Compile Data Set for Download or QSAR
maximum 50k data
Found 19 Enz. Inhib. hit(s) with all data for entry = 10267
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Texas A&M University System

US Patent
LigandPNGBDBM524049(US11136333, Compound 19a)
Affinity DataIC50:  1.27nMAssay Description:IC50 against Abelson kinase ABL1 was determined by Life Technologies corporation though the Z′-LITE biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Texas A&M University System

US Patent
LigandPNGBDBM524050(US11136333, Compound 19bbIC50)
Affinity DataIC50:  2.09nMAssay Description:IC50 against Abelson kinase ABL1 was determined by Life Technologies corporation though the Z′-LITE biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Texas A&M University System

US Patent
LigandPNGBDBM524044(US11136333, Compound 12c)
Affinity DataIC50:  2.13nMAssay Description:IC50 against Abelson kinase ABL1 was determined by Life Technologies corporation though the Z′-LITE biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Texas A&M University System

US Patent
LigandPNGBDBM524048(US11136333, Compound 12g)
Affinity DataIC50:  3.51nMAssay Description:IC50 against Abelson kinase ABL1 was determined by Life Technologies corporation though the Z′-LITE biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Texas A&M University System

US Patent
LigandPNGBDBM524047(US11136333, Compound 12f)
Affinity DataIC50:  15.7nMAssay Description:IC50 against Abelson kinase ABL1 was determined by Life Technologies corporation though the Z′-LITE biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Texas A&M University System

US Patent
LigandPNGBDBM524046(US11136333, Compound 12e)
Affinity DataIC50:  16.1nMAssay Description:IC50 against Abelson kinase ABL1 was determined by Life Technologies corporation though the Z′-LITE biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Texas A&M University System

US Patent
LigandPNGBDBM524042(US11136333, Compound 12a)
Affinity DataIC50:  17.5nMAssay Description:IC50 against Abelson kinase ABL1 was determined by Life Technologies corporation though the Z′-LITE biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Texas A&M University System

US Patent
LigandPNGBDBM524043(US11136333, Compound 12b)
Affinity DataIC50:  18.7nMAssay Description:IC50 against Abelson kinase ABL1 was determined by Life Technologies corporation though the Z′-LITE biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Texas A&M University System

US Patent
LigandPNGBDBM524045(US11136333, Compound 12d)
Affinity DataIC50:  42.6nMAssay Description:IC50 against Abelson kinase ABL1 was determined by Life Technologies corporation though the Z′-LITE biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Texas A&M University System

US Patent
LigandPNGBDBM524050(US11136333, Compound 19bbIC50)
Affinity DataKd:  0.660nMAssay Description:This assay is described in https://www.discoverx.com/kinase-data-sheets/abl1-nonphosphorylated.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Texas A&M University System

US Patent
LigandPNGBDBM524049(US11136333, Compound 19a)
Affinity DataKd:  0.380nMAssay Description:This assay is described in https://www.discoverx.com/kinase-data-sheets/abl1-nonphosphorylated.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Texas A&M University System

US Patent
LigandPNGBDBM524048(US11136333, Compound 12g)
Affinity DataKd:  0.910nMAssay Description:This assay is described in https://www.discoverx.com/kinase-data-sheets/abl1-nonphosphorylated.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Texas A&M University System

US Patent
LigandPNGBDBM524047(US11136333, Compound 12f)
Affinity DataKd:  1.5nMAssay Description:This assay is described in https://www.discoverx.com/kinase-data-sheets/abl1-nonphosphorylated.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Texas A&M University System

US Patent
LigandPNGBDBM524046(US11136333, Compound 12e)
Affinity DataKd:  1.5nMAssay Description:This assay is described in https://www.discoverx.com/kinase-data-sheets/abl1-nonphosphorylated.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Texas A&M University System

US Patent
LigandPNGBDBM524045(US11136333, Compound 12d)
Affinity DataKd:  2.60nMAssay Description:This assay is described in https://www.discoverx.com/kinase-data-sheets/abl1-nonphosphorylated.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Texas A&M University System

US Patent
LigandPNGBDBM524044(US11136333, Compound 12c)
Affinity DataKd:  0.400nMAssay Description:This assay is described in https://www.discoverx.com/kinase-data-sheets/abl1-nonphosphorylated.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Texas A&M University System

US Patent
LigandPNGBDBM524043(US11136333, Compound 12b)
Affinity DataKd:  3.30nMAssay Description:This assay is described in https://www.discoverx.com/kinase-data-sheets/abl1-nonphosphorylated.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Texas A&M University System

US Patent
LigandPNGBDBM6568(6-(2,6-dichlorophenyl)-8-methyl-2-{[3-(methylsulfa...)
Affinity DataKd:  0.580nMAssay Description:This assay is described in https://www.discoverx.com/kinase-data-sheets/abl1-nonphosphorylated.More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
The Texas A&M University System

US Patent
LigandPNGBDBM524042(US11136333, Compound 12a)
Affinity DataKd:  3.5nMAssay Description:This assay is described in https://www.discoverx.com/kinase-data-sheets/abl1-nonphosphorylated.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent