Compile Data Set for Download or QSAR
maximum 50k data
Found 12 Enz. Inhib. hit(s) with all data for entry = 7774
TargetNischarin(Homo sapiens (Human))
Universite De Strasbourg

US Patent
LigandPNGBDBM215802(US9303019, 8)
Affinity DataKi:  0.220nM ΔG°:  -57.3kJ/molepH: 7.35 T: 2°CAssay Description:Binding assays were performed at 37° C. using [125I]LNP 911 as radioligand following the general procedure described but adapted to washed whole ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNischarin(Homo sapiens (Human))
Universite De Strasbourg

US Patent
LigandPNGBDBM215805(US9303019, 20)
Affinity DataKi:  2.80nM ΔG°:  -50.8kJ/molepH: 7.35 T: 2°CAssay Description:Binding assays were performed at 37° C. using [125I]LNP 911 as radioligand following the general procedure described but adapted to washed whole ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNischarin(Homo sapiens (Human))
Universite De Strasbourg

US Patent
LigandPNGBDBM215803(US9303019, 9)
Affinity DataKi:  2.80nM ΔG°:  -50.8kJ/molepH: 7.35 T: 2°CAssay Description:Binding assays were performed at 37° C. using [125I]LNP 911 as radioligand following the general procedure described but adapted to washed whole ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNischarin(Homo sapiens (Human))
Universite De Strasbourg

US Patent
LigandPNGBDBM215800(US9303019, 1)
Affinity DataKi:  8.10nM ΔG°:  -48.0kJ/molepH: 7.35 T: 2°CAssay Description:Binding assays were performed at 37° C. using [125I]LNP 911 as radioligand following the general procedure described but adapted to washed whole ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNischarin(Homo sapiens (Human))
Universite De Strasbourg

US Patent
LigandPNGBDBM215801(US9303019, 5)
Affinity DataKi:  19nM ΔG°:  -45.8kJ/molepH: 7.35 T: 2°CAssay Description:Binding assays were performed at 37° C. using [125I]LNP 911 as radioligand following the general procedure described but adapted to washed whole ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNischarin(Homo sapiens (Human))
Universite De Strasbourg

US Patent
LigandPNGBDBM215804(US9303019, 13)
Affinity DataKi:  120nM ΔG°:  -41.1kJ/molepH: 7.35 T: 2°CAssay Description:Binding assays were performed at 37° C. using [125I]LNP 911 as radioligand following the general procedure described but adapted to washed whole ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Universite De Strasbourg

US Patent
LigandPNGBDBM215805(US9303019, 20)
Affinity DataKi: >1.00E+5nMpH: 7.5Assay Description:The membrane preparation was prepared as described by Newman-Tancredi, A.; Nicolas, J,-P.; Audinot, V.; Gavaudan, S.; Verriele, L.; Touzard, M.; Chap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Universite De Strasbourg

US Patent
LigandPNGBDBM215800(US9303019, 1)
Affinity DataKi: >1.00E+5nMpH: 7.5Assay Description:The membrane preparation was prepared as described by Newman-Tancredi, A.; Nicolas, J,-P.; Audinot, V.; Gavaudan, S.; Verriele, L.; Touzard, M.; Chap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Universite De Strasbourg

US Patent
LigandPNGBDBM215801(US9303019, 5)
Affinity DataKi: >1.00E+5nMpH: 7.5Assay Description:The membrane preparation was prepared as described by Newman-Tancredi, A.; Nicolas, J,-P.; Audinot, V.; Gavaudan, S.; Verriele, L.; Touzard, M.; Chap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Universite De Strasbourg

US Patent
LigandPNGBDBM215802(US9303019, 8)
Affinity DataKi: >1.00E+5nMpH: 7.5Assay Description:The membrane preparation was prepared as described by Newman-Tancredi, A.; Nicolas, J,-P.; Audinot, V.; Gavaudan, S.; Verriele, L.; Touzard, M.; Chap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Universite De Strasbourg

US Patent
LigandPNGBDBM215803(US9303019, 9)
Affinity DataKi: >1.00E+5nMpH: 7.5Assay Description:The membrane preparation was prepared as described by Newman-Tancredi, A.; Nicolas, J,-P.; Audinot, V.; Gavaudan, S.; Verriele, L.; Touzard, M.; Chap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Universite De Strasbourg

US Patent
LigandPNGBDBM215804(US9303019, 13)
Affinity DataKi: >1.00E+5nMpH: 7.5Assay Description:The membrane preparation was prepared as described by Newman-Tancredi, A.; Nicolas, J,-P.; Audinot, V.; Gavaudan, S.; Verriele, L.; Touzard, M.; Chap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent