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Patent code US9353116

Compile Data Set for Download or QSAR
Found 62 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Proto-oncogene tyrosine-protein kinase Src (T338C/V323S)


(Gallus gallus (Chicken))
BDBM234844
PNG
(US9353116, 13)
Show SMILES CC(C)n1nc(Cc2cccc(c2)C(=O)CF)c2c(N)ncnc12
Show InChI InChI=1S/C17H18FN5O/c1-10(2)23-17-15(16(19)20-9-21-17)13(22-23)7-11-4-3-5-12(6-11)14(24)8-18/h3-6,9-10H,7-8H2,1-2H3,(H2,19,20,21)
PDB

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UniChem
US Patent
n/an/a 29n/an/an/an/an/an/a



The Regents of the University of California

US Patent


Assay Description
In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


Citation and Details
More data for this
Ligand-Target Pair
Leucine-rich repeat serine/threonine-protein kinase 2 G2019S


(Homo sapiens (Human))
BDBM234860
PNG
(US9353116, 19 | US9353116, Fig. 16, Compound 1)
Show SMILES COc1cc2ncnc(Nc3cccc(NS(=O)(=O)C=C)c3)c2cc1OC
Show InChI InChI=1S/C18H18N4O4S/c1-4-27(23,24)22-13-7-5-6-12(8-13)21-18-14-9-16(25-2)17(26-3)10-15(14)19-11-20-18/h4-11,22H,1H2,2-3H3,(H,19,20,21)
PDB

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US Patent
n/an/a 45.5n/an/an/an/an/an/a



The Regents of the University of California

US Patent


Assay Description
In vitro kinase assays using LRRK WT and LRRK G2019S.


Citation and Details
More data for this
Ligand-Target Pair
Leucine-rich repeat serine/threonine-protein kinase 2 G2019S


(Homo sapiens (Human))
BDBM234866
PNG
(US9353116, Fig. 16, Compound 5)
Show SMILES COc1cc2ncnc(Nc3cccc(NS(=O)(=O)c4ccccc4)c3)c2cc1OC
Show InChI InChI=1S/C22H20N4O4S/c1-29-20-12-18-19(13-21(20)30-2)23-14-24-22(18)25-15-7-6-8-16(11-15)26-31(27,28)17-9-4-3-5-10-17/h3-14,26H,1-2H3,(H,23,24,25)
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US Patent
n/an/a 46.9n/an/an/an/an/an/a



The Regents of the University of California

US Patent


Assay Description
In vitro kinase assays using LRRK WT and LRRK G2019S.


Citation and Details
More data for this
Ligand-Target Pair
Leucine-rich repeat serine/threonine-protein kinase 2 G2019S


(Homo sapiens (Human))
BDBM234867
PNG
(US9353116, Fig. 16, Compound 6)
Show SMILES COc1cc2ncnc(Nc3cccc(NS(=O)(=O)c4cccs4)c3)c2cc1OC
Show InChI InChI=1S/C20H18N4O4S2/c1-27-17-10-15-16(11-18(17)28-2)21-12-22-20(15)23-13-5-3-6-14(9-13)24-30(25,26)19-7-4-8-29-19/h3-12,24H,1-2H3,(H,21,22,23)
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US Patent
n/an/a 57.7n/an/an/an/an/an/a



The Regents of the University of California

US Patent


Assay Description
In vitro kinase assays using LRRK WT and LRRK G2019S.


Citation and Details
More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (T338C/V323A)


(Gallus gallus (Chicken))
BDBM234843
PNG
(US9353116, 3)
Show SMILES CC(C)n1nc(-c2cccc(NS(=O)(=O)C=C)c2)c2c(N)ncnc12
Show InChI InChI=1S/C16H18N6O2S/c1-4-25(23,24)21-12-7-5-6-11(8-12)14-13-15(17)18-9-19-16(13)22(20-14)10(2)3/h4-10,21H,1H2,2-3H3,(H2,17,18,19)
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US Patent
n/an/a 63n/an/an/an/an/an/a



The Regents of the University of California

US Patent


Assay Description
In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


Citation and Details
More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (T338C/V323A)


(Gallus gallus (Chicken))
BDBM234844
PNG
(US9353116, 13)
Show SMILES CC(C)n1nc(Cc2cccc(c2)C(=O)CF)c2c(N)ncnc12
Show InChI InChI=1S/C17H18FN5O/c1-10(2)23-17-15(16(19)20-9-21-17)13(22-23)7-11-4-3-5-12(6-11)14(24)8-18/h3-6,9-10H,7-8H2,1-2H3,(H2,19,20,21)
PDB

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US Patent
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The Regents of the University of California

US Patent


Assay Description
In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


Citation and Details
More data for this
Ligand-Target Pair
Leucine-rich repeat serine/threonine-protein kinase 2 G2019S


(Homo sapiens (Human))
BDBM234862
PNG
(US9353116, Fig. 16, Compound 4)
Show SMILES COc1cc2ncnc(Nc3cccc(NS(=O)(=O)CC(C)C)c3)c2cc1OC
Show InChI InChI=1S/C20H24N4O4S/c1-13(2)11-29(25,26)24-15-7-5-6-14(8-15)23-20-16-9-18(27-3)19(28-4)10-17(16)21-12-22-20/h5-10,12-13,24H,11H2,1-4H3,(H,21,22,23)
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n/an/a 90.1n/an/an/an/an/an/a



The Regents of the University of California

US Patent


Assay Description
In vitro kinase assays using LRRK WT and LRRK G2019S.


