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Patent code US9403768

Compile Data Set for Download or QSAR
Found 24 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
XIAP protein BIR2


(Artificial Sequence)
BDBM238829
PNG
(US9403768, 1)
Show SMILES CN[C@@H](C)C(=O)N[C@@H](C(C)C)C(=O)N1[C@H](C(=O)Nc2c(F)cccc2F)C(C)(C)c2ccccc12
Show InChI InChI=1S/C26H32F2N4O3/c1-14(2)20(30-23(33)15(3)29-6)25(35)32-19-13-8-7-10-16(19)26(4,5)22(32)24(34)31-21-17(27)11-9-12-18(21)28/h7-15,20,22,29H,1-6H3,(H,30,33)(H,31,34)/t15-,20-,22+/m0/s1
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US Patent
n/an/a 21.2n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Ten nanomolar of 6× Histidine-tagged BIR2 domain, corresponding to amino acids 124-240 of XIAP, or BIR3 domain, corresponding to amino acids 24...


Citation and Details
More data for this
Ligand-Target Pair
XIAP protein BIR2


(Artificial Sequence)
BDBM238840
PNG
(US9403768, 12)
Show SMILES CN[C@@H](C)C(=O)N[C@@H](C(C)C)C(=O)N1[C@@H](Cc2ccccc12)C(=O)Nc1c(F)cccc1F
Show InChI InChI=1S/C24H28F2N4O3/c1-13(2)20(28-22(31)14(3)27-4)24(33)30-18-11-6-5-8-15(18)12-19(30)23(32)29-21-16(25)9-7-10-17(21)26/h5-11,13-14,19-20,27H,12H2,1-4H3,(H,28,31)(H,29,32)/t14-,19-,20-/m0/s1
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US Patent
n/an/a 53n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Ten nanomolar of 6× Histidine-tagged BIR2 domain, corresponding to amino acids 124-240 of XIAP, or BIR3 domain, corresponding to amino acids 24...


Citation and Details
More data for this
Ligand-Target Pair
XIAP protein BIR2


(Artificial Sequence)
BDBM238837
PNG
(US9403768, 9)
Show SMILES CN[C@@H](C)C(=O)N[C@H](C(=O)N1[C@@H](Cc2ccccc12)C(=O)Nc1ccccc1-c1ccccc1)c1ccccc1
Show InChI InChI=1S/C33H32N4O3/c1-22(34-2)31(38)36-30(24-15-7-4-8-16-24)33(40)37-28-20-12-9-17-25(28)21-29(37)32(39)35-27-19-11-10-18-26(27)23-13-5-3-6-14-23/h3-20,22,29-30,34H,21H2,1-2H3,(H,35,39)(H,36,38)/t22-,29-,30-/m0/s1
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US Patent
n/an/a 135n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Ten nanomolar of 6× Histidine-tagged BIR2 domain, corresponding to amino acids 124-240 of XIAP, or BIR3 domain, corresponding to amino acids 24...


Citation and Details
More data for this
Ligand-Target Pair
XIAP protein BIR2


(Artificial Sequence)
BDBM238838
PNG
(US9403768, 10)
Show SMILES CN[C@@H](C)C(=O)N[C@H](C(=O)N1[C@@H](Cc2ccccc12)C(=O)Nc1ccccc1OC)c1ccccc1
Show InChI InChI=1S/C28H30N4O4/c1-18(29-2)26(33)31-25(19-11-5-4-6-12-19)28(35)32-22-15-9-7-13-20(22)17-23(32)27(34)30-21-14-8-10-16-24(21)36-3/h4-16,18,23,25,29H,17H2,1-3H3,(H,30,34)(H,31,33)/t18-,23-,25-/m0/s1
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n/an/a 174n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Ten nanomolar of 6× Histidine-tagged BIR2 domain, corresponding to amino acids 124-240 of XIAP, or BIR3 domain, corresponding to amino acids 24...


