Found 38 Enz. Inhib. hit(s) with all data for entry = 8419 TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Newron Pharmaceuticals
US Patent
Newron Pharmaceuticals
US Patent
Affinity DataKi: 100nMAssay Description:Cells and methods: Functional inhibition of the sodium currents is studied using whole cell patch clamp methods (Hamill O. P., Marty A., Neher E., Sa...More data for this Ligand-Target Pair
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Newron Pharmaceuticals
US Patent
Newron Pharmaceuticals
US Patent
Affinity DataKi: 100nMAssay Description:Cells and methods: Functional inhibition of the sodium currents is studied using whole cell patch clamp methods (Hamill O. P., Marty A., Neher E., Sa...More data for this Ligand-Target Pair
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Newron Pharmaceuticals
US Patent
Newron Pharmaceuticals
US Patent
Affinity DataKi: 100nMAssay Description:Cells and methods: Functional inhibition of the sodium currents is studied using whole cell patch clamp methods (Hamill O. P., Marty A., Neher E., Sa...More data for this Ligand-Target Pair
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Newron Pharmaceuticals
US Patent
Newron Pharmaceuticals
US Patent
Affinity DataKi: 200nMAssay Description:Cells and methods: Functional inhibition of the sodium currents is studied using whole cell patch clamp methods (Hamill O. P., Marty A., Neher E., Sa...More data for this Ligand-Target Pair
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Newron Pharmaceuticals
US Patent
Newron Pharmaceuticals
US Patent
Affinity DataKi: 200nMAssay Description:Cells and methods: Functional inhibition of the sodium currents is studied using whole cell patch clamp methods (Hamill O. P., Marty A., Neher E., Sa...More data for this Ligand-Target Pair
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Newron Pharmaceuticals
US Patent
Newron Pharmaceuticals
US Patent
Affinity DataKi: 300nMAssay Description:Cells and methods: Functional inhibition of the sodium currents is studied using whole cell patch clamp methods (Hamill O. P., Marty A., Neher E., Sa...More data for this Ligand-Target Pair
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Newron Pharmaceuticals
US Patent
Newron Pharmaceuticals
US Patent
Affinity DataKi: 500nMAssay Description:Cells and methods: Functional inhibition of the sodium currents is studied using whole cell patch clamp methods (Hamill O. P., Marty A., Neher E., Sa...More data for this Ligand-Target Pair
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Newron Pharmaceuticals
US Patent
Newron Pharmaceuticals
US Patent
Affinity DataKi: 700nMAssay Description:Cells and methods: Functional inhibition of the sodium currents is studied using whole cell patch clamp methods (Hamill O. P., Marty A., Neher E., Sa...More data for this Ligand-Target Pair
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Newron Pharmaceuticals
US Patent
Newron Pharmaceuticals
US Patent
Affinity DataKi: 1.10E+3nMAssay Description:Cells and methods: Functional inhibition of the sodium currents is studied using whole cell patch clamp methods (Hamill O. P., Marty A., Neher E., Sa...More data for this Ligand-Target Pair
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Newron Pharmaceuticals
US Patent
Newron Pharmaceuticals
US Patent
Affinity DataKi: 1.70E+3nMAssay Description:Cells and methods: Functional inhibition of the sodium currents is studied using whole cell patch clamp methods (Hamill O. P., Marty A., Neher E., Sa...More data for this Ligand-Target Pair
Affinity DataIC50: 700nMT: 2°CAssay Description:Test compound is dissolved in DMSO 500× the highest final concentration desired in the IC50 assay. 30 ml of deionized water is pre-warmed to 37...More data for this Ligand-Target Pair
Affinity DataIC50: 900nMT: 2°CAssay Description:Test compound is dissolved in DMSO 500× the highest final concentration desired in the IC50 assay. 30 ml of deionized water is pre-warmed to 37...More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMT: 2°CAssay Description:Test compound is dissolved in DMSO 500× the highest final concentration desired in the IC50 assay. 30 ml of deionized water is pre-warmed to 37...More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMT: 2°CAssay Description:Test compound is dissolved in DMSO 500× the highest final concentration desired in the IC50 assay. 30 ml of deionized water is pre-warmed to 37...More data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMT: 2°CAssay Description:Test compound is dissolved in DMSO 500× the highest final concentration desired in the IC50 assay. 30 ml of deionized water is pre-warmed to 37...More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMT: 2°CAssay Description:Test compound is dissolved in DMSO 500× the highest final concentration desired in the IC50 assay. 30 ml of deionized water is pre-warmed to 37...More data for this Ligand-Target Pair