Citation and Details
More data for this
Ligand-Target Pair
Leucine-rich repeat serine/threonine-protein kinase 2 G2019S


(Homo sapiens (Human))
BDBM234863
PNG
(US9353116, Fig. 16, Compound 2)
Show SMILES COc1cc2ncnc(Nc3cccc(NS(C)(=O)=O)c3)c2cc1OC
Show InChI InChI=1S/C17H18N4O4S/c1-24-15-8-13-14(9-16(15)25-2)18-10-19-17(13)20-11-5-4-6-12(7-11)21-26(3,22)23/h4-10,21H,1-3H3,(H,18,19,20)
PDB

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The Regents of the University of California

US Patent


Assay Description
In vitro kinase assays using LRRK WT and LRRK G2019S.


Citation and Details
More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (T338C)


(Gallus gallus (Chicken))
BDBM234843
PNG
(US9353116, 3)
Show SMILES CC(C)n1nc(-c2cccc(NS(=O)(=O)C=C)c2)c2c(N)ncnc12
Show InChI InChI=1S/C16H18N6O2S/c1-4-25(23,24)21-12-7-5-6-11(8-12)14-13-15(17)18-9-19-16(13)22(20-14)10(2)3/h4-10,21H,1H2,2-3H3,(H2,17,18,19)
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US Patent
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The Regents of the University of California

US Patent


Assay Description
In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


Citation and Details
More data for this
Ligand-Target Pair
Leucine-rich repeat serine/threonine-protein kinase 2 G2019S


(Homo sapiens (Human))
BDBM234869
PNG
(US9353116, Fig. 16, Compound 8)
Show SMILES CCS(=O)(=O)Nc1cccc(Nc2ncnc3cc(OC)c(OC)cc23)c1
Show InChI InChI=1S/C18H20N4O4S/c1-4-27(23,24)22-13-7-5-6-12(8-13)21-18-14-9-16(25-2)17(26-3)10-15(14)19-11-20-18/h5-11,22H,4H2,1-3H3,(H,19,20,21)
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The Regents of the University of California

US Patent


Assay Description
In vitro kinase assays using LRRK WT and LRRK G2019S.


Citation and Details
More data for this
Ligand-Target Pair
Leucine-rich repeat serine/threonine-protein kinase 2 G2019S


(Homo sapiens (Human))
BDBM234865
PNG
(US9353116, Fig. 16, Compound 3)
Show SMILES CCCS(=O)(=O)Nc1cccc(Nc2ncnc3cc(OC)c(OC)cc23)c1
Show InChI InChI=1S/C19H22N4O4S/c1-4-8-28(24,25)23-14-7-5-6-13(9-14)22-19-15-10-17(26-2)18(27-3)11-16(15)20-12-21-19/h5-7,9-12,23H,4,8H2,1-3H3,(H,20,21,22)
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The Regents of the University of California

US Patent


Assay Description
In vitro kinase assays using LRRK WT and LRRK G2019S.


Citation and Details
More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (T338C/V323S)


(Gallus gallus (Chicken))
BDBM234843
PNG
(US9353116, 3)
Show SMILES CC(C)n1nc(-c2cccc(NS(=O)(=O)C=C)c2)c2c(N)ncnc12
Show InChI InChI=1S/C16H18N6O2S/c1-4-25(23,24)21-12-7-5-6-11(8-12)14-13-15(17)18-9-19-16(13)22(20-14)10(2)3/h4-10,21H,1H2,2-3H3,(H2,17,18,19)
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The Regents of the University of California

US Patent


Assay Description
In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


Citation and Details
More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (T338C)


(Gallus gallus (Chicken))
BDBM234848
PNG
(US9353116, 5)
Show SMILES CC(C)n1nc(-c2ccc(NS(=O)(=O)C=C)cc2)c2c(N)ncnc12
Show InChI InChI=1S/C16H18N6O2S/c1-4-25(23,24)21-12-7-5-11(6-8-12)14-13-15(17)18-9-19-16(13)22(20-14)10(2)3/h4-10,21H,1H2,2-3H3,(H2,17,18,19)
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The Regents of the University of California

US Patent


Assay Description
In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


Citation and Details
More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (T338C)


(Gallus gallus (Chicken))
BDBM50403061
PNG
(CHEMBL2216823 | US9353116, 9)
Show SMILES CC(C)n1nc(Cc2cccc(NS(=O)(=O)C=C)c2)c2c(N)ncnc12
Show InChI InChI=1S/C17H20N6O2S/c1-4-26(24,25)22-13-7-5-6-12(8-13)9-14-15-16(18)19-10-20-17(15)23(21-14)11(2)3/h4-8,10-11,22H,1,9H2,2-3H3,(H2,18,19,20)
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US Patent


Assay Description
In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


Citation and Details
More data for this
Ligand-Target Pair
Leucine-rich repeat serine/threonine-protein kinase 2 (LRRK2)


(Homo sapiens (Human))
BDBM234866
PNG
(US9353116, Fig. 16, Compound 5)
Show SMILES COc1cc2ncnc(Nc3cccc(NS(=O)(=O)c4ccccc4)c3)c2cc1OC
Show InChI InChI=1S/C22H20N4O4S/c1-29-20-12-18-19(13-21(20)30-2)23-14-24-22(18)25-15-7-6-8-16(11-15)26-31(27,28)17-9-4-3-5-10-17/h3-14,26H,1-2H3,(H,23,24,25)
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The Regents of the University of California

US Patent


Assay Description
In vitro kinase assays using LRRK WT and LRRK G2019S.


Citation and Details
More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (T338C)


(Gallus gallus (Chicken))
BDBM234858
PNG
(US9353116, 17)
Show SMILES Nc1ncnc2n(nc(Cc3cccc(NS(=O)(=O)C=C)c3)c12)C1CCCC1
Show InChI InChI=1S/C19H22N6O2S/c1-2-28(26,27)24-14-7-5-6-13(10-14)11-16-17-18(20)21-12-22-19(17)25(23-16)15-8-3-4-9-15/h2,5-7,10,12,15,24H,1,3-4,8-9,11H2,(H2,20,21,22)
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The Regents of the University of California

US Patent


Assay Description
In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


Citation and Details
More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (T338C/V323A)


(Gallus gallus (Chicken))
BDBM50403061
PNG
(CHEMBL2216823 | US9353116, 9)
Show SMILES CC(C)n1nc(Cc2cccc(NS(=O)(=O)C=C)c2)c2c(N)ncnc12
Show InChI InChI=1S/C17H20N6O2S/c1-4-26(24,25)22-13-7-5-6-12(8-13)9-14-15-16(18)19-10-20-17(15)23(21-14)11(2)3/h4-8,10-11,22H,1,9H2,2-3H3,(H2,18,19,20)
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The Regents of the University of California

US Patent


Assay Description
In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


Citation and Details
More data for this
Ligand-Target Pair
Leucine-rich repeat serine/threonine-protein kinase 2 (LRRK2)


(Homo sapiens (Human))
BDBM234860
PNG
(US9353116, 19 | US9353116, Fig. 16, Compound 1)
Show SMILES COc1cc2ncnc(Nc3cccc(NS(=O)(=O)C=C)c3)c2cc1OC
Show InChI InChI=1S/C18H18N4O4S/c1-4-27(23,24)22-13-7-5-6-12(8-13)21-18-14-9-16(25-2)17(26-3)10-15(14)19-11-20-18/h4-11,22H,1H2,2-3H3,(H,19,20,21)
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US Patent


Assay Description
In vitro kinase assays using LRRK WT and LRRK G2019S.


Citation and Details
More data for this
Ligand-Target Pair
Leucine-rich repeat serine/threonine-protein kinase 2 (LRRK2)


(Homo sapiens (Human))
BDBM234862
PNG
(US9353116, Fig. 16, Compound 4)
Show SMILES COc1cc2ncnc(Nc3cccc(NS(=O)(=O)CC(C)C)c3)c2cc1OC
Show InChI InChI=1S/C20H24N4O4S/c1-13(2)11-29(25,26)24-15-7-5-6-14(8-15)23-20-16-9-18(27-3)19(28-4)10-17(16)21-12-22-20/h5-10,12-13,24H,11H2,1-4H3,(H,21,22,23)
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Assay Description
In vitro kinase assays using LRRK WT and LRRK G2019S.


Citation and Details
More data for this
Ligand-Target Pair
Leucine-rich repeat serine/threonine-protein kinase 2 G2019S


(Homo sapiens (Human))
BDBM234868
PNG
(US9353116, Fig. 16, Compound 7)
Show SMILES COc1cc2ncnc(Nc3cccc(NS(=O)(=O)CC(F)(F)F)c3)c2cc1OC
Show InChI InChI=1S/C18H17F3N4O4S/c1-28-15-7-13-14(8-16(15)29-2)22-10-23-17(13)24-11-4-3-5-12(6-11)25-30(26,27)9-18(19,20)21/h3-8,10,25H,9H2,1-2H3,(H,22,23,24)
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US Patent


Assay Description
In vitro kinase assays using LRRK WT and LRRK G2019S.