Citation and Details
More data for this
Ligand-Target Pair
XIAP protein BIR2


(Artificial Sequence)
BDBM238834
PNG
(US9403768, 6)
Show SMILES CN[C@@H](C)C(=O)N[C@H](C(=O)N1[C@@H](Cc2ccccc12)C(=O)NCc1cc(F)ccc1C)c1ccccc1
Show InChI InChI=1S/C29H31FN4O3/c1-18-13-14-23(30)15-22(18)17-32-28(36)25-16-21-11-7-8-12-24(21)34(25)29(37)26(20-9-5-4-6-10-20)33-27(35)19(2)31-3/h4-15,19,25-26,31H,16-17H2,1-3H3,(H,32,36)(H,33,35)/t19-,25-,26-/m0/s1
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US Patent
n/an/a 190n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Ten nanomolar of 6× Histidine-tagged BIR2 domain, corresponding to amino acids 124-240 of XIAP, or BIR3 domain, corresponding to amino acids 24...


Citation and Details
More data for this
Ligand-Target Pair
XIAP protein BIR2


(Artificial Sequence)
BDBM238836
PNG
(US9403768, 8)
Show SMILES CN[C@@H](C)C(=O)N[C@H](C(=O)N1[C@@H](Cc2ccccc12)C(=O)Nc1ccccc1)c1ccccc1
Show InChI InChI=1S/C27H28N4O3/c1-18(28-2)25(32)30-24(19-11-5-3-6-12-19)27(34)31-22-16-10-9-13-20(22)17-23(31)26(33)29-21-14-7-4-8-15-21/h3-16,18,23-24,28H,17H2,1-2H3,(H,29,33)(H,30,32)/t18-,23-,24-/m0/s1
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US Patent
n/an/a 226n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Ten nanomolar of 6× Histidine-tagged BIR2 domain, corresponding to amino acids 124-240 of XIAP, or BIR3 domain, corresponding to amino acids 24...


Citation and Details
More data for this
Ligand-Target Pair
XIAP protein BIR2


(Artificial Sequence)
BDBM238835
PNG
(US9403768, 7)
Show SMILES CN[C@@H](C)C(=O)N[C@H](C(=O)N1[C@@H](Cc2ccccc12)C(N)=O)c1ccccc1
Show InChI InChI=1S/C21H24N4O3/c1-13(23-2)20(27)24-18(14-8-4-3-5-9-14)21(28)25-16-11-7-6-10-15(16)12-17(25)19(22)26/h3-11,13,17-18,23H,12H2,1-2H3,(H2,22,26)(H,24,27)/t13-,17-,18-/m0/s1
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US Patent
n/an/a 368n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Ten nanomolar of 6× Histidine-tagged BIR2 domain, corresponding to amino acids 124-240 of XIAP, or BIR3 domain, corresponding to amino acids 24...


Citation and Details
More data for this
Ligand-Target Pair
XIAP protein BIR2


(Artificial Sequence)
BDBM238839
PNG
(US9403768, 11)
Show SMILES CN[C@@H](C)C(=O)N[C@H](C(=O)N1[C@@H](Cc2ccccc12)C(=O)NCc1ccccc1)c1ccccc1
Show InChI InChI=1S/C28H30N4O3/c1-19(29-2)26(33)31-25(21-13-7-4-8-14-21)28(35)32-23-16-10-9-15-22(23)17-24(32)27(34)30-18-20-11-5-3-6-12-20/h3-16,19,24-25,29H,17-18H2,1-2H3,(H,30,34)(H,31,33)/t19-,24-,25-/m0/s1
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US Patent
n/an/a 723n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Ten nanomolar of 6× Histidine-tagged BIR2 domain, corresponding to amino acids 124-240 of XIAP, or BIR3 domain, corresponding to amino acids 24...


