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Patent code US9469631

Compile Data Set for Download or QSAR
Found 130 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254636
PNG
(US9469631, 33)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1cc(F)c(-c2cnco2)c(F)c1
Show InChI InChI=1S/C23H27F2N3O4/c1-23(2,3)32-22(30)27-8-6-16(7-9-27)28(15-4-5-15)21(29)14-10-17(24)20(18(25)11-14)19-12-26-13-31-19/h10-13,15-16H,4-9H2,1-3H3
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US Patent
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254696
PNG
(US9469631, 97)
Show SMILES CC(C)(C)NS(=O)(=O)c1ccccc1-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C30H41N3O5S/c1-29(2,3)31-39(36,37)26-10-8-7-9-25(26)21-11-13-22(14-12-21)27(34)33(23-15-16-23)24-17-19-32(20-18-24)28(35)38-30(4,5)6/h7-14,23-24,31H,15-20H2,1-6H3
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US Patent
n/an/an/an/a 161n/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254704
PNG
(US9469631, 105)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ccc(cc1)S(N)(=O)=O
Show InChI InChI=1S/C26H33N3O5S/c1-26(2,3)34-25(31)28-16-14-22(15-17-28)29(21-10-11-21)24(30)20-6-4-18(5-7-20)19-8-12-23(13-9-19)35(27,32)33/h4-9,12-13,21-22H,10-11,14-17H2,1-3H3,(H2,27,32,33)
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n/an/an/an/a 115n/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254712
PNG
(US9469631, 113)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1cncc(c1)C#N
Show InChI InChI=1S/C26H30N4O3/c1-26(2,3)33-25(32)29-12-10-23(11-13-29)30(22-8-9-22)24(31)20-6-4-19(5-7-20)21-14-18(15-27)16-28-17-21/h4-7,14,16-17,22-23H,8-13H2,1-3H3
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Boehringer Ingelheim International GmbH

US Patent


Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254613
PNG
(US9469631, 10)
Show SMILES Cc1ncoc1-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C24H31N3O4/c1-16-21(30-15-25-16)17-5-7-18(8-6-17)22(28)27(19-9-10-19)20-11-13-26(14-12-20)23(29)31-24(2,3)4/h5-8,15,19-20H,9-14H2,1-4H3
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n/an/an/an/a 75n/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254629
PNG
(US9469631, 26)
Show SMILES CC1=NNNN1c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C22H32N6O3/c1-15-23-24-25-28(15)19-7-5-16(6-8-19)20(29)27(17-9-10-17)18-11-13-26(14-12-18)21(30)31-22(2,3)4/h5-8,17-18,24-25H,9-14H2,1-4H3
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n/an/an/an/a 224n/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254661
PNG
(US9469631, 62)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1nnco1
Show InChI InChI=1S/C22H28N4O4/c1-22(2,3)30-21(28)25-12-10-18(11-13-25)26(17-8-9-17)20(27)16-6-4-15(5-7-16)19-24-23-14-29-19/h4-7,14,17-18H,8-13H2,1-3H3
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n/an/an/an/a 650n/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254673
PNG
(US9469631, 74)
Show SMILES CC(=O)Nc1nc(ns1)-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C24H31N5O4S/c1-15(30)25-22-26-20(27-34-22)16-5-7-17(8-6-16)21(31)29(18-9-10-18)19-11-13-28(14-12-19)23(32)33-24(2,3)4/h5-8,18-19H,9-14H2,1-4H3,(H,25,26,27,30)
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n/an/an/an/a 886n/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254721
PNG
(US9469631, 122)
Show SMILES O=C(OC1CCCCC1)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1cnco1
Show InChI InChI=1S/C25H31N3O4/c29-24(19-8-6-18(7-9-19)23-16-26-17-31-23)28(20-10-11-20)21-12-14-27(15-13-21)25(30)32-22-4-2-1-3-5-22/h6-9,16-17,20-22H,1-5,10-15H2
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Boehringer Ingelheim International GmbH

US Patent


Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254729
PNG
(US9469631, 130)
Show SMILES CC(C)(OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1cnco1)C(F)(F)F
Show InChI InChI=1S/C23H26F3N3O4/c1-22(2,23(24,25)26)33-21(31)28-11-9-18(10-12-28)29(17-7-8-17)20(30)16-5-3-15(4-6-16)19-13-27-14-32-19/h3-6,13-14,17-18H,7-12H2,1-2H3
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n/an/an/an/a 10n/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254614
PNG
(US9469631, 11)
Show SMILES O=C(OC1CCOCC1)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1cnco1
Show InChI InChI=1S/C24H29N3O5/c28-23(18-3-1-17(2-4-18)22-15-25-16-31-22)27(19-5-6-19)20-7-11-26(12-8-20)24(29)32-21-9-13-30-14-10-21/h1-4,15-16,19-21H,5-14H2
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n/an/an/an/a 516n/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254710
PNG
(US9469631, 111)
Show SMILES CNS(=O)(=O)c1ccc(cc1)-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C27H35N3O5S/c1-27(2,3)35-26(32)29-17-15-23(16-18-29)30(22-11-12-22)25(31)21-7-5-19(6-8-21)20-9-13-24(14-10-20)36(33,34)28-4/h5-10,13-14,22-23,28H,11-12,15-18H2,1-4H3
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n/an/an/an/a 111n/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254615
PNG
(US9469631, 12)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1cn[nH]c1
Show InChI InChI=1S/C23H30N4O3/c1-23(2,3)30-22(29)26-12-10-20(11-13-26)27(19-8-9-19)21(28)17-6-4-16(5-7-17)18-14-24-25-15-18/h4-7,14-15,19-20H,8-13H2,1-3H3,(H,24,25)
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n/an/an/an/a 240n/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254659
PNG
(US9469631, 60)
Show SMILES Cc1noc(n1)-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C23H30N4O4/c1-15-24-20(31-25-15)16-5-7-17(8-6-16)21(28)27(18-9-10-18)19-11-13-26(14-12-19)22(29)30-23(2,3)4/h5-8,18-19H,9-14H2,1-4H3
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Boehringer Ingelheim International GmbH

US Patent


Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254653
PNG
(US9469631, 54)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ccc(cc1)C#N
Show InChI InChI=1S/C27H31N3O3/c1-27(2,3)33-26(32)29-16-14-24(15-17-29)30(23-12-13-23)25(31)22-10-8-21(9-11-22)20-6-4-19(18-28)5-7-20/h4-11,23-24H,12-17H2,1-3H3
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Boehringer Ingelheim International GmbH

US Patent


Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254695
PNG
(US9469631, 96)
Show SMILES COc1ccc(cn1)-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C26H33N3O4/c1-26(2,3)33-25(31)28-15-13-22(14-16-28)29(21-10-11-21)24(30)19-7-5-18(6-8-19)20-9-12-23(32-4)27-17-20/h5-9,12,17,21-22H,10-11,13-16H2,1-4H3
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Boehringer Ingelheim International GmbH