Citation and Details
More data for this
Ligand-Target Pair
Leucine-rich repeat serine/threonine-protein kinase 2 (LRRK2)


(Homo sapiens (Human))
BDBM234867
PNG
(US9353116, Fig. 16, Compound 6)
Show SMILES COc1cc2ncnc(Nc3cccc(NS(=O)(=O)c4cccs4)c3)c2cc1OC
Show InChI InChI=1S/C20H18N4O4S2/c1-27-17-10-15-16(11-18(17)28-2)21-12-22-20(15)23-13-5-3-6-14(9-13)24-30(25,26)19-7-4-8-29-19/h3-12,24H,1-2H3,(H,21,22,23)
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US Patent


Assay Description
In vitro kinase assays using LRRK WT and LRRK G2019S.


Citation and Details
More data for this
Ligand-Target Pair
Leucine-rich repeat serine/threonine-protein kinase 2 (LRRK2)


(Homo sapiens (Human))
BDBM234869
PNG
(US9353116, Fig. 16, Compound 8)
Show SMILES CCS(=O)(=O)Nc1cccc(Nc2ncnc3cc(OC)c(OC)cc23)c1
Show InChI InChI=1S/C18H20N4O4S/c1-4-27(23,24)22-13-7-5-6-12(8-13)21-18-14-9-16(25-2)17(26-3)10-15(14)19-11-20-18/h5-11,22H,4H2,1-3H3,(H,19,20,21)
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The Regents of the University of California

US Patent


Assay Description
In vitro kinase assays using LRRK WT and LRRK G2019S.


Citation and Details
More data for this
Ligand-Target Pair
Leucine-rich repeat serine/threonine-protein kinase 2 (LRRK2)


(Homo sapiens (Human))
BDBM234865
PNG
(US9353116, Fig. 16, Compound 3)
Show SMILES CCCS(=O)(=O)Nc1cccc(Nc2ncnc3cc(OC)c(OC)cc23)c1
Show InChI InChI=1S/C19H22N4O4S/c1-4-8-28(24,25)23-14-7-5-6-13(9-14)22-19-15-10-17(26-2)18(27-3)11-16(15)20-12-21-19/h5-7,9-12,23H,4,8H2,1-3H3,(H,20,21,22)
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US Patent


Assay Description
In vitro kinase assays using LRRK WT and LRRK G2019S.


Citation and Details
More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (T338C)


(Gallus gallus (Chicken))
BDBM234844
PNG
(US9353116, 13)
Show SMILES CC(C)n1nc(Cc2cccc(c2)C(=O)CF)c2c(N)ncnc12
Show InChI InChI=1S/C17H18FN5O/c1-10(2)23-17-15(16(19)20-9-21-17)13(22-23)7-11-4-3-5-12(6-11)14(24)8-18/h3-6,9-10H,7-8H2,1-2H3,(H2,19,20,21)
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The Regents of the University of California

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Assay Description
In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


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More data for this
Ligand-Target Pair
Leucine-rich repeat serine/threonine-protein kinase 2 (LRRK2)


(Homo sapiens (Human))
BDBM234863
PNG
(US9353116, Fig. 16, Compound 2)
Show SMILES COc1cc2ncnc(Nc3cccc(NS(C)(=O)=O)c3)c2cc1OC
Show InChI InChI=1S/C17H18N4O4S/c1-24-15-8-13-14(9-16(15)25-2)18-10-19-17(13)20-11-5-4-6-12(7-11)21-26(3,22)23/h4-10,21H,1-3H3,(H,18,19,20)
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Assay Description
In vitro kinase assays using LRRK WT and LRRK G2019S.


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More data for this
Ligand-Target Pair
Leucine-rich repeat serine/threonine-protein kinase 2 (LRRK2)


(Homo sapiens (Human))
BDBM234868
PNG
(US9353116, Fig. 16, Compound 7)
Show SMILES COc1cc2ncnc(Nc3cccc(NS(=O)(=O)CC(F)(F)F)c3)c2cc1OC
Show InChI InChI=1S/C18H17F3N4O4S/c1-28-15-7-13-14(8-16(15)29-2)22-10-23-17(13)24-11-4-3-5-12(6-11)25-30(26,27)9-18(19,20)21/h3-8,10,25H,9H2,1-2H3,(H,22,23,24)
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In vitro kinase assays using LRRK WT and LRRK G2019S.


