Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 7834
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Xuanzhu Pharma

US Patent
LigandPNGBDBM221893(US9315438, Compound represented by formula (II))
Affinity DataIC50:  2.5nMT: 2°CAssay Description:Human SGLT-2 and SGLT-1 sequences were stably expressed in the CHO cells. The cell culture was conducted in a 96-well plate for 12 hr. The plate was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Xuanzhu Pharma

US Patent
LigandPNGBDBM221897(US9315438, Reference compound 1)
Affinity DataIC50:  3.63nMT: 2°CAssay Description:Human SGLT-2 and SGLT-1 sequences were stably expressed in the CHO cells. The cell culture was conducted in a 96-well plate for 12 hr. The plate was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Xuanzhu Pharma

US Patent
LigandPNGBDBM221894(US9315438, Compound represented by formula (III))
Affinity DataIC50:  7.83nMT: 2°CAssay Description:Human SGLT-2 and SGLT-1 sequences were stably expressed in the CHO cells. The cell culture was conducted in a 96-well plate for 12 hr. The plate was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Xuanzhu Pharma

US Patent
LigandPNGBDBM221896(US9315438, Compound represented by formula (V))
Affinity DataIC50:  282nMT: 2°CAssay Description:Human SGLT-2 and SGLT-1 sequences were stably expressed in the CHO cells. The cell culture was conducted in a 96-well plate for 12 hr. The plate was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Xuanzhu Pharma

US Patent
LigandPNGBDBM221895(US9315438, Compound represented by formula (IV))
Affinity DataIC50:  1.11E+3nMT: 2°CAssay Description:Human SGLT-2 and SGLT-1 sequences were stably expressed in the CHO cells. The cell culture was conducted in a 96-well plate for 12 hr. The plate was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Xuanzhu Pharma

US Patent
LigandPNGBDBM221897(US9315438, Reference compound 1)
Affinity DataIC50:  2.40E+3nMT: 2°CAssay Description:Human SGLT-2 and SGLT-1 sequences were stably expressed in the CHO cells. The cell culture was conducted in a 96-well plate for 12 hr. The plate was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Xuanzhu Pharma

US Patent
LigandPNGBDBM221894(US9315438, Compound represented by formula (III))
Affinity DataIC50:  3.08E+3nMT: 2°CAssay Description:Human SGLT-2 and SGLT-1 sequences were stably expressed in the CHO cells. The cell culture was conducted in a 96-well plate for 12 hr. The plate was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Xuanzhu Pharma

US Patent
LigandPNGBDBM221893(US9315438, Compound represented by formula (II))
Affinity DataIC50:  1.72E+4nMT: 2°CAssay Description:Human SGLT-2 and SGLT-1 sequences were stably expressed in the CHO cells. The cell culture was conducted in a 96-well plate for 12 hr. The plate was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Xuanzhu Pharma

US Patent
LigandPNGBDBM221896(US9315438, Compound represented by formula (V))
Affinity DataIC50:  7.55E+4nMT: 2°CAssay Description:Human SGLT-2 and SGLT-1 sequences were stably expressed in the CHO cells. The cell culture was conducted in a 96-well plate for 12 hr. The plate was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Xuanzhu Pharma

US Patent
LigandPNGBDBM221895(US9315438, Compound represented by formula (IV))
Affinity DataIC50:  1.11E+5nMT: 2°CAssay Description:Human SGLT-2 and SGLT-1 sequences were stably expressed in the CHO cells. The cell culture was conducted in a 96-well plate for 12 hr. The plate was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent