Found 55 Enz. Inhib. hit(s) with all data for entry = 6905 
Affinity DataIC50: 0.834nMAssay Description:The H3 binding assay was/can be used to evaluate the ability of at least one compound in accordance with formula I, Ia, Ib, and/or Ic to inhibit [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 1.37nMAssay Description:The H3 binding assay was/can be used to evaluate the ability of at least one compound in accordance with formula I, Ia, Ib, and/or Ic to inhibit [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 1.63nMAssay Description:The H3 binding assay was/can be used to evaluate the ability of at least one compound in accordance with formula I, Ia, Ib, and/or Ic to inhibit [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 3.41nMpH: 7.4 T: 2°CAssay Description:A GTP gamma S binding assay can be used to investigate antagonist properties of compounds in CHO cells (Chinese Hamster Ovary) transfected with human...More data for this Ligand-Target Pair
Affinity DataIC50: 3.49nMAssay Description:The H3 binding assay was/can be used to evaluate the ability of at least one compound in accordance with formula I, Ia, Ib, and/or Ic to inhibit [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 3.69nMAssay Description:The H3 binding assay was/can be used to evaluate the ability of at least one compound in accordance with formula I, Ia, Ib, and/or Ic to inhibit [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 3.81nMpH: 7.4 T: 2°CAssay Description:A GTP gamma S binding assay can be used to investigate antagonist properties of compounds in CHO cells (Chinese Hamster Ovary) transfected with human...More data for this Ligand-Target Pair
Affinity DataIC50: 5.09nMAssay Description:The H3 binding assay was/can be used to evaluate the ability of at least one compound in accordance with formula I, Ia, Ib, and/or Ic to inhibit [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 5.83nMpH: 7.4 T: 2°CAssay Description:A GTP gamma S binding assay can be used to investigate antagonist properties of compounds in CHO cells (Chinese Hamster Ovary) transfected with human...More data for this Ligand-Target Pair
Affinity DataIC50: 6.19nMpH: 7.4 T: 2°CAssay Description:A GTP gamma S binding assay can be used to investigate antagonist properties of compounds in CHO cells (Chinese Hamster Ovary) transfected with human...More data for this Ligand-Target Pair
Affinity DataIC50: 6.40nMAssay Description:The H3 binding assay was/can be used to evaluate the ability of at least one compound in accordance with formula I, Ia, Ib, and/or Ic to inhibit [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 6.81nMpH: 7.4 T: 2°CAssay Description:A GTP gamma S binding assay can be used to investigate antagonist properties of compounds in CHO cells (Chinese Hamster Ovary) transfected with human...More data for this Ligand-Target Pair
Affinity DataIC50: 7.30nMAssay Description:The H3 binding assay was/can be used to evaluate the ability of at least one compound in accordance with formula I, Ia, Ib, and/or Ic to inhibit [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 7.56nMAssay Description:The H3 binding assay was/can be used to evaluate the ability of at least one compound in accordance with formula I, Ia, Ib, and/or Ic to inhibit [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 8.59nMpH: 7.4 T: 2°CAssay Description:A GTP gamma S binding assay can be used to investigate antagonist properties of compounds in CHO cells (Chinese Hamster Ovary) transfected with human...More data for this Ligand-Target Pair
Affinity DataIC50: 10.2nMAssay Description:The H3 binding assay was/can be used to evaluate the ability of at least one compound in accordance with formula I, Ia, Ib, and/or Ic to inhibit [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 11.6nMpH: 7.4 T: 2°CAssay Description:A GTP gamma S binding assay can be used to investigate antagonist properties of compounds in CHO cells (Chinese Hamster Ovary) transfected with human...More data for this Ligand-Target Pair
Affinity DataIC50: 13.3nMAssay Description:The H3 binding assay was/can be used to evaluate the ability of at least one compound in accordance with formula I, Ia, Ib, and/or Ic to inhibit [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:The H3 binding assay was/can be used to evaluate the ability of at least one compound in accordance with formula I, Ia, Ib, and/or Ic to inhibit [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 14.4nMAssay Description:The H3 binding assay was/can be used to evaluate the ability of at least one compound in accordance with formula I, Ia, Ib, and/or Ic to inhibit [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 16.8nMAssay Description:The H3 binding assay was/can be used to evaluate the ability of at least one compound in accordance with formula I, Ia, Ib, and/or Ic to inhibit [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 17.5nMpH: 7.4 T: 2°CAssay Description:A GTP gamma S binding assay can be used to investigate antagonist properties of compounds in CHO cells (Chinese Hamster Ovary) transfected with human...More data for this Ligand-Target Pair
Affinity DataIC50: 18.2nMpH: 7.4 T: 2°CAssay Description:A GTP gamma S binding assay can be used to investigate antagonist properties of compounds in CHO cells (Chinese Hamster Ovary) transfected with human...More data for this Ligand-Target Pair
Affinity DataIC50: 20.2nMAssay Description:The H3 binding assay was/can be used to evaluate the ability of at least one compound in accordance with formula I, Ia, Ib, and/or Ic to inhibit [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 20.2nMpH: 7.4 T: 2°CAssay Description:A GTP gamma S binding assay can be used to investigate antagonist properties of compounds in CHO cells (Chinese Hamster Ovary) transfected with human...More data for this Ligand-Target Pair