Affinity DataIC50: 3.40E+3nMT: 2°CAssay Description:Test compound is dissolved in DMSO 500× the highest final concentration desired in the IC50 assay. 30 ml of deionized water is pre-warmed to 37...More data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+3nMT: 2°CAssay Description:Test compound is dissolved in DMSO 500× the highest final concentration desired in the IC50 assay. 30 ml of deionized water is pre-warmed to 37...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMT: 2°CAssay Description:Test compound is dissolved in DMSO 500× the highest final concentration desired in the IC50 assay. 30 ml of deionized water is pre-warmed to 37...More data for this Ligand-Target Pair
Affinity DataIC50: 5.80E+3nMT: 2°CAssay Description:Test compound is dissolved in DMSO 500× the highest final concentration desired in the IC50 assay. 30 ml of deionized water is pre-warmed to 37...More data for this Ligand-Target Pair
Affinity DataIC50: 5.80E+3nMT: 2°CAssay Description:Test compound is dissolved in DMSO 500× the highest final concentration desired in the IC50 assay. 30 ml of deionized water is pre-warmed to 37...More data for this Ligand-Target Pair
Affinity DataIC50: 5.80E+3nMT: 2°CAssay Description:Test compound is dissolved in DMSO 500× the highest final concentration desired in the IC50 assay. 30 ml of deionized water is pre-warmed to 37...More data for this Ligand-Target Pair
Affinity DataIC50: 7.30E+3nMT: 2°CAssay Description:Test compound is dissolved in DMSO 500× the highest final concentration desired in the IC50 assay. 30 ml of deionized water is pre-warmed to 37...More data for this Ligand-Target Pair
Affinity DataIC50: 1.06E+4nMT: 2°CAssay Description:Test compound is dissolved in DMSO 500× the highest final concentration desired in the IC50 assay. 30 ml of deionized water is pre-warmed to 37...More data for this Ligand-Target Pair
Affinity DataIC50: 2.39E+4nMT: 2°CAssay Description:Test compound is dissolved in DMSO 500× the highest final concentration desired in the IC50 assay. 30 ml of deionized water is pre-warmed to 37...More data for this Ligand-Target Pair
Affinity DataIC50: 3.40E+4nMT: 2°CAssay Description:Test compound is dissolved in DMSO 500× the highest final concentration desired in the IC50 assay. 30 ml of deionized water is pre-warmed to 37...More data for this Ligand-Target Pair
Affinity DataIC50: 3.78E+4nMT: 2°CAssay Description:Test compound is dissolved in DMSO 500× the highest final concentration desired in the IC50 assay. 30 ml of deionized water is pre-warmed to 37...More data for this Ligand-Target Pair
Affinity DataIC50: 3.83E+4nMT: 2°CAssay Description:Test compound is dissolved in DMSO 500× the highest final concentration desired in the IC50 assay. 30 ml of deionized water is pre-warmed to 37...More data for this Ligand-Target Pair
Affinity DataIC50: >4.00E+4nMT: 2°CAssay Description:Test compound is dissolved in DMSO 500× the highest final concentration desired in the IC50 assay. 30 ml of deionized water is pre-warmed to 37...More data for this Ligand-Target Pair
Affinity DataIC50: >4.00E+4nMT: 2°CAssay Description:Test compound is dissolved in DMSO 500× the highest final concentration desired in the IC50 assay. 30 ml of deionized water is pre-warmed to 37...More data for this Ligand-Target Pair
Affinity DataIC50: >4.00E+4nMT: 2°CAssay Description:Test compound is dissolved in DMSO 500× the highest final concentration desired in the IC50 assay. 30 ml of deionized water is pre-warmed to 37...More data for this Ligand-Target Pair
Affinity DataIC50: >4.00E+4nMT: 2°CAssay Description:Test compound is dissolved in DMSO 500× the highest final concentration desired in the IC50 assay. 30 ml of deionized water is pre-warmed to 37...More data for this Ligand-Target Pair
Affinity DataIC50: >4.00E+4nMT: 2°CAssay Description:Test compound is dissolved in DMSO 500× the highest final concentration desired in the IC50 assay. 30 ml of deionized water is pre-warmed to 37...More data for this Ligand-Target Pair
Affinity DataIC50: >4.00E+4nMT: 2°CAssay Description:Test compound is dissolved in DMSO 500× the highest final concentration desired in the IC50 assay. 30 ml of deionized water is pre-warmed to 37...More data for this Ligand-Target Pair
Affinity DataIC50: >4.00E+4nMT: 2°CAssay Description:Test compound is dissolved in DMSO 500× the highest final concentration desired in the IC50 assay. 30 ml of deionized water is pre-warmed to 37...More data for this Ligand-Target Pair
Affinity DataIC50: >4.00E+4nMT: 2°CAssay Description:Test compound is dissolved in DMSO 500× the highest final concentration desired in the IC50 assay. 30 ml of deionized water is pre-warmed to 37...More data for this Ligand-Target Pair
Affinity DataIC50: >4.00E+4nMT: 2°CAssay Description:Test compound is dissolved in DMSO 500× the highest final concentration desired in the IC50 assay. 30 ml of deionized water is pre-warmed to 37...More data for this Ligand-Target Pair
Affinity DataIC50: >4.00E+4nMT: 2°CAssay Description:Test compound is dissolved in DMSO 500× the highest final concentration desired in the IC50 assay. 30 ml of deionized water is pre-warmed to 37...More data for this Ligand-Target Pair
