Found 17 Enz. Inhib. hit(s) with all data for entry = 8428 TargetGamma-aminobutyric acid receptor subunit alpha-2/delta(Rattus norvegicus (Rat))
Kyowa Hakko Kirin
US Patent
Kyowa Hakko Kirin
US Patent
Affinity DataIC50: 0.700nMT: 2°CAssay Description:A test compound (20 μL) diluted to 5 times of the final concentration with Binding buffer, [3H]-gabapentin diluted to 100 nmol/L with binding buff...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/delta(Rattus norvegicus (Rat))
Kyowa Hakko Kirin
US Patent
Kyowa Hakko Kirin
US Patent
Affinity DataIC50: 1.20nMT: 2°CAssay Description:A test compound (20 μL) diluted to 5 times of the final concentration with Binding buffer, [3H]-gabapentin diluted to 100 nmol/L with binding buff...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/delta(Rattus norvegicus (Rat))
Kyowa Hakko Kirin
US Patent
Kyowa Hakko Kirin
US Patent
Affinity DataIC50: 2.60nMT: 2°CAssay Description:A test compound (20 μL) diluted to 5 times of the final concentration with Binding buffer, [3H]-gabapentin diluted to 100 nmol/L with binding buff...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/delta(Rattus norvegicus (Rat))
Kyowa Hakko Kirin
US Patent
Kyowa Hakko Kirin
US Patent
Affinity DataIC50: 2.60nMT: 2°CAssay Description:A test compound (20 μL) diluted to 5 times of the final concentration with Binding buffer, [3H]-gabapentin diluted to 100 nmol/L with binding buff...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/delta(Rattus norvegicus (Rat))
Kyowa Hakko Kirin
US Patent
Kyowa Hakko Kirin
US Patent
Affinity DataIC50: 2.60nMT: 2°CAssay Description:A test compound (20 μL) diluted to 5 times of the final concentration with Binding buffer, [3H]-gabapentin diluted to 100 nmol/L with binding buff...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/delta(Rattus norvegicus (Rat))
Kyowa Hakko Kirin
US Patent
Kyowa Hakko Kirin
US Patent
Affinity DataIC50: 2.70nMT: 2°CAssay Description:A test compound (20 μL) diluted to 5 times of the final concentration with Binding buffer, [3H]-gabapentin diluted to 100 nmol/L with binding buff...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/delta(Rattus norvegicus (Rat))
Kyowa Hakko Kirin
US Patent
Kyowa Hakko Kirin
US Patent
Affinity DataIC50: 3nMT: 2°CAssay Description:A test compound (20 μL) diluted to 5 times of the final concentration with Binding buffer, [3H]-gabapentin diluted to 100 nmol/L with binding buff...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/delta(Rattus norvegicus (Rat))
Kyowa Hakko Kirin
US Patent
Kyowa Hakko Kirin
US Patent
Affinity DataIC50: 3nMT: 2°CAssay Description:A test compound (20 μL) diluted to 5 times of the final concentration with Binding buffer, [3H]-gabapentin diluted to 100 nmol/L with binding buff...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/delta(Rattus norvegicus (Rat))
Kyowa Hakko Kirin
US Patent
Kyowa Hakko Kirin
US Patent
Affinity DataIC50: 3.60nMT: 2°CAssay Description:A test compound (20 μL) diluted to 5 times of the final concentration with Binding buffer, [3H]-gabapentin diluted to 100 nmol/L with binding buff...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/delta(Rattus norvegicus (Rat))
Kyowa Hakko Kirin
US Patent
Kyowa Hakko Kirin
US Patent
Affinity DataIC50: 3.80nMT: 2°CAssay Description:A test compound (20 μL) diluted to 5 times of the final concentration with Binding buffer, [3H]-gabapentin diluted to 100 nmol/L with binding buff...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/delta(Rattus norvegicus (Rat))
Kyowa Hakko Kirin
US Patent
Kyowa Hakko Kirin
US Patent
Affinity DataIC50: 3.90nMT: 2°CAssay Description:A test compound (20 μL) diluted to 5 times of the final concentration with Binding buffer, [3H]-gabapentin diluted to 100 nmol/L with binding buff...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/delta(Rattus norvegicus (Rat))
Kyowa Hakko Kirin
US Patent
Kyowa Hakko Kirin
US Patent
Affinity DataIC50: 4nMT: 2°CAssay Description:A test compound (20 μL) diluted to 5 times of the final concentration with Binding buffer, [3H]-gabapentin diluted to 100 nmol/L with binding buff...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/delta(Rattus norvegicus (Rat))
Kyowa Hakko Kirin
US Patent
Kyowa Hakko Kirin
US Patent
Affinity DataIC50: 4.10nMT: 2°CAssay Description:A test compound (20 μL) diluted to 5 times of the final concentration with Binding buffer, [3H]-gabapentin diluted to 100 nmol/L with binding buff...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/delta(Rattus norvegicus (Rat))
Kyowa Hakko Kirin
US Patent
Kyowa Hakko Kirin
US Patent
Affinity DataIC50: 4.70nMT: 2°CAssay Description:A test compound (20 μL) diluted to 5 times of the final concentration with Binding buffer, [3H]-gabapentin diluted to 100 nmol/L with binding buff...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/delta(Rattus norvegicus (Rat))
Kyowa Hakko Kirin
US Patent
Kyowa Hakko Kirin
US Patent
Affinity DataIC50: 4.80nMT: 2°CAssay Description:A test compound (20 μL) diluted to 5 times of the final concentration with Binding buffer, [3H]-gabapentin diluted to 100 nmol/L with binding buff...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/delta(Rattus norvegicus (Rat))
Kyowa Hakko Kirin
US Patent
Kyowa Hakko Kirin
US Patent
Affinity DataIC50: 5nMT: 2°CAssay Description:A test compound (20 μL) diluted to 5 times of the final concentration with Binding buffer, [3H]-gabapentin diluted to 100 nmol/L with binding buff...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/delta(Rattus norvegicus (Rat))
Kyowa Hakko Kirin
US Patent
Kyowa Hakko Kirin
US Patent
Affinity DataIC50: 5.20nMT: 2°CAssay Description:A test compound (20 μL) diluted to 5 times of the final concentration with Binding buffer, [3H]-gabapentin diluted to 100 nmol/L with binding buff...More data for this Ligand-Target Pair