US Patent


Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254707
PNG
(US9469631, 108)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ccc(O)nc1
Show InChI InChI=1S/C25H31N3O4/c1-25(2,3)32-24(31)27-14-12-21(13-15-27)28(20-9-10-20)23(30)18-6-4-17(5-7-18)19-8-11-22(29)26-16-19/h4-8,11,16,20-21H,9-10,12-15H2,1-3H3,(H,26,29)
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Boehringer Ingelheim International GmbH

US Patent


Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254727
PNG
(US9469631, 128)
Show SMILES O=C(OC1CCCC1)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1cnco1
Show InChI InChI=1S/C24H29N3O4/c28-23(18-7-5-17(6-8-18)22-15-25-16-30-22)27(19-9-10-19)20-11-13-26(14-12-20)24(29)31-21-3-1-2-4-21/h5-8,15-16,19-21H,1-4,9-14H2
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Boehringer Ingelheim International GmbH

US Patent


Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254604
PNG
(US9469631, 1)
Show SMILES CC1CC(CCN1C(=O)OC(C)(C)C)N(C1CC1)C(=O)c1ccc(cc1)-c1cnco1
Show InChI InChI=1S/C24H31N3O4/c1-16-13-20(11-12-26(16)23(29)31-24(2,3)4)27(19-9-10-19)22(28)18-7-5-17(6-8-18)21-14-25-15-30-21/h5-8,14-16,19-20H,9-13H2,1-4H3
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Boehringer Ingelheim International GmbH

US Patent


Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254640
PNG
(US9469631, 37)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ccc(CS(C)(=O)=O)cc1
Show InChI InChI=1S/C28H36N2O5S/c1-28(2,3)35-27(32)29-17-15-25(16-18-29)30(24-13-14-24)26(31)23-11-9-22(10-12-23)21-7-5-20(6-8-21)19-36(4,33)34/h5-12,24-25H,13-19H2,1-4H3
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n/an/an/an/a 57n/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254676
PNG
(US9469631, 77)
Show SMILES CC(=O)Nc1nnc(s1)-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C24H31N5O4S/c1-15(30)25-22-27-26-20(34-22)16-5-7-17(8-6-16)21(31)29(18-9-10-18)19-11-13-28(14-12-19)23(32)33-24(2,3)4/h5-8,18-19H,9-14H2,1-4H3,(H,25,27,30)
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n/an/an/an/a 394n/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254716
PNG
(US9469631, 117)
Show SMILES CCOC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1cnco1
Show InChI InChI=1S/C21H25N3O4/c1-2-27-21(26)23-11-9-18(10-12-23)24(17-7-8-17)20(25)16-5-3-15(4-6-16)19-13-22-14-28-19/h3-6,13-14,17-18H,2,7-12H2,1H3
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Boehringer Ingelheim International GmbH

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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254621
PNG
(US9469631, 18)
Show SMILES Cn1ncnc1-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C23H31N5O3/c1-23(2,3)31-22(30)27-13-11-19(12-14-27)28(18-9-10-18)21(29)17-7-5-16(6-8-17)20-24-15-25-26(20)4/h5-8,15,18-19H,9-14H2,1-4H3
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n/an/an/an/a 1.00E+3n/an/an/an/a



Boehringer Ingelheim International GmbH

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Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254625
PNG
(US9469631, 22)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)N1NNN=C1
Show InChI InChI=1S/C21H30N6O3/c1-21(2,3)30-20(29)25-12-10-18(11-13-25)27(17-8-9-17)19(28)15-4-6-16(7-5-15)26-14-22-23-24-26/h4-7,14,17-18,23-24H,8-13H2,1-3H3
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Boehringer Ingelheim International GmbH

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Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254665
PNG
(US9469631, 66)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1nnc(N)s1
Show InChI InChI=1S/C22H29N5O3S/c1-22(2,3)30-21(29)26-12-10-17(11-13-26)27(16-8-9-16)19(28)15-6-4-14(5-7-15)18-24-25-20(23)31-18/h4-7,16-17H,8-13H2,1-3H3,(H2,23,25)
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Boehringer Ingelheim International GmbH

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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254693
PNG
(US9469631, 94)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ccccc1C#N
Show InChI InChI=1S/C27H31N3O3/c1-27(2,3)33-26(32)29-16-14-23(15-17-29)30(22-12-13-22)25(31)20-10-8-19(9-11-20)24-7-5-4-6-21(24)18-28/h4-11,22-23H,12-17H2,1-3H3
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Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254722
PNG
(US9469631, 123)
Show SMILES CCCOC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1cnco1
Show InChI InChI=1S/C22H27N3O4/c1-2-13-28-22(27)24-11-9-19(10-12-24)25(18-7-8-18)21(26)17-5-3-16(4-6-17)20-14-23-15-29-20/h3-6,14-15,18-19H,2,7-13H2,1H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254611
PNG
(US9469631, 8)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(-c2cnco2)c(N)c1
Show InChI InChI=1S/C23H30N4O4/c1-23(2,3)31-22(29)26-10-8-17(9-11-26)27(16-5-6-16)21(28)15-4-7-18(19(24)12-15)20-13-25-14-30-20/h4,7,12-14,16-17H,5-6,8-11,24H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254655
PNG
(US9469631, 56)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-n1cnc(c1)-c1ccccc1
Show InChI InChI=1S/C29H34N4O3/c1-29(2,3)36-28(35)31-17-15-25(16-18-31)33(24-13-14-24)27(34)22-9-11-23(12-10-22)32-19-26(30-20-32)21-7-5-4-6-8-21/h4-12,19-20,24-25H,13-18H2,1-3H3
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Boehringer Ingelheim International GmbH

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Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254703
PNG
(US9469631, 104)
Show SMILES CC(=O)NCc1ccc(cc1)-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C29H37N3O4/c1-20(33)30-19-21-5-7-22(8-6-21)23-9-11-24(12-10-23)27(34)32(25-13-14-25)26-15-17-31(18-16-26)28(35)36-29(2,3)4/h5-12,25-26H,13-19H2,1-4H3,(H,30,33)
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Boehringer Ingelheim International GmbH

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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254616
PNG
(US9469631, 13)
Show SMILES Cn1cc(cn1)-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C24H32N4O3/c1-24(2,3)31-23(30)27-13-11-21(12-14-27)28(20-9-10-20)22(29)18-7-5-17(6-8-18)19-15-25-26(4)16-19/h5-8,15-16,20-21H,9-14H2,1-4H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254620
PNG
(US9469631, 17)
Show SMILES Cn1cnc(n1)-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C23H31N5O3/c1-23(2,3)31-22(30)27-13-11-19(12-14-27)28(18-9-10-18)21(29)17-7-5-16(6-8-17)20-24-15-26(4)25-20/h5-8,15,18-19H,9-14H2,1-4H3
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Boehringer Ingelheim International GmbH

