethyl)-5-[4- (1H-pyrazol-1- yl)phenyl][...)
Affinity DataIC50:  8.78nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492503(US10975084, Example 11-66 | {3-[6-(1-methylethyl)-...)
Affinity DataIC50:  8.93nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492492(6-(1-methylethyl)-5-[(E)- 2-phenylethenyl][1,2,4]t...)
Affinity DataIC50:  9.45nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492488(5-[1-(3-chlorophenyl)- 1H-pyrazol-4-yl]-6-(1- meth...)
Affinity DataIC50:  9.66nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492555(6-(1-methylethyl)-5-(4- piperazin-1- ylphenyl)[1,2...)
Affinity DataIC50:  9.79nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492563(6-(1-methylethyl)-5-(6- piperidin-1-ylpyridin-3- y...)
Affinity DataIC50:  10.4nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492515(6-(1-methylethyl)-5-(1- methyl-1H-indazol-5- yl)[1...)
Affinity DataIC50:  10.4nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492564(6-(1-methylethyl)-5-(6- morpholin-4-ylpyridin-3- y...)
Affinity DataIC50:  11.6nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492548(5-[1-(2-hydroxyethyl)- 1H-pyrazol-4-yl]-6-(1- meth...)
Affinity DataIC50:  11.7nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492478(6-(1-methylethyl)-5-(4- piperidin-1- ylphenyl)[1,2...)
Affinity DataIC50:  11.8nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492565(6-(1-methylethyl)-5-[6- (1H-pyrazol-1-yl)pyridin- ...)
Affinity DataIC50:  12.3nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492523(N,N-dimethyl-4-[6-(1- methylethyl)-7-oxo-4,7- dihy...)
Affinity DataIC50:  12.6nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492559(6-(1-methylethyl)-5-(1H- pyrazol-4- yl)[1,2,4]tria...)
Affinity DataIC50:  13.3nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492533(5-[4-(1,1- dioxidothiomorpholin-4- yl)phenyl]-6-(1...)
Affinity DataIC50:  13.5nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492497(5-[4-(hydroxymethyl)phenyl]- 6-(1- methylethyl)[1,...)
Affinity DataIC50:  13.5nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492507(5-(1H-benzimidazol-6-yl)-6-(1- methylethyl)[1,2,4]...)
Affinity DataIC50:  13.5nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492511(6-(1-methylethyl)-5- quinolin-6- yl[1,2,4]triazolo...)
Affinity DataIC50:  14.7nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM492530(6-(1-methylethyl)-5-{4- [4-(1- methylethyl)piperaz...)
Affinity DataIC50:  15.5nMAssay Description:In this assay, the potency (IC50) of each compound was determined from a ten point (1:3 serial dilution; final compound concentration range in assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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