Citation and Details
More data for this
Ligand-Target Pair
XIAP protein BIR2


(Artificial Sequence)
BDBM238832
PNG
(US9403768, 4)
Show SMILES CN[C@@H](C)C(=O)N[C@@H](C(C)C)C(=O)N1[C@@H](Cc2ccccc12)C(=O)NCc1cc(F)ccc1C
Show InChI InChI=1S/C26H33FN4O3/c1-15(2)23(30-24(32)17(4)28-5)26(34)31-21-9-7-6-8-18(21)13-22(31)25(33)29-14-19-12-20(27)11-10-16(19)3/h6-12,15,17,22-23,28H,13-14H2,1-5H3,(H,29,33)(H,30,32)/t17-,22-,23-/m0/s1
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US Patent
n/an/a 884n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Ten nanomolar of 6× Histidine-tagged BIR2 domain, corresponding to amino acids 124-240 of XIAP, or BIR3 domain, corresponding to amino acids 24...


Citation and Details
More data for this
Ligand-Target Pair
XIAP protein BIR2


(Artificial Sequence)
BDBM238833
PNG
(US9403768, 5)
Show SMILES CN[C@@H](C)C(=O)N[C@@H](C(C)C)C(=O)N1[C@@H](Cc2ccccc12)C(=O)Nc1ccccc1C(=O)c1ccccc1
Show InChI InChI=1S/C31H34N4O4/c1-19(2)27(34-29(37)20(3)32-4)31(39)35-25-17-11-8-14-22(25)18-26(35)30(38)33-24-16-10-9-15-23(24)28(36)21-12-6-5-7-13-21/h5-17,19-20,26-27,32H,18H2,1-4H3,(H,33,38)(H,34,37)/t20-,26-,27-/m0/s1
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US Patent
n/an/a 1.48E+3n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Ten nanomolar of 6× Histidine-tagged BIR2 domain, corresponding to amino acids 124-240 of XIAP, or BIR3 domain, corresponding to amino acids 24...


Citation and Details
More data for this
Ligand-Target Pair
XIAP protein BIR2


(Artificial Sequence)
BDBM238830
PNG
(US9403768, 2)
Show SMILES CN[C@@H](C)C(=O)N[C@@H](C(C)C)C(=O)N1[C@@H](Cc2ccccc12)C(N)=O
Show InChI InChI=1S/C18H26N4O3/c1-10(2)15(21-17(24)11(3)20-4)18(25)22-13-8-6-5-7-12(13)9-14(22)16(19)23/h5-8,10-11,14-15,20H,9H2,1-4H3,(H2,19,23)(H,21,24)/t11-,14-,15-/m0/s1
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US Patent
n/an/a 2.18E+3n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Ten nanomolar of 6× Histidine-tagged BIR2 domain, corresponding to amino acids 124-240 of XIAP, or BIR3 domain, corresponding to amino acids 24...


Citation and Details
More data for this
Ligand-Target Pair
XIAP protein BIR2


(Artificial Sequence)
BDBM238831
PNG
(US9403768, 3)
Show SMILES CN[C@@H](C)C(=O)N[C@@H](C(C)C)C(=O)N1[C@@H](Cc2ccccc12)C(=O)NCc1ccccc1
Show InChI InChI=1S/C25H32N4O3/c1-16(2)22(28-23(30)17(3)26-4)25(32)29-20-13-9-8-12-19(20)14-21(29)24(31)27-15-18-10-6-5-7-11-18/h5-13,16-17,21-22,26H,14-15H2,1-4H3,(H,27,31)(H,28,30)/t17-,21-,22-/m0/s1
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US Patent
n/an/a 1.12E+4n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Ten nanomolar of 6× Histidine-tagged BIR2 domain, corresponding to amino acids 124-240 of XIAP, or BIR3 domain, corresponding to amino acids 24...


