Found 27 Enz. Inhib. hit(s) with all data for entry = 7327 
Affinity DataKi: 12.9nMpH: 7.4Assay Description:Membranes from recombinant HEK-293 cells expressing the human κ opioid receptor (cloned in house) were prepared by lysing cells in ice cold hypo...More data for this Ligand-Target Pair
Affinity DataKi: 21.8nMpH: 7.4Assay Description:Membranes from recombinant HEK-293 cells expressing the human κ opioid receptor (cloned in house) were prepared by lysing cells in ice cold hypo...More data for this Ligand-Target Pair
Affinity DataKi: 40.1nMpH: 7.4Assay Description:Membranes from recombinant HEK-293 cells expressing the human κ opioid receptor (cloned in house) were prepared by lysing cells in ice cold hypo...More data for this Ligand-Target Pair
Affinity DataKi: 49.9nM ΔG°: -45.2kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand dose-displacement binding assays for mu-opioid receptors used 0.3 nM [3H]-diprenorphine (Perkin Elmer, Shelton, Conn.), with 5 mg membran...More data for this Ligand-Target Pair
Affinity DataKi: 51.3nMpH: 7.4Assay Description:Membranes from recombinant HEK-293 cells expressing the human κ opioid receptor (cloned in house) were prepared by lysing cells in ice cold hypo...More data for this Ligand-Target Pair
Affinity DataKi: 52.2nMpH: 7.4Assay Description:Membranes from recombinant HEK-293 cells expressing the human κ opioid receptor (cloned in house) were prepared by lysing cells in ice cold hypo...More data for this Ligand-Target Pair
Affinity DataKi: 77.0nM ΔG°: -44.0kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand dose-displacement binding assays for mu-opioid receptors used 0.3 nM [3H]-diprenorphine (Perkin Elmer, Shelton, Conn.), with 5 mg membran...More data for this Ligand-Target Pair
Affinity DataKi: 123nM ΔG°: -42.8kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand dose-displacement binding assays for mu-opioid receptors used 0.3 nM [3H]-diprenorphine (Perkin Elmer, Shelton, Conn.), with 5 mg membran...More data for this Ligand-Target Pair
Affinity DataKi: 138nMpH: 7.4Assay Description:Membranes from recombinant HEK-293 cells expressing the human κ opioid receptor (cloned in house) were prepared by lysing cells in ice cold hypo...More data for this Ligand-Target Pair
Affinity DataKi: 278nM ΔG°: -40.6kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand dose-displacement binding assays for mu-opioid receptors used 0.3 nM [3H]-diprenorphine (Perkin Elmer, Shelton, Conn.), with 5 mg membran...More data for this Ligand-Target Pair
Affinity DataEC50: 745nMpH: 7.4 T: 2°CAssay Description:Membranes from recombinant HEK-293 cells, CHO cells expressing the
recombinant human kappa opioid receptor (kappa) were prepared by lysing
cells in...More data for this Ligand-Target Pair
Affinity DataEC50: 1.64E+3nMpH: 7.4 T: 2°CAssay Description:Membranes from recombinant HEK-293 cells, CHO cells expressing the
recombinant human kappa opioid receptor (kappa) were prepared by lysing
cells in...More data for this Ligand-Target Pair
Affinity DataEC50: 289nMpH: 7.4 T: 2°CAssay Description:Membranes from recombinant HEK-293 cells, CHO cells expressing the
recombinant human kappa opioid receptor (kappa) were prepared by lysing
cells in...More data for this Ligand-Target Pair
Affinity DataEC50: 1.77E+3nMpH: 7.4 T: 2°CAssay Description:Membranes from recombinant HEK-293 cells, CHO cells expressing the
recombinant human kappa opioid receptor (kappa) were prepared by lysing
cells in...More data for this Ligand-Target Pair
Affinity DataEC50: 771nMpH: 7.4 T: 2°CAssay Description:Membranes from recombinant HEK-293 cells, CHO cells expressing the
recombinant human kappa opioid receptor (kappa) were prepared by lysing
cells in...More data for this Ligand-Target Pair
Affinity DataEC50: 399nMpH: 7.4 T: 2°CAssay Description:Membranes from recombinant U-2 OS cells expressing the recombinant human
kappa opioid receptor (kappa) were prepared by lysing cells in ice cold
hy...More data for this Ligand-Target Pair
Affinity DataEC50: 122nMpH: 7.4 T: 2°CAssay Description:Membranes from recombinant HEK-293 cells, CHO cells expressing the
recombinant human kappa opioid receptor (kappa) were prepared by lysing
cells in...More data for this Ligand-Target Pair
Affinity DataEC50: 53nMpH: 7.4 T: 2°CAssay Description:[35S]GTPgammaS functional assays were conducted using freshly thawed
pt-receptor membranes prepared in-house from a cell line expressing
recombinan...More data for this Ligand-Target Pair
Affinity DataEC50: 173nMpH: 7.4 T: 2°CAssay Description:[35S]GTPgammaS functional assays were conducted using freshly thawed
pt-receptor membranes prepared in-house from a cell line expressing
recombinan...More data for this Ligand-Target Pair
Affinity DataEC50: 4.98E+3nMpH: 7.4 T: 2°CAssay Description:[35S]GTPgammaS functional assays were conducted using freshly thawed
pt-receptor membranes prepared in-house from a cell line expressing
recombinan...More data for this Ligand-Target Pair
Affinity DataEC50: 1.50E+4nMpH: 7.4 T: 2°CAssay Description:[35S]GTPgammaS functional assays were conducted using freshly thawed
pt-receptor membranes prepared in-house from a cell line expressing
recombinan...More data for this Ligand-Target Pair
Affinity DataEC50: 656nMpH: 7.4 T: 2°CAssay Description:[35S]GTPgammaS functional assays were conducted using freshly thawed
pt-receptor membranes prepared in-house from a cell line expressing
recombinan...More data for this Ligand-Target Pair
Affinity DataEC50: 68.3nMpH: 7.4 T: 2°CAssay Description:Membranes from recombinant U-2 OS cells expressing the recombinant human
kappa opioid receptor (kappa) were prepared by lysing cells in ice cold
hy...More data for this Ligand-Target Pair
Affinity DataEC50: 379nMpH: 7.4 T: 2°CAssay Description:[35S]GTPgammaS functional assays were conducted using freshly thawed
pt-receptor membranes prepared in-house from a cell line expressing
recombinan...More data for this Ligand-Target Pair
Affinity DataEC50: 174nMpH: 7.4 T: 2°CAssay Description:[35S]GTPgammaS functional assays were conducted using freshly thawed
pt-receptor membranes prepared in-house from a cell line expressing
recombinan...More data for this Ligand-Target Pair
Affinity DataEC50: 196nMpH: 7.4 T: 2°CAssay Description:[35S]GTPgammaS functional assays were conducted using freshly thawed
pt-receptor membranes prepared in-house from a cell line expressing
recombinan...More data for this Ligand-Target Pair
Affinity DataEC50: 457nMpH: 7.4 T: 2°CAssay Description:[35S]GTPgammaS functional assays were conducted using freshly thawed
pt-receptor membranes prepared in-house from a cell line expressing
recombinan...More data for this Ligand-Target Pair