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Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254728
PNG
(US9469631, 129)
Show SMILES CC(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ccc(cc1)C(N)=O
Show InChI InChI=1S/C26H31N3O4/c1-17(2)33-26(32)28-15-13-23(14-16-28)29(22-11-12-22)25(31)21-9-5-19(6-10-21)18-3-7-20(8-4-18)24(27)30/h3-10,17,22-23H,11-16H2,1-2H3,(H2,27,30)
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254642
PNG
(US9469631, 42)
Show SMILES Cn1cncc1-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C24H32N4O3/c1-24(2,3)31-23(30)27-13-11-20(12-14-27)28(19-9-10-19)22(29)18-7-5-17(6-8-18)21-15-25-16-26(21)4/h5-8,15-16,19-20H,9-14H2,1-4H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254646
PNG
(US9469631, 46)
Show SMILES C[C@H]1CN(CC[C@H]1N(C1CC1)C(=O)c1ccc(cc1)-c1cnco1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C24H31N3O4/c1-16-14-26(23(29)31-24(2,3)4)12-11-20(16)27(19-9-10-19)22(28)18-7-5-17(6-8-18)21-13-25-15-30-21/h5-8,13,15-16,19-20H,9-12,14H2,1-4H3/t16-,20+/m0/s1
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254657
PNG
(US9469631, 58)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1cccs1
Show InChI InChI=1S/C24H30N2O3S/c1-24(2,3)29-23(28)25-14-12-20(13-15-25)26(19-10-11-19)22(27)18-8-6-17(7-9-18)21-5-4-16-30-21/h4-9,16,19-20H,10-15H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254622
PNG
(US9469631, 19)
Show SMILES CC1(CC1)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ccc(cn1)S(C)(=O)=O
Show InChI InChI=1S/C26H31N3O5S/c1-26(13-14-26)34-25(31)28-15-11-21(12-16-28)29(20-7-8-20)24(30)19-5-3-18(4-6-19)23-10-9-22(17-27-23)35(2,32)33/h3-6,9-10,17,20-21H,7-8,11-16H2,1-2H3
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Boehringer Ingelheim International GmbH

