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Found 47 Enz. Inhib. hit(s) with all data for entry = 6931
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160301(US9040691, 29)
Affinity DataIC50:  1nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160276(US9040691, 4)
Affinity DataIC50:  1nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160312(US9040691, 40 | US9040691, 41 | US9040691, 42)
Affinity DataIC50:  1.20nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160277(US9040691, 5)
Affinity DataIC50:  1.30nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160283(US9040691, 11)
Affinity DataIC50:  1.90nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160315(US9040691, 43)
Affinity DataIC50:  1.90nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160289(US9040691, 17)
Affinity DataIC50:  2nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160302(US9040691, 30)
Affinity DataIC50:  2nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160273(US9040691, 1)
Affinity DataIC50:  2nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160279(US9040691, 7)
Affinity DataIC50:  2nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160288(US9040691, 16)
Affinity DataIC50:  2.60nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160274(US9040691, 2)
Affinity DataIC50:  2.80nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160309(US9040691, 37)
Affinity DataIC50: <3nMAssay Description:ALKl (Invitrogen, Carlsbad, CA, USA) kinase activity was measured at ProQinase GmbH ( Freiburg. Germany) in a radiometric assay using gamma-33P-ATP a...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160283(US9040691, 11)
Affinity DataIC50:  3nMAssay Description:ALKl (Invitrogen, Carlsbad, CA, USA) kinase activity was measured at ProQinase GmbH ( Freiburg. Germany) in a radiometric assay using gamma-33P-ATP a...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160312(US9040691, 40 | US9040691, 41 | US9040691, 42)
Affinity DataIC50:  3.20nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160312(US9040691, 40 | US9040691, 41 | US9040691, 42)
Affinity DataIC50:  3.5nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160316(US9040691, 44)
Affinity DataIC50:  3.80nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160285(US9040691, 13)
Affinity DataIC50:  4nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160275(US9040691, 3)
Affinity DataIC50:  4nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160310(US9040691, 38)
Affinity DataIC50:  4nMAssay Description:ALKl (Invitrogen, Carlsbad, CA, USA) kinase activity was measured at ProQinase GmbH ( Freiburg. Germany) in a radiometric assay using gamma-33P-ATP a...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160304(US9040691, 32)
Affinity DataIC50:  4nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160303(US9040691, 31)
Affinity DataIC50:  4nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160306(US9040691, 34)
Affinity DataIC50:  4.10nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160280(US9040691, 35 | US9040691, 36 | US9040691, 8)
Affinity DataIC50:  4.40nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160286(US9040691, 14)
Affinity DataIC50:  5.30nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160281(US9040691, 9)
Affinity DataIC50:  5.70nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160311(US9040691, 39)
Affinity DataIC50:  5.70nMAssay Description:ALKl (Invitrogen, Carlsbad, CA, USA) kinase activity was measured at ProQinase GmbH ( Freiburg. Germany) in a radiometric assay using gamma-33P-ATP a...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160284(US9040691, 12)
Affinity DataIC50:  5.90nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160279(US9040691, 7)
Affinity DataIC50:  6.70nMAssay Description:ALKl (Invitrogen, Carlsbad, CA, USA) kinase activity was measured at ProQinase GmbH ( Freiburg. Germany) in a radiometric assay using gamma-33P-ATP a...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160280(US9040691, 35 | US9040691, 36 | US9040691, 8)
Affinity DataIC50:  6.90nMAssay Description:ALKl (Invitrogen, Carlsbad, CA, USA) kinase activity was measured at ProQinase GmbH ( Freiburg. Germany) in a radiometric assay using gamma-33P-ATP a...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160282(US9040691, 10)
Affinity DataIC50:  8nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160305(US9040691, 33)
Affinity DataIC50:  15nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160294(US9040691, 22)
Affinity DataIC50:  17nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160291(US9040691, 19)
Affinity DataIC50:  19nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160280(US9040691, 35 | US9040691, 36 | US9040691, 8)
Affinity DataIC50:  21nMAssay Description:ALKl (Invitrogen, Carlsbad, CA, USA) kinase activity was measured at ProQinase GmbH ( Freiburg. Germany) in a radiometric assay using gamma-33P-ATP a...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM51425(US9040691, 21)
Affinity DataIC50:  25nMAssay Description:ALKl (Invitrogen, Carlsbad, CA, USA) kinase activity was measured at ProQinase GmbH ( Freiburg. Germany) in a radiometric assay using gamma-33P-ATP a...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160298(US9040691, 26)
Affinity DataIC50:  30nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160295(US9040691, 23)
Affinity DataIC50:  30nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160292(US9040691, 20)
Affinity DataIC50:  30nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160278(US9040691, 6)
Affinity DataIC50:  40nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160287(US9040691, 15)
Affinity DataIC50:  60nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160297(US9040691, 25)
Affinity DataIC50:  65nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160299(US9040691, 27)
Affinity DataIC50:  70nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160290(US9040691, 18)
Affinity DataIC50:  80nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160300(US9040691, 28)
Affinity DataIC50:  124nMAssay Description:ALKl (Invitrogen, Carlsbad, CA, USA) kinase activity was measured at ProQinase GmbH ( Freiburg. Germany) in a radiometric assay using gamma-33P-ATP a...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160296(US9040691, 24)
Affinity DataIC50:  140nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM160300(US9040691, 28)
Affinity DataIC50:  170nMAssay Description:In vitro enzyme inhibition using scintillation of incorporated radio label (flashplate assay). Test compounds diluted in DMSO are mixed with a suitab...More data for this Ligand-Target Pair
In DepthDetails US Patent