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More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (T338C)


(Gallus gallus (Chicken))
BDBM234845
PNG
(US9353116, 1)
Show SMILES CC(C)n1nc(-c2cccc(NC(=O)C=C)c2)c2c(N)ncnc12
Show InChI InChI=1S/C17H18N6O/c1-4-13(24)21-12-7-5-6-11(8-12)15-14-16(18)19-9-20-17(14)23(22-15)10(2)3/h4-10H,1H2,2-3H3,(H,21,24)(H2,18,19,20)
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In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


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More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (T338C/V323S)


(Gallus gallus (Chicken))
BDBM50403061
PNG
(CHEMBL2216823 | US9353116, 9)
Show SMILES CC(C)n1nc(Cc2cccc(NS(=O)(=O)C=C)c2)c2c(N)ncnc12
Show InChI InChI=1S/C17H20N6O2S/c1-4-26(24,25)22-13-7-5-6-12(8-13)9-14-15-16(18)19-10-20-17(15)23(21-14)11(2)3/h4-8,10-11,22H,1,9H2,2-3H3,(H2,18,19,20)
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Assay Description
In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


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More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (T338C)


(Gallus gallus (Chicken))
BDBM234861
PNG
(US9353116, 20)
Show SMILES COc1cc2ncnc(Nc3ccc(NS(=O)(=O)C=C)cc3)c2cc1OC
Show InChI InChI=1S/C18H18N4O4S/c1-4-27(23,24)22-13-7-5-12(6-8-13)21-18-14-9-16(25-2)17(26-3)10-15(14)19-11-20-18/h4-11,22H,1H2,2-3H3,(H,19,20,21)
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In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


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More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (T338C)


(Gallus gallus (Chicken))
BDBM234857
PNG
(US9353116, 16)
Show SMILES CC(C)(C)n1nc(Cc2cccc(NS(=O)(=O)C=C)c2)c2c(N)ncnc12
Show InChI InChI=1S/C18H22N6O2S/c1-5-27(25,26)23-13-8-6-7-12(9-13)10-14-15-16(19)20-11-21-17(15)24(22-14)18(2,3)4/h5-9,11,23H,1,10H2,2-4H3,(H2,19,20,21)
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In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


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More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (T338C)


(Gallus gallus (Chicken))
BDBM234849
PNG
(US9353116, 6)
Show SMILES CC(C)n1nc(-c2cccc(NC(=O)CCl)c2)c2c(N)ncnc12
Show InChI InChI=1S/C16H17ClN6O/c1-9(2)23-16-13(15(18)19-8-20-16)14(22-23)10-4-3-5-11(6-10)21-12(24)7-17/h3-6,8-9H,7H2,1-2H3,(H,21,24)(H2,18,19,20)
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In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


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More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (c-Src)


(Gallus gallus (Chicken))
BDBM234848
PNG
(US9353116, 5)
Show SMILES CC(C)n1nc(-c2ccc(NS(=O)(=O)C=C)cc2)c2c(N)ncnc12
Show InChI InChI=1S/C16H18N6O2S/c1-4-25(23,24)21-12-7-5-11(6-8-12)14-13-15(17)18-9-19-16(13)22(20-14)10(2)3/h4-10,21H,1H2,2-3H3,(H2,17,18,19)
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In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


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More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (c-Src)


(Gallus gallus (Chicken))
BDBM234843
PNG
(US9353116, 3)
Show SMILES CC(C)n1nc(-c2cccc(NS(=O)(=O)C=C)c2)c2c(N)ncnc12
Show InChI InChI=1S/C16H18N6O2S/c1-4-25(23,24)21-12-7-5-6-11(8-12)14-13-15(17)18-9-19-16(13)22(20-14)10(2)3/h4-10,21H,1H2,2-3H3,(H2,17,18,19)
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In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


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More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (T338C)


(Gallus gallus (Chicken))
BDBM234860
PNG
(US9353116, 19 | US9353116, Fig. 16, Compound 1)
Show SMILES COc1cc2ncnc(Nc3cccc(NS(=O)(=O)C=C)c3)c2cc1OC
Show InChI InChI=1S/C18H18N4O4S/c1-4-27(23,24)22-13-7-5-6-12(8-13)21-18-14-9-16(25-2)17(26-3)10-15(14)19-11-20-18/h4-11,22H,1H2,2-3H3,(H,19,20,21)
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In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


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More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (T338C)


(Gallus gallus (Chicken))
BDBM234859
PNG
(US9353116, 18)
Show SMILES COc1cc2ncnc(Nc3cccc(NC(=O)C=C)c3)c2cc1OC
Show InChI InChI=1S/C19H18N4O3/c1-4-18(24)22-12-6-5-7-13(8-12)23-19-14-9-16(25-2)17(26-3)10-15(14)20-11-21-19/h4-11H,1H2,2-3H3,(H,22,24)(H,20,21,23)
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In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


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More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (T338C)


(Gallus gallus (Chicken))
BDBM234852
PNG
(US9353116, 10)
Show SMILES CC(C)n1nc(Cc2ccc(NS(=O)(=O)C=C)cc2)c2c(N)ncnc12
Show InChI InChI=1S/C17H20N6O2S/c1-4-26(24,25)22-13-7-5-12(6-8-13)9-14-15-16(18)19-10-20-17(15)23(21-14)11(2)3/h4-8,10-11,22H,1,9H2,2-3H3,(H2,18,19,20)
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Assay Description
In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