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Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254630
PNG
(US9469631, 27)
Show SMILES Cc1cncnc1-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C25H32N4O3/c1-17-15-26-16-27-22(17)18-5-7-19(8-6-18)23(30)29(20-9-10-20)21-11-13-28(14-12-21)24(31)32-25(2,3)4/h5-8,15-16,20-21H,9-14H2,1-4H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254634
PNG
(US9469631, 31)
Show SMILES CC(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ccncc1C#N
Show InChI InChI=1S/C25H28N4O3/c1-17(2)32-25(31)28-13-10-22(11-14-28)29(21-7-8-21)24(30)19-5-3-18(4-6-19)23-9-12-27-16-20(23)15-26/h3-6,9,12,16-17,21-22H,7-8,10-11,13-14H2,1-2H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254638
PNG
(US9469631, 35)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1F)-c1cnco1
Show InChI InChI=1S/C23H28FN3O4/c1-23(2,3)31-22(29)26-10-8-17(9-11-26)27(16-5-6-16)21(28)18-7-4-15(12-19(18)24)20-13-25-14-30-20/h4,7,12-14,16-17H,5-6,8-11H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254643
PNG
(US9469631, 43)
Show SMILES Cc1ncc(o1)-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C24H31N3O4/c1-16-25-15-21(30-16)17-5-7-18(8-6-17)22(28)27(19-9-10-19)20-11-13-26(14-12-20)23(29)31-24(2,3)4/h5-8,15,19-20H,9-14H2,1-4H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254654
PNG
(US9469631, 55)
Show SMILES Cc1cn(c(C)n1)-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C25H34N4O3/c1-17-16-28(18(2)26-17)20-8-6-19(7-9-20)23(30)29(21-10-11-21)22-12-14-27(15-13-22)24(31)32-25(3,4)5/h6-9,16,21-22H,10-15H2,1-5H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254686
PNG
(US9469631, 87)
Show SMILES CCOc1ccc(cc1)-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C28H36N2O4/c1-5-33-25-14-10-21(11-15-25)20-6-8-22(9-7-20)26(31)30(23-12-13-23)24-16-18-29(19-17-24)27(32)34-28(2,3)4/h6-11,14-15,23-24H,5,12-13,16-19H2,1-4H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254694
PNG
(US9469631, 95)
Show SMILES Cc1noc(C)c1-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C25H33N3O4/c1-16-22(17(2)32-26-16)18-6-8-19(9-7-18)23(29)28(20-10-11-20)21-12-14-27(15-13-21)24(30)31-25(3,4)5/h6-9,20-21H,10-15H2,1-5H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254623
PNG
(US9469631, 20)
Show SMILES CC1(CC1)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1cnco1
Show InChI InChI=1S/C23H27N3O4/c1-23(10-11-23)30-22(28)25-12-8-19(9-13-25)26(18-6-7-18)21(27)17-4-2-16(3-5-17)20-14-24-15-29-20/h2-5,14-15,18-19H,6-13H2,1H3
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Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254675
PNG
(US9469631, 76)
Show SMILES CN(C)C(=O)Nc1nnc(s1)-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C25H34N6O4S/c1-25(2,3)35-24(34)30-14-12-19(13-15-30)31(18-10-11-18)21(32)17-8-6-16(7-9-17)20-27-28-22(36-20)26-23(33)29(4)5/h6-9,18-19H,10-15H2,1-5H3,(H,26,28,33)
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254624
PNG
(US9469631, 21)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ccc(cn1)S(C)(=O)=O
Show InChI InChI=1S/C26H33N3O5S/c1-26(2,3)34-25(31)28-15-13-21(14-16-28)29(20-9-10-20)24(30)19-7-5-18(6-8-19)23-12-11-22(17-27-23)35(4,32)33/h5-8,11-12,17,20-21H,9-10,13-16H2,1-4H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254632
PNG
(US9469631, 29)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ccncc1C#N
Show InChI InChI=1S/C26H30N4O3/c1-26(2,3)33-25(32)29-14-11-22(12-15-29)30(21-8-9-21)24(31)19-6-4-18(5-7-19)23-10-13-28-17-20(23)16-27/h4-7,10,13,17,21-22H,8-9,11-12,14-15H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254652
PNG
(US9469631, 53)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1cnco1
Show InChI InChI=1S/C23H29N3O4/c1-23(2,3)30-22(28)25-12-10-19(11-13-25)26(18-8-9-18)21(27)17-6-4-16(5-7-17)20-14-24-15-29-20/h4-7,14-15,18-19H,8-13H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254668
PNG
(US9469631, 69)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1cncnc1
Show InChI InChI=1S/C24H30N4O3/c1-24(2,3)31-23(30)27-12-10-21(11-13-27)28(20-8-9-20)22(29)18-6-4-17(5-7-18)19-14-25-16-26-15-19/h4-7,14-16,20-21H,8-13H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254688
PNG
(US9469631, 89)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ccc(s1)C#N
Show InChI InChI=1S/C25H29N3O3S/c1-25(2,3)31-24(30)27-14-12-20(13-15-27)28(19-8-9-19)23(29)18-6-4-17(5-7-18)22-11-10-21(16-26)32-22/h4-7,10-11,19-20H,8-9,12-15H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254697
PNG
(US9469631, 98)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ccc(CO)cc1
Show InChI InChI=1S/C27H34N2O4/c1-27(2,3)33-26(32)28-16-14-24(15-17-28)29(23-12-13-23)25(31)22-10-8-21(9-11-22)20-6-4-19(18-30)5-7-20/h4-11,23-24,30H,12-18H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254717
PNG
(US9469631, 118)
Show SMILES CC(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1cnco1
Show InChI InChI=1S/C22H27N3O4/c1-15(2)29-22(27)24-11-9-19(10-12-24)25(18-7-8-18)21(26)17-5-3-16(4-6-17)20-13-23-14-28-20/h3-6,13-15,18-19H,7-12H2,1-2H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254725
PNG
(US9469631, 126)
Show SMILES O=C(OCc1ccccc1)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1cnco1
Show InChI InChI=1S/C26H27N3O4/c30-25(21-8-6-20(7-9-21)24-16-27-18-33-24)29(22-10-11-22)23-12-14-28(15-13-23)26(31)32-17-19-4-2-1-3-5-19/h1-9,16,18,22-23H,10-15,17H2
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254618
PNG
(US9469631, 15)
Show SMILES CC(C)(O)COC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1cnco1
Show InChI InChI=1S/C23H29N3O5/c1-23(2,29)14-30-22(28)25-11-9-19(10-12-25)26(18-7-8-18)21(27)17-5-3-16(4-6-17)20-13-24-15-31-20/h3-6,13,15,18-19,29H,7-12,14H2,1-2H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254674
PNG
(US9469631, 75)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1cccnc1
Show InChI InChI=1S/C25H31N3O3/c1-25(2,3)31-24(30)27-15-12-22(13-16-27)28(21-10-11-21)23(29)19-8-6-18(7-9-19)20-5-4-14-26-17-20/h4-9,14,17,21-22H,10-13,15-16H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254726
PNG
(US9469631, 127)
Show SMILES C=CCOC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1cnco1
Show InChI InChI=1S/C22H25N3O4/c1-2-13-28-22(27)24-11-9-19(10-12-24)25(18-7-8-18)21(26)17-5-3-16(4-6-17)20-14-23-15-29-20/h2-6,14-15,18-19H,1,7-13H2
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254667
PNG
(US9469631, 68)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1noc(Cc2ccccc2)n1
Show InChI InChI=1S/C29H34N4O4/c1-29(2,3)36-28(35)32-17-15-24(16-18-32)33(23-13-14-23)27(34)22-11-9-21(10-12-22)26-30-25(37-31-26)19-20-7-5-4-6-8-20/h4-12,23-24H,13-19H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254679
PNG
(US9469631, 80)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ccsc1
Show InChI InChI=1S/C24H30N2O3S/c1-24(2,3)29-23(28)25-13-10-21(11-14-25)26(20-8-9-20)22(27)18-6-4-17(5-7-18)19-12-15-30-16-19/h4-7,12,15-16,20-21H,8-11,13-14H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254719
PNG
(US9469631, 120)
Show SMILES COc1ccc(OC(=O)N2CCC(CC2)N(C2CC2)C(=O)c2ccc(cc2)-c2cnco2)cc1
Show InChI InChI=1S/C26H27N3O5/c1-32-22-8-10-23(11-9-22)34-26(31)28-14-12-21(13-15-28)29(20-6-7-20)25(30)19-4-2-18(3-5-19)24-16-27-17-33-24/h2-5,8-11,16-17,20-21H,6-7,12-15H2,1H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254656
PNG
(US9469631, 57)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ccno1
Show InChI InChI=1S/C23H29N3O4/c1-23(2,3)29-22(28)25-14-11-19(12-15-25)26(18-8-9-18)21(27)17-6-4-16(5-7-17)20-10-13-24-30-20/h4-7,10,13,18-19H,8-9,11-12,14-15H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254672
PNG
(US9469631, 73)
Show SMILES CNC(=O)Nc1nc(ns1)-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C24H32N6O4S/c1-24(2,3)34-23(33)29-13-11-18(12-14-29)30(17-9-10-17)20(31)16-7-5-15(6-8-16)19-26-22(35-28-19)27-21(32)25-4/h5-8,17-18H,9-14H2,1-4H3,(H2,25,26,27,28,32)
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254700
