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Found 22 Enz. Inhib. hit(s) with all data for entry = 849
TargetAcetylcholinesterase(Homo sapiens (Human))
Nobel IlaÇ

US Patent
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  8nMAssay Description:The potential of the compounds of the present invention to inhibit acetylcholinesterase and butyrylcholinesterase enzymes were tested according to th...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Nobel IlaÇ

US Patent
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  700nMAssay Description:The potential of the compounds of the present invention to inhibit acetylcholinesterase and butyrylcholinesterase enzymes were tested according to th...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Nobel IlaÇ

US Patent
LigandPNGBDBM294221((±)-3-(1-(dimethylamino)ethyl)-1-methoxy-6H-benzo[...)
Affinity DataIC50:  2.80E+3nMAssay Description:The potential of the compounds of the present invention to inhibit acetylcholinesterase and butyrylcholinesterase enzymes were tested according to th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCholinesterase(Homo sapiens (Human))
Nobel IlaÇ

US Patent
LigandPNGBDBM294223((±)-3-(1-(dimethylamino)ethyl)-1-hydroxy-6H-benzo[...)
Affinity DataIC50:  4.20E+3nMAssay Description:The potential of the compounds of the present invention to inhibit acetylcholinesterase and butyrylcholinesterase enzymes were tested according to th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCholinesterase(Homo sapiens (Human))
Nobel IlaÇ

US Patent
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  7.10E+3nMAssay Description:The potential of the compounds of the present invention to inhibit acetylcholinesterase and butyrylcholinesterase enzymes were tested according to th...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetylcholinesterase(Homo sapiens (Human))
Nobel IlaÇ

US Patent
LigandPNGBDBM294220((S)-3-(1-(dimethylamino)ethyl)-6H-benzo[c]chromen-...)
Affinity DataIC50:  7.90E+3nMAssay Description:The potential of the compounds of the present invention to inhibit acetylcholinesterase and butyrylcholinesterase enzymes were tested according to th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCholinesterase(Homo sapiens (Human))
Nobel IlaÇ

US Patent
LigandPNGBDBM294226((±)-1-(1-(dimethylamino)ethyl)-6-oxo-6H-benzo[c]ch...)
Affinity DataIC50:  8.50E+3nMAssay Description:The potential of the compounds of the present invention to inhibit acetylcholinesterase and butyrylcholinesterase enzymes were tested according to th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAcetylcholinesterase(Homo sapiens (Human))
Nobel IlaÇ

US Patent
LigandPNGBDBM294219((±)-3-(1-(dimethylamino)ethyl)-6H-benzo[c]chromen-...)
Affinity DataIC50:  1.09E+4nMAssay Description:The potential of the compounds of the present invention to inhibit acetylcholinesterase and butyrylcholinesterase enzymes were tested according to th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCholinesterase(Homo sapiens (Human))
Nobel IlaÇ

US Patent
LigandPNGBDBM11682(2,3-dihydroxybutanedioic acid; 3-[(1S)-1-(dimethyl...)
Affinity DataIC50:  1.10E+4nMAssay Description:The potential of the compounds of the present invention to inhibit acetylcholinesterase and butyrylcholinesterase enzymes were tested according to th...More data for this Ligand-Target Pair
In DepthDetails US PatentDrugBank

TargetCholinesterase(Homo sapiens (Human))
Nobel IlaÇ

US Patent
LigandPNGBDBM294225((±)-3-(1-(dimethylamino)ethyl)-6-oxo-6H-benzo[c]ch...)
Affinity DataIC50:  1.27E+4nMAssay Description:The potential of the compounds of the present invention to inhibit acetylcholinesterase and butyrylcholinesterase enzymes were tested according to th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAcetylcholinesterase(Homo sapiens (Human))
Nobel IlaÇ

US Patent
LigandPNGBDBM294222((±)-1-(1-(dimethylamino)ethyl)-3-methoxy-6H-benzo[...)
Affinity DataIC50:  1.51E+4nMAssay Description:The potential of the compounds of the present invention to inhibit acetylcholinesterase and butyrylcholinesterase enzymes were tested according to th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCholinesterase(Homo sapiens (Human))
Nobel IlaÇ