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More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (c-Src)


(Gallus gallus (Chicken))
BDBM234861
PNG
(US9353116, 20)
Show SMILES COc1cc2ncnc(Nc3ccc(NS(=O)(=O)C=C)cc3)c2cc1OC
Show InChI InChI=1S/C18H18N4O4S/c1-4-27(23,24)22-13-7-5-12(6-8-13)21-18-14-9-16(25-2)17(26-3)10-15(14)19-11-20-18/h4-11,22H,1H2,2-3H3,(H,19,20,21)
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In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


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More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (c-Src)


(Gallus gallus (Chicken))
BDBM234845
PNG
(US9353116, 1)
Show SMILES CC(C)n1nc(-c2cccc(NC(=O)C=C)c2)c2c(N)ncnc12
Show InChI InChI=1S/C17H18N6O/c1-4-13(24)21-12-7-5-6-11(8-12)15-14-16(18)19-9-20-17(14)23(22-15)10(2)3/h4-10H,1H2,2-3H3,(H,21,24)(H2,18,19,20)
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In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


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More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (T338C)


(Gallus gallus (Chicken))
BDBM234850
PNG
(US9353116, 7)
Show SMILES CC(C)n1nc(Cc2cccc(NC(=O)C=C)c2)c2c(N)ncnc12
Show InChI InChI=1S/C18H20N6O/c1-4-15(25)22-13-7-5-6-12(8-13)9-14-16-17(19)20-10-21-18(16)24(23-14)11(2)3/h4-8,10-11H,1,9H2,2-3H3,(H,22,25)(H2,19,20,21)
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In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


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More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (c-Src)


(Gallus gallus (Chicken))
BDBM234852
PNG
(US9353116, 10)
Show SMILES CC(C)n1nc(Cc2ccc(NS(=O)(=O)C=C)cc2)c2c(N)ncnc12
Show InChI InChI=1S/C17H20N6O2S/c1-4-26(24,25)22-13-7-5-12(6-8-13)9-14-15-16(18)19-10-20-17(15)23(21-14)11(2)3/h4-8,10-11,22H,1,9H2,2-3H3,(H2,18,19,20)
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In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


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More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (T338C)


(Gallus gallus (Chicken))
BDBM234856
PNG
(US9353116, 15)
Show SMILES Cn1nc(Cc2cccc(NS(=O)(=O)C=C)c2)c2c(N)ncnc12
Show InChI InChI=1S/C15H16N6O2S/c1-3-24(22,23)20-11-6-4-5-10(7-11)8-12-13-14(16)17-9-18-15(13)21(2)19-12/h3-7,9,20H,1,8H2,2H3,(H2,16,17,18)
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In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


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More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (T338C)


(Gallus gallus (Chicken))
BDBM234853
PNG
(US9353116, 11)
Show SMILES CCS(=O)(=O)Nc1cccc(Cc2nn(C(C)C)c3ncnc(N)c23)c1
Show InChI InChI=1S/C17H22N6O2S/c1-4-26(24,25)22-13-7-5-6-12(8-13)9-14-15-16(18)19-10-20-17(15)23(21-14)11(2)3/h5-8,10-11,22H,4,9H2,1-3H3,(H2,18,19,20)
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Assay Description
In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


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More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (T338C)


(Gallus gallus (Chicken))
BDBM234855
PNG
(US9353116, 14)
Show SMILES CC(C)n1nc(Cc2cccc(c2)C(C)=O)c2c(N)ncnc12
Show InChI InChI=1S/C17H19N5O/c1-10(2)22-17-15(16(18)19-9-20-17)14(21-22)8-12-5-4-6-13(7-12)11(3)23/h4-7,9-10H,8H2,1-3H3,(H2,18,19,20)
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In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


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More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (T338C)


(Gallus gallus (Chicken))
BDBM234851
PNG
(US9353116, 8)
Show SMILES CC(C)n1nc(Cc2ccc(NC(=O)C=C)cc2)c2c(N)ncnc12
Show InChI InChI=1S/C18H20N6O/c1-4-15(25)22-13-7-5-12(6-8-13)9-14-16-17(19)20-10-21-18(16)24(23-14)11(2)3/h4-8,10-11H,1,9H2,2-3H3,(H,22,25)(H2,19,20,21)
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In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


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More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (c-Src)


(Gallus gallus (Chicken))
BDBM234857
PNG
(US9353116, 16)
Show SMILES CC(C)(C)n1nc(Cc2cccc(NS(=O)(=O)C=C)c2)c2c(N)ncnc12
Show InChI InChI=1S/C18H22N6O2S/c1-5-27(25,26)23-13-8-6-7-12(9-13)10-14-15-16(19)20-11-21-17(15)24(22-14)18(2,3)4/h5-9,11,23H,1,10H2,2-4H3,(H2,19,20,21)
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In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