PNG
(US9469631, 101)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ccc(cc1)N1CCOCC1
Show InChI InChI=1S/C30H39N3O4/c1-30(2,3)37-29(35)32-16-14-27(15-17-32)33(26-12-13-26)28(34)24-6-4-22(5-7-24)23-8-10-25(11-9-23)31-18-20-36-21-19-31/h4-11,26-27H,12-21H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254708
PNG
(US9469631, 109)
Show SMILES CCOc1ccc(cn1)-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C27H35N3O4/c1-5-33-24-13-10-21(18-28-24)19-6-8-20(9-7-19)25(31)30(22-11-12-22)23-14-16-29(17-15-23)26(32)34-27(2,3)4/h6-10,13,18,22-23H,5,11-12,14-17H2,1-4H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254720
PNG
(US9469631, 121)
Show SMILES CC(C)(C)COC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1cnco1
Show InChI InChI=1S/C24H31N3O4/c1-24(2,3)15-30-23(29)26-12-10-20(11-13-26)27(19-8-9-19)22(28)18-6-4-17(5-7-18)21-14-25-16-31-21/h4-7,14,16,19-20H,8-13,15H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254637
PNG
(US9469631, 34)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(c(F)c1)-c1ccncc1C#N
Show InChI InChI=1S/C26H29FN4O3/c1-26(2,3)34-25(33)30-12-9-20(10-13-30)31(19-5-6-19)24(32)17-4-7-22(23(27)14-17)21-8-11-29-16-18(21)15-28/h4,7-8,11,14,16,19-20H,5-6,9-10,12-13H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254732
PNG
(US9469631, 38)
Show SMILES CC(C)(C)OC(=O)N1CC[C@@H]([C@@H](F)C1)N(C1CC1)C(=O)c1ccc(cc1)-c1cnco1
Show InChI InChI=1S/C23H28FN3O4/c1-23(2,3)31-22(29)26-11-10-19(18(24)13-26)27(17-8-9-17)21(28)16-6-4-15(5-7-16)20-12-25-14-30-20/h4-7,12,14,17-19H,8-11,13H2,1-3H3/t18-,19-/m0/s1
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254677
PNG
(US9469631, 78)
Show SMILES CCOC(=O)c1cnn(c1C)-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C27H36N4O5/c1-6-35-25(33)23-17-28-31(18(23)2)22-9-7-19(8-10-22)24(32)30(20-11-12-20)21-13-15-29(16-14-21)26(34)36-27(3,4)5/h7-10,17,20-21H,6,11-16H2,1-5H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254681
PNG
(US9469631, 82)
Show SMILES CNC(=O)Nc1nnc(s1)-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C24H32N6O4S/c1-24(2,3)34-23(33)29-13-11-18(12-14-29)30(17-9-10-17)20(31)16-7-5-15(6-8-16)19-27-28-22(35-19)26-21(32)25-4/h5-8,17-18H,9-14H2,1-4H3,(H2,25,26,28,32)
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254689
PNG
(US9469631, 90)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ccoc1
Show InChI InChI=1S/C24H30N2O4/c1-24(2,3)30-23(28)25-13-10-21(11-14-25)26(20-8-9-20)22(27)18-6-4-17(5-7-18)19-12-15-29-16-19/h4-7,12,15-16,20-21H,8-11,13-14H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254713
PNG
(US9469631, 114)
Show SMILES CN(C)c1ccc(cn1)-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C27H36N4O3/c1-27(2,3)34-26(33)30-16-14-23(15-17-30)31(22-11-12-22)25(32)20-8-6-19(7-9-20)21-10-13-24(28-18-21)29(4)5/h6-10,13,18,22-23H,11-12,14-17H2,1-5H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254658
PNG
(US9469631, 59)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1nccs1
Show InChI InChI=1S/C23H29N3O3S/c1-23(2,3)29-22(28)25-13-10-19(11-14-25)26(18-8-9-18)21(27)17-6-4-16(5-7-17)20-24-12-15-30-20/h4-7,12,15,18-19H,8-11,13-14H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254662
PNG
(US9469631, 63)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-n1cncn1
Show InChI InChI=1S/C22H29N5O3/c1-22(2,3)30-21(29)25-12-10-19(11-13-25)27(18-8-9-18)20(28)16-4-6-17(7-5-16)26-15-23-14-24-26/h4-7,14-15,18-19H,8-13H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254670
PNG
(US9469631, 71)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-n1cccn1
Show InChI InChI=1S/C23H30N4O3/c1-23(2,3)30-22(29)25-15-11-20(12-16-25)27(19-9-10-19)21(28)17-5-7-18(8-6-17)26-14-4-13-24-26/h4-8,13-14,19-20H,9-12,15-16H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254702
PNG
(US9469631, 103)
Show SMILES CCNC(=O)c1ccc(cc1)-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C29H37N3O4/c1-5-30-26(33)22-10-6-20(7-11-22)21-8-12-23(13-9-21)27(34)32(24-14-15-24)25-16-18-31(19-17-25)28(35)36-29(2,3)4/h6-13,24-25H,5,14-19H2,1-4H3,(H,30,33)
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254718
PNG
(US9469631, 119)
Show SMILES Fc1ccc(OC(=O)N2CCC(CC2)N(C2CC2)C(=O)c2ccc(cc2)-c2cnco2)cc1
Show InChI InChI=1S/C25H24FN3O4/c26-19-5-9-22(10-6-19)33-25(31)28-13-11-21(12-14-28)29(20-7-8-20)24(30)18-3-1-17(2-4-18)23-15-27-16-32-23/h1-6,9-10,15-16,20-21H,7-8,11-14H2
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254619
PNG
(US9469631, 16)
Show SMILES Cc1ccc(nn1)-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C25H32N4O3/c1-17-5-12-22(27-26-17)18-6-8-19(9-7-18)23(30)29(20-10-11-20)21-13-15-28(16-14-21)24(31)32-25(2,3)4/h5-9,12,20-21H,10-11,13-16H2,1-4H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254730
PNG
(US9469631, 40)
Show SMILES CC(C)(C)OC(=O)N1CC[C@@H]([C@H](F)C1)N(C1CC1)C(=O)c1ccc(cc1)-c1cnco1
Show InChI InChI=1S/C23H28FN3O4/c1-23(2,3)31-22(29)26-11-10-19(18(24)13-26)27(17-8-9-17)21(28)16-6-4-15(5-7-16)20-12-25-14-30-20/h4-7,12,14,17-19H,8-11,13H2,1-3H3/t18-,19+/m1/s1
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254687
PNG
(US9469631, 88)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ccc(OC(F)(F)F)cc1
Show InChI InChI=1S/C27H31F3N2O4/c1-26(2,3)36-25(34)31-16-14-22(15-17-31)32(21-10-11-21)24(33)20-6-4-18(5-7-20)19-8-12-23(13-9-19)35-27(28,29)30/h4-9,12-13,21-22H,10-11,14-17H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254723
PNG
(US9469631, 124)
Show SMILES O=C(Oc1ccccc1)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1cnco1
Show InChI InChI=1S/C25H25N3O4/c29-24(19-8-6-18(7-9-19)23-16-26-17-31-23)28(20-10-11-20)21-12-14-27(15-13-21)25(30)32-22-4-2-1-3-5-22/h1-9,16-17,20-21H,10-15H2
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254648
PNG
(US9469631, 49)
Show SMILES CC(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(c(F)c1)-n1cncn1
Show InChI InChI=1S/C21H26FN5O3/c1-14(2)30-21(29)25-9-7-17(8-10-25)27(16-4-5-16)20(28)15-3-6-19(18(22)11-15)26-13-23-12-24-26/h3,6,11-14,16-17H,4-5,7-10H2,1-2H3
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Quantitative detection of cAMP accumulation from cells expressing human GPR119 receptor is achieved using Perkin Elmer's LANCE cAMP-384 Kit (Cat#AD02...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254645
PNG
(US9469631, 45)
Show SMILES COC1CN(CCC1N(C1CC1)C(=O)c1ccc(cc1)-c1cnco1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C24H31N3O5/c1-24(2,3)32-23(29)26-12-11-19(21(14-26)30-4)27(18-9-10-18)22(28)17-7-5-16(6-8-17)20-13-25-15-31-20/h5-8,13,15,18-19,21H,9-12,14H2,1-4H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254680
PNG
(US9469631, 81)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(c(Cl)c1)-n1cnc(c1)-c1ccccc1
Show InChI InChI=1S/C29H33ClN4O3/c1-29(2,3)37-28(36)32-15-13-23(14-16-32)34(22-10-11-22)27(35)21-9-12-26(24(30)17-21)33-18-25(31-19-33)20-7-5-4-6-8-20/h4-9,12,17-19,22-23H,10-11,13-16H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254684
PNG
(US9469631, 85)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-n1cnc(c1)-c1ccncn1
Show InChI InChI=1S/C27H32N6O3/c1-27(2,3)36-26(35)31-14-11-22(12-15-31)33(21-8-9-21)25(34)19-4-6-20(7-5-19)32-16-24(30-18-32)23-10-13-28-17-29-23/h4-7,10,13,16-18,21-22H,8-9,11-12,14-15H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254724
PNG
(US9469631, 125)
Show SMILES CC(C)COC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1cnco1
Show InChI InChI=1S/C23H29N3O4/c1-16(2)14-29-23(28)25-11-9-20(10-12-25)26(19-7-8-19)22(27)18-5-3-17(4-6-18)21-13-24-15-30-21/h3-6,13,15-16,19-20H,7-12,14H2,1-2H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254605
PNG
(US9469631, 2)
Show SMILES CC1CN(CCC1N(C1CC1)C(=O)c1ccc(cc1)-c1cnco1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C24H31N3O4/c1-16-14-26(23(29)31-24(2,3)4)12-11-20(16)27(19-9-10-19)22(28)18-7-5-17(6-8-18)21-13-25-15-30-21/h5-8,13,15-16,19-20H,9-12,14H2,1-4H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254609
