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Found 27 Enz. Inhib. hit(s) with all data for entry = 7291
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Merck Canada

US Patent
LigandPNGBDBM186602(US9168248, 75)
Affinity DataIC50:  1nMpH: 7.5Assay Description:The potency of compounds of formula I against the stearoyl-CoA desaturase was determined by measuring the conversion of radiolabeled stearoyl-CoA to ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Merck Canada

US Patent
LigandPNGBDBM186603(US9168248, 76)
Affinity DataIC50:  1nMpH: 7.5Assay Description:The potency of compounds of formula I against the stearoyl-CoA desaturase was determined by measuring the conversion of radiolabeled stearoyl-CoA to ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Merck Canada

US Patent
LigandPNGBDBM186597(US9168248, 42)
Affinity DataIC50:  1nMpH: 7.5Assay Description:The potency of compounds of formula I against the stearoyl-CoA desaturase was determined by measuring the conversion of radiolabeled stearoyl-CoA to ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Merck Canada

US Patent
LigandPNGBDBM186593(US9168248, 17)
Affinity DataIC50:  1nMpH: 7.5Assay Description:The potency of compounds of formula I against the stearoyl-CoA desaturase was determined by measuring the conversion of radiolabeled stearoyl-CoA to ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Merck Canada

US Patent
LigandPNGBDBM186592(US9168248, 16)
Affinity DataIC50:  1nMpH: 7.5Assay Description:The potency of compounds of formula I against the stearoyl-CoA desaturase was determined by measuring the conversion of radiolabeled stearoyl-CoA to ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Merck Canada

US Patent
LigandPNGBDBM186596(US9168248, 28)
Affinity DataIC50:  1nMpH: 7.5Assay Description:The potency of compounds of formula I against the stearoyl-CoA desaturase was determined by measuring the conversion of radiolabeled stearoyl-CoA to ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Merck Canada

US Patent
LigandPNGBDBM186595(US9168248, 22)
Affinity DataIC50:  1nMpH: 7.5Assay Description:The potency of compounds of formula I against the stearoyl-CoA desaturase was determined by measuring the conversion of radiolabeled stearoyl-CoA to ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Merck Canada

US Patent
LigandPNGBDBM186594(US9168248, 18)
Affinity DataIC50:  1nMpH: 7.5Assay Description:The potency of compounds of formula I against the stearoyl-CoA desaturase was determined by measuring the conversion of radiolabeled stearoyl-CoA to ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Merck Canada

US Patent
LigandPNGBDBM186600(US9168248, 68)
Affinity DataIC50:  3nMpH: 7.5Assay Description:The potency of compounds of formula I against the stearoyl-CoA desaturase was determined by measuring the conversion of radiolabeled stearoyl-CoA to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Merck Canada

US Patent
LigandPNGBDBM186577(US9168248, 1 | US9168248, 72)
Affinity DataIC50:  3nMpH: 7.5Assay Description:The potency of compounds of formula I against the stearoyl-CoA desaturase was determined by measuring the conversion of radiolabeled stearoyl-CoA to ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Merck Canada

US Patent
LigandPNGBDBM186578(US9168248, 2)
Affinity DataIC50:  11nMpH: 7.5Assay Description:The potency of compounds of formula I against the stearoyl-CoA desaturase was determined by measuring the conversion of radiolabeled stearoyl-CoA to ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Merck Canada

US Patent
LigandPNGBDBM186577(US9168248, 1 | US9168248, 72)
Affinity DataIC50:  12nMpH: 7.5Assay Description:The potency of compounds of formula I against the stearoyl-CoA desaturase was determined by measuring the conversion of radiolabeled stearoyl-CoA to ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Merck Canada

US Patent
LigandPNGBDBM186590(US9168248, 14)
Affinity DataIC50:  12nMpH: 7.5Assay Description:The potency of compounds of formula I against the stearoyl-CoA desaturase was determined by measuring the conversion of radiolabeled stearoyl-CoA to ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Merck Canada