Citation and Details
More data for this
Ligand-Target Pair
XIAP protein BIR3


(Artificial Sequence)
BDBM238839
PNG
(US9403768, 11)
Show SMILES CN[C@@H](C)C(=O)N[C@H](C(=O)N1[C@@H](Cc2ccccc12)C(=O)NCc1ccccc1)c1ccccc1
Show InChI InChI=1S/C28H30N4O3/c1-19(29-2)26(33)31-25(21-13-7-4-8-14-21)28(35)32-23-16-10-9-15-22(23)17-24(32)27(34)30-18-20-11-5-3-6-12-20/h3-16,19,24-25,29H,17-18H2,1-2H3,(H,30,34)(H,31,33)/t19-,24-,25-/m0/s1
PDB

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US Patent
n/an/a 3.32E+4n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Ten nanomolar of 6× Histidine-tagged BIR2 domain, corresponding to amino acids 124-240 of XIAP, or BIR3 domain, corresponding to amino acids 24...


Citation and Details
More data for this
Ligand-Target Pair
XIAP protein BIR3


(Artificial Sequence)
BDBM238829
PNG
(US9403768, 1)
Show SMILES CN[C@@H](C)C(=O)N[C@@H](C(C)C)C(=O)N1[C@H](C(=O)Nc2c(F)cccc2F)C(C)(C)c2ccccc12
Show InChI InChI=1S/C26H32F2N4O3/c1-14(2)20(30-23(33)15(3)29-6)25(35)32-19-13-8-7-10-16(19)26(4,5)22(32)24(34)31-21-17(27)11-9-12-18(21)28/h7-15,20,22,29H,1-6H3,(H,30,33)(H,31,34)/t15-,20-,22+/m0/s1
PDB

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UniChem
US Patent
n/an/a>5.48E+4n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Ten nanomolar of 6× Histidine-tagged BIR2 domain, corresponding to amino acids 124-240 of XIAP, or BIR3 domain, corresponding to amino acids 24...


Citation and Details
More data for this
Ligand-Target Pair
XIAP protein BIR3


(Artificial Sequence)
BDBM238840
PNG
(US9403768, 12)
Show SMILES CN[C@@H](C)C(=O)N[C@@H](C(C)C)C(=O)N1[C@@H](Cc2ccccc12)C(=O)Nc1c(F)cccc1F
Show InChI InChI=1S/C24H28F2N4O3/c1-13(2)20(28-22(31)14(3)27-4)24(33)30-18-11-6-5-8-15(18)12-19(30)23(32)29-21-16(25)9-7-10-17(21)26/h5-11,13-14,19-20,27H,12H2,1-4H3,(H,28,31)(H,29,32)/t14-,19-,20-/m0/s1
PDB

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UniChem
US Patent
n/an/a>5.48E+4n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Ten nanomolar of 6× Histidine-tagged BIR2 domain, corresponding to amino acids 124-240 of XIAP, or BIR3 domain, corresponding to amino acids 24...


Citation and Details
More data for this
Ligand-Target Pair
XIAP protein BIR3


(Artificial Sequence)
BDBM238836
PNG
(US9403768, 8)
Show SMILES CN[C@@H](C)C(=O)N[C@H](C(=O)N1[C@@H](Cc2ccccc12)C(=O)Nc1ccccc1)c1ccccc1
Show InChI InChI=1S/C27H28N4O3/c1-18(28-2)25(32)30-24(19-11-5-3-6-12-19)27(34)31-22-16-10-9-13-20(22)17-23(31)26(33)29-21-14-7-4-8-15-21/h3-16,18,23-24,28H,17H2,1-2H3,(H,29,33)(H,30,32)/t18-,23-,24-/m0/s1
PDB

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UniChem
US Patent
n/an/a>5.48E+4n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Ten nanomolar of 6× Histidine-tagged BIR2 domain, corresponding to amino acids 124-240 of XIAP, or BIR3 domain, corresponding to amino acids 24...