PNG
(US9469631, 6)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1cncs1
Show InChI InChI=1S/C23H29N3O3S/c1-23(2,3)29-22(28)25-12-10-19(11-13-25)26(18-8-9-18)21(27)17-6-4-16(5-7-17)20-14-24-15-30-20/h4-7,14-15,18-19H,8-13H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254617
PNG
(US9469631, 14)
Show SMILES O=C(OCC1CCOCC1)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1cnco1
Show InChI InChI=1S/C25H31N3O5/c29-24(20-3-1-19(2-4-20)23-15-26-17-33-23)28(21-5-6-21)22-7-11-27(12-8-22)25(30)32-16-18-9-13-31-14-10-18/h1-4,15,17-18,21-22H,5-14,16H2
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Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254669
PNG
(US9469631, 70)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ccncc1
Show InChI InChI=1S/C25H31N3O3/c1-25(2,3)31-24(30)27-16-12-22(13-17-27)28(21-8-9-21)23(29)20-6-4-18(5-7-20)19-10-14-26-15-11-19/h4-7,10-11,14-15,21-22H,8-9,12-13,16-17H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254685
PNG
(US9469631, 86)
Show SMILES COc1ccc(cc1)-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C27H34N2O4/c1-27(2,3)33-26(31)28-17-15-23(16-18-28)29(22-11-12-22)25(30)21-7-5-19(6-8-21)20-9-13-24(32-4)14-10-20/h5-10,13-14,22-23H,11-12,15-18H2,1-4H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254705
PNG
(US9469631, 106)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ccc(C#N)c(F)c1
Show InChI InChI=1S/C27H30FN3O3/c1-27(2,3)34-26(33)30-14-12-23(13-15-30)31(22-10-11-22)25(32)19-6-4-18(5-7-19)20-8-9-21(17-29)24(28)16-20/h4-9,16,22-23H,10-15H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254606
PNG
(US9469631, 3)
Show SMILES CC(=C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1cnco1
Show InChI InChI=1S/C22H25N3O4/c1-15(2)29-22(27)24-11-9-19(10-12-24)25(18-7-8-18)21(26)17-5-3-16(4-6-17)20-13-23-14-28-20/h3-6,13-14,18-19H,1,7-12H2,2H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254626
PNG
(US9469631, 23)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ccnnc1
Show InChI InChI=1S/C24H30N4O3/c1-24(2,3)31-23(30)27-14-11-21(12-15-27)28(20-8-9-20)22(29)18-6-4-17(5-7-18)19-10-13-25-26-16-19/h4-7,10,13,16,20-21H,8-9,11-12,14-15H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254678
PNG
(US9469631, 79)
Show SMILES CCOC(=O)c1c(C)nn(c1C)-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C28H38N4O5/c1-7-36-26(34)24-18(2)29-32(19(24)3)23-10-8-20(9-11-23)25(33)31(21-12-13-21)22-14-16-30(17-15-22)27(35)37-28(4,5)6/h8-11,21-22H,7,12-17H2,1-6H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254682
PNG
(US9469631, 83)
Show SMILES Cc1c(ncn1-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C)-c1ccccc1
Show InChI InChI=1S/C30H36N4O3/c1-21-27(22-8-6-5-7-9-22)31-20-33(21)24-12-10-23(11-13-24)28(35)34(25-14-15-25)26-16-18-32(19-17-26)29(36)37-30(2,3)4/h5-13,20,25-26H,14-19H2,1-4H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254690
PNG
(US9469631, 91)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ccc(CC#N)cc1
Show InChI InChI=1S/C28H33N3O3/c1-28(2,3)34-27(33)30-18-15-25(16-19-30)31(24-12-13-24)26(32)23-10-8-22(9-11-23)21-6-4-20(5-7-21)14-17-29/h4-11,24-25H,12-16,18-19H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254698
PNG
(US9469631, 99)
Show SMILES COc1ncc(cn1)-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C25H32N4O4/c1-25(2,3)33-24(31)28-13-11-21(12-14-28)29(20-9-10-20)22(30)18-7-5-17(6-8-18)19-15-26-23(32-4)27-16-19/h5-8,15-16,20-21H,9-14H2,1-4H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254706
PNG
(US9469631, 107)
Show SMILES COC(=O)c1ccc(cn1)-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C27H33N3O5/c1-27(2,3)35-26(33)29-15-13-22(14-16-29)30(21-10-11-21)24(31)19-7-5-18(6-8-19)20-9-12-23(28-17-20)25(32)34-4/h5-9,12,17,21-22H,10-11,13-16H2,1-4H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254644
PNG
(US9469631, 44)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1cocn1
Show InChI InChI=1S/C23H29N3O4/c1-23(2,3)30-22(28)25-12-10-19(11-13-25)26(18-8-9-18)21(27)17-6-4-16(5-7-17)20-14-29-15-24-20/h4-7,14-15,18-19H,8-13H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254663
PNG
(US9469631, 64)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-n1cccc1
Show InChI InChI=1S/C24H31N3O3/c1-24(2,3)30-23(29)26-16-12-21(13-17-26)27(20-10-11-20)22(28)18-6-8-19(9-7-18)25-14-4-5-15-25/h4-9,14-15,20-21H,10-13,16-17H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254671
PNG
(US9469631, 72)
Show SMILES CN(C)C(=O)Nc1nc(ns1)-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C25H34N6O4S/c1-25(2,3)35-24(34)30-14-12-19(13-15-30)31(18-10-11-18)21(32)17-8-6-16(7-9-17)20-26-22(36-28-20)27-23(33)29(4)5/h6-9,18-19H,10-15H2,1-5H3,(H,26,27,28,33)
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Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254608
PNG
(US9469631, 5)
Show SMILES Cc1nc(co1)-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C24H31N3O4/c1-16-25-21(15-30-16)17-5-7-18(8-6-17)22(28)27(19-9-10-19)20-11-13-26(14-12-20)23(29)31-24(2,3)4/h5-8,15,19-20H,9-14H2,1-4H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254612
PNG
(US9469631, 9)
Show SMILES COc1cc(ccc1-c1cnco1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C24H31N3O5/c1-24(2,3)32-23(29)26-11-9-18(10-12-26)27(17-6-7-17)22(28)16-5-8-19(20(13-16)30-4)21-14-25-15-31-21/h5,8,13-15,17-18H,6-7,9-12H2,1-4H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254628
PNG
(US9469631, 25)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ncon1
Show InChI InChI=1S/C22H28N4O4/c1-22(2,3)30-21(28)25-12-10-18(11-13-25)26(17-8-9-17)20(27)16-6-4-15(5-7-16)19-23-14-29-24-19/h4-7,14,17-18H,8-13H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254660
PNG
(US9469631, 61)
Show SMILES Cc1nnc(o1)-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C23H30N4O4/c1-15-24-25-20(30-15)16-5-7-17(8-6-16)21(28)27(18-9-10-18)19-11-13-26(14-12-19)22(29)31-23(2,3)4/h5-8,18-19H,9-14H2,1-4H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254664
PNG
(US9469631, 65)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ccco1
Show InChI InChI=1S/C24H30N2O4/c1-24(2,3)30-23(28)25-14-12-20(13-15-25)26(19-10-11-19)22(27)18-8-6-17(7-9-18)21-5-4-16-29-21/h4-9,16,19-20H,10-15H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254692
PNG
(US9469631, 93)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ccc(cc1)S(C)(=O)=O
Show InChI InChI=1S/C27H34N2O5S/c1-27(2,3)34-26(31)28-17-15-23(16-18-28)29(22-11-12-22)25(30)21-7-5-19(6-8-21)20-9-13-24(14-10-20)35(4,32)33/h5-10,13-14,22-23H,11-12,15-18H2,1-4H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254701
PNG
(US9469631, 102)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ccc(cc1)C(N)=O
Show InChI InChI=1S/C27H33N3O4/c1-27(2,3)34-26(33)29-16-14-23(15-17-29)30(22-12-13-22)25(32)21-10-6-19(7-11-21)18-4-8-20(9-5-18)24(28)31/h4-11,22-23H,12-17H2,1-3H3,(H2,28,31)
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254610
PNG
(US9469631, 7)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(-c2cnco2)c(c1)[N+]([O-])=O
Show InChI InChI=1S/C23H28N4O6/c1-23(2,3)33-22(29)25-10-8-17(9-11-25)26(16-5-6-16)21(28)15-4-7-18(19(12-15)27(30)31)20-13-24-14-32-20/h4,7,12-14,16-17H,5-6,8-11H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254731
PNG
(US9469631, 39)
Show SMILES CC(C)(C)OC(=O)N1CC[C@H]([C@H](F)C1)N(C1CC1)C(=O)c1ccc(cc1)-c1cnco1
Show InChI InChI=1S/C23H28FN3O4/c1-23(2,3)31-22(29)26-11-10-19(18(24)13-26)27(17-8-9-17)21(28)16-6-4-15(5-7-16)20-12-25-14-30-20/h4-7,12,14,17-19H,8-11,13H2,1-3H3/t18-,19-/m1/s1
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254714
PNG
(US9469631, 115)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ccc(nc1)C(O)=O
Show InChI InChI=1S/C26H31N3O5/c1-26(2,3)34-25(33)28-14-12-21(13-15-28)29(20-9-10-20)23(30)18-6-4-17(5-7-18)19-8-11-22(24(31)32)27-16-19/h4-8,11,16,20-21H,9-10,12-15H2,1-3H3,(H,31,32)
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n/an/an/an/a 1.09E+3n/an/an/an/a