Affinity DataIC50: 21.3nMAssay Description:The H3 binding assay was/can be used to evaluate the ability of at least one compound in accordance with formula I, Ia, Ib, and/or Ic to inhibit [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 23.9nMpH: 7.4 T: 2°CAssay Description:A GTP gamma S binding assay can be used to investigate antagonist properties of compounds in CHO cells (Chinese Hamster Ovary) transfected with human...More data for this Ligand-Target Pair
Affinity DataIC50: 29.1nMAssay Description:The H3 binding assay was/can be used to evaluate the ability of at least one compound in accordance with formula I, Ia, Ib, and/or Ic to inhibit [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 30.4nMAssay Description:The H3 binding assay was/can be used to evaluate the ability of at least one compound in accordance with formula I, Ia, Ib, and/or Ic to inhibit [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 33.9nMpH: 7.4 T: 2°CAssay Description:A GTP gamma S binding assay can be used to investigate antagonist properties of compounds in CHO cells (Chinese Hamster Ovary) transfected with human...More data for this Ligand-Target Pair
Affinity DataIC50: 39.7nMpH: 7.4 T: 2°CAssay Description:A GTP gamma S binding assay can be used to investigate antagonist properties of compounds in CHO cells (Chinese Hamster Ovary) transfected with human...More data for this Ligand-Target Pair
Affinity DataIC50: 44.7nMAssay Description:The H3 binding assay was/can be used to evaluate the ability of at least one compound in accordance with formula I, Ia, Ib, and/or Ic to inhibit [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 45.3nMAssay Description:The H3 binding assay was/can be used to evaluate the ability of at least one compound in accordance with formula I, Ia, Ib, and/or Ic to inhibit [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 62.5nMAssay Description:The H3 binding assay was/can be used to evaluate the ability of at least one compound in accordance with formula I, Ia, Ib, and/or Ic to inhibit [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 88.3nMAssay Description:The H3 binding assay was/can be used to evaluate the ability of at least one compound in accordance with formula I, Ia, Ib, and/or Ic to inhibit [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 105nMAssay Description:The H3 binding assay was/can be used to evaluate the ability of at least one compound in accordance with formula I, Ia, Ib, and/or Ic to inhibit [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 127nMpH: 7.4 T: 2°CAssay Description:A GTP gamma S binding assay can be used to investigate antagonist properties of compounds in CHO cells (Chinese Hamster Ovary) transfected with human...More data for this Ligand-Target Pair
Affinity DataIC50: 146nMAssay Description:The H3 binding assay was/can be used to evaluate the ability of at least one compound in accordance with formula I, Ia, Ib, and/or Ic to inhibit [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 197nMpH: 7.4 T: 2°CAssay Description:A GTP gamma S binding assay can be used to investigate antagonist properties of compounds in CHO cells (Chinese Hamster Ovary) transfected with human...More data for this Ligand-Target Pair
Affinity DataIC50: 262nMpH: 7.4 T: 2°CAssay Description:A GTP gamma S binding assay can be used to investigate antagonist properties of compounds in CHO cells (Chinese Hamster Ovary) transfected with human...More data for this Ligand-Target Pair
Affinity DataIC50: 351nMAssay Description:The H3 binding assay was/can be used to evaluate the ability of at least one compound in accordance with formula I, Ia, Ib, and/or Ic to inhibit [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 433nMAssay Description:The H3 binding assay was/can be used to evaluate the ability of at least one compound in accordance with formula I, Ia, Ib, and/or Ic to inhibit [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 441nMAssay Description:The H3 binding assay was/can be used to evaluate the ability of at least one compound in accordance with formula I, Ia, Ib, and/or Ic to inhibit [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 733nMpH: 7.4 T: 2°CAssay Description:A GTP gamma S binding assay can be used to investigate antagonist properties of compounds in CHO cells (Chinese Hamster Ovary) transfected with human...More data for this Ligand-Target Pair
Affinity DataIC50: 834nMpH: 7.4 T: 2°CAssay Description:A GTP gamma S binding assay can be used to investigate antagonist properties of compounds in CHO cells (Chinese Hamster Ovary) transfected with human...More data for this Ligand-Target Pair
Affinity DataIC50: 870nMpH: 7.4 T: 2°CAssay Description:A GTP gamma S binding assay can be used to investigate antagonist properties of compounds in CHO cells (Chinese Hamster Ovary) transfected with human...More data for this Ligand-Target Pair
Affinity DataIC50: >1.05E+3nMpH: 7.4 T: 2°CAssay Description:A GTP gamma S binding assay can be used to investigate antagonist properties of compounds in CHO cells (Chinese Hamster Ovary) transfected with human...More data for this Ligand-Target Pair
Affinity DataIC50: 1.63E+3nMAssay Description:The H3 binding assay was/can be used to evaluate the ability of at least one compound in accordance with formula I, Ia, Ib, and/or Ic to inhibit [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: >1.80E+3nMpH: 7.4 T: 2°CAssay Description:A GTP gamma S binding assay can be used to investigate antagonist properties of compounds in CHO cells (Chinese Hamster Ovary) transfected with human...More data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+3nMAssay Description:The H3 binding assay was/can be used to evaluate the ability of at least one compound in accordance with formula I, Ia, Ib, and/or Ic to inhibit [3H]...More data for this Ligand-Target Pair