Citation and Details
More data for this
Ligand-Target Pair
XIAP protein BIR3


(Artificial Sequence)
BDBM238830
PNG
(US9403768, 2)
Show SMILES CN[C@@H](C)C(=O)N[C@@H](C(C)C)C(=O)N1[C@@H](Cc2ccccc12)C(N)=O
Show InChI InChI=1S/C18H26N4O3/c1-10(2)15(21-17(24)11(3)20-4)18(25)22-13-8-6-5-7-12(13)9-14(22)16(19)23/h5-8,10-11,14-15,20H,9H2,1-4H3,(H2,19,23)(H,21,24)/t11-,14-,15-/m0/s1
PDB

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UniChem
US Patent
n/an/a>5.48E+4n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Ten nanomolar of 6× Histidine-tagged BIR2 domain, corresponding to amino acids 124-240 of XIAP, or BIR3 domain, corresponding to amino acids 24...


Citation and Details
More data for this
Ligand-Target Pair
XIAP protein BIR3


(Artificial Sequence)
BDBM238838
PNG
(US9403768, 10)
Show SMILES CN[C@@H](C)C(=O)N[C@H](C(=O)N1[C@@H](Cc2ccccc12)C(=O)Nc1ccccc1OC)c1ccccc1
Show InChI InChI=1S/C28H30N4O4/c1-18(29-2)26(33)31-25(19-11-5-4-6-12-19)28(35)32-22-15-9-7-13-20(22)17-23(32)27(34)30-21-14-8-10-16-24(21)36-3/h4-16,18,23,25,29H,17H2,1-3H3,(H,30,34)(H,31,33)/t18-,23-,25-/m0/s1
PDB

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UniChem
US Patent
n/an/a>5.48E+4n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Ten nanomolar of 6× Histidine-tagged BIR2 domain, corresponding to amino acids 124-240 of XIAP, or BIR3 domain, corresponding to amino acids 24...


Citation and Details
More data for this
Ligand-Target Pair
XIAP protein BIR3


(Artificial Sequence)
BDBM238834
PNG
(US9403768, 6)
Show SMILES CN[C@@H](C)C(=O)N[C@H](C(=O)N1[C@@H](Cc2ccccc12)C(=O)NCc1cc(F)ccc1C)c1ccccc1
Show InChI InChI=1S/C29H31FN4O3/c1-18-13-14-23(30)15-22(18)17-32-28(36)25-16-21-11-7-8-12-24(21)34(25)29(37)26(20-9-5-4-6-10-20)33-27(35)19(2)31-3/h4-15,19,25-26,31H,16-17H2,1-3H3,(H,32,36)(H,33,35)/t19-,25-,26-/m0/s1
PDB

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n/an/a>5.48E+4n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Ten nanomolar of 6× Histidine-tagged BIR2 domain, corresponding to amino acids 124-240 of XIAP, or BIR3 domain, corresponding to amino acids 24...


Citation and Details
More data for this
Ligand-Target Pair
XIAP protein BIR3


(Artificial Sequence)
BDBM238837
PNG
(US9403768, 9)
Show SMILES CN[C@@H](C)C(=O)N[C@H](C(=O)N1[C@@H](Cc2ccccc12)C(=O)Nc1ccccc1-c1ccccc1)c1ccccc1
Show InChI InChI=1S/C33H32N4O3/c1-22(34-2)31(38)36-30(24-15-7-4-8-16-24)33(40)37-28-20-12-9-17-25(28)21-29(37)32(39)35-27-19-11-10-18-26(27)23-13-5-3-6-14-23/h3-20,22,29-30,34H,21H2,1-2H3,(H,35,39)(H,36,38)/t22-,29-,30-/m0/s1
PDB

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UniChem
US Patent
n/an/a>5.48E+4n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Ten nanomolar of 6× Histidine-tagged BIR2 domain, corresponding to amino acids 124-240 of XIAP, or BIR3 domain, corresponding to amino acids 24...