Boehringer Ingelheim International GmbH

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Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254607
PNG
(US9469631, 4)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ocnc1I
Show InChI InChI=1S/C23H28IN3O4/c1-23(2,3)31-22(29)26-12-10-18(11-13-26)27(17-8-9-17)21(28)16-6-4-15(5-7-16)19-20(24)25-14-30-19/h4-7,14,17-18H,8-13H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254631
PNG
(US9469631, 28)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(-c2cnco2)c(F)c1
Show InChI InChI=1S/C23H28FN3O4/c1-23(2,3)31-22(29)26-10-8-17(9-11-26)27(16-5-6-16)21(28)15-4-7-18(19(24)12-15)20-13-25-14-30-20/h4,7,12-14,16-17H,5-6,8-11H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254635
PNG
(US9469631, 32)
Show SMILES CC1(CC1)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ccncc1C#N
Show InChI InChI=1S/C26H28N4O3/c1-26(11-12-26)33-25(32)29-14-9-22(10-15-29)30(21-6-7-21)24(31)19-4-2-18(3-5-19)23-8-13-28-17-20(23)16-27/h2-5,8,13,17,21-22H,6-7,9-12,14-15H2,1H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254639
PNG
(US9469631, 36)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1c(F)cc(cc1F)-c1cnco1
Show InChI InChI=1S/C23H27F2N3O4/c1-23(2,3)32-22(30)27-8-6-16(7-9-27)28(15-4-5-15)21(29)20-17(24)10-14(11-18(20)25)19-12-26-13-31-19/h10-13,15-16H,4-9H2,1-3H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254683
PNG
(US9469631, 84)
Show SMILES Cc1nc(cn1-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C)-c1ccccc1
Show InChI InChI=1S/C30H36N4O3/c1-21-31-27(22-8-6-5-7-9-22)20-33(21)24-12-10-23(11-13-24)28(35)34(25-14-15-25)26-16-18-32(19-17-26)29(36)37-30(2,3)4/h5-13,20,25-26H,14-19H2,1-4H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254691
PNG
(US9469631, 92)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ccc(NS(C)(=O)=O)cc1
Show InChI InChI=1S/C27H35N3O5S/c1-27(2,3)35-26(32)29-17-15-24(16-18-29)30(23-13-14-23)25(31)21-7-5-19(6-8-21)20-9-11-22(12-10-20)28-36(4,33)34/h5-12,23-24,28H,13-18H2,1-4H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254715
PNG
(US9469631, 116)
Show SMILES COC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1cnco1
Show InChI InChI=1S/C20H23N3O4/c1-26-20(25)22-10-8-17(9-11-22)23(16-6-7-16)19(24)15-4-2-14(3-5-15)18-12-21-13-27-18/h2-5,12-13,16-17H,6-11H2,1H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254649
PNG
(US9469631, 50)
Show SMILES CC(C)OC(=O)N1CC[C@H]([C@@H](F)C1)N(C1CC1)C(=O)c1ccc(c(F)c1)-n1cncn1
Show InChI InChI=1S/C21H25F2N5O3/c1-13(2)31-21(30)26-8-7-19(17(23)10-26)28(15-4-5-15)20(29)14-3-6-18(16(22)9-14)27-12-24-11-25-27/h3,6,9,11-13,15,17,19H,4-5,7-8,10H2,1-2H3/t17-,19+/m0/s1
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n/an/an/an/a 1.02E+3n/an/an/an/a



