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Found 2 Enz. Inhib. hit(s) with all data for entry = 6484
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
Vertex Pharmaceuticals

US Patent
LigandPNGBDBM50437436(CHEMBL2409216 | US8841450, I-1)
Affinity DataKi:  16nMpH: 7.5Assay Description:Compounds were screened for their ability to inhibit ATR kinase using a radioactive-phosphate incorporation assay. Assays were carried out in a mixtu...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
Vertex Pharmaceuticals

US Patent
LigandPNGBDBM50437437(CHEMBL2409217 | US8841450, I-2)
Affinity DataKi:  90nMpH: 7.5Assay Description:Compounds were screened for their ability to inhibit ATR kinase using a radioactive-phosphate incorporation assay. Assays were carried out in a mixtu...More data for this Ligand-Target Pair
In DepthDetails US Patent