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More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (c-Src)


(Gallus gallus (Chicken))
BDBM234850
PNG
(US9353116, 7)
Show SMILES CC(C)n1nc(Cc2cccc(NC(=O)C=C)c2)c2c(N)ncnc12
Show InChI InChI=1S/C18H20N6O/c1-4-15(25)22-13-7-5-6-12(8-13)9-14-16-17(19)20-10-21-18(16)24(23-14)11(2)3/h4-8,10-11H,1,9H2,2-3H3,(H,22,25)(H2,19,20,21)
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In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


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More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (c-Src)


(Gallus gallus (Chicken))
BDBM234854
PNG
(US9353116, 12)
Show SMILES CC(C)n1nc(Cc2cccc(NC(=O)CCl)c2)c2c(N)ncnc12
Show InChI InChI=1S/C17H19ClN6O/c1-10(2)24-17-15(16(19)20-9-21-17)13(23-24)7-11-4-3-5-12(6-11)22-14(25)8-18/h3-6,9-10H,7-8H2,1-2H3,(H,22,25)(H2,19,20,21)
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In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


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More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (c-Src)


(Gallus gallus (Chicken))
BDBM234860
PNG
(US9353116, 19 | US9353116, Fig. 16, Compound 1)
Show SMILES COc1cc2ncnc(Nc3cccc(NS(=O)(=O)C=C)c3)c2cc1OC
Show InChI InChI=1S/C18H18N4O4S/c1-4-27(23,24)22-13-7-5-6-12(8-13)21-18-14-9-16(25-2)17(26-3)10-15(14)19-11-20-18/h4-11,22H,1H2,2-3H3,(H,19,20,21)
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In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


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More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (c-Src)


(Gallus gallus (Chicken))
BDBM234846
PNG
(US9353116, 2)
Show SMILES CC(C)n1nc(-c2cccc(NC(=O)C=C)c2)c2cncnc12
Show InChI InChI=1S/C17H17N5O/c1-4-15(23)20-13-7-5-6-12(8-13)16-14-9-18-10-19-17(14)22(21-16)11(2)3/h4-11H,1H2,2-3H3,(H,20,23)
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Assay Description
In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


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More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (c-Src)


(Gallus gallus (Chicken))
BDBM234859
PNG
(US9353116, 18)
Show SMILES COc1cc2ncnc(Nc3cccc(NC(=O)C=C)c3)c2cc1OC
Show InChI InChI=1S/C19H18N4O3/c1-4-18(24)22-12-6-5-7-13(8-12)23-19-14-9-16(25-2)17(26-3)10-15(14)20-11-21-19/h4-11H,1H2,2-3H3,(H,22,24)(H,20,21,23)
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In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


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More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (c-Src)


(Gallus gallus (Chicken))
BDBM234858
PNG
(US9353116, 17)
Show SMILES Nc1ncnc2n(nc(Cc3cccc(NS(=O)(=O)C=C)c3)c12)C1CCCC1
Show InChI InChI=1S/C19H22N6O2S/c1-2-28(26,27)24-14-7-5-6-13(10-14)11-16-17-18(20)21-12-22-19(17)25(23-16)15-8-3-4-9-15/h2,5-7,10,12,15,24H,1,3-4,8-9,11H2,(H2,20,21,22)
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Assay Description
In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


Citation and Details
More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (T338C)


(Gallus gallus (Chicken))
BDBM234854
PNG
(US9353116, 12)
Show SMILES CC(C)n1nc(Cc2cccc(NC(=O)CCl)c2)c2c(N)ncnc12
Show InChI InChI=1S/C17H19ClN6O/c1-10(2)24-17-15(16(19)20-9-21-17)13(23-24)7-11-4-3-5-12(6-11)22-14(25)8-18/h3-6,9-10H,7-8H2,1-2H3,(H,22,25)(H2,19,20,21)
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Assay Description
In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


Citation and Details
More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (T338C)


(Gallus gallus (Chicken))
BDBM234846
PNG
(US9353116, 2)
Show SMILES CC(C)n1nc(-c2cccc(NC(=O)C=C)c2)c2cncnc12
Show InChI InChI=1S/C17H17N5O/c1-4-15(23)20-13-7-5-6-12(8-13)16-14-9-18-10-19-17(14)22(21-16)11(2)3/h4-11H,1H2,2-3H3,(H,20,23)
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Assay Description
In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


Citation and Details
More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (c-Src)