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Assay Description
Quantitative detection of cAMP accumulation from cells expressing human GPR119 receptor is achieved using Perkin Elmer's LANCE cAMP-384 Kit (Cat#AD02...


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More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254650
PNG
(US9469631, 51)
Show SMILES CC(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-n1ccnc1C
Show InChI InChI=1S/C23H30N4O3/c1-16(2)30-23(29)25-13-10-21(11-14-25)27(20-8-9-20)22(28)18-4-6-19(7-5-18)26-15-12-24-17(26)3/h4-7,12,15-16,20-21H,8-11,13-14H2,1-3H3
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Assay Description
Quantitative detection of cAMP accumulation from cells expressing human GPR119 receptor is achieved using Perkin Elmer's LANCE cAMP-384 Kit (Cat#AD02...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254647
PNG
(US9469631, 48)
Show SMILES CC(C)OC(=O)N1CC[C@@H]([C@H](F)C1)N(C1CC1)C(=O)c1ccc(c(F)c1)-n1cncn1
Show InChI InChI=1S/C21H25F2N5O3/c1-13(2)31-21(30)26-8-7-19(17(23)10-26)28(15-4-5-15)20(29)14-3-6-18(16(22)9-14)27-12-24-11-25-27/h3,6,9,11-13,15,17,19H,4-5,7-8,10H2,1-2H3/t17-,19+/m1/s1
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Assay Description
Quantitative detection of cAMP accumulation from cells expressing human GPR119 receptor is achieved using Perkin Elmer's LANCE cAMP-384 Kit (Cat#AD02...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254641
PNG
(US9469631, 41)
Show SMILES CC(C)(C)OC(=O)N1CC[C@H]([C@@H](F)C1)N(C1CC1)C(=O)c1ccc(cc1)-c1cnco1
Show InChI InChI=1S/C23H28FN3O4/c1-23(2,3)31-22(29)26-11-10-19(18(24)13-26)27(17-8-9-17)21(28)16-6-4-15(5-7-16)20-12-25-14-30-20/h4-7,12,14,17-19H,8-11,13H2,1-3H3/t18-,19+/m0/s1
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254633
PNG
(US9469631, 30)
Show SMILES CNC(=O)c1ccc(nc1)-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C27H34N4O4/c1-27(2,3)35-26(34)30-15-13-22(14-16-30)31(21-10-11-21)25(33)19-7-5-18(6-8-19)23-12-9-20(17-29-23)24(32)28-4/h5-9,12,17,21-22H,10-11,13-16H2,1-4H3,(H,28,32)
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Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254709
PNG
(US9469631, 110)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ccc(cc1F)S(C)(=O)=O
Show InChI InChI=1S/C27H33FN2O5S/c1-27(2,3)35-26(32)29-15-13-21(14-16-29)30(20-9-10-20)25(31)19-7-5-18(6-8-19)23-12-11-22(17-24(23)28)36(4,33)34/h5-8,11-12,17,20-21H,9-10,13-16H2,1-4H3
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MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254733
PNG
(US9469631, 47)
Show SMILES C[C@@H]1CN(CC[C@@H]1N(C1CC1)C(=O)c1ccc(cc1)-c1cnco1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C24H31N3O4/c1-16-14-26(23(29)31-24(2,3)4)12-11-20(16)27(19-9-10-19)22(28)18-7-5-17(6-8-18)21-13-25-15-30-21/h5-8,13,15-16,19-20H,9-12,14H2,1-4H3/t16-,20+/m1/s1
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Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254666
PNG
(US9469631, 67)
Show SMILES Cc1nc(no1)-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C23H30N4O4/c1-15-24-20(25-31-15)16-5-7-17(8-6-16)21(28)27(18-9-10-18)19-11-13-26(14-12-19)22(29)30-23(2,3)4/h5-8,18-19H,9-14H2,1-4H3
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Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254627
PNG
(US9469631, 24)
Show SMILES Cc1cc(ccc1-c1cnco1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C24H31N3O4/c1-16-13-17(5-8-20(16)21-14-25-15-30-21)22(28)27(18-6-7-18)19-9-11-26(12-10-19)23(29)31-24(2,3)4/h5,8,13-15,18-19H,6-7,9-12H2,1-4H3
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Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254651
PNG
(US9469631, 52)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-n1ccnc1
Show InChI InChI=1S/C23H30N4O3/c1-23(2,3)30-22(29)25-13-10-20(11-14-25)27(19-8-9-19)21(28)17-4-6-18(7-5-17)26-15-12-24-16-26/h4-7,12,15-16,19-20H,8-11,13-14H2,1-3H3
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Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254699
PNG
(US9469631, 100)
Show SMILES CC(C)(C)OC(=O)N1CCC(CC1)N(C1CC1)C(=O)c1ccc(cc1)-c1ccc(nc1)C#N
Show InChI InChI=1S/C26H30N4O3/c1-26(2,3)33-25(32)29-14-12-23(13-15-29)30(22-10-11-22)24(31)19-6-4-18(5-7-19)20-8-9-21(16-27)28-17-20/h4-9,17,22-23H,10-15H2,1-3H3
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Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


Citation and Details
More data for this
Ligand-Target Pair
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM254711
PNG
(US9469631, 112)
Show SMILES CN(C)Cc1ccc(cc1)-c1ccc(cc1)C(=O)N(C1CC1)C1CCN(CC1)C(=O)OC(C)(C)C
Show InChI InChI=1S/C29H39N3O3/c1-29(2,3)35-28(34)31-18-16-26(17-19-31)32(25-14-15-25)27(33)24-12-10-23(11-13-24)22-8-6-21(7-9-22)20-30(4)5/h6-13,25-26H,14-20H2,1-5H3
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n/an/an/an/a 1.74E+3n/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] are stably transfected with an expression vector for human GPR119 cDNA (Acc. N...


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More data for this
Ligand-Target Pair
* indicates data uncertainty>20%