Found 18 Enz. Inhib. hit(s) with all data for entry = 8183 TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University
US Patent
Washington University
US Patent
Affinity DataIC50: 14nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University
US Patent
Washington University
US Patent
Affinity DataIC50: 29nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University
US Patent
Washington University
US Patent
Affinity DataIC50: 43nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University
US Patent
Washington University
US Patent
Affinity DataIC50: 46nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University
US Patent
Washington University
US Patent
Affinity DataIC50: 52nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University
US Patent
Washington University
US Patent
Affinity DataIC50: 61nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University
US Patent
Washington University
US Patent
Affinity DataIC50: 62nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University
US Patent
Washington University
US Patent
Affinity DataIC50: 65nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University
US Patent
Washington University
US Patent
Affinity DataIC50: 147nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University
US Patent
Washington University
US Patent
Affinity DataIC50: 282nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University
US Patent
Washington University
US Patent
Affinity DataIC50: 748nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University
US Patent
Washington University
US Patent
Affinity DataIC50: 1.06E+3nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University
US Patent
Washington University
US Patent
Affinity DataIC50: 1.33E+3nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University
US Patent
Washington University
US Patent
Affinity DataIC50: 1.58E+3nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University
US Patent
Washington University
US Patent
Affinity DataIC50: 1.73E+3nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University
US Patent
Washington University
US Patent
Affinity DataIC50: 1.99E+3nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University
US Patent
Washington University
US Patent
Affinity DataIC50: 3.63E+3nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University
US Patent
Washington University
US Patent
Affinity DataIC50: 5.86E+3nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