US Patent
LigandPNGBDBM294220((S)-3-(1-(dimethylamino)ethyl)-6H-benzo[c]chromen-...)
Affinity DataIC50:  1.62E+4nMAssay Description:The potential of the compounds of the present invention to inhibit acetylcholinesterase and butyrylcholinesterase enzymes were tested according to th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCholinesterase(Homo sapiens (Human))
Nobel IlaÇ

US Patent
LigandPNGBDBM294219((±)-3-(1-(dimethylamino)ethyl)-6H-benzo[c]chromen-...)
Affinity DataIC50:  1.79E+4nMAssay Description:The potential of the compounds of the present invention to inhibit acetylcholinesterase and butyrylcholinesterase enzymes were tested according to th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAcetylcholinesterase(Homo sapiens (Human))
Nobel IlaÇ

US Patent
LigandPNGBDBM294223((±)-3-(1-(dimethylamino)ethyl)-1-hydroxy-6H-benzo[...)
Affinity DataIC50:  1.89E+4nMAssay Description:The potential of the compounds of the present invention to inhibit acetylcholinesterase and butyrylcholinesterase enzymes were tested according to th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCholinesterase(Homo sapiens (Human))
Nobel IlaÇ

US Patent
LigandPNGBDBM294221((±)-3-(1-(dimethylamino)ethyl)-1-methoxy-6H-benzo[...)
Affinity DataIC50:  2.11E+4nMAssay Description:The potential of the compounds of the present invention to inhibit acetylcholinesterase and butyrylcholinesterase enzymes were tested according to th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCholinesterase(Homo sapiens (Human))
Nobel IlaÇ

US Patent
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  2.19E+4nMAssay Description:The potential of the compounds of the present invention to inhibit acetylcholinesterase and butyrylcholinesterase enzymes were tested according to th...More data for this Ligand-Target Pair
In DepthDetails US PatentDrugBank

TargetCholinesterase(Homo sapiens (Human))
Nobel IlaÇ

US Patent
LigandPNGBDBM294222((±)-1-(1-(dimethylamino)ethyl)-3-methoxy-6H-benzo[...)
Affinity DataIC50:  2.47E+4nMAssay Description:The potential of the compounds of the present invention to inhibit acetylcholinesterase and butyrylcholinesterase enzymes were tested according to th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAcetylcholinesterase(Homo sapiens (Human))
Nobel IlaÇ

US Patent
LigandPNGBDBM294224((±)-1-(1-(dimethylamino)ethyl)-3-hydroxy-6H-benzo[...)
Affinity DataIC50:  3.31E+4nMAssay Description:The potential of the compounds of the present invention to inhibit acetylcholinesterase and butyrylcholinesterase enzymes were tested according to th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAcetylcholinesterase(Homo sapiens (Human))
Nobel IlaÇ

US Patent
LigandPNGBDBM11682(2,3-dihydroxybutanedioic acid; 3-[(1S)-1-(dimethyl...)
Affinity DataIC50:  3.52E+4nMAssay Description:The potential of the compounds of the present invention to inhibit acetylcholinesterase and butyrylcholinesterase enzymes were tested according to th...More data for this Ligand-Target Pair
In DepthDetails US PatentDrugBank

TargetAcetylcholinesterase(Homo sapiens (Human))
Nobel IlaÇ

US Patent
LigandPNGBDBM294226((±)-1-(1-(dimethylamino)ethyl)-6-oxo-6H-benzo[c]ch...)
Affinity DataIC50: >4.00E+4nMAssay Description:The potential of the compounds of the present invention to inhibit acetylcholinesterase and butyrylcholinesterase enzymes were tested according to th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAcetylcholinesterase(Homo sapiens (Human))
Nobel IlaÇ

US Patent
LigandPNGBDBM294225((±)-3-(1-(dimethylamino)ethyl)-6-oxo-6H-benzo[c]ch...)
Affinity DataIC50:  4.00E+4nMAssay Description:The potential of the compounds of the present invention to inhibit acetylcholinesterase and butyrylcholinesterase enzymes were tested according to th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCholinesterase(Homo sapiens (Human))
Nobel IlaÇ

US Patent
LigandPNGBDBM294224((±)-1-(1-(dimethylamino)ethyl)-3-hydroxy-6H-benzo[...)
Affinity DataIC50: >4.00E+4nMAssay Description:The potential of the compounds of the present invention to inhibit acetylcholinesterase and butyrylcholinesterase enzymes were tested according to th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent