Compile Data Set for Download or QSAR
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Found 26 Enz. Inhib. hit(s) with all data for entry = 8185
TargetHistamine H3 receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM50088162(CHEMBL3427228 | US9365511, 4)
Affinity DataIC50:  0.670nMAssay Description:Compounds of the present invention were evaluated using the human H3 receptor (H3R) HTRF cAMP assay. In this assay, HEK293 cells expressing the human...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM50088061(CHEMBL3427242 | US9365511, 37)
Affinity DataIC50:  0.780nMAssay Description:Compounds of the present invention were evaluated using the human H3 receptor (H3R) HTRF cAMP assay. In this assay, HEK293 cells expressing the human...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM235922(US9365511, 18)
Affinity DataIC50:  0.790nMAssay Description:Compounds of the present invention were evaluated using the human H3 receptor (H3R) HTRF cAMP assay. In this assay, HEK293 cells expressing the human...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM50088141(CHEMBL3427230 | US9365511, 7)
Affinity DataIC50:  0.930nMAssay Description:Compounds of the present invention were evaluated using the human H3 receptor (H3R) HTRF cAMP assay. In this assay, HEK293 cells expressing the human...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM235919(US9365511, 12)
Affinity DataIC50:  0.950nMAssay Description:Compounds of the present invention were evaluated using the human H3 receptor (H3R) HTRF cAMP assay. In this assay, HEK293 cells expressing the human...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM235928(US9365511, 35)
Affinity DataIC50:  0.960nMAssay Description:Compounds of the present invention were evaluated using the human H3 receptor (H3R) HTRF cAMP assay. In this assay, HEK293 cells expressing the human...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM50088058(CHEMBL3427245 | US9365511, 45)
Affinity DataIC50:  0.970nMAssay Description:Compounds of the present invention were evaluated using the human H3 receptor (H3R) HTRF cAMP assay. In this assay, HEK293 cells expressing the human...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM235924(US9365511, 24)
Affinity DataIC50:  0.990nMAssay Description:Compounds of the present invention were evaluated using the human H3 receptor (H3R) HTRF cAMP assay. In this assay, HEK293 cells expressing the human...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM50088139(CHEMBL3427232 | US9365511, 9)
Affinity DataIC50:  1.10nMAssay Description:Compounds of the present invention were evaluated using the human H3 receptor (H3R) HTRF cAMP assay. In this assay, HEK293 cells expressing the human...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM50088140(CHEMBL3427231 | US9365511, 8)
Affinity DataIC50:  1.20nMAssay Description:Compounds of the present invention were evaluated using the human H3 receptor (H3R) HTRF cAMP assay. In this assay, HEK293 cells expressing the human...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM235929(US9365511, 38)
Affinity DataIC50:  1.20nMAssay Description:Compounds of the present invention were evaluated using the human H3 receptor (H3R) HTRF cAMP assay. In this assay, HEK293 cells expressing the human...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM235921(US9365511, 16)
Affinity DataIC50:  1.5nMAssay Description:Compounds of the present invention were evaluated using the human H3 receptor (H3R) HTRF cAMP assay. In this assay, HEK293 cells expressing the human...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM50088137(CHEMBL3427234 | US9365511, 11)
Affinity DataIC50:  1.80nMAssay Description:Compounds of the present invention were evaluated using the human H3 receptor (H3R) HTRF cAMP assay. In this assay, HEK293 cells expressing the human...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM235926(US9365511, 27)
Affinity DataIC50:  1.90nMAssay Description:Compounds of the present invention were evaluated using the human H3 receptor (H3R) HTRF cAMP assay. In this assay, HEK293 cells expressing the human...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM235927(US9365511, 33)
Affinity DataIC50:  2.10nMAssay Description:Compounds of the present invention were evaluated using the human H3 receptor (H3R) HTRF cAMP assay. In this assay, HEK293 cells expressing the human...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM235920(US9365511, 13)
Affinity DataIC50:  2.10nMAssay Description:Compounds of the present invention were evaluated using the human H3 receptor (H3R) HTRF cAMP assay. In this assay, HEK293 cells expressing the human...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM50088163(CHEMBL3427227 | US9365511, 3)
Affinity DataIC50:  2.5nMAssay Description:Compounds of the present invention were evaluated using the human H3 receptor (H3R) HTRF cAMP assay. In this assay, HEK293 cells expressing the human...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM235930(US9365511, 43)
Affinity DataIC50:  2.5nMAssay Description:Compounds of the present invention were evaluated using the human H3 receptor (H3R) HTRF cAMP assay. In this assay, HEK293 cells expressing the human...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM235923(US9365511, 20)
Affinity DataIC50:  3nMAssay Description:Compounds of the present invention were evaluated using the human H3 receptor (H3R) HTRF cAMP assay. In this assay, HEK293 cells expressing the human...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM50088138(CHEMBL3427233 | US9365511, 10)
Affinity DataIC50:  3.10nMAssay Description:Compounds of the present invention were evaluated using the human H3 receptor (H3R) HTRF cAMP assay. In this assay, HEK293 cells expressing the human...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM50088132(CHEMBL3427239 | US9365511, 25)
Affinity DataIC50:  3.30nMAssay Description:Compounds of the present invention were evaluated using the human H3 receptor (H3R) HTRF cAMP assay. In this assay, HEK293 cells expressing the human...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM50088166(CHEMBL3427225 | US9365511, 1)
Affinity DataIC50:  3.80nMAssay Description:Compounds of the present invention were evaluated using the human H3 receptor (H3R) HTRF cAMP assay. In this assay, HEK293 cells expressing the human...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM235925(US9365511, 26)
Affinity DataIC50:  3.80nMAssay Description:Compounds of the present invention were evaluated using the human H3 receptor (H3R) HTRF cAMP assay. In this assay, HEK293 cells expressing the human...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM50088160(CHEMBL3427229 | US9365511, 5)
Affinity DataIC50:  5.5nMAssay Description:Compounds of the present invention were evaluated using the human H3 receptor (H3R) HTRF cAMP assay. In this assay, HEK293 cells expressing the human...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM235931(US9365511, 44)
Affinity DataIC50:  6.90nMAssay Description:Compounds of the present invention were evaluated using the human H3 receptor (H3R) HTRF cAMP assay. In this assay, HEK293 cells expressing the human...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM50088165(CHEMBL3427226 | US9365511, 2)
Affinity DataIC50:  8.10nMAssay Description:Compounds of the present invention were evaluated using the human H3 receptor (H3R) HTRF cAMP assay. In this assay, HEK293 cells expressing the human...More data for this Ligand-Target Pair
In DepthDetails US Patent