(Gallus gallus (Chicken))
BDBM50403061
PNG
(CHEMBL2216823 | US9353116, 9)
Show SMILES CC(C)n1nc(Cc2cccc(NS(=O)(=O)C=C)c2)c2c(N)ncnc12
Show InChI InChI=1S/C17H20N6O2S/c1-4-26(24,25)22-13-7-5-6-12(8-13)9-14-15-16(18)19-10-20-17(15)23(21-14)11(2)3/h4-8,10-11,22H,1,9H2,2-3H3,(H2,18,19,20)
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Assay Description
In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


Citation and Details
More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (c-Src)


(Gallus gallus (Chicken))
BDBM234847
PNG
(US9353116, 4)
Show SMILES CC(C)n1nc(-c2cccc(NS(=O)(=O)C=C)c2)c2cncnc12
Show InChI InChI=1S/C16H17N5O2S/c1-4-24(22,23)20-13-7-5-6-12(8-13)15-14-9-17-10-18-16(14)21(19-15)11(2)3/h4-11,20H,1H2,2-3H3
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Assay Description
In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


Citation and Details
More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (c-Src)


(Gallus gallus (Chicken))
BDBM234851
PNG
(US9353116, 8)
Show SMILES CC(C)n1nc(Cc2ccc(NC(=O)C=C)cc2)c2c(N)ncnc12
Show InChI InChI=1S/C18H20N6O/c1-4-15(25)22-13-7-5-12(6-8-13)9-14-16-17(19)20-10-21-18(16)24(23-14)11(2)3/h4-8,10-11H,1,9H2,2-3H3,(H,22,25)(H2,19,20,21)
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Assay Description
In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


Citation and Details
More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (T338C)


(Gallus gallus (Chicken))
BDBM234847
PNG
(US9353116, 4)
Show SMILES CC(C)n1nc(-c2cccc(NS(=O)(=O)C=C)c2)c2cncnc12
Show InChI InChI=1S/C16H17N5O2S/c1-4-24(22,23)20-13-7-5-6-12(8-13)15-14-9-17-10-18-16(14)21(19-15)11(2)3/h4-11,20H,1H2,2-3H3
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Assay Description
In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


Citation and Details
More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (c-Src)


(Gallus gallus (Chicken))
BDBM234855
PNG
(US9353116, 14)
Show SMILES CC(C)n1nc(Cc2cccc(c2)C(C)=O)c2c(N)ncnc12
Show InChI InChI=1S/C17H19N5O/c1-10(2)22-17-15(16(18)19-9-20-17)14(21-22)8-12-5-4-6-13(7-12)11(3)23/h4-7,9-10H,8H2,1-3H3,(H2,18,19,20)
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Assay Description
In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


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More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (c-Src)


(Gallus gallus (Chicken))
BDBM234849
PNG
(US9353116, 6)
Show SMILES CC(C)n1nc(-c2cccc(NC(=O)CCl)c2)c2c(N)ncnc12
Show InChI InChI=1S/C16H17ClN6O/c1-9(2)23-16-13(15(18)19-8-20-16)14(22-23)10-4-3-5-11(6-10)21-12(24)7-17/h3-6,8-9H,7H2,1-2H3,(H,21,24)(H2,18,19,20)
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Assay Description
In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


Citation and Details
More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (c-Src)


(Gallus gallus (Chicken))
BDBM234856
PNG
(US9353116, 15)
Show SMILES Cn1nc(Cc2cccc(NS(=O)(=O)C=C)c2)c2c(N)ncnc12
Show InChI InChI=1S/C15H16N6O2S/c1-3-24(22,23)20-11-6-4-5-10(7-11)8-12-13-14(16)17-9-18-15(13)21(2)19-12/h3-7,9,20H,1,8H2,2H3,(H2,16,17,18)
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Assay Description
In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


Citation and Details
More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (c-Src)


(Gallus gallus (Chicken))
BDBM234853
PNG
(US9353116, 11)
Show SMILES CCS(=O)(=O)Nc1cccc(Cc2nn(C(C)C)c3ncnc(N)c23)c1
Show InChI InChI=1S/C17H22N6O2S/c1-4-26(24,25)22-13-7-5-6-12(8-13)9-14-15-16(18)19-10-20-17(15)23(21-14)11(2)3/h5-8,10-11,22H,4,9H2,1-3H3,(H2,18,19,20)
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Assay Description
In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


Citation and Details
More data for this
Ligand-Target Pair
3D
3D Structure (crystal)
Proto-oncogene tyrosine-protein kinase Src (c-Src)


(Gallus gallus (Chicken))
BDBM234844
PNG
(US9353116, 13)
Show SMILES CC(C)n1nc(Cc2cccc(c2)C(=O)CF)c2c(N)ncnc12
Show InChI InChI=1S/C17H18FN5O/c1-10(2)23-17-15(16(19)20-9-21-17)13(22-23)7-11-4-3-5-12(6-11)14(24)8-18/h3-6,9-10H,7-8H2,1-2H3,(H2,19,20,21)
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Assay Description
In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...


Citation and Details
More data for this
Ligand-Target Pair
* indicates data uncertainty>20%