Citation and Details
More data for this
Ligand-Target Pair
XIAP protein BIR3


(Artificial Sequence)
BDBM238835
PNG
(US9403768, 7)
Show SMILES CN[C@@H](C)C(=O)N[C@H](C(=O)N1[C@@H](Cc2ccccc12)C(N)=O)c1ccccc1
Show InChI InChI=1S/C21H24N4O3/c1-13(23-2)20(27)24-18(14-8-4-3-5-9-14)21(28)25-16-11-7-6-10-15(16)12-17(25)19(22)26/h3-11,13,17-18,23H,12H2,1-2H3,(H2,22,26)(H,24,27)/t13-,17-,18-/m0/s1
PDB

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PC sid
UniChem
US Patent
n/an/a>5.48E+4n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Ten nanomolar of 6× Histidine-tagged BIR2 domain, corresponding to amino acids 124-240 of XIAP, or BIR3 domain, corresponding to amino acids 24...


Citation and Details
More data for this
Ligand-Target Pair
XIAP protein BIR3


(Artificial Sequence)
BDBM238832
PNG
(US9403768, 4)
Show SMILES CN[C@@H](C)C(=O)N[C@@H](C(C)C)C(=O)N1[C@@H](Cc2ccccc12)C(=O)NCc1cc(F)ccc1C
Show InChI InChI=1S/C26H33FN4O3/c1-15(2)23(30-24(32)17(4)28-5)26(34)31-21-9-7-6-8-18(21)13-22(31)25(33)29-14-19-12-20(27)11-10-16(19)3/h6-12,15,17,22-23,28H,13-14H2,1-5H3,(H,29,33)(H,30,32)/t17-,22-,23-/m0/s1
PDB

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PC cid
PC sid
UniChem
US Patent
n/an/a>5.48E+4n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Ten nanomolar of 6× Histidine-tagged BIR2 domain, corresponding to amino acids 124-240 of XIAP, or BIR3 domain, corresponding to amino acids 24...


Citation and Details
More data for this
Ligand-Target Pair
XIAP protein BIR3


(Artificial Sequence)
BDBM238831
PNG
(US9403768, 3)
Show SMILES CN[C@@H](C)C(=O)N[C@@H](C(C)C)C(=O)N1[C@@H](Cc2ccccc12)C(=O)NCc1ccccc1
Show InChI InChI=1S/C25H32N4O3/c1-16(2)22(28-23(30)17(3)26-4)25(32)29-20-13-9-8-12-19(20)14-21(29)24(31)27-15-18-10-6-5-7-11-18/h5-13,16-17,21-22,26H,14-15H2,1-4H3,(H,27,31)(H,28,30)/t17-,21-,22-/m0/s1
PDB

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a>5.48E+4n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Ten nanomolar of 6× Histidine-tagged BIR2 domain, corresponding to amino acids 124-240 of XIAP, or BIR3 domain, corresponding to amino acids 24...


Citation and Details
More data for this
Ligand-Target Pair
XIAP protein BIR3


(Artificial Sequence)
BDBM238833
PNG
(US9403768, 5)
Show SMILES CN[C@@H](C)C(=O)N[C@@H](C(C)C)C(=O)N1[C@@H](Cc2ccccc12)C(=O)Nc1ccccc1C(=O)c1ccccc1
Show InChI InChI=1S/C31H34N4O4/c1-19(2)27(34-29(37)20(3)32-4)31(39)35-25-17-11-8-14-22(25)18-26(35)30(38)33-24-16-10-9-15-23(24)28(36)21-12-6-5-7-13-21/h5-17,19-20,26-27,32H,18H2,1-4H3,(H,33,38)(H,34,37)/t20-,26-,27-/m0/s1
PDB

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a>5.48E+4n/an/an/an/an/an/a



Hoffmann-La Roche Inc.

US Patent


Assay Description
Ten nanomolar of 6× Histidine-tagged BIR2 domain, corresponding to amino acids 124-240 of XIAP, or BIR3 domain, corresponding to amino acids 24...


Citation and Details
More data for this
Ligand-Target Pair
* indicates data uncertainty>20%