US Patent
LigandPNGBDBM186587(US9168248, 11)
Affinity DataIC50:  13nMpH: 7.5Assay Description:The potency of compounds of formula I against the stearoyl-CoA desaturase was determined by measuring the conversion of radiolabeled stearoyl-CoA to ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Merck Canada

US Patent
LigandPNGBDBM186579(US9168248, 3)
Affinity DataIC50:  13nMpH: 7.5Assay Description:The potency of compounds of formula I against the stearoyl-CoA desaturase was determined by measuring the conversion of radiolabeled stearoyl-CoA to ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Merck Canada

US Patent
LigandPNGBDBM186591(US9168248, 15)
Affinity DataIC50:  17nMpH: 7.5Assay Description:The potency of compounds of formula I against the stearoyl-CoA desaturase was determined by measuring the conversion of radiolabeled stearoyl-CoA to ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Merck Canada

US Patent
LigandPNGBDBM186598(US9168248, 46)
Affinity DataIC50:  21nMpH: 7.5Assay Description:The potency of compounds of formula I against the stearoyl-CoA desaturase was determined by measuring the conversion of radiolabeled stearoyl-CoA to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Merck Canada

US Patent
LigandPNGBDBM186589(US9168248, 13)
Affinity DataIC50:  24nMpH: 7.5Assay Description:The potency of compounds of formula I against the stearoyl-CoA desaturase was determined by measuring the conversion of radiolabeled stearoyl-CoA to ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Merck Canada

US Patent
LigandPNGBDBM186580(US9168248, 4)
Affinity DataIC50:  41nMpH: 7.5Assay Description:The potency of compounds of formula I against the stearoyl-CoA desaturase was determined by measuring the conversion of radiolabeled stearoyl-CoA to ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Merck Canada

US Patent
LigandPNGBDBM186581(US9168248, 5)
Affinity DataIC50:  49nMpH: 7.5Assay Description:The potency of compounds of formula I against the stearoyl-CoA desaturase was determined by measuring the conversion of radiolabeled stearoyl-CoA to ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Merck Canada

US Patent
LigandPNGBDBM186599(US9168248, 54)
Affinity DataIC50:  62nMpH: 7.5Assay Description:The potency of compounds of formula I against the stearoyl-CoA desaturase was determined by measuring the conversion of radiolabeled stearoyl-CoA to ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Merck Canada

US Patent
LigandPNGBDBM186582(US9168248, 6)
Affinity DataIC50:  65nMpH: 7.5Assay Description:The potency of compounds of formula I against the stearoyl-CoA desaturase was determined by measuring the conversion of radiolabeled stearoyl-CoA to ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Merck Canada

US Patent
LigandPNGBDBM186585(US9168248, 9)
Affinity DataIC50:  181nMpH: 7.5Assay Description:The potency of compounds of formula I against the stearoyl-CoA desaturase was determined by measuring the conversion of radiolabeled stearoyl-CoA to ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Merck Canada

US Patent
LigandPNGBDBM186583(US9168248, 7)
Affinity DataIC50:  244nMpH: 7.5Assay Description:The potency of compounds of formula I against the stearoyl-CoA desaturase was determined by measuring the conversion of radiolabeled stearoyl-CoA to ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Merck Canada

US Patent
LigandPNGBDBM186586(US9168248, 10)
Affinity DataIC50:  338nMpH: 7.5Assay Description:The potency of compounds of formula I against the stearoyl-CoA desaturase was determined by measuring the conversion of radiolabeled stearoyl-CoA to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Merck Canada

US Patent
LigandPNGBDBM186588(US9168248, 12)
Affinity DataIC50:  366nMpH: 7.5Assay Description:The potency of compounds of formula I against the stearoyl-CoA desaturase was determined by measuring the conversion of radiolabeled stearoyl-CoA to ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Merck Canada

US Patent
LigandPNGBDBM186584(US9168248, 8)
Affinity DataIC50:  708nMpH: 7.5Assay Description:The potency of compounds of formula I against the stearoyl-CoA desaturase was determined by measuring the conversion of radiolabeled stearoyl-CoA to ...More data for this Ligand-Target Pair
In DepthDetails US Patent